IRIS
CAMPIANI, GIUSEPPE
 Distribuzione geografica
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Continente #
NA - Nord America 15.626
EU - Europa 13.827
AS - Asia 2.189
AF - Africa 77
OC - Oceania 26
SA - Sud America 24
Continente sconosciuto - Info sul continente non disponibili 13
Totale 31.782
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Nazione #
US - Stati Uniti d'America 15.562
GB - Regno Unito 4.107
IE - Irlanda 2.299
IT - Italia 1.854
CN - Cina 1.628
UA - Ucraina 1.221
SE - Svezia 1.198
DE - Germania 914
RU - Federazione Russa 797
FR - Francia 667
FI - Finlandia 395
SG - Singapore 225
TR - Turchia 157
ES - Italia 96
CA - Canada 59
CZ - Repubblica Ceca 53
CI - Costa d'Avorio 51
BE - Belgio 47
IN - India 43
AT - Austria 35
VN - Vietnam 27
GR - Grecia 26
IR - Iran 26
RO - Romania 25
NL - Olanda 24
AU - Australia 22
PT - Portogallo 13
EU - Europa 12
JP - Giappone 12
PL - Polonia 11
NG - Nigeria 9
BR - Brasile 8
EG - Egitto 8
CL - Cile 7
HU - Ungheria 7
IL - Israele 7
KR - Corea 7
SA - Arabia Saudita 7
ID - Indonesia 6
LA - Repubblica Popolare Democratica del Laos 6
LV - Lettonia 6
BG - Bulgaria 5
PK - Pakistan 5
ZA - Sudafrica 5
BD - Bangladesh 4
NO - Norvegia 4
NZ - Nuova Zelanda 4
PA - Panama 4
AZ - Azerbaigian 3
CH - Svizzera 3
DK - Danimarca 3
EE - Estonia 3
HK - Hong Kong 3
KH - Cambogia 3
KW - Kuwait 3
MA - Marocco 3
MY - Malesia 3
RS - Serbia 3
AE - Emirati Arabi Uniti 2
AL - Albania 2
BO - Bolivia 2
CO - Colombia 2
GE - Georgia 2
HR - Croazia 2
IM - Isola di Man 2
KG - Kirghizistan 2
PE - Perù 2
SK - Slovacchia (Repubblica Slovacca) 2
TH - Thailandia 2
A2 - ???statistics.table.value.countryCode.A2??? 1
AR - Argentina 1
EC - Ecuador 1
GH - Ghana 1
JM - Giamaica 1
JO - Giordania 1
KZ - Kazakistan 1
LK - Sri Lanka 1
LT - Lituania 1
MC - Monaco 1
MD - Moldavia 1
SY - Repubblica araba siriana 1
TM - Turkmenistan 1
TW - Taiwan 1
VE - Venezuela 1
Totale 31.782
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Città #
Southend 3.822
Fairfield 2.762
Dublin 2.280
Ashburn 1.466
Chandler 1.250
Woodbridge 1.196
Jacksonville 1.006
Seattle 984
Wilmington 979
Cambridge 926
Houston 909
Siena 751
Ann Arbor 654
Princeton 396
Beijing 375
Nanjing 344
Boardman 181
Dearborn 164
Fremont 156
Singapore 150
Helsinki 144
San Diego 136
Izmir 134
New York 133
Nanchang 127
Shanghai 123
Moscow 119
Florence 108
San Mateo 90
Washington 80
Menlo Park 77
Málaga 77
Shenyang 69
Hebei 68
Lappeenranta 63
Jiaxing 57
Kunming 57
Rome 55
Venezia 55
Lancaster 54
Abidjan 51
Redwood City 51
Milan 47
Düsseldorf 46
Brno 43
London 43
Tianjin 43
Brussels 42
Ningbo 41
Changsha 40
Jinan 40
Norwalk 39
Aachen 34
Guangzhou 30
Vienna 28
Ottawa 24
San Francisco 24
Dong Ket 23
Hangzhou 22
Hanover 21
Los Angeles 20
Hefei 19
Philadelphia 19
Toronto 19
Frankfurt am Main 18
Munich 17
Turin 17
Zhengzhou 17
Prato 16
Parma 15
Timisoara 15
Avellino 14
Pisa 14
Salerno 14
Taizhou 14
Marietta 12
Rende 12
San Giovanni Valdarno 12
Changchun 11
Amsterdam 10
Lanzhou 10
Leawood 10
Palermo 10
Arezzo 9
Dallas 9
Fisciano 9
Haikou 9
Lastra a Signa 9
Maletto 9
Mestre 9
Naples 9
Bologna 8
Borgo San Lorenzo 8
Catanzaro 8
Kilburn 8
Lagos 8
Palo Alto 8
Santa Clara 8
Ventimiglia 8
Bari 7
Totale 23.787
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Nome #
Development of Potent Inhibitors of the Mycobacterium tuberculosis Virulence Factor Zmp1 and Evaluation of Their Effect on Mycobacterial Survival inside Macrophages 290
