SAVINI, LUISA
SAVINI, LUISA
Dipartimento di Biotecnologie, Chimica e Farmacia
ANTIMALARIAL AGENTS HAVING POLYAROMATIC STRUCTURE
2007-01-01 Campiani, Giuseppe; Gemma, Sandra; C., Fattorusso; G., Kukreja; B. P., Joshi; O., TAGLIALATELA SCAFATI; Savini, Luisa; M., DE ANGELIS; E., Fattorusso
Application of near infrared reflectance spectroscopy (NIRS) to several antibiotic compounds
1992-01-01 Corti, Piero; Savini, Luisa; Dreassi, Elena; S., Petriconi; R., Genga; L., Montecchi; S., Lonardi
Application of Near-Infrared Reflectance Analysis (NIRA) to the integrated control of antibiotics tablet production
1995-01-01 Dreassi, Elena; G., Ceramelli; Savini, Luisa; Corti, Piero; P. L., Perruccio; S., Lonardi
Application of NIRS to the control of pharmaceuticals identification and assay of several primary materials
1992-01-01 Corti, Piero; Savini, Luisa; Dreassi, Elena; G., Ceramelli; L., Montecchi; S., Lonardi
Chelating agents as potential antitumorals. 2-quinolylhydrazones and bis-2-quinolylhydrazones. I
1995-01-01 Savini, Luisa; Massarelli, Paola; Chiasserini, Luisa; Sega, Alessandro; Pellerano, Cesare; Barzi, A; Nocentini, G.
Chelating agents as potential antitumorals: alfa-(N)-heterocyclic hydrazones and bis-alfa-(N)-heterocyclic hydrazones
1997-01-01 Savini, Luisa; Massarelli, Paola; Chiasserini, Luisa; Nencini, Cristina; Pellerano, Cesare
Chelating Properties of New Series of Heterocyclic hydrazones. X-ray Crystallography and Mass Spectrometry of Their Metal Complexes
1998-01-01 Giorgi, Gianluca; Savini, Luisa; Chiasserini, Luisa; Nencini, Cristina; Pellerano, Cesare
Clotrimazole Scaffold as an Innovative Pharmacophore Towards Potent Antimalarial Agents: Design, Synthesis, Biological and Structure-Activity Relationship Studies.
2008-01-01 Gemma, Sandra; Campiani, Giuseppe; Butini, Stefania; G., Kukreja; SANNA COCCONE, Salvatore; B., Joshi; M., Persico; Nacci, Vito; Fiorini, Isabella; E., Novellino; Fattorusso, E; O., TAGLIALATELA SCAFATI; Savini, Luisa; D., Taramelli; N., Basilico; S., Parapini; G., Morace; V., Yardley; S., Croft; M., Coletta; S., Marini; Fattorusso, Caterina
Design and Synthesis of Potent Antimalarial Agents Based on Clotrimazole Scaffold: Exploring an Innovative Pharmacophore.
2007-01-01 Gemma, Sandra; Campiani, Giuseppe; Butini, Stefania; B., Joshi; G., Kukreja; M., Persico; B., Catalanotti; E., Novellino; Fattorusso, E; Nacci, Vito; Savini, Luisa; D., Taramelli; N., Basilico; G., Morace; V., Yardley; C., Fattorusso
Design, synthesis, and structure-activity relationship studies of 4-quinolinyl- and 9-acrydinylhydrazones as potent antimalarial agents.
2008-01-01 C., Fattorusso; Campiani, Giuseppe; G., Kukreja; M., Persico; Butini, Stefania; Romano, MARIA PIA; Altarelli, Maria; S., Ros; Brindisi, Margherita; Savini, Luisa; E., Novellino; Nacci, Vito; E., Fattorusso; S., Parapini; N., Basilico; D., Taramelli; V., Yardley; S., Croft; M., Borriello; Gemma, Sandra
Development of Antitubercular Compounds Based on a 4-Quinolylhydrazone Scaffold. Further Structure-activity Relationship Studies.
