IRIS
TAFI, ANDREA
 Distribuzione geografica
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Continente #
NA - Nord America 5.591
EU - Europa 4.846
AS - Asia 796
AF - Africa 16
SA - Sud America 11
OC - Oceania 8
Continente sconosciuto - Info sul continente non disponibili 4
Totale 11.272
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Nazione #
US - Stati Uniti d'America 5.571
GB - Regno Unito 1.626
IE - Irlanda 805
CN - Cina 690
UA - Ucraina 556
SE - Svezia 472
IT - Italia 414
FR - Francia 311
DE - Germania 293
RU - Federazione Russa 128
FI - Finlandia 125
SG - Singapore 60
ES - Italia 28
CA - Canada 18
BE - Belgio 15
RO - Romania 15
TR - Turchia 13
CZ - Repubblica Ceca 12
CI - Costa d'Avorio 11
NL - Olanda 8
VN - Vietnam 8
PL - Polonia 7
AU - Australia 6
AT - Austria 5
BR - Brasile 5
EU - Europa 4
JP - Giappone 4
GR - Grecia 3
IM - Isola di Man 3
IN - India 3
RS - Serbia 3
ZA - Sudafrica 3
AZ - Azerbaigian 2
BG - Bulgaria 2
CH - Svizzera 2
CL - Cile 2
HK - Hong Kong 2
HU - Ungheria 2
KH - Cambogia 2
KR - Corea 2
LK - Sri Lanka 2
LU - Lussemburgo 2
NG - Nigeria 2
NZ - Nuova Zelanda 2
PT - Portogallo 2
AL - Albania 1
AM - Armenia 1
BD - Bangladesh 1
BO - Bolivia 1
DK - Danimarca 1
FK - Isole Falkland (Malvinas) 1
GE - Georgia 1
HR - Croazia 1
IL - Israele 1
IR - Iran 1
KZ - Kazakistan 1
LT - Lituania 1
LV - Lettonia 1
MK - Macedonia 1
OM - Oman 1
PA - Panama 1
PE - Perù 1
PR - Porto Rico 1
SI - Slovenia 1
SY - Repubblica araba siriana 1
VE - Venezuela 1
Totale 11.272
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Città #
Southend 1.520
Fairfield 832
Dublin 805
Menlo Park 468
Jacksonville 452
Chandler 413
Woodbridge 410
Wilmington 344
Ashburn 343
Houston 323
Seattle 306
Cambridge 285
Beijing 212
Ann Arbor 191
Siena 150
Princeton 143
Nanjing 140
New York 72
Boardman 68
San Diego 61
Nanchang 60
San Mateo 51
Fremont 36
Venezia 35
Helsinki 32
Changsha 29
Shenyang 29
Singapore 29
Hebei 25
Kunming 25
Dearborn 24
Düsseldorf 23
Hangzhou 23
Málaga 23
Tianjin 23
Moscow 22
Florence 19
Jinan 19
London 19
Lancaster 18
Jiaxing 17
Rome 16
Shanghai 15
Brussels 14
Ningbo 14
Zhengzhou 12
Abidjan 11
Milan 11
Redwood City 11
Timisoara 11
Brno 10
Izmir 10
Rende 10
San Francisco 10
Toronto 10
Changchun 9
Norwalk 9
Taizhou 9
Falls Church 8
Kilburn 7
Lanzhou 7
Mestre 6
Philadelphia 6
Bellante 5
Indiana 5
Vienna 5
Chicago 4
Dong Ket 4
Grünheide 4
Guangzhou 4
Konstanz 4
Kostomloty Drugie 4
Madrid 4
Montreal 4
Naples 4
Paris 4
Pavia 4
Saint Petersburg 4
São Paulo 4
Tappahannock 4
Atlanta 3
Auburn Hills 3
Aversa 3
Belgrade 3
Buffalo 3
Catanzaro 3
Detroit 3
Haikou 3
Hefei 3
Ho Chi Minh City 3
Lanuvio 3
Southwark 3
Stellenbosch 3
Sydney 3
Villingen-schwenningen 3
Amsterdam 2
Andover 2
Anguillara Sabazia 2
Campi Bisenzio 2
Cardiff 2
Totale 8.471
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Nome #
1-[(3-Aryloxy-3-aryl)propyl]-2H-imidazoles, new imidazoles with potent activity against Candida albicans and dermatophytes. Synthesis, structure-activity relationship, and molecular modeling studies 276
Ruthenium-catalyzed synthesis of 5-amino-1,2,3-triazole-4-carboxylates for triazole-based scaffolds: Beyond the Dimroth rearrangement 245
Valutazione della specificità di substrato delle lipasi da Candida rugosa e Rhizomucor miehei 219
Discovery of GPCR ligands for probing signal transduction pathways 208
Discovery and cardioprotective effects of the first non-peptide agonists of the G protein-coupled prokineticin receptor-1 204
Investigations on the 4-quinolone-3-carboxylic acid motif part 5: modulation of the physicochemical profile of a set of potent and selective cannabinoid-2 receptor ligands through a bioisosteric approach 199
