NACCI, VITO

NACCI, VITO  

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Titolo Data di pubblicazione Autore(i) File Abstract
Activation of the c-Jun NH2 Terminal Kinase (JNK) Signalling Pathway is Essential During PBOX-6-Induced Apoptosis in Chronic Myelogenous leukemia (CML) Cells 1-gen-2002 MC GEE, M.; Campiani, G.; Ramunno, A.; Williams, C; Zisterer, D; Nacci, V.; Lawler, M. -
Antiproliferative action of pyrrolobenzoxazepine derivatives in cultured cells: Absence of correlation with binding to the peripheral-type benzodiazepine binding site 1-gen-1998 Daniela M., Zisterer; Nicole, Hance; Campiani, Giuseppe; Antonio, Garofalo; Nacci, Vito; D., Clive Williams -
An approach to modified heterocyclic analogues of huperzine A and isohuperzine A. Synthesis of the pyrimidone and pyrazole analogues, and their anticholinesterase activity 1-gen-1996 Alan P., Kozikowski; Campiani, Giuseppe; Nacci, Vito; Sega, Alessandro; Ashima, Saxena; Bhupendra P., Doctor -
Benzothiazine and Benzothiazepine derivatives: synthesis and preliminary biological evaluation 1-gen-1993 A., Garofalo; Campiani, Giuseppe; Fiorini, Isabella; Nacci, Vito -
Cardiovascular Characterization of Pyrrolo[2,1-d][1,5]benzothiazepine Derivatives Binding Selectively to the Peripheral-Type Benzodiazepine Receptor (PBR):  From Dual PBR Affinity and Calcium Antagonist Activity to Novel and Selective Calcium Entry Blockers 1-gen-1996 Campiani, Giuseppe; Fiorini, Isabella; Maria P., De Filippis; Silvia M., Ciani; Antonio, Garofalo; Nacci, Vito; Giorgi, Gianluca; Sega, Alessandro; Botta, Maurizio; Alberto, Chiarini; Roberta, Budriesi; Giancarlo, Bruni; Maria R., Romeo; Cristina, Manzoni; Tiziana, Mennini -
Caspase-3 is not essential for DNA fragmentation in MCF-7 cells during apoptosis induced by the pyrrolo-1,5-benzoxazepine, PBOX-6 1-gen-2002 M., MC GEE; E., Hyland; Campiani, Giuseppe; A., Ramunno; Nacci, Vito; Dm, Zisterer -
Characterisation of 1H-cyclopentapyrimidine-2,4(1H,3H)-dione derivative (S)-CPW399 as a novel, potent and subtype-selective AMPA receptor full agonist with partial desensitization properties 1-gen-2001 Campiani, Giuseppe; E., Morelli; Nacci, Vito; C., Fattorusso; A., Ramunno; E., Novellino; J., Greenwood; T., Liljefors; R., Griffiths; C., Sinclair; H., Reavy; A. S., Kristensen; D. S., Pickering; A., Schousboe; A., Cagnotto; E., Fumagalli; T., Mennini -
Clotrimazole Scaffold as an Innovative Pharmacophore Towards Potent Antimalarial Agents: Design, Synthesis, Biological and Structure-Activity Relationship Studies. 1-gen-2008 Gemma, Sandra; Campiani, Giuseppe; Butini, Stefania; G., Kukreja; SANNA COCCONE, Salvatore; B., Joshi; M., Persico; Nacci, Vito; Fiorini, Isabella; E., Novellino; Fattorusso, E; O., TAGLIALATELA SCAFATI; Savini, Luisa; D., Taramelli; N., Basilico; S., Parapini; G., Morace; V., Yardley; S., Croft; M., Coletta; S., Marini; Fattorusso, Caterina -
Combining 4-Aminoquinoline- and Clotrimazole-based Pharmacophores towards Innovative and Potent Hybrid Antimalarials. 1-gen-2009 Gemma, Sandra; Campiani, Giuseppe; Butini, Stefania; B. P., Joshi; G., Kukreja; SANNA COCCONE, Salvatore; Bernetti, Matteo; M., Persico; Nacci, Vito; Fiorini, Isabella; E., Novellino; D., Taramelli; N., Basilico; S., Parapini; V., Yardley; S., Croft; S., KELLER MAERKI; M., Rottmann; R., Brun; M., Coletta; S., Marini; G., Guiso; S., Caccia; C., Fattorusso -
A Comparative Molecular Field Analysis Model for 6-Arylpyrrolo[2,1-d][1,5]benzothiazepines Binding Selectively to the Mitochondrial Benzodiazepine Receptor 1-gen-1994 Giovanni, Greco; Ettore, Novellino; Fiorini, Isabella; Nacci, Vito; Campiani, Giuseppe; Silvia M., Ciani; Antonio, Garofalo; Paola, Bernasconi; Tiziana, Mennini -
