Sfoglia per Autore
Development of Potent and Selective Monoacylglycerol Lipase Inhibitors. SARs, Structural Analysis, and Biological Characterization
2024-01-01 Butini, Stefania; Grether, Uwe; Jung, Kwang-Mook; Ligresti, Alessia; Allarà, Marco; Postmus, Annemarieke G. J.; Maramai, Samuele; Brogi, Simone; Papa, Alessandro; Carullo, Gabriele; Sykes, David; Veprintsev, Dmitry; Federico, Stefano; Grillo, Alessandro; Di Guglielmo, Bruno; Ramunno, Anna; Stevens, Anna Floor; Heer, Dominik; Lamponi, Stefania; Gemma, Sandra; Benz, Jörg; Di Marzo, Vincenzo; van der Stelt, Mario; Piomelli, Daniele; Campiani, Giuseppe
Development of potent and selective FAAH inhibitors with improved drug-like properties as potential tools to treat neuroinflammatory conditions
2023-01-01 Papa, Alessandro; Pasquini, Silvia; Galvani, Francesca; Cammarota, Mariarosaria; Contri, Chiara; Carullo, Gabriele; Gemma, Sandra; Ramunno, Anna; Lamponi, Stefania; Gorelli, Beatrice; Saponara, Simona; Varani, Katia; Mor, Marco; Campiani, Giuseppe; Boscia, Francesca; Vincenzi, Fabrizio; Lodola, Alessio; Butini, Stefania
A Comparative Study between Lycorine and Galantamine Abilities to Interact with AMYLOID β and Reduce In Vitro Neurotoxicity
2023-01-01 Kola, Arian; Lamponi, Stefania; Currò, Francesco; Valensin, Daniela
Design and synthesis of multifunctional microtubule targeting agents endowed with dual pro-apoptotic and anti-autophagic efficacy
2022-01-01 Campiani, Giuseppe; Khan, Tuhina; Ulivieri, Cristina; Staiano, Leopoldo; Papulino, Chiara; Magnano, Stefania; Nathwani, Seema; Ramunno, Anna; Lucena-Agell, Daniel; Relitti, Nicola; Federico, Stefano; Pozzetti, Luca; Carullo, Gabriele; Casagni, Alice; Brogi, Simone; Vanni, Francesca; Galatello, Paola; Ghanim, Magda; Mccabe, Niamh; Lamponi, Stefania; Valoti, Massimo; Ibrahim, Ola; O'Sullivan, Jeffrey; Turkington, Richard; Kelly, Vincent P.; Vanwemmel, Ruben; Díaz, J. Fernando; Gemma, Sandra; Zisterer, Daniela; Altucci, Lucia; De Matteis, Antonella; Butini, Stefania; Benedetti, Rosaria
Structuring and de-structuring of nanovectors from algal lipids: simulated digestion, preliminary antioxidant capacity and in vitro tests
2022-01-01 Clemente, Ilaria; Lamponi, Stefania; Tamasi, Gabriella; Rodolfi, Liliana; Rossi, Claudio; Ristori, Sandra
Preliminary in vitro cytotoxicity, mutagenicity and antitumoral activity evaluation of graphene flake and aqueous graphene paste
2022-01-01 Lamponi, S.
Click-Chemistry Cross-Linking of Hyaluronan Graft Copolymers
2022-01-01 Saletti, Mario; Paolino, Marco; Ballerini, Lavinia; Giuliani, Germano; Leone, Gemma; Lamponi, Stefania; Andreassi, Marco; Bonechi, Claudia; Donati, Alessandro; Piovani, Daniele; Schieroni, Alberto Giacometti; Magnani, Agnese; Cappelli, Andrea
Functionalized Hyaluronic Acid for “In Situ” Matrix Metalloproteinase Inhibition: A Bioactive Material to Treat the Dry Eye Sydrome
2022-01-01 Burgalassi, Susi; Fragai, Marco; Francesconi, Oscar; Cerofolini, Linda; Monti, Daniela; Leone, Gemma; Lamponi, Stefania; Greco, Giuseppe; Magnani, Agnese; Nativi, Cristina
Calcium ions hyaluronan/gellan gum protective shell for delivery of oleuropein in the knee
2022-01-01 Consumi, M.; Leone, G.; Pepi, S.; Pardini, A.; Lamponi, S.; Bonechi, C.; Tamasi, G.; Rossi, C.; Magnani, A.