Structure-activity relationships, biological evaluation and structural studies of novel pyrrolonaphthoxazepines as antitumor agents 266
Development of novel cyclic peptides as pro-apoptotic agents 264
Antimalarial agents against both sexual and asexual parasites stages: structure-activity relationships and biological studies of the Malaria Box compound 1-[5-(4-bromo-2-chlorophenyl)furan-2-yl]- N -[(piperidin-4-yl)methyl]methanamine (MMV019918) and analogues 258
(S)-2-Amino-3-(5-methyl-3-hydroxyisoxazol-4-yl)propanoic Acid (AMPA) and Kainate Receptor Ligands: further exploration of bioisosteric replacements and structural and biological investigation 252
Development and Pharmacological Characterization of Selective Blockers of 2-Arachidonoyl Glycerol Degradation with Efficacy in Rodent Models of Multiple Sclerosis and Pain 247
iPSC-derived neurons profiling reveals GABAergic circuit disruption and acetylated α-tubulin defect which improves after iHDAC6 treatment in Rett syndrome 245
Novel spiroindoline HDAC inhibitors: Synthesis, molecular modelling and biological studies 227
Synthetic spirocyclic endoperoxides: new antimalarial scaffolds 225
A new microtubule-targeting compound PBOX-15 inhibits T-cell migration via post-translational modifications of tubulin 217
The 1-(2,3-dichlorophenyl)-piperazine-to-aripiprazole ratio at steady state in rats and schizophrenic patients 217
Bridged bicyclic 2,3-dioxabicyclo[3.3.1]nonanes as antiplasmodial agents: Synthesis, structure-activity relationships and studies on their biomimetic reaction with Fe(II) 212
Development of Potent Inhibitors of Fatty Acid Amide Hydrolase Useful for the Treatment of Neuropathic Pain 210
First dual AK/GSK-3β inhibitors endowed with antioxidant properties as multifunctional, potential neuroprotective agents 210
Natural Compounds and Synthetic Drugs to Target FAAH Enzyme 209
Synthesis, Molecular Modelling and Biological Studies of 3-hydroxy-pyrane-4-one and 3-hydroxy-pyridine-4-one Derivatives as HIV-1 Integrase Inhibitors 208
Development of novel multipotent compounds modulating endocannabinoid and dopaminergic systems 208
Old but gold: tracking the new guise of Histone Deacetylase 6 (HDAC6) enzyme as a biomarker and therapeutic target in rare diseases 207
Identification of novel fluorescent probes preventing PrP(Sc) replication in prion diseases 197
Targeting Dopamine D3and Serotonin 5-HT1Aand 5-HT2AReceptors for Developing Effective Antipsychotics: Synthesis, Biological Characterization, and Behavioral Studies 196
null 195
A Jocic-type approach for a practical and scalable synthesis of pyrrolonaphthoxazepine (PNOX)-based potent proapoptotic agents 195
Structure-based discovery of the first non-covalent inhibitors of Leishmania major tryparedoxin peroxidase by high throughput docking 193
Activation of the Wnt pathway by small peptides: rational design, synthesis and biological evaluation 193
Targeting clinically-relevant metallo-β-lactamases: from high-throughput docking to broad-spectrum inhibitors 184
Discovery of a new class of potential multifunctional atypical antipsychotic agents targeting dopamine d3 and serotonin 5-HT 1A and 5-HT2A receptors: Design, synthesis, and effects on behavior 184
Selective Kainate Receptor (GluK1) Ligands Structurally Based upon 1H-Cyclopentapyrimidin-2,4(1H,3H)-dione: Synthesis, Molecular Modeling, and Pharmacological and Biostructural Characterization 183
Structural characterization of Giardia duodenalis thioredoxin reductase (gTrxR) and computational analysis of its interaction with NBDHEX 183
