IRIS
BRIZZI, ANTONELLA
 Distribuzione geografica
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Continente #
EU - Europa 3.809
NA - Nord America 3.244
AS - Asia 501
AF - Africa 13
OC - Oceania 11
SA - Sud America 10
Continente sconosciuto - Info sul continente non disponibili 1
Totale 7.589
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Nazione #
US - Stati Uniti d'America 3.226
GB - Regno Unito 1.148
IT - Italia 805
IE - Irlanda 619
CN - Cina 333
SE - Svezia 293
UA - Ucraina 229
DE - Germania 190
FR - Francia 187
RU - Federazione Russa 179
FI - Finlandia 86
SG - Singapore 81
TR - Turchia 28
BE - Belgio 13
ES - Italia 13
IN - India 12
AU - Australia 11
CA - Canada 11
CI - Costa d'Avorio 10
VN - Vietnam 10
JP - Giappone 7
CL - Cile 6
CZ - Repubblica Ceca 6
PK - Pakistan 6
PL - Polonia 6
HK - Hong Kong 5
MX - Messico 5
NL - Olanda 5
SI - Slovenia 5
SK - Slovacchia (Repubblica Slovacca) 4
TW - Taiwan 4
AT - Austria 3
GR - Grecia 3
KR - Corea 3
SA - Arabia Saudita 3
CH - Svizzera 2
EE - Estonia 2
EG - Egitto 2
HU - Ungheria 2
NO - Norvegia 2
RO - Romania 2
AM - Armenia 1
AR - Argentina 1
BR - Brasile 1
CO - Colombia 1
DK - Danimarca 1
DZ - Algeria 1
EU - Europa 1
IL - Israele 1
IM - Isola di Man 1
IR - Iran 1
JM - Giamaica 1
JO - Giordania 1
KG - Kirghizistan 1
KZ - Kazakistan 1
LK - Sri Lanka 1
LT - Lituania 1
LV - Lettonia 1
MY - Malesia 1
PA - Panama 1
PE - Perù 1
PT - Portogallo 1
UZ - Uzbekistan 1
Totale 7.589
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Città #
Southend 1.081
Dublin 617
Fairfield 498
Siena 283
Menlo Park 252
Chandler 251
Ashburn 236
Woodbridge 231
Wilmington 196
Jacksonville 183
Seattle 162
Houston 155
Cambridge 143
Ann Arbor 138
Princeton 108
Beijing 106
Nanjing 77
Singapore 55
Fremont 52
Helsinki 48
Florence 46
Milan 46
Boardman 40
San Mateo 38
Dearborn 30
Rome 27
Izmir 25
San Diego 25
Moscow 24
New York 23
Nanchang 21
Shanghai 18
Shenyang 18
Düsseldorf 15
London 15
Naples 13
Brussels 12
Hebei 11
Tianjin 11
Abidjan 10
Dong Ket 10
Kunming 10
Norwalk 10
Redwood City 10
Guangzhou 9
Mogliano 9
Candiolo 8
Chicago 8
Santa Clara 8
Venezia 8
Aligarh 7
Anguillara Sabazia 7
Melbourne 7
Mestre 7
Paris 7
Málaga 6
Ningbo 6
Palermo 6
Washington 6
Bari 5
Cardiff 5
Galatone 5
Hong Kong 5
Jinan 5
Los Angeles 5
San Francisco 5
Valencia 5
Arconate 4
Como 4
Empoli 4
Falkenstein 4
Jiaxing 4
Lastra a Signa 4
Livorno 4
Mestrino 4
Munich 4
Philadelphia 4
Port Talbot 4
Tokyo 4
Turku 4
Zhengzhou 4
Bologna 3
Brno 3
Cascina 3
Gavirate 3
Grünheide 3
Gunzenhausen 3
Hangzhou 3
Krakow 3
Menges 3
Montemiletto 3
Montreal 3
Multan 3
Nuremberg 3
Ottawa 3
Porto San Giorgio 3
Prague 3
Sesto Fiorentino 3
Southwark 3
Taichung 3
Totale 5.642
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Nome #
Ligandi TRPV1 328
Design and Synthesis of New Transient Receptor Potential Vanilloid Type-1 (TRPV1) Channel Modulators: Identification, Molecular Modeling Analysis, and Pharmacological Characterization of the N-(4-Hydroxy-3-methoxybenzyl)-4-(thiophen-2-yl)butanamide, a Small Molecule Endowed with Agonist TRPV1 Activity and Protective Effects against Oxidative Stress 280
Quercetin/oleic acid-based G-protein-coupled receptor 40 ligands as new insulin secretion modulators 238
Synthesis of novel 2-(1-adamantanylcarboxamido)thiophene derivatives. Selective cannabinoid type 2 (CB2) receptor agonists as potential agents for the treatment of skin inflammatory disease 222
Cytotoxic effects of cannabinoids on human HT-29 colorectal adenocarcinoma cells: different mechanisms of THC, CBD, and CB83 207
Investigations on the 4-Quinolone-3-carboxylic Acid Motif. 7. Synthesis and Pharmacological Evaluation of 4-Quinolone-3-carboxamides and 4-Hydroxy-2-quinolone-3-carboxamides as High Affinity Cannabinoid Receptor 2 (CB2R) Ligands with Improved Aqueous Solubility 200
1-Aryl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide: An effective scaffold for the design of either CB1 and CB2 receptor ligands 192