Azetidin-2-one-based small molecules as dual hHDAC6/HDAC8 inhibitors: Investigation of their mechanism of action and impact of dual inhibition profile on cell viability
2022-01-01 Federico, S.; Khan, T.; Fontana, A.; Brogi, S.; Benedetti, R.; Sarno, F.; Carullo, G.; Pezzotta, A.; Saraswati, A. P.; Passaro, E.; Pozzetti, L.; Papa, A.; Relitti, N.; Gemma, S.; Butini, S.; Pistocchi, A.; Ramunno, A.; Vincenzi, F.; Varani, K.; Tatangelo, V.; Patrussi, L.; Baldari, C. T.; Saponara, S.; Gorelli, B.; Lamponi, S.; Valoti, M.; Saccoccia, F.; Giannaccari, M.; Ruberti, G.; Herp, D.; Jung, M.; Altucci, L.; Campiani, G.
Synthesis and biological evaluation of benzhydryl-based antiplasmodial agents possessing Plasmodium falciparum chloroquine resistance transporter (PfCRT) inhibitory activity
2021-01-01 Relitti, N.; Federico, S.; Pozzetti, L.; Butini, S.; Lamponi, S.; Taramelli, D.; D'Alessandro, S.; Martin, R. E.; Shafik, S. H.; Summers, R. L.; Babij, S. K.; Habluetzel, A.; Tapanelli, S.; Caldelari, R.; Gemma, S.; Campiani, G.
Harnessing the role of HDAC6 in Idiopathic Pulmonary Fibrosis: design, synthesis, structural analysis, and biological evaluation of potent inhibitors
2021-01-01 Campiani, Giuseppe; Cavella, Caterina; Osko, Jeremy D; Brindisi, Margherita; Relitti, Nicola; Brogi, Simone; Saraswati, A Prasanth; Federico, Stefano; Chemi, Giulia; Maramai, Samuele; Carullo, Gabriele; Jaeger, Benedikt; Carleo, Alfonso; Benedetti, Rosaria; Sarno, Federica; Lamponi, Stefania; Rottoli, Paola; Bargagli, Elena; Bertucci, Carlo; Tedesco, Daniele; Herp, Daniel; Senger, Johanna; Ruberti, Giovina; Saccoccia, Fulvio; Saponara, Simona; Gorelli, Beatrice; Valoti, Massimo; Kennedy, Breándan; Sundaramurthi, Husvinee; Butini, Stefania; Jung, Manfred; Roach, Katy M; Altucci, Lucia; Bradding, Peter; Christianson, David W; Gemma, Sandra; Prasse, Antje
Bioactive natural compounds with antiplatelet and anticoagulant activity and their potential role in the treatment of thrombotic disorders
2021-01-01 Lamponi, S.
Sodium hyaluronate-g-2-((N-(6-aminohexyl)-4-methoxyphenyl)sulfonamido)-N-hydroxyacetamide with enhanced affinity towards MMP12 catalytic domain to be used as visco-supplement with increased degradation resistance
2021-01-01 Leone, G.; Pepi, S.; Consumi, M.; Lamponi, S.; Fragai, M.; Martinucci, M.; Baldoneschi, V.; Francesconi, O.; Nativi, C.; Magnani, A.
Phosphorylated xanthan gum-Ag(I) complex as antibacterial viscosity enhancer for eye drops formulation
2021-01-01 Leone, G.; Pepi, S.; Consumi, M.; Mahdizadeh, F. F.; Lamponi, S.; Magnani, A.