2009-01-01 Gemma, Sandra; Savini, Luisa; Altarelli, Maria; Tripaldi, Pierangela; Chiasserini, Luisa; SANNA COCCONE, Salvatore; Vinod, Kumar; Camodeca, Caterina; Campiani, Giuseppe; Ettore, Novellino; Sandra, Clarizio; Giovanni, Delogu; Butini, Stefania
Development of molecular probes for the identification of extra interaction sites in the mid-gorge and peripheral sites of butyrylcholinesterase (BuChE). Rational design of novel, selective, and highly potent BuChE inhibitors.
2005-01-01 Campiani, Giuseppe; Fattorusso, C; Butini, Stefania; Gaeta, A; Agnusdei, M; Gemma, Sandra; Persico, M; Catalanotti, B; Savini, Luisa; Nacci, Vito; Novellino, E; Holloway, Hw; Greig, Nh; Belinskaya, T; Fedorko, Jm; Saxena, A.
Development of piperazine-tethered heterodimers as potent antimalarials against chloroquine-resistant P. falciparum strains. Synthesis and molecular modeling.
2007-01-01 Gemma, Sandra; Kukreja, G; Campiani, Giuseppe; Butini, Stefania; Bernetti, Matteo; Joshi, Bp; Savini, Luisa; Basilico, N; Taramelli, D; Yardley, V; Bertamino, A; Novellino, E; Persico, M; Catalanotti, B; Fattorusso, C.
High affinity central benzodiazepine receptor ligands: synthesis and structure-activity relationship studies of a new series of pyrazolo[4,3-c]quinolin-3-ones
1998-01-01 Savini, Luisa; Massarelli, Paola; Nencini, Cristina; Pellerano, Cesare; Biggio, G.; Maciocco, A.; Tuligi, G.; Carrieri, A.; Cinone, N.; Carotti, A.
Malaria chemotherapy: recent advances in drug development
2010-01-01 Gemma, Sandra; Travagli, Valter; Savini, Luisa; Novellino, E; Campiani, Giuseppe; Butini, Stefania
Microwave-assisted synthesis of 4-quinolylhydrazines followed by nickel boride reduction: a convenient approach to 4-aminoquinolines and derivatives
2008-01-01 Gemma, Sandra; G., Kukreja; Tripaldi, Pierangela; Altarelli, Maria; Bernetti, Matteo; Franceschini, Silvia; Savini, Luisa; Campiani, Giuseppe; C., Fattorusso; Butini, Stefania
Mimicking the Intramolecular Hydrogen Bond: Synthesis, Biological Evaluation, and Molecular Modeling of Benzoxazines and Quinazolines as Potential Antimalarial Agents
2012-01-01 Gemma, Sandra; Camodeca, Caterina; Brindisi, Margherita; Brogi, Simone; Gagan, Kukreja; Kunjir, SANIL ASHOK; Emanuele, Gabellieri; Leonardo, Lucantoni; Annette, Habluetzel; Donatella, Taramelli; Nicoletta, Basilico; Roberta, Gualdani; Francesco Tadini, Buoninsegni; Gianluca, Bartolommei; Maria Rosa, Moncelli; Rowena E., Martin; Robert L., Summers; Lamponi, Stefania; Savini, Luisa; Fiorini, Isabella; Valoti, Massimo; Ettore, Novellino; Campiani, Giuseppe; Butini, Stefania
Near Infrared Reflectance Spectroscopy in the determination of the physical state of primary materials in pharmaceutical production
1995-01-01 Dreassi, Elena; G., Ceramelli; Savini, Luisa; Corti, Piero; P. L., Perruccio
New 1-[quinolyl(4)]-1,2,3-triazoles: synthesis and evaluation of antiinflammatory and analgesic properties. II
1994-01-01 Savini, Luisa; Massarelli, Paola; Chiasserini, Luisa; Pellerano, Cesare; Bruni, Giancarlo
New alpha-(N)-heterocyclichydrazones: evaluation of anticancer, anti-HIV and antimicrobial activity.
2004-01-01 Savini, Luisa; Chiasserini, Luisa; Travagli, Valter; Pellerano, Cesare; Novellino, E.; Cosentino, S.; Pisano, M. B.