Cinnamic acids derived compounds with antileishmanial activity target Leishmania amazonensis arginase 180
A stereoselective route to 6-substituted pyrrolo-1,5-benzoxazepinones and their analogues 179
1H-Cyclopentapyrimidine-2,4(1H,3H)-dione-Related Ionotropic Glutamate Receptors Ligands. Structure-Activity Relationships and Identification of Potent and Selective iGluR5 Modulators 176
Optimization of 4-Aminoquinoline/Clotrimazole-Based Hybrid Antimalarials: Further Structure-Activity Relationships, in vivo Studies, and Preliminary Toxicity Profiling 173
Synthesis and structure-activity relationship studies in serotonin 5-HT4 receptor ligands based on a benzo[de][2,6]naphthridine scaffold 172
Synthetic studies toward 1,2-dioxanes as precursors of potential endoperoxide-containing antimalarials 170
Multitarget compounds bearing tacrine- and donepezil-like structural and functional motifs for the potential treatment of Alzheimer's disease 170
The FAAH inhibitor URB597 suppresses hippocampal maximal dentate afterdischarges and restores seizure-induced impairment of short and long-term synaptic plasticity 170
Pyrrolo 1,3 benzothiazepine-based Atypical Antipsychotic Agents. Synthesis, Structure-Activity Relationship, Molecular Modeling, and Biological Studies 168
Telomerase-based cancer therapeutics: a review on their clinical trials 168
Discovery of Potent Inhibitors of Human and Mouse Fatty Acid Amide Hydrolases 167
A light in the dark: State of the art and perspectives in optogenetics and optopharmacology for restoring vision 166
Non-Nucleoside Inhibitors of Human Adenosine Kinase: Synthesis, Molecular Modeling, and Biological Studies 165
Discovery of Bishomo(hetero)arylpiperazines as Novel Multifunctional Ligands Targeting Dopamine D-3 and Serotonin 5-HT1A and 5-HT2A Receptors 165
Cardiovascular Characterization of Pyrrolo[2,1-d][1,5]benzothiazepine Derivatives Binding Selectively to the Peripheral-Type Benzodiazepine Receptor (PBR):  From Dual PBR Affinity and Calcium Antagonist Activity to Novel and Selective Calcium Entry Blockers 165
Synthesis and Antiplasmodial Activity of Bicyclic Dioxanes as Simplified Dihydroplakortin Analogues 164
Novel Ligands Specific for Mitochondrial Benzodiazepine Receptors: 6-arylpyrrolo[2,1-d][1,5]benzothiazepine Derivatives. Synthesis, Structure-Activity Relationships, and Molecular Modeling Studies 164
Exploiting Protein Fluctuations at the Active-Site Gorge of Human Cholinesterases: Further Optimization of the Design Strategy to Develop Extremely Potent Inhibitors 162
Mimicking the Intramolecular Hydrogen Bond: Synthesis, Biological Evaluation, and Molecular Modeling of Benzoxazines and Quinazolines as Potential Antimalarial Agents 162
Synthesis and structure–activity relationship studies in serotonin 5-HT1A receptor agonists based on fused pyrrolidone scaffolds 162
Microwave-assisted synthesis of 4-quinolylhydrazines followed by nickel boride reduction: a convenient approach to 4-aminoquinolines and derivatives 161
The Interactions of the 5-HT3 Receptor with Quipazine-Like Arylpiperazine Ligands. The Journey Track at the End of the First Decade of the Third Millennium 161
A synthetic strategy to bridged 2,3,8-trioxabicyclo[3,3,1]nonane endoperoxides 161
Synthesis of Dihydroplakortin, 6-epi-Dihydroplakortin, and Their C10-Desethyl Analogues 161
Quinolylhydrazones as novel inhibitors of Plasmodium falciparum serine protease PfSUB1 159