Structural and Functional Analysis of Extracts in Plants
2021-01-01 Lamponi, Stefania
Selective Fatty Acid Amide Hydrolase Inhibitors as Potential Novel Antiepileptic Agents
2021-01-01 Grillo, Alessandro; Fezza, Filomena; Chemi, Giulia; Colangeli, Roberto; Brogi, Simone; Fazio, Domenico; Federico, Stefano; Papa, Alessandro; Relitti, Nicola; Di Maio, Roberto; Giorgi, Gianluca; Lamponi, Stefania; Valoti, Massimo; Gorelli, Beatrice; Saponara, Simona; Benedusi, Mascia; Pecorelli, Alessandra; Minetti, Patrizia; Valacchi, Giuseppe; Butini, Stefania; Campiani, Giuseppe; Gemma, Sandra; Maccarrone, Mauro; Di Giovanni, Giuseppe
The importance of structural and functional analysis of extracts in plants
2021-01-01 Lamponi, S.
Novel quinolone-based potent and selective HDAC6 inhibitors: synthesis, molecular modeling studies and biological investigation
2021-01-01 Relitti, N.; Saraswati, A. P.; Chemi, G.; Brindisi, M.; Brogi, S.; Herp, D.; Schmidtkunz, K.; Saccoccia, F.; Ruberti, G.; Ulivieri, C.; Vanni, F.; Sarno, F.; Altucci, L.; Lamponi, S.; Jung, M.; Gemma, S.; Butini, S.; Campiani, G.
Chemical profile, antioxidant, anti-proliferative, anticoagulant and mutagenic effects of a hydroalcoholic extract of Tuscan Rosmarinus officinalis
2021-01-01 Lamponi, Stefania; Baratto, Maria Camilla; Miraldi, Elisabetta; Baini, Giulia; Biagi, Marco
Titolo | Data di pubblicazione | Autore(i) | File | Abstract |
---|---|---|---|---|
Development of Potent and Selective Monoacylglycerol Lipase Inhibitors. SARs, Structural Analysis, and Biological Characterization | 1-gen-2024 | Butini, Stefania; Grether, Uwe; Jung, Kwang-Mook; Ligresti, Alessia; Allarà, Marco; Postmus, Annemarieke G. J.; Maramai, Samuele; Brogi, Simone; Papa, Alessandro; Carullo, Gabriele; Sykes, David; Veprintsev, Dmitry; Federico, Stefano; Grillo, Alessandro; Di Guglielmo, Bruno; Ramunno, Anna; Stevens, Anna Floor; Heer, Dominik; Lamponi, Stefania; Gemma, Sandra; Benz, Jörg; Di Marzo, Vincenzo; van der Stelt, Mario; Piomelli, Daniele; Campiani, Giuseppe | - | |
Development of potent and selective FAAH inhibitors with improved drug-like properties as potential tools to treat neuroinflammatory conditions | 1-gen-2023 | Papa, Alessandro; Pasquini, Silvia; Galvani, Francesca; Cammarota, Mariarosaria; Contri, Chiara; Carullo, Gabriele; Gemma, Sandra; Ramunno, Anna; Lamponi, Stefania; Gorelli, Beatrice; Saponara, Simona; Varani, Katia; Mor, Marco; Campiani, Giuseppe; Boscia, Francesca; Vincenzi, Fabrizio; Lodola, Alessio; Butini, Stefania | - | |
A Comparative Study between Lycorine and Galantamine Abilities to Interact with AMYLOID β and Reduce In Vitro Neurotoxicity | 1-gen-2023 | Kola, Arian; Lamponi, Stefania; Currò, Francesco; Valensin, Daniela | - | |
