CARULLO, GABRIELE
CARULLO, GABRIELE
Dipartimento di Biotecnologie, Chimica e Farmacia
3-Amino-alkylated indoles: Unexplored green products acting as anti-inflammatory agents
2020-01-01 Mazzotta, S.; Frattaruolo, L.; Brindisi, M.; Ulivieri, C.; Vanni, F.; Brizzi, A.; Carullo, G.; Cappello, A. R.; Aiello, F.
7-docosahexaenoyl-quercetin
2021-01-01 Mazzotta, S.; Carullo, G.; Sciubba, F.; Di Cocco, M. E.; Aiello, F.
A multitarget semi-synthetic derivative of the flavonoid morin with improved in vitro vasorelaxant activity: Role of CaV1.2 and KCa1.1 channels
2021-01-01 Carullo, G.; Ahmed, A.; Trezza, A.; Spiga, O.; Brizzi, A.; Saponara, S.; Fusi, F.; Aiello, F.
A novel potent class I HDAC inhibitor reverses the STAT4/p66Shc apoptotic defect in B cells from chronic lymphocytic leukemia patients
2024-01-01 Rossi, Sara; Tatangelo, Vanessa; Dichiara, Maria; Butini, Stefania; Gemma, Sandra; Brogi, Simone; Pasquini, Silvia; Cappello, Martina; Vincenzi, Fabrizio; Varani, Katia; Lopresti, Ludovica; Malchiodi, Margherita; Carrara, Chiara; Gozzetti, Alessandro; Bocchia, Monica; Marotta, Giuseppe; Patrussi, Laura; Carullo, Gabriele; Baldari, Cosima T.; Campiani, Giuseppe
A Therapeutic Perspective of HDAC8 in Different Diseases: An Overview of Selective Inhibitors
2022-01-01 Fontana, A.; Cursaro, I.; Carullo, G.; Gemma, S.; Butini, S.; Campiani, G.
An ancient remedial repurposing: synthesis of new pinocembrin fatty acid acyl derivatives as potential antimicrobial/anti-inflammatory agents
2019-01-01 Tundis, Rosa; Frattaruolo, Luca; Carullo, Gabriele; Armentano, Biagio; Badolato, Mariateresa; Rosa Loizzo, Monica; Aiello, Francesca; Rita Cappello, Anna
Anti-Inflammatory and Antinociceptive Properties of the Quercetin-3-Oleate AV2, a Novel FFAR1 Partial Agonist
2024-01-01 Pessina, Federica; Casini, Ilenia; Gamberucci, Alessandra; Carullo, Gabriele; Signorini, Cinzia; Brizzi, Antonella; Aiello, Francesca; Aloisi, Anna Maria; Pieretti, Stefano
Antioxidant and Anti-Inflammatory Activities of Flavanones from Glycyrrhiza glabra L. (licorice) Leaf Phytocomplexes: Identification of Licoflavanone as a Modulator of NF-kB/MAPK Pathway
2019-01-01 Frattaruolo, Luca; Carullo, Gabriele; Brindisi, Matteo; Mazzotta, Sarah; Bellissimo, Luca; Rago, Vittoria; Curcio, Rosita; Dolce, Vincenza; Aiello, Francesca; Cappello, Anna Rita
Artificial intelligence-driven identification of morin analogues acting as CaV1.2 channel blockers: synthesis and biological evaluation
2023-01-01 Carullo, G.; Falbo, F.; Ahmed, A.; Trezza, A.; Gianibbi, B.; Nicolotti, O.; Campiani, G.; Aiello, F.; Saponara, S.; Fusi, F.
Autochthonous white grape pomaces as bioactive source for functional jams
2019-01-01 Restuccia, D.; Giorgi, G.; Gianfranco Spizzirri, U.; Sciubba, F.; Capuani, G.; Rago, V.; Carullo, G.; Aiello, F.