A stereoselective approach to peptidomimetic BACE1 inhibitors 159
Unravelling the response of chronic lymphocytic leukemia to a novel class of anticancer agents, the pyrrolonaphthoxazepines (PNOXs) 159
Synthetic studies toward bicyclic endoperoxides presenting polar side chains 158
Design and Synthesis of Potent Antimalarial Agents Based on Clotrimazole Scaffold: Exploring an Innovative Pharmacophore 157
Pyrroloquinoxaline Derivatives as High-Affinity and Selective 5-HT3 Receptor Agonists: Synthesis, Further Structure-Activity Relationships, and Biological Studies 156
Donepezil-like multifunctional agents: Design, synthesis, molecular modeling and biological evaluation 155
Novel quinolone-based potent and selective HDAC6 inhibitors: synthesis, molecular modeling studies and biological investigation 155
Diltiazem-like calcium entry blockers: a hypothesis of the receptor-binding site based on a comparative molecular field analysis model 153
ANTIMALARIAL AGENTS HAVING POLYAROMATIC STRUCTURE 153
Endocannabinoid Modulation of Predator Stress-Induced Long-Term Anxiety in Rats 153
Dopamine D3 receptor antagonists as potential therapeutics for the treatment of neurological diseases 153
Pyrrolo[2,1-c][1,4]benzothiazines: Synthesis, Structure-Activity Relationships, Molecular Modeling Studies, and Cardiovascular Activity 152
Development of a multiplexed activity-based protein profiling assay to evaluate activity of endocannabinoid hydrolase inhibitors 152
ARYL PIPERAZINE DERIVATIVES USEFUL FOR THE TREATMENT OF NEUROPSYCHIATRY DISORDERS. 151
Novel peptidomimetics as BACE-1 inhibitors: synthesis, molecular modeling, and biological studies 150
Development of piperazine-tethered heterodimers as potent antimalarials against chloroquine-resistant P. falciparum strains. Synthesis and molecular modeling 150
Synthesis of N1-arylidene-N2-quinolyl- and N2-acrydinylhydrazones as potent antimalarial agents active against CQ-resistant P. falciparum strains 149
Development of Antitubercular Compounds Based on a 4-Quinolylhydrazone Scaffold. Further Structure-activity Relationship Studies 149
Design, synthesis, and structure-activity relationship studies of 4-quinolinyl- and 9-acrydinylhydrazones as potent antimalarial agents 148
A Concerted Study Using Binding Measurements, X-ray Structural Data, and Molecular Modeling on the Stereochemical Features Responsible for the Affinity of 6-Arylpyrrolo[2,1-d][1,5]benzothiazepines toward Mitochondrial Benzodiazepine Receptors 148
New Antipsychotic Agents with Serotonin and Dopamine Antagonist Properties Based on a Pyrrolo[2,1-b][1,3]benzothiazepine Structure 147
A Comparative Molecular Field Analysis Model for 6-Arylpyrrolo[2,1-d][1,5]benzothiazepines Binding Selectively to the Mitochondrial Benzodiazepine Receptor 147
Pyrrolobenzoxazepinone Derivatives as Non-Nucleoside HIV-1 RT Inhibitors: Further Structure-Activity Relationship Studies and Identification of More Potent Broad-Spectrum HIV-1 RT Inhibitors with Antiviral Activity 146
Raising the bar in anticancer therapy: recent advances in, and perspectives on, telomerase inhibitors 146
A palladium-catalyzed synthetic approach to new Huperzine A analogues modified at the pyridone ring 145
Quinoxalinylethylpyridylthioureas (QXPTs) as Potent Non-nucleoside HIV-1 Reverse Transcriptase (RT) Inhibitors. Further SAR Studies and Identification of a Novel Orally Bioavailable Hydrazine-Based Antiviral Agent 145