Design and synthesis of multifunctional microtubule targeting agents endowed with dual pro-apoptotic and anti-autophagic efficacy | 1-gen-2022 | Campiani, Giuseppe; Khan, Tuhina; Ulivieri, Cristina; Staiano, Leopoldo; Papulino, Chiara; Magnano, Stefania; Nathwani, Seema; Ramunno, Anna; Lucena-Agell, Daniel; Relitti, Nicola; Federico, Stefano; Pozzetti, Luca; Carullo, Gabriele; Casagni, Alice; Brogi, Simone; Vanni, Francesca; Galatello, Paola; Ghanim, Magda; Mccabe, Niamh; Lamponi, Stefania; Valoti, Massimo; Ibrahim, Ola; O'Sullivan, Jeffrey; Turkington, Richard; Kelly, Vincent P.; Vanwemmel, Ruben; Díaz, J. Fernando; Gemma, Sandra; Zisterer, Daniela; Altucci, Lucia; De Matteis, Antonella; Butini, Stefania; Benedetti, Rosaria | - | |
Structuring and de-structuring of nanovectors from algal lipids: simulated digestion, preliminary antioxidant capacity and in vitro tests | 1-gen-2022 | Clemente, Ilaria; Lamponi, Stefania; Tamasi, Gabriella; Rodolfi, Liliana; Rossi, Claudio; Ristori, Sandra | - | |
Preliminary in vitro cytotoxicity, mutagenicity and antitumoral activity evaluation of graphene flake and aqueous graphene paste | 1-gen-2022 | Lamponi, S. | - | |
Click-Chemistry Cross-Linking of Hyaluronan Graft Copolymers | 1-gen-2022 | Saletti, Mario; Paolino, Marco; Ballerini, Lavinia; Giuliani, Germano; Leone, Gemma; Lamponi, Stefania; Andreassi, Marco; Bonechi, Claudia; Donati, Alessandro; Piovani, Daniele; Schieroni, Alberto Giacometti; Magnani, Agnese; Cappelli, Andrea | - | |
Functionalized Hyaluronic Acid for “In Situ” Matrix Metalloproteinase Inhibition: A Bioactive Material to Treat the Dry Eye Sydrome | 1-gen-2022 | Burgalassi, Susi; Fragai, Marco; Francesconi, Oscar; Cerofolini, Linda; Monti, Daniela; Leone, Gemma; Lamponi, Stefania; Greco, Giuseppe; Magnani, Agnese; Nativi, Cristina | - | |
Calcium ions hyaluronan/gellan gum protective shell for delivery of oleuropein in the knee | 1-gen-2022 | Consumi, M.; Leone, G.; Pepi, S.; Pardini, A.; Lamponi, S.; Bonechi, C.; Tamasi, G.; Rossi, C.; Magnani, A. | - | |
Azetidin-2-one-based small molecules as dual hHDAC6/HDAC8 inhibitors: Investigation of their mechanism of action and impact of dual inhibition profile on cell viability | 1-gen-2022 | Federico, S.; Khan, T.; Fontana, A.; Brogi, S.; Benedetti, R.; Sarno, F.; Carullo, G.; Pezzotta, A.; Saraswati, A. P.; Passaro, E.; Pozzetti, L.; Papa, A.; Relitti, N.; Gemma, S.; Butini, S.; Pistocchi, A.; Ramunno, A.; Vincenzi, F.; Varani, K.; Tatangelo, V.; Patrussi, L.; Baldari, C. T.; Saponara, S.; Gorelli, B.; Lamponi, S.; Valoti, M.; Saccoccia, F.; Giannaccari, M.; Ruberti, G.; Herp, D.; Jung, M.; Altucci, L.; Campiani, G. | - | |
Synthesis and biological evaluation of benzhydryl-based antiplasmodial agents possessing Plasmodium falciparum chloroquine resistance transporter (PfCRT) inhibitory activity | 1-gen-2021 | Relitti, N.; Federico, S.; Pozzetti, L.; Butini, S.; Lamponi, S.; Taramelli, D.; D'Alessandro, S.; Martin, R. E.; Shafik, S. H.; Summers, R. L.; Babij, S. K.; Habluetzel, A.; Tapanelli, S.; Caldelari, R.; Gemma, S.; Campiani, G. | - | |