Nuclear magnetic resonance for studying recognition processes between anandamide and cannabinoid receptors 191
Suppressing effect of COR659 on alcohol, sucrose, and chocolate self-administration in rats: Involvement of the GABAB and cannabinoid CB1 receptors 190
New fluoroquinolones active against fluoroquinolones-resistant Mycobacterium tuberculosis strains 169
Screen of unfocused libraries identified compounds with direct or synergistic antibacterial activity 169
Dihydro-alkylthio-benzyl-oxopyrimidines as Inhibitors of Reverse Transcriptase: Synthesis and Rationalization of the Biological Data on Both Wild-Type Enzyme and Relevant Clinical Mutants 165
The Interactions of the 5-HT3 Receptor with Quipazine-Like Arylpiperazine Ligands. The Journey Track at the End of the First Decade of the Third Millennium 161
Synthesis, Cannabinoid Receptor Affinity, and Molecular Modeling Studies of Substituted 1-Aryl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamides 153
Synthesis and biological evaluation of New N-alkyl 1-aryl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamides as cannabinoid receptor ligands 149
Rapid combinatorial access to a library of 1,5-disubstituted-3-indole-N-alkylacetamides as CB2 receptor ligands 149
Investigations on the 4-Quinolone-3-carboxylic Acid Motif. 6. Synthesis and Pharmacological Evaluation of 7-Substituted 4-Quinolone-3-carboxamide Derivatives as High Affinity Ligands for Cannabinoid Receptors 147
Synthetic bioactive olivetol-related amides: the influence of the phenolic group in cannabinoid receptor activity 146
Nuovi Potenti e Selettivi ligandi dei recettori dei cannabinoidi 144
Development and characterization of immobilized cannabinoid receptor (CB1/CB2) open tubular column for on-line screening 142
Synthesis and antitumor activities of a series of novel quinoxalinhydrazides 140
Regioselective functionalization of quinolin-4(1H)-ones via sequential palladium-catalyzed reactions 140
New Resorcinol-Anandamide "Hybrids" as Potent Cannabinoid Receptor Ligands Endowed with antinociceptive activity in vivo 140
Synthesis and in vitro pharmacological activity of oxypropanol analogs of labetalol 139
TRPV1-FAAH-COX: The Couples Game in Pain Treatment 137
Active manganese dioxide promoted cyclization of ortho-(1H-pyrrol-1-yl)aryl and heteroaryl carboxylic acids to 5H-pyrrolo[1,2-a][3,1]benzoxazin-5-one derivatives 136
HIV-Reverse Transcriptase Inhibition: Inclusion of Ligand-Induced Fit by Cross-Docking Studies 130
Design, synthesis, binding, and molecular modeling studies of new potent ligands of cannabinoid receptors 129
Resorcinol-sn-Glycerol Derivatives: Novel 2-Arachidonoylglycerol (2-AG) Mimetics Endowed with High Affinity and Selectivity for Cannabinoid Type 1 (CB1) Receptor 128
Structure-affinity relationships and pharmacological characterization of new alkyl-resorcinol cannabinoid receptor ligands: Identification of a dual cannabinoid receptor/TRPA1 channel agonist 128
Synthesis, cannabinoid receptor affinity, molecular modeling studies and in vivo pharmacological evaluation of new substituted 1-aryl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamides. 2. Effect of the 3-carboxamide substituent on the affinity and selectivity profile. 127
Thiazolothiazepine Inhibitors of HIV-1 Integrase 118
Polycondensed Heterocycles. Part 11: Preparation and Regioselective Reductions of 5-Phenyl-4H-pyrrolo[1,2-a][1]benzazepin-4-one 115
Synthesis of pyrazolo[1,5-a]pyrimidine ring as a possible bioisosteric replacement of the 5-(1H-pyrrol-1-yl)pyrazole scaffold 114
Design, Synthesis, and Binding Studies of New Potent Ligands of Cannabinoids Receptors 112
Pinocembrin and its linolenoyl ester derivative induce wound healing activity in HaCaT cell line potentially involving a GPR120/FFA4 mediated pathway 109
