IRIS
ANZINI, MAURIZIO
 Distribuzione geografica
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Continente #
NA - Nord America 10.617
EU - Europa 9.466
AS - Asia 4.931
SA - Sud America 752
AF - Africa 185
OC - Oceania 12
Continente sconosciuto - Info sul continente non disponibili 8
Totale 25.971
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Nazione #
US - Stati Uniti d'America 10.464
GB - Regno Unito 2.372
CN - Cina 1.942
SG - Singapore 1.439
RU - Federazione Russa 1.413
IT - Italia 1.111
IE - Irlanda 1.071
DE - Germania 950
UA - Ucraina 740
SE - Svezia 665
BR - Brasile 620
FR - Francia 539
VN - Vietnam 415
HK - Hong Kong 398
FI - Finlandia 326
KR - Corea 267
IN - India 136
CA - Canada 75
ES - Italia 72
TR - Turchia 65
ZA - Sudafrica 65
AR - Argentina 59
BD - Bangladesh 47
IQ - Iraq 44
MX - Messico 40
JP - Giappone 36
PL - Polonia 32
CI - Costa d'Avorio 28
NL - Olanda 28
RO - Romania 28
NG - Nigeria 25
BE - Belgio 24
AT - Austria 21
ID - Indonesia 21
CZ - Repubblica Ceca 19
EC - Ecuador 19
CL - Cile 16
KE - Kenya 15
DZ - Algeria 14
MA - Marocco 14
CO - Colombia 12
SA - Arabia Saudita 12
AE - Emirati Arabi Uniti 11
AZ - Azerbaigian 10
EE - Estonia 10
PK - Pakistan 10
UZ - Uzbekistan 10
EG - Egitto 9
PH - Filippine 9
AU - Australia 8
CR - Costa Rica 8
EU - Europa 8
UY - Uruguay 8
KZ - Kazakistan 7
LT - Lituania 7
NP - Nepal 7
PY - Paraguay 7
VE - Venezuela 7
CH - Svizzera 6
IR - Iran 6
JO - Giordania 6
TN - Tunisia 6
DO - Repubblica Dominicana 5
DK - Danimarca 4
GR - Grecia 4
HN - Honduras 4
HU - Ungheria 4
IL - Israele 4
LK - Sri Lanka 4
NI - Nicaragua 4
NZ - Nuova Zelanda 4
PT - Portogallo 4
AL - Albania 3
BB - Barbados 3
BG - Bulgaria 3
BH - Bahrain 3
GT - Guatemala 3
JM - Giamaica 3
MY - Malesia 3
OM - Oman 3
PS - Palestinian Territory 3
AO - Angola 2
GE - Georgia 2
HR - Croazia 2
KG - Kirghizistan 2
PA - Panama 2
PE - Perù 2
SK - Slovacchia (Repubblica Slovacca) 2
SY - Repubblica araba siriana 2
TH - Thailandia 2
TT - Trinidad e Tobago 2
AM - Armenia 1
BO - Bolivia 1
BS - Bahamas 1
BZ - Belize 1
CG - Congo 1
CV - Capo Verde 1
CY - Cipro 1
ET - Etiopia 1
GA - Gabon 1
Totale 25.956
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Città #
Southend 2.124
Dallas 1.201
Fairfield 1.160
Dublin 1.064
Singapore 827
Ashburn 742
Chandler 607
Jacksonville 604
Santa Clara 503
Woodbridge 501
Wilmington 478
Beijing 427
Seattle 412
Houston 397
Cambridge 391
Moscow 380
Hong Kong 376
Milan 372
Hefei 346
Ann Arbor 324
San Jose 315
Seoul 264
Munich 253
Siena 231
Princeton 224
Nanjing 214
Helsinki 178
Los Angeles 151
Ho Chi Minh City 138
Council Bluffs 135
The Dalles 125
Menlo Park 123
Lauterbourg 119
Hanoi 117
Rome 108
Boardman 103
Fremont 89
New York 85
Buffalo 75
Shanghai 71
Shenyang 69
Nanchang 67
San Diego 67
São Paulo 67
Dearborn 57
Bengaluru 56
Málaga 48
Johannesburg 47
Lancaster 47
Orem 42
San Mateo 42
Tianjin 42
Izmir 40
Hebei 39
Düsseldorf 38
London 36
Frankfurt am Main 32
Norwalk 31
Changsha 30
Jiaxing 29
Abidjan 28
Florence 28
Jinan 27
San Francisco 27
Turin 27
Kunming 26
Venezia 25
Brussels 24
Tokyo 24
Figino 23
Redwood City 23
Mestre 22
Philadelphia 22
Stockholm 22
Turku 21
Abuja 20
Vienna 20
Washington 20
Zhengzhou 20
Ningbo 19
Toronto 18
Amsterdam 17
Atlanta 17
Haiphong 17
Timisoara 17
Belo Horizonte 16
Chicago 16
Montreal 16
Rio de Janeiro 16
Baghdad 15
Guangzhou 15
Warsaw 15
Brno 14
Hangzhou 14
Chennai 13
Dong Ket 13
Phoenix 13
Mumbai 12
Nuremberg 12
Boston 11
Totale 18.045
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Nome #
1,5-Diarylpyrrole-3-acetic Acids and Esters as Novel Classes of Potent and Highly Selective Cyclooxygenase-2 Inhibitors 537
