CAPPELLI, ANDREA
CAPPELLI, ANDREA
Dipartimento di Biotecnologie, Chimica e Farmacia
1,5-Diarylpyrrole-3-acetic Acids and Esters as Novel Classes of Potent and Highly Selective Cyclooxygenase-2 Inhibitors
2005-01-01 Biava, M.; Porretta, G. C.; Cappelli, Andrea; Vomero, S.; Manetti, Fabrizio; Botta, Maurizio; Sautebin, L.; Rossi, A.; Makovec, F.; Anzini, Maurizio
11C-Labelling of the 5-HT3 Antagonist VC125 for PET Distribution Studies
1997-01-01 Sharon Stone, Elander; Jan Olov, Thorell; Martin, Ingvar; Cappelli, Andrea; Anzini, Maurizio; Vomero, Salvatore
3-Substituted-1,5-diarly-2-alkyl-pyrroles Highly Selective and Orally Effective COX-2 Inhibitors
2006-01-01 Cappelli, Andrea; Anzini, Maurizio; G., Caselli; A., Giordani; F., Makovec; L. C., Rovati; M., Biava
5-HT and Benzodiazepine Receptor Ligands. III. Synthesis and Receptor Affinities of 1,2,4,-Triazolo[4',3':1,6]pyridazino[4,5-b]quinoline and 2,3-Dihydro-9-phenyl-1H-pyrrolo[3,4-b]quinoline-1-one Derivatives
1990-01-01 Anzini, Maurizio; Cappelli, Andrea; Vomero, Salvatore; Botta, Maurizio; A., Cagnotto
6-(1-Piperazinyl)-7H-indeno[2,1-c]quinoline Derivatives with High Affinity and Selectivity for 5-HT3 Serotonin Sites
1993-01-01 Anzini, Maurizio; Cappelli, Andrea; Vomero, Salvatore; A., Cagnotto; M., Skorupska
A Click Chemistry-Based “Grafting Through” Approach to the Synthesis of a Biorelevant Polymer Brush
2011-01-01 Cappelli, A.; Paolino, M.; Grisci, G.; Giuliani, G.; Donati, A.; Mendichi, R.; Boccia, A. C.; Samperi, F.; Battiato, S.; Paccagnini, E.; Giacomello, E.; Sorrentino, V.; Licciardi, M.; Giammona, G.; Vomero, S.
A Computational Model of the 5-HT3 Receptor Extracellular Domain: Search for Ligand Binding Sites.
2001-01-01 Menziani, M. C.; DE RIENZO, F.; Cappelli, Andrea; Anzini, Maurizio; DE BENEDETTI, P. G.
A Nanocomposite Material Formed by Benzofulvene Polymer Nanoparticles Loaded with a Potent 5-HT3 Receptor Antagonist (CR3124)
2010-01-01 Cappelli, Andrea; Galeazzi, S; Zanardi, Iacopo; Travagli, Valter; Anzini, Maurizio; Mendichi, R; Petralito, S; Memoli, A; Paccagnini, Eugenio; Peris, W; Giordani, A; Makovec, F; Fresta, M; Vomero, Salvatore
A Non-Peptide NK1 Receptor Agonist Showing Subpicomolar Affinity
2004-01-01 Cappelli, Andrea; Giuliani, Germano; PERICOT MOHR GL, G; Gallelli, A; Anzini, Maurizio; Vomero, Salvatore; Cupello, A; Scarrone, S; Matarrese, M; Moresco, Rm; Fazio, F; Finetti, Federica; Morbidelli, Lucia; Ziche, Marina
A non-toxic, reversibly released imaging probe for oral cancer that is derived from natural compounds
2021-01-01 Ghanim, Magda; Relitti, Nicola; Mcmanus, Gavin; Butini, Stefania; Cappelli, Andrea; Campiani, Giuseppe; Mok, K H; Kelly, Vincent P
A stereoselective approach to peptidomimetic BACE1 inhibitors
2013-01-01 Butini, Stefania; Emanuele, Gabellieri; Brindisi, Margherita; Giovani, Simone; Maramai, Samuele; Kshirsagar, Giridhar; Egeria, Guarino; Brogi, Simone; Valeria La, Pietra; Mariateresa, Giustiniano; Luciana, Marinelli; Ettore, Novellino; Campiani, Giuseppe; Cappelli, Andrea; Gemma, Sandra
Age and Sex Influence the Neuro-inflammatory Response to a Peripheral Acute LPS Challenge
2019-01-01 Murtaj, V.; Belloli, S.; Di Grigoli, G.; Pannese, M.; Ballarini, E.; Rodriguez-Menendez, V.; Marmiroli, P.; Cappelli, A.; Masiello, V.; Monterisi, C.; Bellelli, G.; Panina-Bordignon, P.; Moresco, R. M.
