IRIS
ANZINI, MAURIZIO
 Distribuzione geografica
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Continente #
NA - Nord America 7.144
EU - Europa 6.677
AS - Asia 1.099
SA - Sud America 12
AF - Africa 11
OC - Oceania 10
Continente sconosciuto - Info sul continente non disponibili 8
Totale 14.961
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Nazione #
US - Stati Uniti d'America 7.119
GB - Regno Unito 2.306
IE - Irlanda 1.070
CN - Cina 955
UA - Ucraina 730
DE - Germania 650
SE - Svezia 647
IT - Italia 470
FR - Francia 381
FI - Finlandia 193
RU - Federazione Russa 65
ES - Italia 54
SG - Singapore 51
TR - Turchia 44
RO - Romania 24
CA - Canada 23
BE - Belgio 18
CZ - Repubblica Ceca 15
PL - Polonia 15
AT - Austria 14
VN - Vietnam 13
IN - India 11
EU - Europa 8
NL - Olanda 7
AU - Australia 6
BR - Brasile 6
JP - Giappone 6
EE - Estonia 5
IR - Iran 5
NG - Nigeria 4
NZ - Nuova Zelanda 4
ZA - Sudafrica 4
CL - Cile 3
HK - Hong Kong 3
AE - Emirati Arabi Uniti 2
CH - Svizzera 2
DK - Danimarca 2
DZ - Algeria 2
GR - Grecia 2
HU - Ungheria 2
KR - Corea 2
LK - Sri Lanka 2
AL - Albania 1
BG - Bulgaria 1
CR - Costa Rica 1
EC - Ecuador 1
EG - Egitto 1
GE - Georgia 1
HR - Croazia 1
IL - Israele 1
KZ - Kazakistan 1
LI - Liechtenstein 1
MN - Mongolia 1
MX - Messico 1
PE - Perù 1
PY - Paraguay 1
SA - Arabia Saudita 1
SK - Slovacchia (Repubblica Slovacca) 1
Totale 14.961
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Città #
Southend 2.124
Fairfield 1.160
Dublin 1.063
Chandler 606
Jacksonville 601
Ashburn 559
Woodbridge 501
Wilmington 477
Seattle 409
Cambridge 390
Houston 387
Ann Arbor 324
Princeton 224
Beijing 218
Nanjing 213
Siena 210
Menlo Park 123
Boardman 102
Fremont 89
Helsinki 75
Shenyang 67
Nanchang 66
San Diego 64
Shanghai 59
Dearborn 57
Moscow 50
Málaga 48
Lancaster 46
San Mateo 42
Izmir 40
Hebei 39
New York 37
Düsseldorf 36
Tianjin 35
Milan 34
Norwalk 31
Singapore 31
Jiaxing 29
Changsha 26
Jinan 26
Kunming 25
Venezia 25
London 23
Redwood City 23
Mestre 22
San Francisco 20
Ningbo 19
Washington 19
Brussels 18
Philadelphia 18
Timisoara 17
Zhengzhou 17
Brno 14
Vienna 14
Dong Ket 13
Hangzhou 12
Florence 11
Gdynia 10
Eboli 8
Guangzhou 8
Lanzhou 8
Rome 8
Saint Petersburg 8
Bonndorf 7
Changchun 7
Hefei 7
Montréal 7
Mumbai 7
Munich 7
Taizhou 7
Toronto 7
Leawood 6
Amsterdam 5
Edinburgh 5
Frankfurt am Main 5
Fuzhou 5
Los Angeles 5
Ottawa 5
Tallinn 5
Auburn Hills 4
Auckland 4
Carmignano 4
Chicago 4
Kilburn 4
Lagos 4
Las Vegas 4
Latina 4
New Bedfont 4
Sala Bolognese 4
Santa Clara 4
Stockholm 4
São Paulo 4
West Jordan 4
Bucharest 3
Durban 3
Grünheide 3
Haikou 3
Hounslow 3
Madrid 3
Paris 3
Totale 11.252
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Nome #
1,5-Diarylpyrrole-3-acetic Acids and Esters as Novel Classes of Potent and Highly Selective Cyclooxygenase-2 Inhibitors 353
Development of Potent Inhibitors of the Mycobacterium tuberculosis Virulence Factor Zmp1 and Evaluation of Their Effect on Mycobacterial Survival inside Macrophages 286
Design, Synthesis, and Biological Evaluation of Imidazo[1,5-a]quinoline as Highly Potent Ligands of Central Benzodiazepine Receptors 251
Synthesis and biological evaluation of a new class of benzothiazines as neuroprotective agents 234
Synthesis and Biological Evaluation of Novel Neuroprotective Pyridazine Derivatives as Excitatory Amino Acid Transporter 2 (EAAT2) Activators 233
Aromatase and 5-alpha reductase gene expression: modulation by pain and morphine treatment in male rats 188
