Sfoglia per Autore
Novel multitarget directed ligands inspired by riluzole: A serendipitous synthesis of substituted benzo[b][1,4]thiazepines potentially useful as neuroprotective agents
2024-01-01 Maramai, S.; Saletti, M.; Paolino, M.; Giuliani, G.; Cazzola, J.; Spaiardi, P.; Talpo, F.; Frosini, M.; Pifferi, A.; Ballarotto, M.; Carotti, A.; Poggialini, F.; Vagaggini, C.; Dreassi, E.; Giorgi, G.; Dondio, G.; Cappelli, A.; Rosario Biella, G.; Anzini, M.
Reactivity of a Morita–Baylis–Hillman Adduct Derivative Bearing a Triphenylamine Moiety with Lysine Models
2024-01-01 Venditti, Jacopo; Saletti, Mario; Paolino, Marco; Contena, Stefano; Bonechi, Claudia; Giuliani, Germano; Giorgi, Gianluca; Boccia, Antonella Caterina; Botta, Chiara; Blancafort, Lluís; Cappelli, Andrea
Systematic Modification of the Substitution Pattern of the 7-Hydroxy-5-oxopyrazolo[4,3-b]pyridine-6-carboxamide Scaffold Enabled the Discovery of New Ligands with High Affinity and Selectivity for the Cannabinoid Type 2 Receptor
2023-01-01 Mugnaini, Claudia; Kostrzewa, Magdalena; Casini, Marta; Kumar, Poulami; Catallo, Valeria; Allarà, Marco; Guastaferro, Laura; Brizzi, Antonella; Paolino, Marco; Tafi, Andrea; Kapatais, Christelos; Giorgi, Gianluca; Vacondio, Federica; Mor, Marco; Corelli, Federico; Ligresti, Alessia
Spontaneous polymerization of benzofulvene monomers bearing a 4-Pyri- dylacetylene substituent in different positions of the benzofulvene scaffold
2023-01-01 Paolino, M; Saletti, M; Reale, A; Razzano, V; Giuliani, G; Donati, A; Bonechi, C; Giorgi, G; Mercorillo, G; Samperi, F; Mroz, W; Botta, C; Cappelli, A
A tri(ethylene glycol)-tethered Morita-Baylis-Hillman dimer in the formation of macrocyclic crown ether-paracyclophane hybrid structures
2023-01-01 Saletti, Mario; Venditti, Jacopo; Paolino, Marco; Zacchei, Arianna; Giuliani, Germano; Giorgi, Gianluca; Bonechi, Claudia; Donati, Alessandro; Cappelli, Andrea
Reactivity of ethyl nitrosoacrylate toward pyrrole, indole and pyrrolo[3,2-c]carbazole: an experimental and theoretical study
2023-01-01 Benzi, Alice; Lopes Susana, M. M.; Nunes Sandra, C. C.; Giorgi, Gianluca; Bianchi, Lara; Tavani, Cinzia; Pais Alberto, A. C. C.; Petrillo, Giovanni; Pinho e Melo Teresa, M. V. D.
Spontaneous polymerization of benzofulvene derivatives bearing complexed or un-complexed pyridine rings
2022-01-01 Paolino, Marco; Saletti, Mario; Reale, Annalisa; Razzano, Vincenzo; Giuliani, Germano; Donati, Alessandro; Bonechi, Claudia; Giorgi, Gianluca; Atrei, Andrea; Mauro, Matteo; Scamporrino, Andrea; Samperi, Filippo; Fois, Ettore; Tabacchi, Gloria; Botta, Chiara; Cappelli, Andrea
Xanthopsin-like systems via site-specific click-functionalization of a retinoic acid binding protein
2022-01-01 Tassone, G.; Paolino, M.; Pozzi, C.; Reale, A.; Salvini, L.; Giorgi, G.; Orlandini, M.; Galvagni, F.; Mangani, S.; Yang, X.; Carlotti, B.; Ortica, F.; Latterini, L.; Olivucci, M.; Cappelli, A.