Aggregation-Induced Förster Resonance Energy Transfer in Polybenzofulvene/Dye Nanoparticles
2015-01-01 Villafiorita Monteleone, Francesca; Cappelli, Andrea; Paolino, Marco; Colombo, Miriam; Cariati, Elena; Mura, Andrea; Bongiovanni, Giovanni; Botta, Chiara
Amidine, Thiourea and Guanidine Derivatives of 2-Aminobenzothiazoles and Aminobenzothiazines, Novel Pharmacological Agents for the Treatment of Neurodegenerative Pathologies
2007-01-01 Anzini, Maurizio; A., Giordani; F., Makovec; Cappelli, Andrea; Vomero, Salvatore; G., Caselli; L. C., Rovati
Anionic Polymerization of a Benzofulvene Monomer Leading to a Thermoreversible π-Stacked Polymer. Studies in Macromolecular and Aggregate Structure
2008-01-01 Cappelli, Andrea; Galeazzi, S; Giuliani, Germano; Anzini, Maurizio; Aggravi, M; Donati, Alessandro; Zetta, L; Boccia, A; Mendichi, R; Giorgi, Gianluca; Paccagnini, Eugenio; Vomero, Salvatore
Antiamnestic Effect of the Two Novel k-Opioid Agonists, VA-100 and VA-101, in the Mouse Passive Avoidance Test
2001-01-01 Ghelardini, C.; Galeotti, N.; DI CESARE MANNELLI, L.; Cappelli, Andrea; Anzini, Maurizio; Bartolini, A.
Antiproliferative effect of two novel COX-2 inhibitors on human keratinocytes
2013-01-01 Sticozzi, Claudia; Belmonte, Giuseppe; Cervellati, Franco; Di Capua, Angela; Maioli, Emanuela; Cappelli, Andrea; Giordani, Antonio; Biava, Mariangela; Anzini, Maurizio; Valacchi, Giuseppe
Aromatase and 5-alpha reductase gene expression: modulation by pain and morphine treatment in male rats
2010-01-01 Aloisi, ANNA MARIA; Ceccarelli, I; Fiorenzani, P; Maddalena, M; Rossi, A; Tomei, V; Sorda, G; Danielli, B; Rovini, M; Cappelli, Andrea; Anzini, Maurizio; Giordano, Antonio
Bithiophene-based polybenzofulvene derivatives with high stacking and hole mobility
2015-01-01 Cappelli, Andrea; Razzano, Vincenzo; Paolino, Marco; Grisci, Giorgio; Giuliani, Germano; Donati, Alessandro; Mendichi, Raniero; Samperi, Filippo; Battiato, Salvatore; Boccia, Antonella Caterina; Mura, Andrea; Bongiovanni, Giovanni; Mróz, Wojciech; Botta, Chiara
Bivalent Ligands for the Serotonin 5-HT3 Receptor
2011-01-01 Cappelli, Andrea; Manini, Monica; Paolino, Marco; A., Gallelli; Anzini, Maurizio; L., Mennuni; M., DEL CADIA; F., DE RIENZO; M. C., Menziani; Vomero, Salvatore
Titolo | Data di pubblicazione | Autore(i) | File | Abstract |
---|---|---|---|---|
1,5-Diarylpyrrole-3-acetic Acids and Esters as Novel Classes of Potent and Highly Selective Cyclooxygenase-2 Inhibitors | 1-gen-2005 | Biava, M.; Porretta, G. C.; Cappelli, Andrea; Vomero, S.; Manetti, Fabrizio; Botta, Maurizio; Sautebin, L.; Rossi, A.; Makovec, F.; Anzini, Maurizio | - | |
