MANGANI, STEFANO
MANGANI, STEFANO
Dipartimento di Biotecnologie, Chimica e Farmacia
1,2,4-Triazole-3-Thione Analogues with a 2-Ethylbenzoic Acid at Position 4 as VIM-type Metallo-β-Lactamase Inhibitors
2022-01-01 Verdirosa, Federica; Gavara, Laurent; Sevaille, Laurent; Tassone, Giusy; Corsica, Giuseppina; Legru, Alice; Feller, Georges; Chelini, Giulia; Mercuri, Paola Sandra; Tanfoni, Silvia; Sannio, Filomena; Benvenuti, Manuela; Cerboni, Giulia; De Luca, Filomena; Bouajila, Ezeddine; Vo Hoang, Yen; Licznar-Fajardo, Patricia; Galleni, Moreno; Pozzi, Cecilia; Mangani, Stefano; Docquier, Jean-Denis; Hernandez, Jean-François
1,2,4-Triazole-3-thione compounds with a 4-ethyl alkyl/aryl sulfide substituent are broad-spectrum metallo-β-lactamase inhibitors with re-sensitization activity
2021-01-01 Legru, Alice; Verdirosa, Federica; Hernandez, Jean-François; Tassone, Giusy; Sannio, Filomena; Benvenuti, Manuela; Conde, Pierre-Alexis; Bossis, Guillaume; Thomas, Caitlyn A; Crowder, Michael W; Dillenberger, Melissa; Becker, Katja; Pozzi, Cecilia; Mangani, Stefano; Docquier, Jean-Denis; Gavara, Laurent
2'-Deoxyuridine 5'-monophosphate substrate displacement in thymidylate synthase through 6-hydroxy-2H-naphtho[1,8-bc]furan-2-one derivatives
2013-01-01 Ferrari, Stefania; Calò, Samuele; Leone, Rosalida; Luciani, Rosaria; Costantino, Luca; Sammak, Susan; DI PISA, Flavio; Pozzi, Cecilia; Mangani, Stefano; Costi, M. Paola
4-Amino-1,2,4-triazole-3-thione-derived Schiff bases as metallo-β-lactamase inhibitors
2020-01-01 Gavara, L.; Sevaille, L.; De Luca, F.; Mercuri, P.; Bebrone, C.; Feller, G.; Legru, A.; Cerboni, G.; Tanfoni, S.; Baud, D.; Cutolo, G.; Bestgen, B.; Chelini, G.; Verdirosa, F.; Sannio, F.; Pozzi, C.; Benvenuti, M.; Kwapien, K.; Fischer, M.; Becker, K.; Frere, J. -M.; Mangani, S.; Gresh, N.; Berthomieu, D.; Galleni, M.; Docquier, Jd; Hernandez, J. -F.
4-Chlorocatechol 1,2-dioxygenase from the chlorophenol-utilizing Gram-positive Rhodococcus opacus 1CP: crystallization and preliminary crystallographic analysis
2002-01-01 M., Ferraroni; M. Y., R.; F., Briganti; A., Scozzafava; Mangani, Stefano; I. P., Solyanikova; M. P., Kolomysteva; L., Golovleva
A copper(I) protein possibly involved in the assembly of Cu-A center of bacterial cytochrome c oxidase
2005-01-01 L., Banci; I., Bertini; S., Ciofi Baffoni; E., Katsari; N., Katsaros; K., Kubicek; Mangani, Stefano
A hint for the function of human Sco1 from different structures
2006-01-01 L., Banci; I., Bertini; V., Calderone; S., Ciofi Baffoni; Mangani, Stefano; M., Martinelli; P., Palumaa; S. L., Wang
A hint for the function of human Sco1 from different structures (vol 103, pg 8595, 2006)
2006-01-01 L., Banci; I., Bertini; V., Calderone; S., Ciofi Baffoni; Mangani, Stefano; M., Martinelli; P., Palumaa; S. L., Wang
A new proposal for urease mechanism based on the crystal structures of the native and inhibited enzyme from Bacillus pasteurii: why urea hydrolysis casts two nickels
1999-01-01 S., Benini; W. R., Rypniewski; K. S., Wilson; S., Miletti; S., Ciurli; Mangani, Stefano
A prokaryotic superoxide dismutase paralog lacking two Cu ligands: From largely unstructured in solution to ordered in the crystal
2005-01-01 L., Banci; I., Bertini; V., Calderone; F., Cramaro; R. D., Conte; A., Fantoni; Mangani, Stefano; A., Quattrone; M. S., Viezzoli