Molecular recognition of natural products by resorc[4]arene receptors 190
In Memory of Maurizio Botta: His Contribution to the Development of Computer-Aided Drug Design 181
Characterization of COR627 and COR628, two novel positive allosteric modulators of the GABA B receptor 172
Antifungal agents. 10. New derivatives of 1-[(Aryl)[4-aryl-1H-pyrrol-3-yl]methyl]-1H-imidazole, synthesis, anti-Candida activity and Quantitative Structure-Analysis Relationship studies 165
Dihydro-alkylthio-benzyl-oxopyrimidines as Inhibitors of Reverse Transcriptase: Synthesis and Rationalization of the Biological Data on Both Wild-Type Enzyme and Relevant Clinical Mutants 160
Computational studies of competitive inhibitors of nitric oxide synthase (NOS) enzymes: towards the development of powerful and isoform-selective inhibitors 150
Diltiazem-like calcium entry blockers: a hypothesis of the receptor-binding site based on a comparative molecular field analysis model 150
Pyrrolo[2,1-c][1,4]benzothiazines: Synthesis, Structure-Activity Relationships, Molecular Modeling Studies, and Cardiovascular Activity 150
Stereoretentive Chlorination of Cyclic Alcohols Catalyzed by Titanium(IV) Tetrachloride: Evidence for a Front Side Attack Mechanism 148
α1-Adrenoceptor antagonists. 5. Pyridazinone-arylpiperazines. Probing the influence on affinity and selectivity of both ortho-Alkoxy groups at the arylpiperazine moiety and cyclic substituents at the pyridazinone nucleus 147
Pharmacophore Modelling: A Forty Year Old Approach and its Modern Synergies 146
Synthesis and Interaction with Copper(II) Cations of Cyano- and Aminoresorcin[4]arenes 144
3D-QSAR using pharmacophore-based alignment and virtual screening for discovery of novel MCF-7 cell line inhibitors 144
Synthesis, molecular modeling studies, and pharmacological activity of selective A1 receptor antagonists 143
Unconventional Plasticity of HIV-1 Reverse Transcriptase: How Inhibitors Could Open a Connection "Gate" between Allosteric and Catalytic Sites. 142
Pyrrolobenzodiazepines and related systems. 2. Synthesis and biological properties of isonoraptazepine derivatives 141
A Novel Route to Calix[4]arenes. 2. Solution- and Solid-State Structural Analyses and Molecular Modeling Studies 137
Metadynamics Simulations of Enantioselective Acylation Give Insights into the Catalytic Mechanism of Burkholderia cepacia Lipase 137
Design, Synthesis, and Pharmacological Characterization of Indole-3-ylacetamides, Indole-3-yloxoacetamides, and Indole-3-ylcarboxamides: Potent and Selective CB2 Cannabinoid Receptor Inverse Agonists 136
Synthesis and preliminary biological evaluation of 1-aminomethyl-4-substituted-4-H-pyrrolo[2,1-C][1,4] benzothiazines, a new class of calcium antagonists 134
A dynamic target-based pharmacophoric model mapping the CD4 binding site on HIV-1 gp120 to identify new inhibitors of gp120-CD4 protein-protein interactions 133
Synthesis and “in vitro” cardiovascular activity of 4-aryl-2,3,3a,4-tetrahydro-1h-pyrrolo[2,1-c][1,4]benzothiazin-1-ones and 7-acetoxy-6-phenyl-7a,8,9,10-tetrahydropyrrolo [2,1,-d][1,5]benzothiazepin-10-one 133
Antifungal Agents. 11.N-Substituted Derivatives of 1-[(Aryl)(4-aryl-1H-pyrrol-3yl)methyl]-1H-imidazole: Synthesis, Anti-Candida Activity, and QSAR Studies 132
Stereochemical Preference of 2'-Deoxycytidine for Chiral Bis(diamido)-bridged Basket Resorcin[4]arenes 131
Interactions of vinca alkaloid subunits with chiral amido[4]resorcinarenes: a dynamic, kinetic and spectroscopic study 131
A drop of enantioselectivity in the Pseudomonas cepacia lipase-catalyzed ester hydrolysis is influenced by the chain length of the fatty acid 127