11C-Labelling of the 5-HT3 Antagonist VC125 for PET Distribution Studies | 1-gen-1997 | Sharon Stone, Elander; Jan Olov, Thorell; Martin, Ingvar; Cappelli, Andrea; Anzini, Maurizio; Vomero, Salvatore | - | |
3-Substituted-1,5-diarly-2-alkyl-pyrroles Highly Selective and Orally Effective COX-2 Inhibitors | 1-gen-2006 | Cappelli, Andrea; Anzini, Maurizio; G., Caselli; A., Giordani; F., Makovec; L. C., Rovati; M., Biava | - | |
5-HT and Benzodiazepine Receptor Ligands. III. Synthesis and Receptor Affinities of 1,2,4,-Triazolo[4',3':1,6]pyridazino[4,5-b]quinoline and 2,3-Dihydro-9-phenyl-1H-pyrrolo[3,4-b]quinoline-1-one Derivatives | 1-gen-1990 | Anzini, Maurizio; Cappelli, Andrea; Vomero, Salvatore; Botta, Maurizio; A., Cagnotto | - | |
6-(1-Piperazinyl)-7H-indeno[2,1-c]quinoline Derivatives with High Affinity and Selectivity for 5-HT3 Serotonin Sites | 1-gen-1993 | Anzini, Maurizio; Cappelli, Andrea; Vomero, Salvatore; A., Cagnotto; M., Skorupska | - | |
A Click Chemistry-Based “Grafting Through” Approach to the Synthesis of a Biorelevant Polymer Brush | 1-gen-2011 | Cappelli, A.; Paolino, M.; Grisci, G.; Giuliani, G.; Donati, A.; Mendichi, R.; Boccia, A. C.; Samperi, F.; Battiato, S.; Paccagnini, E.; Giacomello, E.; Sorrentino, V.; Licciardi, M.; Giammona, G.; Vomero, S. | - | |
A Computational Model of the 5-HT3 Receptor Extracellular Domain: Search for Ligand Binding Sites. | 1-gen-2001 | Menziani, M. C.; DE RIENZO, F.; Cappelli, Andrea; Anzini, Maurizio; DE BENEDETTI, P. G. | - | |
A Nanocomposite Material Formed by Benzofulvene Polymer Nanoparticles Loaded with a Potent 5-HT3 Receptor Antagonist (CR3124) | 1-gen-2010 | Cappelli, Andrea; Galeazzi, S; Zanardi, Iacopo; Travagli, Valter; Anzini, Maurizio; Mendichi, R; Petralito, S; Memoli, A; Paccagnini, Eugenio; Peris, W; Giordani, A; Makovec, F; Fresta, M; Vomero, Salvatore | - | |
A Non-Peptide NK1 Receptor Agonist Showing Subpicomolar Affinity | 1-gen-2004 | Cappelli, Andrea; Giuliani, Germano; PERICOT MOHR GL, G; Gallelli, A; Anzini, Maurizio; Vomero, Salvatore; Cupello, A; Scarrone, S; Matarrese, M; Moresco, Rm; Fazio, F; Finetti, Federica; Morbidelli, Lucia; Ziche, Marina | - | |
A non-toxic, reversibly released imaging probe for oral cancer that is derived from natural compounds | 1-gen-2021 | Ghanim, Magda; Relitti, Nicola; Mcmanus, Gavin; Butini, Stefania; Cappelli, Andrea; Campiani, Giuseppe; Mok, K H; Kelly, Vincent P | - | |
A stereoselective approach to peptidomimetic BACE1 inhibitors | 1-gen-2013 | Butini, Stefania; Emanuele, Gabellieri; Brindisi, Margherita; Giovani, Simone; Maramai, Samuele; Kshirsagar, Giridhar; Egeria, Guarino; Brogi, Simone; Valeria La, Pietra; Mariateresa, Giustiniano; Luciana, Marinelli; Ettore, Novellino; Campiani, Giuseppe; Cappelli, Andrea; Gemma, Sandra | - | |