Azetidin-2-one-based small molecules as dual hHDAC6/HDAC8 inhibitors: Investigation of their mechanism of action and impact of dual inhibition profile on cell viability
2022-01-01 Federico, S.; Khan, T.; Fontana, A.; Brogi, S.; Benedetti, R.; Sarno, F.; Carullo, G.; Pezzotta, A.; Saraswati, A. P.; Passaro, E.; Pozzetti, L.; Papa, A.; Relitti, N.; Gemma, S.; Butini, S.; Pistocchi, A.; Ramunno, A.; Vincenzi, F.; Varani, K.; Tatangelo, V.; Patrussi, L.; Baldari, C. T.; Saponara, S.; Gorelli, B.; Lamponi, S.; Valoti, M.; Saccoccia, F.; Giannaccari, M.; Ruberti, G.; Herp, D.; Jung, M.; Altucci, L.; Campiani, G.
Biostimulants for Sustainable Food Production: Effects of Wood Distillate to Fortify Chickpea Flour for Development of Functional Bakery Products
2024-01-01 Fedeli, Riccardo; Spizzirri, Umile Gianfranco; Aquino, Giovanna; Basilicata, Manuela Giovanna; Pepe, Giacomo; Campiglia, Pietro; Celletti, Silvia; Tudino, Valeria; Dichiara, Maria; Gemma, Sandra; Butini, Stefania; Carullo, Gabriele; Aiello, Francesca; Restuccia, Donatella; Campiani, Giuseppe; Loppi, Stefano
Design and synthesis of multifunctional microtubule targeting agents endowed with dual pro-apoptotic and anti-autophagic efficacy
2022-01-01 Campiani, Giuseppe; Khan, Tuhina; Ulivieri, Cristina; Staiano, Leopoldo; Papulino, Chiara; Magnano, Stefania; Nathwani, Seema; Ramunno, Anna; Lucena-Agell, Daniel; Relitti, Nicola; Federico, Stefano; Pozzetti, Luca; Carullo, Gabriele; Casagni, Alice; Brogi, Simone; Vanni, Francesca; Galatello, Paola; Ghanim, Magda; Mccabe, Niamh; Lamponi, Stefania; Valoti, Massimo; Ibrahim, Ola; O'Sullivan, Jeffrey; Turkington, Richard; Kelly, Vincent P.; Vanwemmel, Ruben; Díaz, J. Fernando; Gemma, Sandra; Zisterer, Daniela; Altucci, Lucia; De Matteis, Antonella; Butini, Stefania; Benedetti, Rosaria
Design and Synthesis of Oligopeptidic Parvulin Inhibitors
2022-01-01 Relitti, N.; Prasanth Saraswati, A.; Carullo, G.; Papa, A.; Monti, A.; Benedetti, R.; Passaro, E.; Brogi, S.; Calderone, V.; Butini, S.; Gemma, S.; Altucci, L.; Campiani, G.; Doti, N.
Design, synthesis and in vitro experimental validation of novel TRPV4 antagonists inspired by labdane diterpenes
2020-01-01 Mazzotta, S.; Carullo, G.; Schiano Moriello, A.; Amodeo, P.; Di Marzo, V.; Vega-Holm, M.; Vitale, R. M.; Aiello, F.; Brizzi, A.; De Petrocellis, L.
Design, synthesis and pharmacological evaluation of ester-based quercetin derivatives as selective vascular KCa1.1 channel stimulators
2020-01-01 Carullo, G.; Ahmed, A.; Trezza, A.; Spiga, O.; Brizzi, A.; Saponara, S.; Fusi, F.; Aiello, F.