Novel analgesic/anti-inflammatory agents: 1,5-Diarylpyrrole nitrooxyethyl sulfides and related compounds as Cyclooxygenase-2 inhibitors containing a nitric oxide donor moiety endowed with vasorelaxant properties
2022-01-01 Saletti, Mario; Maramai, Samuele; Reale, Annalisa; Paolino, Marco; Brogi, Simone; Di Capua, Angela; Cappelli, Andrea; Giorgi, Gianluca; D'Avino, Danilo; Rossi, Antonietta; Ghelardini, Carla; Di Cesare Mannelli, Lorenzo; Sardella, Roccaldo; Carotti, Andrea; Woelkart, Gerald; Klösch, Burkhard; Bigogno, Chiara; Dondio, Giulio; Anzini, Maurizio
Design, Synthesis and Characterization of a Visible-Light-Sensitive Molecular Switch and Its PEGylation Towards a Self-Assembling Molecule
2022-01-01 Paolino, Marco; Saletti, Mario; Reale, Annalisa; Licciardi, Mariano; Varvarà, Paola; Marquette, Arnaud; Léonard, Jérémie; Bonechi, Claudia; Donati, Alessandro; Giorgi, Gianluca; Giuliani, Germano; Carlotti, Benedetta; Ortica, Fausto; Latterini, Loredana; Gentile, Mariangela; Paccagnini, Eugenio; Olivucci, Massimo; Cappelli, Andrea
Towards the engineering of a photon-only two-stroke rotary molecular motor
2022-01-01 Filatov Gulak, Michael; Paolino, Marco; Pierron, Robin; Cappelli, Andrea; Giorgi, Gianluca; Léonard, Jérémie; Huix-Rotllant, Miquel; Ferré, Nicolas; Yang, Xuchun; Kaliakin, Danil; Blanco-González, Alejandro; Olivucci, Massimo
Milk kefir enriched with inulin-grafted seed extract from white wine pomace: chemical characterisation, antioxidant profile and in vitro gastrointestinal digestion
2022-01-01 Carullo, G.; Spizzirri, U. G.; Montopoli, M.; Cocetta, V.; Armentano, B.; Tinazzi, M.; Sciubba, F.; Giorgi, G.; Enrica Di Cocco, M.; Bohn, T.; Aiello, F.; Restuccia, D.
An easy access to furan fused polyheterocyclic systems
2022-01-01 Benzi, Alice; Bianchi, Lara; Giorgi, Gianluca; Maccagno, Massimo; Petrillo, Giovanni; Spinelli, Domenico; Tavani, Cinzia
Selective Fatty Acid Amide Hydrolase Inhibitors as Potential Novel Antiepileptic Agents
2021-01-01 Grillo, Alessandro; Fezza, Filomena; Chemi, Giulia; Colangeli, Roberto; Brogi, Simone; Fazio, Domenico; Federico, Stefano; Papa, Alessandro; Relitti, Nicola; Di Maio, Roberto; Giorgi, Gianluca; Lamponi, Stefania; Valoti, Massimo; Gorelli, Beatrice; Saponara, Simona; Benedusi, Mascia; Pecorelli, Alessandra; Minetti, Patrizia; Valacchi, Giuseppe; Butini, Stefania; Campiani, Giuseppe; Gemma, Sandra; Maccarrone, Mauro; Di Giovanni, Giuseppe
On the Transition from a Biomimetic Molecular Switch to a Rotary Molecular Motor
2021-01-01 Paolino, Marco; Giovannini, Tommaso; Manathunga, Madushanka; Latterini, Loredana; Zampini, Giulia; Pierron, Robin; Léonard, Jérémie; Fusi, Stefania; Giorgi, Gianluca; Giuliani, Germano; Cappelli, Andrea; Cappelli, Chiara; Olivucci, Massimo
In memory of Giovanni Sindona
2021-01-01 Giorgi, G.; Napoli, A.
Laccase-Catalyzed 1,4-Dioxane-Mediated synthesis of Belladine N-Oxides with anti-influenza a virus activity
2021-01-01 Zippilli, Claudio; Botta, Lorenzo; Mattia Bizzarri, Bruno; Nencioni, Lucia; De Angelis, Marta; Protto, Virginia; Giorgi, Gianluca; Baratto, MARIA CAMILLA; Pogni, Rebecca; Saladino, Raffaele
In search for novel liver X receptors modulators by extending the structure–activity relationships of cholenamide derivatives
2021-01-01 Pontini, L.; Palazzoli, P.; Maggioni, D.; Damiano, G.; Giorgi, G.; Russo, V.; Marinozzi, M.
Design, synthesis, and physicochemical and pharmacological profiling of 7‐Hydroxy-5-oxopyrazolo[4,3‐b]pyridine-6-carboxamide derivatives with antiosteoarthritic activity in vivo
2020-01-01 Mugnaini, Claudia; Kostrzewa, Magdalena; Bryk, Marta; Mokhtar Mahmoud, Ali; Brizzi, Antonella; Lamponi, Stefania; Giorgi, Gianluca; Ferlenghi, Francesca; Vacondio, Federica; Maccioni, Paola; Colombo, Giancarlo; Mor, Marco; Starowicz, Katarzyna; Di Marzo, Vincenzo; Ligresti, Alessia; Corelli, Federico
2-Aryl-3-Vinyl Substituted Imidazo[1,2-a]pyridines and fluorescent electrocyclization derivatives therefrom
2020-01-01 Benzi, A.; Bianchi, L.; Giorgi, G.; Maccagno, M.; Petrillo, G.; Tavani, C.