A redox switch in CopC: An intriguing copper trafficking protein that binds copper(I) and copper(II) at different sites
2003-01-01 F., Arnesano; L., Banci; I., Bertini; Mangani, Stefano; A. R., Thompsett
A structure-based proposal for the catalytic mechanism of the bacterial acid phosphatase AphA belonging to the DDDD superfamily of phosphohydrolases
2006-01-01 V., Calderone; C., Forleo; Benvenuti, Manuela; M. C., Thaller; Rossolini, GIAN MARIA; Mangani, Stefano
A ternary complex of carbonic anhydrase: X-ray crystallographic structure of the adduct of human carbonic anhydrase II with the activator phenylalanine and the inhibitor azide
1998-01-01 F., Briganti; V., Iaconi; Mangani, Stefano; P., Orioli; A., Scozzafava; G., Vernaglione; C. T., Supuran
Accelerating Drug Discovery Efforts for Trypanosomatidic Infections Using an Integrated Transnational Academic Drug Discovery Platform
2019-01-01 Moraes, Carolina B.; Witt, Gesa; Kuzikov, Maria; Ellinger, Bernhard; Calogeropoulou, Theodora; Prousis, Kyriakos C.; Mangani, Stefano; Di Pisa, Flavio; Landi, Giacomo; Iacono, Lucia Dello; Pozzi, Cecilia; Freitas-Junior, Lucio H.; dos Santos Pascoalino, Bruno; Bertolacini, Claudia P.; Behrens, Birte; Keminer, Oliver; Leu, Jennifer; Wolf, Markus; Reinshagen, Jeanette; Cordeiro-da-Silva, Anabela; Santarem, Nuno; Venturelli, Alberto; Wrigley, Stephen; Karunakaran, Deepa; Kebede, Bethlehem; Pöhner, Ina; Müller, Wolfgang; Panecka-Hofman, Joanna; Wade, Rebecca C.; Fenske, Martina; Clos, Joachim; Alunda, José María; Corral, María Jesús; Uliassi, Elisa; Bolognesi, Maria Laura; Linciano, Pasquale; Quotadamo, Antonio; Ferrari, Stefania; Santucci, Matteo; Borsari, Chiara; Costi, Maria Paola; Gul, Sheraz
Amino-thiadiazole as innovative inhibitors of human glutaminyl cyclase for the treatment of Alzheimer disease
2018-01-01 Pozzi, Cecilia; Tassone, Giusy; Linciano, Pasquale; Costi, MARIA PAOLA; Mangani, Stefano
Amino-thiadiazole as innovative inhibitors of human glutaminyl cyclase, a validated target towards Alzheimer disease
2018-01-01 Pozzi, Cecilia; Tassone, Giusy; Linciano, Pasquale; Benvenuti, Manuela; Costi, MARIA PAOLA; Mangani, Stefano
An Italian contribution to structural genomics: Understanding metalloproteins
2006-01-01 F., Arnesano; L., Banci; I., Bertini; F., Capozzi; S., Ciofi Baffoni; S., Ciurli; C., Luchinat; Mangani, Stefano; A., Rosato; P., Turano; M. S., Viezzoli
An update on β-lactamase inhibitor discovery and development
2018-01-01 Docquier, Jean-Denis; Mangani, Stefano
Anion Coordination Chemistry - Crystal-structure of the Super Complex - [h81,4,7,10,13,16,19,22,25,28-deca-azacyclotriacontane][co(cn)6]2cl2.10h 2o
1987-01-01 Bianchi, Antonio; Garcia-España, Enrique; Mangani, Stefano; Micheloni, Mauro; Orioli, Pierluigi; Paoletti, Piero
Anion Coordination Chemistry .2. Electrochemical, Thermodynamic, and Structural Studies On Supercomplex Formation Between Large Polyammonium Cycloalkanes and the 2 Complex Anions Hexacyanoferrate(ii) and Hexacyanocobaltate(iii)
1987-01-01 Bencini, Andrea; Bianchi, Antonio; Garcia-españa, Enrique; Giusti, Mauro; Mangani, Stefano; Micheloni, Mauro; Orioli, Pierluigi; Paoletti, Piero
Titolo | Data di pubblicazione | Autore(i) | File | Abstract |
---|---|---|---|---|