Diastereoselective gas-phase ion/molecule reactions of ethanolamine neurotransmitter/amido[4]resorcinarene adducts 126
Prokineticin 1 receptor agonists and their uses 125
Rational design and synthesis of homochiral azole antifungal agents 124
Synthesis and biological evaluation of conformationally restricted analogs of tolmetin and ketorolac 124
Pharmacophore Modeling for Qualitative Prediction of Antiestrogenic Activity 122
Three-Dimensional Quantitative Structure-Selectivity Relationships (3D-QSSR) Analysis Guided Rational Design of a Highly Selective Ligand for the Cannabinoid Receptor 2 122
The tetramerization of 2,4-dimethoxycinnamates. A novel route to calixarenes 122
Vibrational relaxation in crystal SO2 122
Chiral Recognition by Resorcin[4]arene Receptors: Intrinsic Kinetics and Dynamics 120
Microwave-assisted intramolecular huisgen cycloaddition of azido alkynes derived from α-amino acids 120
Application of pharmacophore models in medicinal chemistry 120
AMBER force field implementation of the boronate function to simulate the inhibition of β-lactamases by alkyl and aryl boronic acids 119
Polar phonons in SO2 single crystal 119
Cavity Effects on the Enantioselectivity of Chiral Amido[4]resorcinarene Stereoisomers 119
Bis(diamido)-bridged basket resorcin[4]arenes as enantioselective receptors for amino acids and amines 118
An approach to address Candida rugosa lipase regioselectivity in the acylation reactions of trytilated glucosides 118
Importance of the Thiomorpholine Introduction in New Pyrrole Derivatives as Antimycobacterial Agents Analogues of BM 212 115
Molecular modeling as a powerful technique for understanding small-large molecules interactions 113
Modelling Amphetamine/Receptor Interactions: A Gas-Phase Study of Complexes Formed between Amphetamine and Some Chiral Amido[4]resorcinarenes 111
Antimycobacterial compounds. Optimization of the BM212 structure, the lead compound for a new pyrrole derivative class 111
Lipase-catalyzed regioselective acylation of resorcin[4]arenes 111
Molecular modeling of azole antifungal agents active against Candida albicans .1. A comparative molecular field analysis study 111
Flattened Cone 2,8,14,20-Tetrakis(l-valinamido)-[4]resorcinarene: An Enantioselective Allosteric Receptor in the Gas Phase 111
Cyclic dipeptides. 4. On the Pummerer rearrangement of diastereomeric dehydrocyclolanthionine sulfoxides 110
Antimycobacterial compounds. New pyrrole derivatives of BM212 110
Pharmacophore Based Receptor Modeling: The Case of Adenosine A3 Receptor Antagonists. An Approach to the Optimization of Protein Models 109
Synthesis and Preliminary Biological Evaluation of 4,6-Disubstituted 3-Cyanopyridin-2(1H)-ones, a New Class of Calcium Entry Blockers 109
N-Linked Peptidoresorc[4]arene-Based Receptors as Noncompetitive Inhibitors for alpha-Chymotrypsin 108
Discovery of Chiral Cyclopropyl Dihydro-Alkylthio-Benzyl-Oxopyrimidine (S-DABO) Derivatives as Potent HIV-1 Reverse Transcriptase Inhibitors with High Activity Against Clinically Relevant Mutants 107
Chair-boat equilibrium as driving force in epimerization of 3,7-dimethylbicyclo[3.3.1]nonan-2,9-dione derivatives. Stereocontrolled synthesis of 3-exo,7-exo- and 3-endo,7-exo-3,7-dimethylbicyclo[3.3.1]nonan-9-ones 106
Desymmetrisation of meso-methylcyclooctanones. Highly Enantioselective Synthesis of C8 syn-Isoprenoid and syn,syn-Deoxypropionate Subunits from a Bicyclo[3.3.1]nonane Precursor 106
Conformational search of antisense nucleotides. Part. 2 105
Conformational search of antisense nucleotides 104
Chalcone Prenyltransferase from Morus nigra cell cultures. Substrate specificity studies 103