Development of 1-(2-aminophenyl)pyrrole-based amides acting as human topoisomerase I inhibitors
2023-01-01 Carullo, Gabriele; Mazzotta, Sarah; Ceramella, Jessica; Iacopetta, Domenico; Ramunno, Anna; Rosano, Camillo; Brizzi, Antonella; Campiani, Giuseppe; Aiello, Francesca; Sinicropi, Maria S
Development of Epigenetic Modifiers with Therapeutic Potential in FMS-Related Tyrosine Kinase 3/Internal Tandem Duplication (FLT3/ITD) Acute Myeloid Leukemia and Other Blood Malignancies
2024-01-01 Carullo, Gabriele; Rossi, Sara; Giudice, Valentina; Pezzotta, Alex; Chianese, Ugo; Scala, Pasqualina; Carbone, Sabrina; Fontana, Anna; Panzeca, Giovanna; Pasquini, Silvia; Contri, Chiara; Gemma, Sandra; Ramunno, Anna; Saponara, Simona; Galvani, Francesca; Lodola, Alessio; Mor, Marco; Benedetti, Rosaria; Selleri, Carmine; Varani, Katia; Butini, Stefania; Altucci, Lucia; Vincenzi, Fabrizio; Pistocchi, Anna; Campiani, Giuseppe
Development of potent and selective FAAH inhibitors with improved drug-like properties as potential tools to treat neuroinflammatory conditions
2023-01-01 Papa, Alessandro; Pasquini, Silvia; Galvani, Francesca; Cammarota, Mariarosaria; Contri, Chiara; Carullo, Gabriele; Gemma, Sandra; Ramunno, Anna; Lamponi, Stefania; Gorelli, Beatrice; Saponara, Simona; Varani, Katia; Mor, Marco; Campiani, Giuseppe; Boscia, Francesca; Vincenzi, Fabrizio; Lodola, Alessio; Butini, Stefania
Development of Potent and Selective Monoacylglycerol Lipase Inhibitors. SARs, Structural Analysis, and Biological Characterization
2024-01-01 Butini, Stefania; Grether, Uwe; Jung, Kwang-Mook; Ligresti, Alessia; Allarà, Marco; Postmus, Annemarieke G. J.; Maramai, Samuele; Brogi, Simone; Papa, Alessandro; Carullo, Gabriele; Sykes, David; Veprintsev, Dmitry; Federico, Stefano; Grillo, Alessandro; Di Guglielmo, Bruno; Ramunno, Anna; Stevens, Anna Floor; Heer, Dominik; Lamponi, Stefania; Gemma, Sandra; Benz, Jörg; Di Marzo, Vincenzo; van der Stelt, Mario; Piomelli, Daniele; Campiani, Giuseppe
| Titolo | Data di pubblicazione | Autore(i) | File | Abstract |
|---|---|---|---|---|
| 3-Amino-alkylated indoles: Unexplored green products acting as anti-inflammatory agents | 1-gen-2020 | Mazzotta, S.; Frattaruolo, L.; Brindisi, M.; Ulivieri, C.; Vanni, F.; Brizzi, A.; Carullo, G.; Cappello, A. R.; Aiello, F. | - | |
| 7-docosahexaenoyl-quercetin | 1-gen-2021 | Mazzotta, S.; Carullo, G.; Sciubba, F.; Di Cocco, M. E.; Aiello, F. | - | |
| A multitarget semi-synthetic derivative of the flavonoid morin with improved in vitro vasorelaxant activity: Role of CaV1.2 and KCa1.1 channels | 1-gen-2021 | Carullo, G.; Ahmed, A.; Trezza, A.; Spiga, O.; Brizzi, A.; Saponara, S.; Fusi, F.; Aiello, F. | - | |
| A novel potent class I HDAC inhibitor reverses the STAT4/p66Shc apoptotic defect in B cells from chronic lymphocytic leukemia patients | 1-gen-2024 | Rossi, Sara; Tatangelo, Vanessa; Dichiara, Maria; Butini, Stefania; Gemma, Sandra; Brogi, Simone; Pasquini, Silvia; Cappello, Martina; Vincenzi, Fabrizio; Varani, Katia; Lopresti, Ludovica; Malchiodi, Margherita; Carrara, Chiara; Gozzetti, Alessandro; Bocchia, Monica; Marotta, Giuseppe; Patrussi, Laura; Carullo, Gabriele; Baldari, Cosima T.; Campiani, Giuseppe | - | |