Development of Potent Inhibitors of the Mycobacterium tuberculosis Virulence Factor Zmp1 and Evaluation of Their Effect on Mycobacterial Survival inside Macrophages 398
Design, Synthesis, and Biological Evaluation of Imidazo[1,5-a]quinoline as Highly Potent Ligands of Central Benzodiazepine Receptors 393
Anionic Polymerization of a Benzofulvene Monomer Leading to a Thermoreversible π-Stacked Polymer. Studies in Macromolecular and Aggregate Structure 352
Synthesis and biological evaluation of a new class of benzothiazines as neuroprotective agents 348
Novel analgesic/anti-inflammatory agents: 1,5-Diarylpyrrole nitrooxyethyl sulfides and related compounds as Cyclooxygenase-2 inhibitors containing a nitric oxide donor moiety endowed with vasorelaxant properties 339
Aromatase and 5-alpha reductase gene expression: modulation by pain and morphine treatment in male rats 331
Synthesis and Biological Evaluation of Novel Neuroprotective Pyridazine Derivatives as Excitatory Amino Acid Transporter 2 (EAAT2) Activators 331
A Nanocomposite Material Formed by Benzofulvene Polymer Nanoparticles Loaded with a Potent 5-HT3 Receptor Antagonist (CR3124) 324
Carborane-Conjugated 2-Quinolinecarboxamide Ligands of the Translocator Protein for Boron Neutron Capture Therapy 305
A Non-Peptide NK1 Receptor Agonist Showing Subpicomolar Affinity 297
Development of subnanomolar-affinity serotonin 5-HT4 receptor ligands based on quinoline structures 296
Synthesis, biological evaluation and molecular modeling of novel selective COX-2 inhibitors: sulfide, sulfoxide, and sulfone derivatives of 1,5-diarylpyrrol-3-substituted scaffold 292
Synthesis and biological evaluation of fluorinated 1,5-diarylpyrrole-3-alkoxyethyl ether derivatives as selective COX-2 inhibitors endowed with anti-inflammatory activity 273
Exploring Translocator Protein (TSPO) Medicinal Chemistry: An Approach for Targeting Radionuclides and Boron Atoms to Mitochondria 271
Bivalent Ligands for the Serotonin 5-HT3 Receptor 265
Characterization of Quinoline Derivatives. II. 7-(4-methyl-1-piperazinyl)-6H-[1]benzopyrano[3,4-c]quinoline 263
Multivalent ligands for the serotonin 5-HT4 receptor 260
Antiproliferative effect of two novel COX-2 inhibitors on human keratinocytes 253
3-Substituted-1,5-diarly-2-alkyl-pyrroles Highly Selective and Orally Effective COX-2 Inhibitors 252
Synthesis and structure-activity relationship studies in serotonin 5-HT4 receptor ligands based on a benzo[de][2,6]naphthridine scaffold 252
Characterization of persistent intramolecular C-H⋅⋅⋅X(N,O) bonds in solid state and solution 249
Synthesis and Spontaneous Polymerization of Oligo(ethylene glycol)-Conjugated Benzofulvene Macromonomers. A Polymer Brush Forming a Physical Hydrogel 248
Synthesis and structure–activity relationship studies in serotonin 5-HT1A receptor agonists based on fused pyrrolidone scaffolds 248
5-HT and Benzodiazepine Receptor Ligands. III. Synthesis and Receptor Affinities of 1,2,4,-Triazolo[4',3':1,6]pyridazino[4,5-b]quinoline and 2,3-Dihydro-9-phenyl-1H-pyrrolo[3,4-b]quinoline-1-one Derivatives 247
Novel Analgesic/Anti-inflammatory Agents: 1,5-Diarylpyrrole Nitrooxyalkyl Ethers and Related Compounds as Cyclooxygenase-2 Inhibiting Nitric Oxide Donors 244
Design, Synthesis, and Biological Evaluation of AT1 Angiotensin II Receptor Antagonists Based on the Pyrazolo[3,4-b]pyridine and related Heteroaromatic Bicyclic Systems 243
6-(1-Piperazinyl)-7H-indeno[2,1-c]quinoline Derivatives with High Affinity and Selectivity for 5-HT3 Serotonin Sites 242
The novel anti-inflammatory agent VA694, endowed with both NO-releasing and COX2-selective inhibiting properties, exhibits NO-mediated positive effects on blood pressure, coronary flow and endothelium in an experimental model of hypertension and endothelial dysfunction 242