A Concerted Study Using Binding Measurements, X-ray Structural Data, and Molecular Modeling on the Stereochemical Features Responsible for the Affinity of 6-Arylpyrrolo[2,1-d][1,5]benzothiazepines toward Mitochondrial Benzodiazepine Receptors 1-gen-1995 Alessandro, Dalpiaz; Valerio, Bertolasi; Pier Andrea, Borea; Nacci, Vito; Fiorini, Isabella; Campiani, Giuseppe; Tiziana, Mennini; Cristina, Manzoni; Ettore, Novellino; Giovanni, Greco -
Design and Synthesis of Potent Antimalarial Agents Based on Clotrimazole Scaffold: Exploring an Innovative Pharmacophore. 1-gen-2007 Gemma, Sandra; Campiani, Giuseppe; Butini, Stefania; B., Joshi; G., Kukreja; M., Persico; B., Catalanotti; E., Novellino; Fattorusso, E; Nacci, Vito; Savini, Luisa; D., Taramelli; N., Basilico; G., Morace; V., Yardley; C., Fattorusso -
Design, synthesis, and structure-activity relationship studies of 4-quinolinyl- and 9-acrydinylhydrazones as potent antimalarial agents. 1-gen-2008 C., Fattorusso; Campiani, Giuseppe; G., Kukreja; M., Persico; Butini, Stefania; Romano, MARIA PIA; Altarelli, Maria; S., Ros; Brindisi, Margherita; Savini, Luisa; E., Novellino; Nacci, Vito; E., Fattorusso; S., Parapini; N., Basilico; D., Taramelli; V., Yardley; S., Croft; M., Borriello; Gemma, Sandra -
Development of molecular probes for the identification of extra interaction sites in the mid-gorge and peripheral sites of butyrylcholinesterase (BuChE). Rational design of novel, selective, and highly potent BuChE inhibitors. 1-gen-2005 Campiani, Giuseppe; Fattorusso, C; Butini, Stefania; Gaeta, A; Agnusdei, M; Gemma, Sandra; Persico, M; Catalanotti, B; Savini, Luisa; Nacci, Vito; Novellino, E; Holloway, Hw; Greig, Nh; Belinskaya, T; Fedorko, Jm; Saxena, A. -
Discovery of a new class of potential multifunctional atypical antipsychotic agents targeting dopamine d3 and serotonin 5-HT 1A and 5-HT2A receptors: Design, synthesis, and effects on behavior 1-gen-2009 Butini, Stefania; Gemma, Sandra; Campiani, Giuseppe; Franceschini, Silvia; Trotta, Francesco; Marianna, Borriello; Nicoleta, Ceres; Sindu, Ros; SANNA COCCONE, Salvatore; Bernetti, Matteo; MERI DE, Angelis; Brindisi, Margherita; Nacci, Vito; Fiorini, Isabella; Ettore, Novellino; Alfredo, Cagnotto; Tiziana, Mennini; KARIN SANDAGER, Nielsen; JESPER TOBIAS, Andreasen; JORGEN SCHEEL, Kruger; JENS D., Mikkelsen; AND CATERINA, Fattorusso -
Discovery of Huperzine A/Tacrine Hybrids as Potent Inhibitors of Human Cholinesterases Targeting Their Mid-gorge Recognition Sites 1-gen-2006 Gemma, Sandra; Gabellieri, Emanuele; Huleatt, P.; C., Fattorusso; M., Borriello; B., Catalanotti; Butini, Stefania; M., DE ANGELIS; E., Novellino; Nacci, Vito; T., Belinskaya; Saxena, Ashima; Campiani, Giuseppe -
Exploiting Protein Fluctuations at the Active-Site Gorge of Human Cholinesterases: Further Optimization of the Design Strategy to Develop Extremely Potent Inhibitors 1-gen-2008 Butini, Stefania; Campiani, Giuseppe; M., Borriello; Gemma, Sandra; Panico, Alessandro; M., Persico; B., Catalanotti; S., Ros; Brindisi, Margherita; M., Agnusdei; Fiorini, Isabella; Nacci, Vito; E., Novellino; T., Belinskaya; A., Saxena; C., Fattorusso -
Inhibition of G1 cyclin-dependent kinase activity during growth arrest of human astrocytoma cells by the pyrrolo-1,5-benzoxazepine, PBOX-21 1-gen-2003 J. M., Mulligan; Campiani, Giuseppe; A., Ramunno; Nacci, Vito; D. M., Zisterer -
Neuronal high affinity sodium-dependent glutamate transporters (EAATs): targets for the development of novel therapeutics against neurodegenerative diseases. 1-gen-2003 Campiani, Giuseppe; Fattorusso, C.; DE ANGELIS, M.; Catalanotti, B.; Butini, Stefania; Fattorusso, R.; Fiorini, Isabella; Nacci, Vito; Novellino, E. -
New Antipsychotic Agents with Serotonin and Dopamine Antagonist Properties Based on a Pyrrolo[2,1-b][1,3]benzothiazepine Structure 1-gen-1998 Campiani, Giuseppe; Nacci, Vito; Bechelli, Susanna; Silvia M., Ciani; Antonio, Garofalo; Fiorini, Isabella; Håkan, Wikström; Peter de, Boer; Yi, Liao; Pieter G., Tepper; Alfredo, Cagnotto; Tiziana, Mennini -