Titolo | Data di pubblicazione | Autore(i) | File | Abstract |
---|---|---|---|---|
ANTIMALARIAL AGENTS HAVING POLYAROMATIC STRUCTURE | 1-gen-2007 | Campiani, Giuseppe; Gemma, Sandra; C., Fattorusso; G., Kukreja; B. P., Joshi; O., TAGLIALATELA SCAFATI; Savini, Luisa; M., DE ANGELIS; E., Fattorusso | - | |
Application of near infrared reflectance spectroscopy (NIRS) to several antibiotic compounds | 1-gen-1992 | Corti, Piero; Savini, Luisa; Dreassi, Elena; S., Petriconi; R., Genga; L., Montecchi; S., Lonardi | - | |
Application of Near-Infrared Reflectance Analysis (NIRA) to the integrated control of antibiotics tablet production | 1-gen-1995 | Dreassi, Elena; G., Ceramelli; Savini, Luisa; Corti, Piero; P. L., Perruccio; S., Lonardi | - | |
Application of NIRS to the control of pharmaceuticals identification and assay of several primary materials | 1-gen-1992 | Corti, Piero; Savini, Luisa; Dreassi, Elena; G., Ceramelli; L., Montecchi; S., Lonardi | - | |
Chelating agents as potential antitumorals. 2-quinolylhydrazones and bis-2-quinolylhydrazones. I | 1-gen-1995 | Savini, Luisa; Massarelli, Paola; Chiasserini, Luisa; Sega, Alessandro; Pellerano, Cesare; Barzi, A; Nocentini, G. | - | |
Chelating agents as potential antitumorals: alfa-(N)-heterocyclic hydrazones and bis-alfa-(N)-heterocyclic hydrazones | 1-gen-1997 | Savini, Luisa; Massarelli, Paola; Chiasserini, Luisa; Nencini, Cristina; Pellerano, Cesare | - | |
Chelating Properties of New Series of Heterocyclic hydrazones. X-ray Crystallography and Mass Spectrometry of Their Metal Complexes | 1-gen-1998 | Giorgi, Gianluca; Savini, Luisa; Chiasserini, Luisa; Nencini, Cristina; Pellerano, Cesare | - | |
Clotrimazole Scaffold as an Innovative Pharmacophore Towards Potent Antimalarial Agents: Design, Synthesis, Biological and Structure-Activity Relationship Studies. | 1-gen-2008 | Gemma, Sandra; Campiani, Giuseppe; Butini, Stefania; G., Kukreja; SANNA COCCONE, Salvatore; B., Joshi; M., Persico; Nacci, Vito; Fiorini, Isabella; E., Novellino; Fattorusso, E; O., TAGLIALATELA SCAFATI; Savini, Luisa; D., Taramelli; N., Basilico; S., Parapini; G., Morace; V., Yardley; S., Croft; M., Coletta; S., Marini; Fattorusso, Caterina | - | |
Design and Synthesis of Potent Antimalarial Agents Based on Clotrimazole Scaffold: Exploring an Innovative Pharmacophore. | 1-gen-2007 | Gemma, Sandra; Campiani, Giuseppe; Butini, Stefania; B., Joshi; G., Kukreja; M., Persico; B., Catalanotti; E., Novellino; Fattorusso, E; Nacci, Vito; Savini, Luisa; D., Taramelli; N., Basilico; G., Morace; V., Yardley; C., Fattorusso | - | |
Design, synthesis, and structure-activity relationship studies of 4-quinolinyl- and 9-acrydinylhydrazones as potent antimalarial agents. | 1-gen-2008 | C., Fattorusso; Campiani, Giuseppe; G., Kukreja; M., Persico; Butini, Stefania; Romano, MARIA PIA; Altarelli, Maria; S., Ros; Brindisi, Margherita; Savini, Luisa; E., Novellino; Nacci, Vito; E., Fattorusso; S., Parapini; N., Basilico; D., Taramelli; V., Yardley; S., Croft; M., Borriello; Gemma, Sandra | - | |
Development of Antitubercular Compounds Based on a 4-Quinolylhydrazone Scaffold. Further Structure-activity Relationship Studies. | 1-gen-2009 | Gemma, Sandra; Savini, Luisa; Altarelli, Maria; Tripaldi, Pierangela; Chiasserini, Luisa; SANNA COCCONE, Salvatore; Vinod, Kumar; Camodeca, Caterina; Campiani, Giuseppe; Ettore, Novellino; Sandra, Clarizio; Giovanni, Delogu; Butini, Stefania | - | |