Dendrimeric tetravalent ligands for the serotonin-gated ion channel 239
Amidine, Thiourea and Guanidine Derivatives of 2-Aminobenzothiazoles and Aminobenzothiazines, Novel Pharmacological Agents for the Treatment of Neurodegenerative Pathologies 237
A Computational Model of the 5-HT3 Receptor Extracellular Domain: Search for Ligand Binding Sites 231
Design, Synthesis, and Preliminary Biological Evaluation of Pyrrolo[3,4-c]quinolin-1-one and Oxoisoindoline Derivatives as Aggrecanase Inhibitors 231
Development of a CE method for the determination of mycophenolic acid in human plasma: A comparison with HPLC 230
The Interactions of the 5-HT3 Receptor with Quipazine-Like Arylpiperazine Ligands. The Journey Track at the End of the First Decade of the Third Millennium 230
Design, Synthesis, and Structure-Affinity Relationship Studies in NK1 Receptor Ligands Based on Azole-Fused Quinolinecarboxamide Moieties 227
Physicochemical and biopharmaceutical characterization of endo-2-(8-methyl-8-azabicyclo[3.2.1]oct-3-yl)-2,3-dihydro-1H-benz[e]isoindol-1-one (CR3124) a novel potent 5-HT3 receptor antagonist 227
Structural Manipulation of Benzofulvene Derivatives Showing Spontaneous Thermoreversible Polymerization. Role of the Substituents in the Modulation of Polymer Properties 222
5,6-Dihydro-5-[4-[4-(2-methoxyphenyl)-1- piperazinyl]butyl]-4H- pyrrolo[1,2-a][1,4]benzodiazepine-4,6-dione and Related Compounds as New 5-HT1A Receptor Ligands 222
Phenylindenone isomers as divergent modulators of p38α MAP kinase 220
Characterization of Quinoline Derivatives. I. 6,7-Dihydro-8-(4-methyl-1-piperazinyl)[1]benzoxepino[4,5-c]quinoline 0.13-Hydrate 218
11C-Labelling of the 5-HT3 Antagonist VC125 for PET Distribution Studies 217
Synthesis, biological evaluation and docking analysis of a new series of methylsulfonyl and sulfamoyl acetamides and ethyl acetates as potent COX-2 inhibitors 216
Enlarging the NSAIDs Family: Ether, Ester and Acid Derivatives of the 1,5-Diarrylpyrrole Scaffold as novel anti-inflammatory and analgesic agents 212
Nitroesteri di 1,5-Diaril-2-alchil-pirroli-3-sostituiti,Inibitori Selettivi di COX-2 e Donatori di Ossido Nitrico 208
Novel multitarget directed ligands inspired by riluzole: A serendipitous synthesis of substituted benzo[b][1,4]thiazepines potentially useful as neuroprotective agents 207
Synthesis and Structure-Activity Relationship Studies in Translocator Protein Ligands Based on a Pyrazolo[3,4-b]quinoline Scaffold 206
Antiamnestic Effect of the Two Novel k-Opioid Agonists, VA-100 and VA-101, in the Mouse Passive Avoidance Test 204
Synthesis and biological evaluation of amidine, guanidine, and thiourea derivatives of 2-amino(6-trifluoromethoxy)benzothiazole as neuroprotective agents potentially useful in brain diseases 202
Chondroprotective effect of three different classes of anti-inflammatory agents on human osteoarthritic chondrocytes exposed to IL-1β. S. Cheleschi, N. A. Pascarelli, G. Valacchi, A. Di Capua, M. Biava, G. belmonte, A. Giordani, C. Sticozzi, M. Anzini, A. Fioravanti 199
Mapping the Peripheral Benzodiazepine Receptor Binding Site by Conformationally Restrained Derivatives of 1-(2-Chlorophenyl)-N-methyl-N-(1-methylpropyl)-3-isoquinolinecarboxamide (PK11195) 198
Synthesis of 6,7-Dihydro-8-(4-methyl-1-piperazinyl)-[1]benzoxepino[4,5-c]quinoline as Potential 5-HT3 Receptor Ligand 198
Synthesis of 2-Substituted-2,3-dihydro-9-phenyl-1H-pyrrolo[3,4-b]quinolin-3-ones as Potential Peripheral Benzodiazepine-receptor Ligands 197
Non-peptide NK1 receptor ligands based on the 4-phenylpyridine moiety 195
Synthesis of trifluoromethyl-substituted pyrazolo[4,3-c]pyridines - Sequential versus multicomponent reaction approach 195