Synthesis, biological evaluation and molecular modeling of novel selective COX-2 inhibitors: sulfide, sulfoxide, and sulfone derivatives of 1,5-diarylpyrrol-3-substituted scaffold 183
Synthesis and biological evaluation of fluorinated 1,5-diarylpyrrole-3-alkoxyethyl ether derivatives as selective COX-2 inhibitors endowed with anti-inflammatory activity 182
Carborane-Conjugated 2-Quinolinecarboxamide Ligands of the Translocator Protein for Boron Neutron Capture Therapy 171
Synthesis and structure-activity relationship studies in serotonin 5-HT4 receptor ligands based on a benzo[de][2,6]naphthridine scaffold 170
Multivalent ligands for the serotonin 5-HT4 receptor 169
Anionic Polymerization of a Benzofulvene Monomer Leading to a Thermoreversible π-Stacked Polymer. Studies in Macromolecular and Aggregate Structure 168
Physicochemical and biopharmaceutical characterization of endo-2-(8-methyl-8-azabicyclo[3.2.1]oct-3-yl)-2,3-dihydro-1H-benz[e]isoindol-1-one (CR3124) a novel potent 5-HT3 receptor antagonist 165
Development of subnanomolar-affinity serotonin 5-HT4 receptor ligands based on quinoline structures 165
Synthesis and structure–activity relationship studies in serotonin 5-HT1A receptor agonists based on fused pyrrolidone scaffolds 159
The Interactions of the 5-HT3 Receptor with Quipazine-Like Arylpiperazine Ligands. The Journey Track at the End of the First Decade of the Third Millennium 158
A Nanocomposite Material Formed by Benzofulvene Polymer Nanoparticles Loaded with a Potent 5-HT3 Receptor Antagonist (CR3124) 155
Synthesis, biological evaluation and docking analysis of a new series of methylsulfonyl and sulfamoyl acetamides and ethyl acetates as potent COX-2 inhibitors 154
Enlarging the NSAIDs Family: Ether, Ester and Acid Derivatives of the 1,5-Diarrylpyrrole Scaffold as novel anti-inflammatory and analgesic agents 152
Nitroesteri di 1,5-Diaril-2-alchil-pirroli-3-sostituiti,Inibitori Selettivi di COX-2 e Donatori di Ossido Nitrico 151
The novel anti-inflammatory agent VA694, endowed with both NO-releasing and COX2-selective inhibiting properties, exhibits NO-mediated positive effects on blood pressure, coronary flow and endothelium in an experimental model of hypertension and endothelial dysfunction 151
Synthesis, Biological Evaluation, and Quantitative Receptor Docking Simulations of 2-Acylaminoethyl-1,4-benzodiazepines as novel Tifluadom-Like Ligands with High Affinity and Selectivity for k-Opioid Receptors 149
Characterization of persistent intramolecular C-H⋅⋅⋅X(N,O) bonds in solid state and solution 145
Synthesis and Structure-Activity Relationship Studies in Translocator Protein Ligands Based on a Pyrazolo[3,4-b]quinoline Scaffold 145
Novel Analgesic/Anti-inflammatory Agents: 1,5-Diarylpyrrole Nitrooxyalkyl Ethers and Related Compounds as Cyclooxygenase-2 Inhibiting Nitric Oxide Donors 144
Synthesis of trifluoromethyl-substituted pyrazolo[4,3-c]pyridines - Sequential versus multicomponent reaction approach 144
Phenylindenone isomers as divergent modulators of p38α MAP kinase 143
Structural Manipulation of Benzofulvene Derivatives Showing Spontaneous Thermoreversible Polymerization. Role of the Substituents in the Modulation of Polymer Properties 140
Bivalent Ligands for the Serotonin 5-HT3 Receptor 140
3-Substituted-1,5-diarly-2-alkyl-pyrroles Highly Selective and Orally Effective COX-2 Inhibitors 140
Characterization of Quinoline Derivatives. II. 7-(4-methyl-1-piperazinyl)-6H-[1]benzopyrano[3,4-c]quinoline 139
A Non-Peptide NK1 Receptor Agonist Showing Subpicomolar Affinity 139