A multitarget semi-synthetic derivative of the flavonoid morin with improved in vitro vasorelaxant activity: Role of CaV1.2 and KCa1.1 channels 108
3-Amino-alkylated indoles: Unexplored green products acting as anti-inflammatory agents 105
In Silico-Guided Rational Drug Design and Synthesis of Novel 4-(Thiophen-2-yl)butanamides as Potent and Selective TRPV1 Agonists 99
In vitro and in vivo pharmacology of synthetic olivetol- or resorcinol-derived cannabinoid receptor ligands 99
Design, synthesis and pharmacological evaluation of ester-based quercetin derivatives as selective vascular KCa1.1 channel stimulators 99
Identification and Quantification of Trans-Resveratrol in Dietary Supplements by a Rapid and Straightforward RP-HPLC Method 98
Conformational Analysis of the N-Arachinylethanolamide (Anandamide) using Nuclear Magnetic Resonance and Theoretical Calculations 94
Anti-addictive properties of COR659 – Additional pharmacological evidence and comparison with a series of novel analogues 92
An approach to the stereo-controlled synthesis of polycyclic derivatives of L-4-thiazolidinecarboxilic acid active against HIV-1 integrase 89
Targeting neuropathic pain: pathobiology, current treatment and peptidomimetics as a new therapeutic opportunity 84
Design, synthesis and biological evaluation of light-driven on-off multitarget AChE and MAO-B inhibitors 82
Suppressing effect of the novel positive allosteric modulator of the GABAB receptor, COR659, on locomotor hyperactivity induced by different drugs of abuse 81
Design, synthesis, and physicochemical and pharmacological profiling of 7‐Hydroxy-5-oxopyrazolo[4,3‐b]pyridine-6-carboxamide derivatives with antiosteoarthritic activity in vivo 79
Computational drug repurposing for the identification of SARS-CoV-2 main protease inhibitors 79
Napthoxazepine Inhibitors of HIV-1 Integrase: Synthesis and Biological Evaluation 78
Old strategies and new perspectives in modulating the endocannabinoid system 73
GPR120/FFAR4 pharmacology: focus on agonists in Type 2 diabetes mellitus drug discovery 72
New synthesis of N1- and N2-substituted pyrazolo[4,3-b]pyridine-5-one derivatives as CB2 receptor ligands 69
Design, synthesis and in vitro experimental validation of novel TRPV4 antagonists inspired by labdane diterpenes 64
2-Hydroxy-5-(3,5,7-trihydroxy-4-oxo-4H-chromen-2-yl)phenyl(E)-3-(4-hydroxy-3-methoxyphenyl)acrylate: synthesis, in silico analysis and in vitro pharmacological evaluation 62
Optimization of Pyrazole Compounds as Antibiotic Adjuvants Active against Colistin- and Carbapenem-Resistant Acinetobacter baumannii 59
Lipoic/Capsaicin-Related Amides: Synthesis and Biological Characterization of New TRPV1 Agonists Endowed with Protective Properties against Oxidative Stress 59
Structure optimization of positive allosteric modulators of GABAB receptors led to the unexpected discovery of antagonists/potential negative allosteric modulators 55
The GABAB receptor positive allosteric modulator COR659: in vitro metabolism, in vivo pharmacokinetics in rats, synthesis and pharmacological characterization of metabolically protected derivatives 47
Development of 1-(2-aminophenyl)pyrrole-based amides acting as human topoisomerase I inhibitors 39
Totale 7.749
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Categoria #
all - tutte 24.692
article - articoli 0
book - libri 0
conference - conferenze 0
curatela - curatele 0
other - altro 0
patent - brevetti 0
selected - selezionate 0
volume - volumi 0
Totale 24.692
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Totale Lug Ago Sett Ott Nov Dic Gen Feb Mar Apr Mag Giu
2019/2020994 0 0 63 179 87 107 89 129 86 127 48 79
2020/20211.320 42 101 38 122 64 134 91 169 125 245 116 73
2021/20221.054 84 121 97 102 64 41 50 55 45 113 96 186
2022/20231.150 81 88 177 136 100 225 45 92 91 29 60 26
2023/20241.133 58 24 92 63 63 236 363 36 17 40 28 113
2024/2025328 59 98 171 0 0 0 0 0 0 0 0 0
Totale 7.749