Development of molecular probes for the identification of extra interaction sites in the mid-gorge and peripheral sites of butyrylcholinesterase (BuChE). Rational design of novel, selective, and highly potent BuChE inhibitors. | 1-gen-2005 | Campiani, Giuseppe; Fattorusso, C; Butini, Stefania; Gaeta, A; Agnusdei, M; Gemma, Sandra; Persico, M; Catalanotti, B; Savini, Luisa; Nacci, Vito; Novellino, E; Holloway, Hw; Greig, Nh; Belinskaya, T; Fedorko, Jm; Saxena, A. | - | |
Development of piperazine-tethered heterodimers as potent antimalarials against chloroquine-resistant P. falciparum strains. Synthesis and molecular modeling. | 1-gen-2007 | Gemma, Sandra; Kukreja, G; Campiani, Giuseppe; Butini, Stefania; Bernetti, Matteo; Joshi, Bp; Savini, Luisa; Basilico, N; Taramelli, D; Yardley, V; Bertamino, A; Novellino, E; Persico, M; Catalanotti, B; Fattorusso, C. | - | |
High affinity central benzodiazepine receptor ligands: synthesis and structure-activity relationship studies of a new series of pyrazolo[4,3-c]quinolin-3-ones | 1-gen-1998 | Savini, Luisa; Massarelli, Paola; Nencini, Cristina; Pellerano, Cesare; Biggio, G.; Maciocco, A.; Tuligi, G.; Carrieri, A.; Cinone, N.; Carotti, A. | - | |
Malaria chemotherapy: recent advances in drug development | 1-gen-2010 | Gemma, Sandra; Travagli, Valter; Savini, Luisa; Novellino, E; Campiani, Giuseppe; Butini, Stefania | - | |
Microwave-assisted synthesis of 4-quinolylhydrazines followed by nickel boride reduction: a convenient approach to 4-aminoquinolines and derivatives | 1-gen-2008 | Gemma, Sandra; G., Kukreja; Tripaldi, Pierangela; Altarelli, Maria; Bernetti, Matteo; Franceschini, Silvia; Savini, Luisa; Campiani, Giuseppe; C., Fattorusso; Butini, Stefania | - | |
Mimicking the Intramolecular Hydrogen Bond: Synthesis, Biological Evaluation, and Molecular Modeling of Benzoxazines and Quinazolines as Potential Antimalarial Agents | 1-gen-2012 | Gemma, Sandra; Camodeca, Caterina; Brindisi, Margherita; Brogi, Simone; Gagan, Kukreja; Kunjir, SANIL ASHOK; Emanuele, Gabellieri; Leonardo, Lucantoni; Annette, Habluetzel; Donatella, Taramelli; Nicoletta, Basilico; Roberta, Gualdani; Francesco Tadini, Buoninsegni; Gianluca, Bartolommei; Maria Rosa, Moncelli; Rowena E., Martin; Robert L., Summers; Lamponi, Stefania; Savini, Luisa; Fiorini, Isabella; Valoti, Massimo; Ettore, Novellino; Campiani, Giuseppe; Butini, Stefania | - | |
Near Infrared Reflectance Spectroscopy in the determination of the physical state of primary materials in pharmaceutical production | 1-gen-1995 | Dreassi, Elena; G., Ceramelli; Savini, Luisa; Corti, Piero; P. L., Perruccio | - | |
New 1-[quinolyl(4)]-1,2,3-triazoles: synthesis and evaluation of antiinflammatory and analgesic properties. II | 1-gen-1994 | Savini, Luisa; Massarelli, Paola; Chiasserini, Luisa; Pellerano, Cesare; Bruni, Giancarlo | - | |
New alpha-(N)-heterocyclichydrazones: evaluation of anticancer, anti-HIV and antimicrobial activity. | 1-gen-2004 | Savini, Luisa; Chiasserini, Luisa; Travagli, Valter; Pellerano, Cesare; Novellino, E.; Cosentino, S.; Pisano, M. B. | - |