Crystal structure of the OXA-48 beta-lactamase reveals mechanistic diversity among class D carbapenemases 103
Inhibition of Amine Oxidases Activity by 1-acetyl-3,5-diphenyl-4,5-dihydro-(1H)-Pyrazole Derivatives 99
Alpha1-Adrenoceptor Antagonists. 4. Pharmacophore-based Design, Synthesis, and Biological Evaluation of New Imidazo-, Benzimidazo-, and Indoloarylpiperazine Derivatives 97
Gas-phase enantioselectivity of chiral amido[4]resorcinarene receptors 97
Tetrahydrofuran Acetogenins from Laurencia glandulifera 94
Synthesis of Calix[4]arenes. 4. Design, Synthesis, Computational Studies and Homodimerization of Polymethylene Bridged Resorc[4]arenes 93
Towards the modelling of glycosaminoglycan-protein interactions. A comprehensive study of the conformational properties of hyaluronan 93
Synthesis of Calix[4]arenes. 5. Design, Synthesis and Computational Studies of Chiral Amidoresorc[4]arenes 91
Erratum: Lipase-catalyzed regioselective acylation of resorcin[4]arenes 85
Novel hypotensive agents from Verbesina caracasana. 8. Synthesis and pharmacology of (3,4-dimethoxycinnamoyl)-N1-agmatine and synthetic analogues 82
Pharmacophore modeling: a continuously evolving tool for computational drug design 81
Synthesis, antitubercular activity and pharmacophore fitting of new derivatives of toluidine 81
Cyclic Dipeptides. 3. Synthesis of Methyl (R)-6-[(tert-Butoxycarbonyl)amino]-4,5,6,7-tetrahydro-2-methyl-5-oxo-1,4-thiazepine-3-carboxylate and Its Hexahydro Analogs. Elaboration of a Novel Dual ACE/NEP Inhibitor 81
Nuovi derivati 1,2-difenilpirrolici attivi come agenti antitubercolari. 80
New derivatives of toluidine: synthesis, antitubercular activity and pharmacophore hypothesis 80
Synthesis and molecular modelling studies of resorcin[4]arene-capped porphyrins 78
STRUCTURE AND CONFORMATION OF STEREOISOMERIC C-ISOPROPOXYCARBONYLMETHYLCALIX[4]RESORCINARENES 77
SYNTHESIS AND MOLECULAR MODELING OF TAXANES MODIFIED AT RING-C 77
Nuovi derivati 1,5-difenilpirrolici derivati del BM212 come agenti antitubercolari 76
Computer Simulations of Enantioselective Ester Hydrolyses Catalyzed by Pseudomonas cepacia Lipase 76
Issues inherent in the rational design of azole antifungal agents 75
Molecular Modelling as a powerful technique for understanding small-large molecule interactions 75
Enantioselective guest exchange in a chiral resorcin[4]arenes cavity 73
Novel Hypotensive Agents from Verbesina caracasana. 6. Synthesis and Pharmacology of Caracasandiamide 72
CONFORMATIONAL EFFECTS ON THE STEREOCHEMICAL COURSE OF THE NABH4 REDUCTION OF SUBSTITUTED BICYCLO[3.3.1]NONAN-2-ONES 71
structure-activity relationship studies of a new series of imidazi[2,1-f]purinones as potent and selective A3 adenosine receptor antagonists 65
Pharmacophore optimization for antitubercular pyrrole active compounds 63
Structural flexibility of hyaluronan oligomers as probed by molecular modeling 59
Totale 11.329
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Categoria #
all - tutte 34.699
article - articoli 0
book - libri 0
conference - conferenze 0
curatela - curatele 0
other - altro 0
patent - brevetti 0
selected - selezionate 0
volume - volumi 0
Totale 34.699
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Totale Lug Ago Sett Ott Nov Dic Gen Feb Mar Apr Mag Giu
2019/20202.078 0 73 151 408 133 162 214 307 181 229 73 147
2020/20211.670 95 165 21 179 102 246 58 244 234 88 143 95
2021/20221.156 77 211 78 53 52 31 70 45 53 129 104 253
2022/20231.797 108 124 254 249 169 352 55 154 207 44 59 22
2023/20241.065 44 27 54 63 23 355 390 23 1 18 7 60
2024/2025173 59 114 0 0 0 0 0 0 0 0 0 0
Totale 11.329