| A Therapeutic Perspective of HDAC8 in Different Diseases: An Overview of Selective Inhibitors | 1-gen-2022 | Fontana, A.; Cursaro, I.; Carullo, G.; Gemma, S.; Butini, S.; Campiani, G. | - | |
| An ancient remedial repurposing: synthesis of new pinocembrin fatty acid acyl derivatives as potential antimicrobial/anti-inflammatory agents | 1-gen-2019 | Tundis, Rosa; Frattaruolo, Luca; Carullo, Gabriele; Armentano, Biagio; Badolato, Mariateresa; Rosa Loizzo, Monica; Aiello, Francesca; Rita Cappello, Anna | - | |
| Anti-Inflammatory and Antinociceptive Properties of the Quercetin-3-Oleate AV2, a Novel FFAR1 Partial Agonist | 1-gen-2024 | Pessina, Federica; Casini, Ilenia; Gamberucci, Alessandra; Carullo, Gabriele; Signorini, Cinzia; Brizzi, Antonella; Aiello, Francesca; Aloisi, Anna Maria; Pieretti, Stefano | - | |
| Antioxidant and Anti-Inflammatory Activities of Flavanones from Glycyrrhiza glabra L. (licorice) Leaf Phytocomplexes: Identification of Licoflavanone as a Modulator of NF-kB/MAPK Pathway | 1-gen-2019 | Frattaruolo, Luca; Carullo, Gabriele; Brindisi, Matteo; Mazzotta, Sarah; Bellissimo, Luca; Rago, Vittoria; Curcio, Rosita; Dolce, Vincenza; Aiello, Francesca; Cappello, Anna Rita | - | |
| Artificial intelligence-driven identification of morin analogues acting as CaV1.2 channel blockers: synthesis and biological evaluation | 1-gen-2023 | Carullo, G.; Falbo, F.; Ahmed, A.; Trezza, A.; Gianibbi, B.; Nicolotti, O.; Campiani, G.; Aiello, F.; Saponara, S.; Fusi, F. | - | |
| Autochthonous white grape pomaces as bioactive source for functional jams | 1-gen-2019 | Restuccia, D.; Giorgi, G.; Gianfranco Spizzirri, U.; Sciubba, F.; Capuani, G.; Rago, V.; Carullo, G.; Aiello, F. | - | |
| Azetidin-2-one-based small molecules as dual hHDAC6/HDAC8 inhibitors: Investigation of their mechanism of action and impact of dual inhibition profile on cell viability | 1-gen-2022 | Federico, S.; Khan, T.; Fontana, A.; Brogi, S.; Benedetti, R.; Sarno, F.; Carullo, G.; Pezzotta, A.; Saraswati, A. P.; Passaro, E.; Pozzetti, L.; Papa, A.; Relitti, N.; Gemma, S.; Butini, S.; Pistocchi, A.; Ramunno, A.; Vincenzi, F.; Varani, K.; Tatangelo, V.; Patrussi, L.; Baldari, C. T.; Saponara, S.; Gorelli, B.; Lamponi, S.; Valoti, M.; Saccoccia, F.; Giannaccari, M.; Ruberti, G.; Herp, D.; Jung, M.; Altucci, L.; Campiani, G. | - | |
| Biostimulants for Sustainable Food Production: Effects of Wood Distillate to Fortify Chickpea Flour for Development of Functional Bakery Products | 1-gen-2024 | Fedeli, Riccardo; Spizzirri, Umile Gianfranco; Aquino, Giovanna; Basilicata, Manuela Giovanna; Pepe, Giacomo; Campiglia, Pietro; Celletti, Silvia; Tudino, Valeria; Dichiara, Maria; Gemma, Sandra; Butini, Stefania; Carullo, Gabriele; Aiello, Francesca; Restuccia, Donatella; Campiani, Giuseppe; Loppi, Stefano | - | |
| Design and synthesis of multifunctional microtubule targeting agents endowed with dual pro-apoptotic and anti-autophagic efficacy | 1-gen-2022 | Campiani, Giuseppe; Khan, Tuhina; Ulivieri, Cristina; Staiano, Leopoldo; Papulino, Chiara; Magnano, Stefania; Nathwani, Seema; Ramunno, Anna; Lucena-Agell, Daniel; Relitti, Nicola; Federico, Stefano; Pozzetti, Luca; Carullo, Gabriele; Casagni, Alice; Brogi, Simone; Vanni, Francesca; Galatello, Paola; Ghanim, Magda; Mccabe, Niamh; Lamponi, Stefania; Valoti, Massimo; Ibrahim, Ola; O'Sullivan, Jeffrey; Turkington, Richard; Kelly, Vincent P.; Vanwemmel, Ruben; Díaz, J. Fernando; Gemma, Sandra; Zisterer, Daniela; Altucci, Lucia; De Matteis, Antonella; Butini, Stefania; Benedetti, Rosaria | - | |