Dendrimeric tetravalent ligands for the serotonin-gated ion channel 139
Cyclooxygenase-2 Inhibitors. 1,5-Diarylpyrrol-3-acetic Esters with Enhanced Inhibitory Activity Toward Cyclooxygenase-2 and Improved Cyclooxygenase-2/Cyclooxygenase-1 Selectivity 138
Novel Analgesic/Anti-inflammatory Agents: Diarylpyrrole Acetic Esters Endowed with Nitric Oxide Releasing Properties 136
Antiproliferative effect of two novel COX-2 inhibitors on human keratinocytes 135
Synthesis of 1,2,4,-Triazolo[4',3':1,6]pyridazino[4,5-b]quinoline Derivatives 134
Synthesis, Biological Evaluation, and Enzyme Docking Simulations of 1,5-Diarylpyrrole-3-Alkoxyethyl Ethers as Selective Cyclooxygenase-2 Inhibitors Endowed with Anti-inflammatory and Antinociceptive Activity 133
Design, Synthesis, and Biological Evaluation of AT1 Angiotensin II Receptor Antagonists Based on the Pyrazolo[3,4-b]pyridine and related Heteroaromatic Bicyclic Systems 133
Synthesis of 6,7-Dihydro-8-(4-methyl-1-piperazinyl)-[1]benzoxepino[4,5-c]quinoline as Potential 5-HT3 Receptor Ligand 132
A Computational Model of the 5-HT3 Receptor Extracellular Domain: Search for Ligand Binding Sites 132
Molecular Basis of Peripheral vs Central Benzodiazepine Receptor Selectivity in a New Class of Peripheral Benzodiazepine Receptor Ligands Related to Alpidem 132
Synthesis and Spontaneous Polymerization of Oligo(ethylene glycol)-Conjugated Benzofulvene Macromonomers. A Polymer Brush Forming a Physical Hydrogel 130
Heterotricyclic Amide Derivatives as Neurokinin-1 (NK1) Receptor Ligands 128
Enantioresolution and stereochemical characterization of two chiral sulfoxides endowed with COX-2 inhibitory activity 128
Amidine, Thiourea and Guanidine Derivatives of 2-Aminobenzothiazoles and Aminobenzothiazines, Novel Pharmacological Agents for the Treatment of Neurodegenerative Pathologies 128
Synthesis of 2-Substituted-2,3-dihydro-9-phenyl-1H-pyrrolo[3,4-b]quinolin-3-ones as Potential Peripheral Benzodiazepine-receptor Ligands 127
New red-shifted coelenterazine analogues with an extended electronic conjugation 127
Synthesis, Labeling, and Biological Evaluation of Halogenated 2-Quinolinecarboxamides as Potential Radioligands for the Visualization of Peripheral Benzodiazepine Receptors 126
Synthesis of 6-(4-Methyl-1-piperazinyl)-7H-indeno[2,1-c]quinoline Derivatives as Potential 5-HT Receptor Ligands 125
Design, Synthesis, and Structure-Affinity Relationship Studies in NK1 Receptor Ligands Based on Azole-Fused Quinolinecarboxamide Moieties 124
Novel and Highly Potent 5-HT3 Receptor Agonists Based on a Pyrroloquinoxaline Structure 123
Synthesis and Characterization of a New Benzofulvene Polymer Showing a Thermoreversible Polymerization Behavior 123
Synthesis, in vitro, and in vivo biological evaluation and molecular docking simulations of chiral alcohol and ether derivatives of the 1,5-diarylpyrrole scaffold as novel anti-inflammatory and analgesic agents 123
Further studies on imidazo[4,5-b]pyridine AT1 angiotensin II receptor antagonists. Effects of the transformation of the 4-phenylquinoline backbone into 4-phenylisoquinolinone or 1-phenylindene scaffolds 122
Synthesis and biological evaluation of amidine, guanidine, and thiourea derivatives of 2-amino(6-trifluoromethoxy)benzothiazole as neuroprotective agents potentially useful in brain diseases 122
Polycondensed heterocycles. III. Synthesis of 5,11-dioxo-1,2,3,11a-tetrahydro-5H,11H- and 5-oxo-2,3,11,11a-tetrahydro-1H,5H-pyrrolo[2,1-c][1,4]benzothiazepine 122