1,2,4-Triazole-3-Thione Analogues with a 2-Ethylbenzoic Acid at Position 4 as VIM-type Metallo-β-Lactamase Inhibitors | 1-gen-2022 | Verdirosa, Federica; Gavara, Laurent; Sevaille, Laurent; Tassone, Giusy; Corsica, Giuseppina; Legru, Alice; Feller, Georges; Chelini, Giulia; Mercuri, Paola Sandra; Tanfoni, Silvia; Sannio, Filomena; Benvenuti, Manuela; Cerboni, Giulia; De Luca, Filomena; Bouajila, Ezeddine; Vo Hoang, Yen; Licznar-Fajardo, Patricia; Galleni, Moreno; Pozzi, Cecilia; Mangani, Stefano; Docquier, Jean-Denis; Hernandez, Jean-François | - | |
1,2,4-Triazole-3-thione compounds with a 4-ethyl alkyl/aryl sulfide substituent are broad-spectrum metallo-β-lactamase inhibitors with re-sensitization activity | 1-gen-2021 | Legru, Alice; Verdirosa, Federica; Hernandez, Jean-François; Tassone, Giusy; Sannio, Filomena; Benvenuti, Manuela; Conde, Pierre-Alexis; Bossis, Guillaume; Thomas, Caitlyn A; Crowder, Michael W; Dillenberger, Melissa; Becker, Katja; Pozzi, Cecilia; Mangani, Stefano; Docquier, Jean-Denis; Gavara, Laurent | - | |
2'-Deoxyuridine 5'-monophosphate substrate displacement in thymidylate synthase through 6-hydroxy-2H-naphtho[1,8-bc]furan-2-one derivatives | 1-gen-2013 | Ferrari, Stefania; Calò, Samuele; Leone, Rosalida; Luciani, Rosaria; Costantino, Luca; Sammak, Susan; DI PISA, Flavio; Pozzi, Cecilia; Mangani, Stefano; Costi, M. Paola | - | |
4-Amino-1,2,4-triazole-3-thione-derived Schiff bases as metallo-β-lactamase inhibitors | 1-gen-2020 | Gavara, L.; Sevaille, L.; De Luca, F.; Mercuri, P.; Bebrone, C.; Feller, G.; Legru, A.; Cerboni, G.; Tanfoni, S.; Baud, D.; Cutolo, G.; Bestgen, B.; Chelini, G.; Verdirosa, F.; Sannio, F.; Pozzi, C.; Benvenuti, M.; Kwapien, K.; Fischer, M.; Becker, K.; Frere, J. -M.; Mangani, S.; Gresh, N.; Berthomieu, D.; Galleni, M.; Docquier, Jd; Hernandez, J. -F. | - | |
4-Chlorocatechol 1,2-dioxygenase from the chlorophenol-utilizing Gram-positive Rhodococcus opacus 1CP: crystallization and preliminary crystallographic analysis | 1-gen-2002 | M., Ferraroni; M. Y., R.; F., Briganti; A., Scozzafava; Mangani, Stefano; I. P., Solyanikova; M. P., Kolomysteva; L., Golovleva | - | |
A copper(I) protein possibly involved in the assembly of Cu-A center of bacterial cytochrome c oxidase | 1-gen-2005 | L., Banci; I., Bertini; S., Ciofi Baffoni; E., Katsari; N., Katsaros; K., Kubicek; Mangani, Stefano | - | |
A hint for the function of human Sco1 from different structures | 1-gen-2006 | L., Banci; I., Bertini; V., Calderone; S., Ciofi Baffoni; Mangani, Stefano; M., Martinelli; P., Palumaa; S. L., Wang | - | |
A hint for the function of human Sco1 from different structures (vol 103, pg 8595, 2006) | 1-gen-2006 | L., Banci; I., Bertini; V., Calderone; S., Ciofi Baffoni; Mangani, Stefano; M., Martinelli; P., Palumaa; S. L., Wang | - | |
A new proposal for urease mechanism based on the crystal structures of the native and inhibited enzyme from Bacillus pasteurii: why urea hydrolysis casts two nickels | 1-gen-1999 | S., Benini; W. R., Rypniewski; K. S., Wilson; S., Miletti; S., Ciurli; Mangani, Stefano | - | |
A prokaryotic superoxide dismutase paralog lacking two Cu ligands: From largely unstructured in solution to ordered in the crystal | 1-gen-2005 | L., Banci; I., Bertini; V., Calderone; F., Cramaro; R. D., Conte; A., Fantoni; Mangani, Stefano; A., Quattrone; M. S., Viezzoli | - | |