| Design and Synthesis of Oligopeptidic Parvulin Inhibitors | 1-gen-2022 | Relitti, N.; Prasanth Saraswati, A.; Carullo, G.; Papa, A.; Monti, A.; Benedetti, R.; Passaro, E.; Brogi, S.; Calderone, V.; Butini, S.; Gemma, S.; Altucci, L.; Campiani, G.; Doti, N. | - | |
| Design, synthesis and in vitro experimental validation of novel TRPV4 antagonists inspired by labdane diterpenes | 1-gen-2020 | Mazzotta, S.; Carullo, G.; Schiano Moriello, A.; Amodeo, P.; Di Marzo, V.; Vega-Holm, M.; Vitale, R. M.; Aiello, F.; Brizzi, A.; De Petrocellis, L. | - | |
| Design, synthesis and pharmacological evaluation of ester-based quercetin derivatives as selective vascular KCa1.1 channel stimulators | 1-gen-2020 | Carullo, G.; Ahmed, A.; Trezza, A.; Spiga, O.; Brizzi, A.; Saponara, S.; Fusi, F.; Aiello, F. | - | |
| Development of 1-(2-aminophenyl)pyrrole-based amides acting as human topoisomerase I inhibitors | 1-gen-2023 | Carullo, Gabriele; Mazzotta, Sarah; Ceramella, Jessica; Iacopetta, Domenico; Ramunno, Anna; Rosano, Camillo; Brizzi, Antonella; Campiani, Giuseppe; Aiello, Francesca; Sinicropi, Maria S | - | |
| Development of Epigenetic Modifiers with Therapeutic Potential in FMS-Related Tyrosine Kinase 3/Internal Tandem Duplication (FLT3/ITD) Acute Myeloid Leukemia and Other Blood Malignancies | 1-gen-2024 | Carullo, Gabriele; Rossi, Sara; Giudice, Valentina; Pezzotta, Alex; Chianese, Ugo; Scala, Pasqualina; Carbone, Sabrina; Fontana, Anna; Panzeca, Giovanna; Pasquini, Silvia; Contri, Chiara; Gemma, Sandra; Ramunno, Anna; Saponara, Simona; Galvani, Francesca; Lodola, Alessio; Mor, Marco; Benedetti, Rosaria; Selleri, Carmine; Varani, Katia; Butini, Stefania; Altucci, Lucia; Vincenzi, Fabrizio; Pistocchi, Anna; Campiani, Giuseppe | - | |
| Development of potent and selective FAAH inhibitors with improved drug-like properties as potential tools to treat neuroinflammatory conditions | 1-gen-2023 | Papa, Alessandro; Pasquini, Silvia; Galvani, Francesca; Cammarota, Mariarosaria; Contri, Chiara; Carullo, Gabriele; Gemma, Sandra; Ramunno, Anna; Lamponi, Stefania; Gorelli, Beatrice; Saponara, Simona; Varani, Katia; Mor, Marco; Campiani, Giuseppe; Boscia, Francesca; Vincenzi, Fabrizio; Lodola, Alessio; Butini, Stefania | - | |
| Development of Potent and Selective Monoacylglycerol Lipase Inhibitors. SARs, Structural Analysis, and Biological Characterization | 1-gen-2024 | Butini, Stefania; Grether, Uwe; Jung, Kwang-Mook; Ligresti, Alessia; Allarà, Marco; Postmus, Annemarieke G. J.; Maramai, Samuele; Brogi, Simone; Papa, Alessandro; Carullo, Gabriele; Sykes, David; Veprintsev, Dmitry; Federico, Stefano; Grillo, Alessandro; Di Guglielmo, Bruno; Ramunno, Anna; Stevens, Anna Floor; Heer, Dominik; Lamponi, Stefania; Gemma, Sandra; Benz, Jörg; Di Marzo, Vincenzo; van der Stelt, Mario; Piomelli, Daniele; Campiani, Giuseppe | - |