Development of molecular probes for the identification of extra interaction sites in the mid-gorge and peripheral sites of butyrylcholinesterase (BuChE). Rational design of novel, selective, and highly potent BuChE inhibitors 145
Allosteric Modulation of Ionotropic Glutamate Receptors: An Outlook on New Therapeutic Approaches To Treat Central Nervous System Disorders 144
Novel aryl piperazine derivatives with medical utility 141
Malaria chemotherapy: recent advances in drug development 141
An approach to modified heterocyclic analogues of huperzine A and isohuperzine A. Synthesis of the pyrimidone and pyrazole analogues, and their anticholinesterase activity 141
Azetidin-2-one-based small molecules as dual hHDAC6/HDAC8 inhibitors: Investigation of their mechanism of action and impact of dual inhibition profile on cell viability 141
Pyrroloquinoxaline hydrazones as fluorescent probes for amyloid fibrils 140
Multifunctional Cholinesterase and Amyloid Beta Fibrillization Modulators. Synthesis and Biological Investigation 140
Selective Fatty Acid Amide Hydrolase Inhibitors as Potential Novel Antiepileptic Agents 140
Pyrrolo[1,5]benzoxa(thia)zepines as a New Class of Potent Apoptotic Agents. Biological Studies and Identification of an Intracellular Location of Their Drug Target 139
Harnessing the role of HDAC6 in Idiopathic Pulmonary Fibrosis: design, synthesis, structural analysis, and biological evaluation of potent inhibitors 139
Specific Targeting of Hepatitis C Virus NS3 RNA Helicase. Discovery of the Potent and Selective Competitive Nucleotide-Mimicking Inhibitor QU663 136
Polycondensed heterocycles. IV. Synthesis of 1,4-Dioxo-2,3,3a,4-tetrahydro-1H-pyrrolo[2,1-c][1,4]benzothiazine 136
Identification of a novel arylpiperazine scaffold for fatty acid amide hydrolase inhibition with improved drug disposition properties 135
Discovery of Huperzine A/Tacrine Hybrids as Potent Inhibitors of Human Cholinesterases Targeting Their Mid-gorge Recognition Sites 134
Synthesis and preliminary biological evaluation of 1-aminomethyl-4-substituted-4-H-pyrrolo[2,1-C][1,4] benzothiazines, a new class of calcium antagonists 134
A Straightforward Approach for Engineering Efficacy and Selectivity at GPCRs 134
Synthesis, Biological Activity, and SARs of Pyrrolobenzoxazepine Derivatives, a New Class of Specific “Peripheral-Type” Benzodiazepine Receptor Ligands 134
Specific Targeting of Peripheral Serotonin 5-HT3 Receptors. Synthesis, Biological Investigation and Structure Activity Relationships 134
Inhibition of G1 cyclin-dependent kinase activity during growth arrest of human astrocytoma cells by the pyrrolo-1,5-benzoxazepine, PBOX-21 133
Polycondensed heterocycles. V. Synthesis of 5H,11H-Pyrrolo[2,1-c][1,4]benzothiazepine 133
Totale 17.076
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Categoria #
all - tutte 99.575
article - articoli 0
book - libri 0
conference - conferenze 0
curatela - curatele 0
other - altro 0
patent - brevetti 0
selected - selezionate 0
volume - volumi 0
Totale 99.575
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Totale Lug Ago Sett Ott Nov Dic Gen Feb Mar Apr Mag Giu
2019/20205.677 0 0 416 1.093 456 603 612 801 553 572 163 408
2020/20215.596 239 500 254 515 364 874 383 693 516 557 440 261
2021/20223.544 302 526 243 194 174 82 200 140 170 437 390 686
2022/20234.785 284 398 635 661 534 960 117 387 427 135 157 90
2023/20243.997 157 81 351 177 214 1.084 1.234 69 34 119 139 338
2024/20251.139 197 342 600 0 0 0 0 0 0 0 0 0
Totale 32.388