Cyclooxygenase-2 Inhibitors. 1,5-Diarylpyrrol-3-acetic Esters with Enhanced Inhibitory Activity Toward Cyclooxygenase-2 and Improved Cyclooxygenase-2/Cyclooxygenase-1 Selectivity 195
Synthesis, Biological Evaluation, and Quantitative Receptor Docking Simulations of 2-Acylaminoethyl-1,4-benzodiazepines as novel Tifluadom-Like Ligands with High Affinity and Selectivity for k-Opioid Receptors 195
Novel and Highly Potent 5-HT3 Receptor Agonists Based on a Pyrroloquinoxaline Structure 194
Novel Analgesic/Anti-inflammatory Agents: Diarylpyrrole Acetic Esters Endowed with Nitric Oxide Releasing Properties 194
Synthesis of 6-(4-Methyl-1-piperazinyl)-7H-indeno[2,1-c]quinoline Derivatives as Potential 5-HT Receptor Ligands 193
Synthesis, Labeling, and Biological Evaluation of Halogenated 2-Quinolinecarboxamides as Potential Radioligands for the Visualization of Peripheral Benzodiazepine Receptors 193
Novel Basic Derivatives of Benz[e]isoindol-1-ones and Pyrrolo[3,4-c]quinolin-1-ones with 5-HT3 Antagonistic Activity, their Preparation and their Therapeutic Use 193
Mapping and Fitting the Peripheral Benzodiazepine Receptor Binding Site by Carboxamide Derivatives. Comparison of Different Approaches to Quantitative Ligand-Receptor Interaction Modeling 191
Molecular Basis of Peripheral vs Central Benzodiazepine Receptor Selectivity in a New Class of Peripheral Benzodiazepine Receptor Ligands Related to Alpidem 190
Synthesis, Biological Evaluation, and Enzyme Docking Simulations of 1,5-Diarylpyrrole-3-Alkoxyethyl Ethers as Selective Cyclooxygenase-2 Inhibitors Endowed with Anti-inflammatory and Antinociceptive Activity 189
Further studies on imidazo[4,5-b]pyridine AT1 angiotensin II receptor antagonists. Effects of the transformation of the 4-phenylquinoline backbone into 4-phenylisoquinolinone or 1-phenylindene scaffolds 188
Structure-Activity Relationships in Carboxamide Derivatives Based on the Targeted Delivery of Radionuclides and Boron Atoms by Means of Peripheral Benzodiazepine Receptor Ligands 188
New red-shifted coelenterazine analogues with an extended electronic conjugation 187
Synthesis of 1,2,4,-Triazolo[4',3':1,6]pyridazino[4,5-b]quinoline Derivatives 186
Synthesis and Characterization of a New Benzofulvene Polymer Showing a Thermoreversible Polymerization Behavior 186
Heterotricyclic Amide Derivatives as Neurokinin-1 (NK1) Receptor Ligands 185
In Vitro Effects of VA441, a New Selective Cyclooxygenase-2 Inhibitor, on Human Osteoarthritic Chondrocytes exposed to IL-1β 184
New π-stacked benzofulvene polymer showing thermoreversible polymerization: studies in macromolecular and aggregate structures and polymerization mechanism 184
Characterization of Quinoline Derivatives. Part 3. Mass Spectrometry and X-ray Crystallography of Biologically Interesting Arylquinolines 183
Characterization and Differentiation of Heterocyclic Isomers. Part 2. Mass Spectrometry and Molecular Orbital Calculations on Pyrrolo[1,2-a][1,4]benzodiazepin-4-one, -6-one, -4,6-dione 183
Synthesis, in vitro, and in vivo biological evaluation and molecular docking simulations of chiral alcohol and ether derivatives of the 1,5-diarylpyrrole scaffold as novel anti-inflammatory and analgesic agents 181
Multivalent Supramolecular Dendrimer-Based Drugs 179
Determination of a novel angiotensin-AT1 Antagonist CR3210, in biological samples by HPLC 179
Radiosynthesis of [11C]-Labelled COX-2 Selective Inhibitor as a Potential PET Tracer Candidate for Cyclooxigenase-2 Expression 179
New Insight into the Central Benzodiazepine Receptor-Ligand Interactions: Design, Synthesis, Biological Evaluation, and Molecular Modeling of 3-Substituted 6-Phenyl-4H-imidazo[1,5-a][1,4]benzodiazepines and Related Compounds 177