A redox switch in CopC: An intriguing copper trafficking protein that binds copper(I) and copper(II) at different sites | 1-gen-2003 | F., Arnesano; L., Banci; I., Bertini; Mangani, Stefano; A. R., Thompsett | - | |
A structure-based proposal for the catalytic mechanism of the bacterial acid phosphatase AphA belonging to the DDDD superfamily of phosphohydrolases | 1-gen-2006 | V., Calderone; C., Forleo; Benvenuti, Manuela; M. C., Thaller; Rossolini, GIAN MARIA; Mangani, Stefano | - | |
A ternary complex of carbonic anhydrase: X-ray crystallographic structure of the adduct of human carbonic anhydrase II with the activator phenylalanine and the inhibitor azide | 1-gen-1998 | F., Briganti; V., Iaconi; Mangani, Stefano; P., Orioli; A., Scozzafava; G., Vernaglione; C. T., Supuran | - | |
Accelerating Drug Discovery Efforts for Trypanosomatidic Infections Using an Integrated Transnational Academic Drug Discovery Platform | 1-gen-2019 | Moraes, Carolina B.; Witt, Gesa; Kuzikov, Maria; Ellinger, Bernhard; Calogeropoulou, Theodora; Prousis, Kyriakos C.; Mangani, Stefano; Di Pisa, Flavio; Landi, Giacomo; Iacono, Lucia Dello; Pozzi, Cecilia; Freitas-Junior, Lucio H.; dos Santos Pascoalino, Bruno; Bertolacini, Claudia P.; Behrens, Birte; Keminer, Oliver; Leu, Jennifer; Wolf, Markus; Reinshagen, Jeanette; Cordeiro-da-Silva, Anabela; Santarem, Nuno; Venturelli, Alberto; Wrigley, Stephen; Karunakaran, Deepa; Kebede, Bethlehem; Pöhner, Ina; Müller, Wolfgang; Panecka-Hofman, Joanna; Wade, Rebecca C.; Fenske, Martina; Clos, Joachim; Alunda, José María; Corral, María Jesús; Uliassi, Elisa; Bolognesi, Maria Laura; Linciano, Pasquale; Quotadamo, Antonio; Ferrari, Stefania; Santucci, Matteo; Borsari, Chiara; Costi, Maria Paola; Gul, Sheraz | - | |
Amino-thiadiazole as innovative inhibitors of human glutaminyl cyclase for the treatment of Alzheimer disease | 1-gen-2018 | Pozzi, Cecilia; Tassone, Giusy; Linciano, Pasquale; Costi, MARIA PAOLA; Mangani, Stefano | - | |
Amino-thiadiazole as innovative inhibitors of human glutaminyl cyclase, a validated target towards Alzheimer disease | 1-gen-2018 | Pozzi, Cecilia; Tassone, Giusy; Linciano, Pasquale; Benvenuti, Manuela; Costi, MARIA PAOLA; Mangani, Stefano | - | |
An Italian contribution to structural genomics: Understanding metalloproteins | 1-gen-2006 | F., Arnesano; L., Banci; I., Bertini; F., Capozzi; S., Ciofi Baffoni; S., Ciurli; C., Luchinat; Mangani, Stefano; A., Rosato; P., Turano; M. S., Viezzoli | - | |
An update on β-lactamase inhibitor discovery and development | 1-gen-2018 | Docquier, Jean-Denis; Mangani, Stefano | - | |
Anion Coordination Chemistry - Crystal-structure of the Super Complex - [h81,4,7,10,13,16,19,22,25,28-deca-azacyclotriacontane][co(cn)6]2cl2.10h 2o | 1-gen-1987 | Bianchi, Antonio; Garcia-España, Enrique; Mangani, Stefano; Micheloni, Mauro; Orioli, Pierluigi; Paoletti, Piero | - | |
Anion Coordination Chemistry .2. Electrochemical, Thermodynamic, and Structural Studies On Supercomplex Formation Between Large Polyammonium Cycloalkanes and the 2 Complex Anions Hexacyanoferrate(ii) and Hexacyanocobaltate(iii) | 1-gen-1987 | Bencini, Andrea; Bianchi, Antonio; Garcia-españa, Enrique; Giusti, Mauro; Mangani, Stefano; Micheloni, Mauro; Orioli, Pierluigi; Paoletti, Piero | - |