Age and Sex Influence the Neuro-inflammatory Response to a Peripheral Acute LPS Challenge | 1-gen-2019 | Murtaj, V.; Belloli, S.; Di Grigoli, G.; Pannese, M.; Ballarini, E.; Rodriguez-Menendez, V.; Marmiroli, P.; Cappelli, A.; Masiello, V.; Monterisi, C.; Bellelli, G.; Panina-Bordignon, P.; Moresco, R. M. | - | |
Aggregation-Induced Förster Resonance Energy Transfer in Polybenzofulvene/Dye Nanoparticles | 1-gen-2015 | Villafiorita Monteleone, Francesca; Cappelli, Andrea; Paolino, Marco; Colombo, Miriam; Cariati, Elena; Mura, Andrea; Bongiovanni, Giovanni; Botta, Chiara | - | |
Amidine, Thiourea and Guanidine Derivatives of 2-Aminobenzothiazoles and Aminobenzothiazines, Novel Pharmacological Agents for the Treatment of Neurodegenerative Pathologies | 1-gen-2007 | Anzini, Maurizio; A., Giordani; F., Makovec; Cappelli, Andrea; Vomero, Salvatore; G., Caselli; L. C., Rovati | - | |
Anionic Polymerization of a Benzofulvene Monomer Leading to a Thermoreversible π-Stacked Polymer. Studies in Macromolecular and Aggregate Structure | 1-gen-2008 | Cappelli, Andrea; Galeazzi, S; Giuliani, Germano; Anzini, Maurizio; Aggravi, M; Donati, Alessandro; Zetta, L; Boccia, A; Mendichi, R; Giorgi, Gianluca; Paccagnini, Eugenio; Vomero, Salvatore | - | |
Antiamnestic Effect of the Two Novel k-Opioid Agonists, VA-100 and VA-101, in the Mouse Passive Avoidance Test | 1-gen-2001 | Ghelardini, C.; Galeotti, N.; DI CESARE MANNELLI, L.; Cappelli, Andrea; Anzini, Maurizio; Bartolini, A. | - | |
Antiproliferative effect of two novel COX-2 inhibitors on human keratinocytes | 1-gen-2013 | Sticozzi, Claudia; Belmonte, Giuseppe; Cervellati, Franco; Di Capua, Angela; Maioli, Emanuela; Cappelli, Andrea; Giordani, Antonio; Biava, Mariangela; Anzini, Maurizio; Valacchi, Giuseppe | - | |
Aromatase and 5-alpha reductase gene expression: modulation by pain and morphine treatment in male rats | 1-gen-2010 | Aloisi, ANNA MARIA; Ceccarelli, I; Fiorenzani, P; Maddalena, M; Rossi, A; Tomei, V; Sorda, G; Danielli, B; Rovini, M; Cappelli, Andrea; Anzini, Maurizio; Giordano, Antonio | - | |
Bithiophene-based polybenzofulvene derivatives with high stacking and hole mobility | 1-gen-2015 | Cappelli, Andrea; Razzano, Vincenzo; Paolino, Marco; Grisci, Giorgio; Giuliani, Germano; Donati, Alessandro; Mendichi, Raniero; Samperi, Filippo; Battiato, Salvatore; Boccia, Antonella Caterina; Mura, Andrea; Bongiovanni, Giovanni; Mróz, Wojciech; Botta, Chiara | - | |
Bivalent Ligands for the Serotonin 5-HT3 Receptor | 1-gen-2011 | Cappelli, Andrea; Manini, Monica; Paolino, Marco; A., Gallelli; Anzini, Maurizio; L., Mennuni; M., DEL CADIA; F., DE RIENZO; M. C., Menziani; Vomero, Salvatore | - |