Harnessing the role of HDAC6 in Idiopathic Pulmonary Fibrosis: design, synthesis, structural analysis, and biological evaluation of potent inhibitors | 1-gen-2021 | Campiani, Giuseppe; Cavella, Caterina; Osko, Jeremy D; Brindisi, Margherita; Relitti, Nicola; Brogi, Simone; Saraswati, A Prasanth; Federico, Stefano; Chemi, Giulia; Maramai, Samuele; Carullo, Gabriele; Jaeger, Benedikt; Carleo, Alfonso; Benedetti, Rosaria; Sarno, Federica; Lamponi, Stefania; Rottoli, Paola; Bargagli, Elena; Bertucci, Carlo; Tedesco, Daniele; Herp, Daniel; Senger, Johanna; Ruberti, Giovina; Saccoccia, Fulvio; Saponara, Simona; Gorelli, Beatrice; Valoti, Massimo; Kennedy, Breándan; Sundaramurthi, Husvinee; Butini, Stefania; Jung, Manfred; Roach, Katy M; Altucci, Lucia; Bradding, Peter; Christianson, David W; Gemma, Sandra; Prasse, Antje | - | |
Bioactive natural compounds with antiplatelet and anticoagulant activity and their potential role in the treatment of thrombotic disorders | 1-gen-2021 | Lamponi, S. | - | |
Sodium hyaluronate-g-2-((N-(6-aminohexyl)-4-methoxyphenyl)sulfonamido)-N-hydroxyacetamide with enhanced affinity towards MMP12 catalytic domain to be used as visco-supplement with increased degradation resistance | 1-gen-2021 | Leone, G.; Pepi, S.; Consumi, M.; Lamponi, S.; Fragai, M.; Martinucci, M.; Baldoneschi, V.; Francesconi, O.; Nativi, C.; Magnani, A. | - | |
Phosphorylated xanthan gum-Ag(I) complex as antibacterial viscosity enhancer for eye drops formulation | 1-gen-2021 | Leone, G.; Pepi, S.; Consumi, M.; Mahdizadeh, F. F.; Lamponi, S.; Magnani, A. | - | |
Structural and Functional Analysis of Extracts in Plants | 1-gen-2021 | Lamponi, Stefania | - | |
Selective Fatty Acid Amide Hydrolase Inhibitors as Potential Novel Antiepileptic Agents | 1-gen-2021 | Grillo, Alessandro; Fezza, Filomena; Chemi, Giulia; Colangeli, Roberto; Brogi, Simone; Fazio, Domenico; Federico, Stefano; Papa, Alessandro; Relitti, Nicola; Di Maio, Roberto; Giorgi, Gianluca; Lamponi, Stefania; Valoti, Massimo; Gorelli, Beatrice; Saponara, Simona; Benedusi, Mascia; Pecorelli, Alessandra; Minetti, Patrizia; Valacchi, Giuseppe; Butini, Stefania; Campiani, Giuseppe; Gemma, Sandra; Maccarrone, Mauro; Di Giovanni, Giuseppe | - | |
The importance of structural and functional analysis of extracts in plants | 1-gen-2021 | Lamponi, S. | - | |
Novel quinolone-based potent and selective HDAC6 inhibitors: synthesis, molecular modeling studies and biological investigation | 1-gen-2021 | Relitti, N.; Saraswati, A. P.; Chemi, G.; Brindisi, M.; Brogi, S.; Herp, D.; Schmidtkunz, K.; Saccoccia, F.; Ruberti, G.; Ulivieri, C.; Vanni, F.; Sarno, F.; Altucci, L.; Lamponi, S.; Jung, M.; Gemma, S.; Butini, S.; Campiani, G. | - | |
Chemical profile, antioxidant, anti-proliferative, anticoagulant and mutagenic effects of a hydroalcoholic extract of Tuscan Rosmarinus officinalis | 1-gen-2021 | Lamponi, Stefania; Baratto, Maria Camilla; Miraldi, Elisabetta; Baini, Giulia; Biagi, Marco | - |
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