Ethyl 8-Fluoro-6-(3-nitrophenyl)-4H-imidazo[1,5-a][1,4]benzodiazepine-3-carboxylate as Novel, Highly Potent, and Safe Antianxiety Agent 177
Polycondensed heterocycles. III. Synthesis of 5,11-dioxo-1,2,3,11a-tetrahydro-5H,11H- and 5-oxo-2,3,11,11a-tetrahydro-1H,5H-pyrrolo[2,1-c][1,4]benzothiazepine 174
Esteri di Acidi Grassi Insaturi e Ormoni Androgeni Potenzialmente utili nel Trattamento del Dolore 172
CoMFA Analysis of Ligands of the Mitochondrial Benzodiazepine Receptor: A Versatile Tool for the Design of New Lead Compounds 171
Enantioresolution and stereochemical characterization of two chiral sulfoxides endowed with COX-2 inhibitory activity 170
Hyaluronan graft copolymers bearing fatty-acid residues as self-assembling nanoparticles for olanzapine delivery 170
Molecular Structure and Dynamics of Some Potent 5-HT3 Receptor Antagonists. Insight into the Interaction with the Receptor 168
Design, Synthesis, Structural Studies, Biological Evaluation, and Computational Simulations of Novel Potent AT1 Angiotensin II Receptor Antagonists Based on the 4-Phenylquinoline Structure 166
Further Studies on the Interaction of 5-Hydroxytryptamine3 (5-HT3) Receptor with Arylpiperazine Ligands. Development of a New 5-HT3 Receptor Ligand Showing Potent Acetylcholinesterase Inhibitory Properties 165
Polycondensed heterocycles. VII. A convenient synthesis of pyrrolo[1,2-a]quinoxaline derivatives by intramolecular aromatic nucleophilic displacement 164
Structure–affinity relationship studies on arylpiperazine derivatives related to quipazine as serotonin transporter ligands. Molecular basis of the selectivity SERT/5-HT3 receptor 164
Use of imidazo[1,5-a]quinoline scaffold as the pharmacophore in the design of bivalent ligands of central benzodiazepine receptors 162
Novel polybenzofulvene derivatives: synthesis and uses thereof 161
Synthesis, Resolution, and Absolute Configuration of Two Novel and Selective Cyclooxygenase-2 Inhibitors Based on 1,5-Diarylpyrrole Structure 160
Novel potent 5-HT3 receptor ligands based on the pyrrolidone structure: synthesis, biological evaluation, and computational rationalization of the ligand-receptor interaction modalities 159
Synthesis, Biological Evaluation and Receptor Docking Simulations of 2-[(Acylamino)ethyl]-1,4-benzodiazepines as k-Opioid Receptor Agonists Endowed with Antinociceptive and Antiamnestic Activity 158
Synthesis and structure-activity relationship studies in peripheral benzodiazepine receptor ligands related to alpidem 158
Synthesis and Biological Characterization of Novel 2-Quinolinecarboxamide Ligands of the Peripheral Benzodiazepine Receptors Bearing Technetium-99m or Rhenium 157
Radiosynthesis and preclinical evaluation of 11C-VA426, a cyclooxygenase-2 selective ligand 155
Novel Potent and Selective 5-HT3 Receptor Antagonists Based on Arylpiperazine Skeleton: Synthesis, Structure, Biological Activity and CoMFA Studies 154
Totale 22.144
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Categoria #
all - tutte 77.524
article - articoli 0
book - libri 0
conference - conferenze 0
curatela - curatele 0
other - altro 0
patent - brevetti 0
selected - selezionate 0
volume - volumi 0
Totale 77.524
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Totale Lug Ago Sett Ott Nov Dic Gen Feb Mar Apr Mag Giu
2021/20221.557 116 220 57 200 64 35 79 47 67 201 147 324
2022/20232.291 136 171 301 344 241 458 50 193 209 64 85 39
2023/20241.583 55 25 186 65 46 438 517 63 0 20 18 150
2024/20253.415 69 174 290 171 395 202 142 208 303 136 337 988
2025/20267.494 564 1.142 956 796 1.311 269 832 187 273 413 152 599
2026/2027159 159 0 0 0 0 0 0 0 0 0 0 0
Totale 26.088