Novel Basic Derivatives of Benz[e]isoindol-1-ones and Pyrrolo[3,4-c]quinolin-1-ones with 5-HT3 Antagonistic Activity, their Preparation and their Therapeutic Use 122
Mapping the Peripheral Benzodiazepine Receptor Binding Site by Conformationally Restrained Derivatives of 1-(2-Chlorophenyl)-N-methyl-N-(1-methylpropyl)-3-isoquinolinecarboxamide (PK11195) 121
Development of a CE method for the determination of mycophenolic acid in human plasma: A comparison with HPLC 120
Structure-Activity Relationships in Carboxamide Derivatives Based on the Targeted Delivery of Radionuclides and Boron Atoms by Means of Peripheral Benzodiazepine Receptor Ligands 120
Non-peptide NK1 receptor ligands based on the 4-phenylpyridine moiety 119
Synthesis, Resolution, and Absolute Configuration of Two Novel and Selective Cyclooxygenase-2 Inhibitors Based on 1,5-Diarylpyrrole Structure 118
Multivalent Supramolecular Dendrimer-Based Drugs 116
5-HT and Benzodiazepine Receptor Ligands. III. Synthesis and Receptor Affinities of 1,2,4,-Triazolo[4',3':1,6]pyridazino[4,5-b]quinoline and 2,3-Dihydro-9-phenyl-1H-pyrrolo[3,4-b]quinoline-1-one Derivatives 115
Structure–affinity relationship studies on arylpiperazine derivatives related to quipazine as serotonin transporter ligands. Molecular basis of the selectivity SERT/5-HT3 receptor 114
Design, Synthesis, and Preliminary Biological Evaluation of Pyrrolo[3,4-c]quinolin-1-one and Oxoisoindoline Derivatives as Aggrecanase Inhibitors 114
New Insight into the Central Benzodiazepine Receptor-Ligand Interactions: Design, Synthesis, Biological Evaluation, and Molecular Modeling of 3-Substituted 6-Phenyl-4H-imidazo[1,5-a][1,4]benzodiazepines and Related Compounds 113
Characterization of Quinoline Derivatives. I. 6,7-Dihydro-8-(4-methyl-1-piperazinyl)[1]benzoxepino[4,5-c]quinoline 0.13-Hydrate 111
Polycondensed heterocycles. VII. A convenient synthesis of pyrrolo[1,2-a]quinoxaline derivatives by intramolecular aromatic nucleophilic displacement 111
Improving the Solubility of a New Class of Antiinflammatory Pharmacodynamic Hybrids, that Release Nitric Oxide and Inhibit Cycloxygenase-2 Isoenzyme 111
New π-stacked benzofulvene polymer showing thermoreversible polymerization: studies in macromolecular and aggregate structures and polymerization mechanism 111
Synthesis and structure-activity relationship studies in peripheral benzodiazepine receptor ligands related to alpidem 111
Chondroprotective effect of three different classes of anti-inflammatory agents on human osteoarthritic chondrocytes exposed to IL-1β. S. Cheleschi, N. A. Pascarelli, G. Valacchi, A. Di Capua, M. Biava, G. belmonte, A. Giordani, C. Sticozzi, M. Anzini, A. Fioravanti 111
Molecular Structure and Dynamics of Some Potent 5-HT3 Receptor Antagonists. Insight into the Interaction with the Receptor 110
Ethyl 8-Fluoro-6-(3-nitrophenyl)-4H-imidazo[1,5-a][1,4]benzodiazepine-3-carboxylate as Novel, Highly Potent, and Safe Antianxiety Agent 107
Further Studies on the Interaction of 5-Hydroxytryptamine3 (5-HT3) Receptor with Arylpiperazine Ligands. Development of a New 5-HT3 Receptor Ligand Showing Potent Acetylcholinesterase Inhibitory Properties 102
Determination of a novel angiotensin-AT1 Antagonist CR3210, in biological samples by HPLC 101
5,6-Dihydro-5-[4-[4-(2-methoxyphenyl)-1- piperazinyl]butyl]-4H- pyrrolo[1,2-a][1,4]benzodiazepine-4,6-dione and Related Compounds as New 5-HT1A Receptor Ligands 101
Esteri di Acidi Grassi Insaturi e Ormoni Androgeni Potenzialmente utili nel Trattamento del Dolore 100
Design, Synthesis, Structural Studies, Biological Evaluation, and Computational Simulations of Novel Potent AT1 Angiotensin II Receptor Antagonists Based on the 4-Phenylquinoline Structure 99
Hyaluronan graft copolymers bearing fatty-acid residues as self-assembling nanoparticles for olanzapine delivery 99
Antiamnestic Effect of the Two Novel k-Opioid Agonists, VA-100 and VA-101, in the Mouse Passive Avoidance Test 98
Synthesis and Biological Characterization of Novel 2-Quinolinecarboxamide Ligands of the Peripheral Benzodiazepine Receptors Bearing Technetium-99m or Rhenium 98
6-(1-Piperazinyl)-7H-indeno[2,1-c]quinoline Derivatives with High Affinity and Selectivity for 5-HT3 Serotonin Sites 97
Mapping and Fitting the Peripheral Benzodiazepine Receptor Binding Site by Carboxamide Derivatives. Comparison of Different Approaches to Quantitative Ligand-Receptor Interaction Modeling 97
11C-Labelling of the 5-HT3 Antagonist VC125 for PET Distribution Studies 97
Characterization and Differentiation of Heterocyclic Isomers. Part 2. Mass Spectrometry and Molecular Orbital Calculations on Pyrrolo[1,2-a][1,4]benzodiazepin-4-one, -6-one, -4,6-dione 97
Characterization of Quinoline Derivatives. Part 3. Mass Spectrometry and X-ray Crystallography of Biologically Interesting Arylquinolines 96
Synthesis of 6-[N-Alkyl-N-(4-hidroxybutyl)amino]pyrimidine Derivatives- Simplified Analogues of Acyclonucleosides 95
In Vitro Effects of VA441, a New Selective Cyclooxygenase-2 Inhibitor, on Human Osteoarthritic Chondrocytes exposed to IL-1β 94
Novel potent 5-HT3 receptor ligands based on the pyrrolidone structure: synthesis, biological evaluation, and computational rationalization of the ligand-receptor interaction modalities 94
Novel polybenzofulvene derivatives: synthesis and uses thereof 93
Radiosynthesis of [11C]-Labelled COX-2 Selective Inhibitor as a Potential PET Tracer Candidate for Cyclooxigenase-2 Expression 92
Radiosynthesis and preclinical evaluation of 11C-VA426, a cyclooxygenase-2 selective ligand 91
Sensitive SPE-HPLC Method to Determine a Novel Angiotensin-AT1 Antagonist in Biological Samples 90
Novel Potent and Selective Central 5-HT3 Receptor Ligands Provided with Different Intrinsic Efficacy. 2. Molecular Basis of the Intrinsic Efficacy of Arylpiperazine Derivatives at the Central 5-HT3 Receptors 90
Novel Potent 5-HT3 Receptor Ligands Based on the Pyrrolidone Structure. Effects of the Quaternization of the Basic Nitrogen on the Interaction with 5-HT3 Receptor 88
Synthesis and 5-HT Receptors Binding Studies of Some 3-Substituted-2-(4-methyl-1-piperazinyl)-4-phenylquinolines 86
Novel Potent and Selective 5-HT3 Receptor Antagonists Based on Arylpiperazine Skeleton: Synthesis, Structure, Biological Activity and CoMFA Studies 84
Totale 13.242
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Categoria #
all - tutte 44.560
article - articoli 0
book - libri 0
conference - conferenze 0
curatela - curatele 0
other - altro 0
patent - brevetti 0
selected - selezionate 0
volume - volumi 0
Totale 44.560
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Totale Lug Ago Sett Ott Nov Dic Gen Feb Mar Apr Mag Giu
2019/20203.240 442 116 213 542 202 251 252 422 240 282 70 208
2020/20212.348 136 232 49 263 153 341 76 339 306 160 185 108
2021/20221.557 116 220 57 200 64 35 79 47 67 201 147 324
2022/20232.291 136 171 301 344 241 458 50 193 209 64 85 39
2023/20241.583 55 25 186 65 46 438 517 63 0 20 18 150
2024/202545 45 0 0 0 0 0 0 0 0 0 0 0
Totale 15.065