Titolo | Data di pubblicazione | Autore(i) | File | Abstract |
---|---|---|---|---|
Novel multitarget directed ligands inspired by riluzole: A serendipitous synthesis of substituted benzo[b][1,4]thiazepines potentially useful as neuroprotective agents | 1-gen-2024 | Maramai, S.; Saletti, M.; Paolino, M.; Giuliani, G.; Cazzola, J.; Spaiardi, P.; Talpo, F.; Frosini, M.; Pifferi, A.; Ballarotto, M.; Carotti, A.; Poggialini, F.; Vagaggini, C.; Dreassi, E.; Giorgi, G.; Dondio, G.; Cappelli, A.; Rosario Biella, G.; Anzini, M. | - | |
Reactivity of a Morita–Baylis–Hillman Adduct Derivative Bearing a Triphenylamine Moiety with Lysine Models | 1-gen-2024 | Venditti, Jacopo; Saletti, Mario; Paolino, Marco; Contena, Stefano; Bonechi, Claudia; Giuliani, Germano; Giorgi, Gianluca; Boccia, Antonella Caterina; Botta, Chiara; Blancafort, Lluís; Cappelli, Andrea | - | |
Systematic Modification of the Substitution Pattern of the 7-Hydroxy-5-oxopyrazolo[4,3-b]pyridine-6-carboxamide Scaffold Enabled the Discovery of New Ligands with High Affinity and Selectivity for the Cannabinoid Type 2 Receptor | 1-gen-2023 | Mugnaini, Claudia; Kostrzewa, Magdalena; Casini, Marta; Kumar, Poulami; Catallo, Valeria; Allarà, Marco; Guastaferro, Laura; Brizzi, Antonella; Paolino, Marco; Tafi, Andrea; Kapatais, Christelos; Giorgi, Gianluca; Vacondio, Federica; Mor, Marco; Corelli, Federico; Ligresti, Alessia | - | |
Spontaneous polymerization of benzofulvene monomers bearing a 4-Pyri- dylacetylene substituent in different positions of the benzofulvene scaffold | 1-gen-2023 | Paolino, M; Saletti, M; Reale, A; Razzano, V; Giuliani, G; Donati, A; Bonechi, C; Giorgi, G; Mercorillo, G; Samperi, F; Mroz, W; Botta, C; Cappelli, A | - | |
A tri(ethylene glycol)-tethered Morita-Baylis-Hillman dimer in the formation of macrocyclic crown ether-paracyclophane hybrid structures | 1-gen-2023 | Saletti, Mario; Venditti, Jacopo; Paolino, Marco; Zacchei, Arianna; Giuliani, Germano; Giorgi, Gianluca; Bonechi, Claudia; Donati, Alessandro; Cappelli, Andrea | - | |
Reactivity of ethyl nitrosoacrylate toward pyrrole, indole and pyrrolo[3,2-c]carbazole: an experimental and theoretical study | 1-gen-2023 | Benzi, Alice; Lopes Susana, M. M.; Nunes Sandra, C. C.; Giorgi, Gianluca; Bianchi, Lara; Tavani, Cinzia; Pais Alberto, A. C. C.; Petrillo, Giovanni; Pinho e Melo Teresa, M. V. D. | - | |
Spontaneous polymerization of benzofulvene derivatives bearing complexed or un-complexed pyridine rings | 1-gen-2022 | Paolino, Marco; Saletti, Mario; Reale, Annalisa; Razzano, Vincenzo; Giuliani, Germano; Donati, Alessandro; Bonechi, Claudia; Giorgi, Gianluca; Atrei, Andrea; Mauro, Matteo; Scamporrino, Andrea; Samperi, Filippo; Fois, Ettore; Tabacchi, Gloria; Botta, Chiara; Cappelli, Andrea | - | |
Xanthopsin-like systems via site-specific click-functionalization of a retinoic acid binding protein | 1-gen-2022 | Tassone, G.; Paolino, M.; Pozzi, C.; Reale, A.; Salvini, L.; Giorgi, G.; Orlandini, M.; Galvagni, F.; Mangani, S.; Yang, X.; Carlotti, B.; Ortica, F.; Latterini, L.; Olivucci, M.; Cappelli, A. | - | |
Novel analgesic/anti-inflammatory agents: 1,5-Diarylpyrrole nitrooxyethyl sulfides and related compounds as Cyclooxygenase-2 inhibitors containing a nitric oxide donor moiety endowed with vasorelaxant properties | 1-gen-2022 | Saletti, Mario; Maramai, Samuele; Reale, Annalisa; Paolino, Marco; Brogi, Simone; Di Capua, Angela; Cappelli, Andrea; Giorgi, Gianluca; D'Avino, Danilo; Rossi, Antonietta; Ghelardini, Carla; Di Cesare Mannelli, Lorenzo; Sardella, Roccaldo; Carotti, Andrea; Woelkart, Gerald; Klösch, Burkhard; Bigogno, Chiara; Dondio, Giulio; Anzini, Maurizio | - | |
Design, Synthesis and Characterization of a Visible-Light-Sensitive Molecular Switch and Its PEGylation Towards a Self-Assembling Molecule | 1-gen-2022 | Paolino, Marco; Saletti, Mario; Reale, Annalisa; Licciardi, Mariano; Varvarà, Paola; Marquette, Arnaud; Léonard, Jérémie; Bonechi, Claudia; Donati, Alessandro; Giorgi, Gianluca; Giuliani, Germano; Carlotti, Benedetta; Ortica, Fausto; Latterini, Loredana; Gentile, Mariangela; Paccagnini, Eugenio; Olivucci, Massimo; Cappelli, Andrea | - | |
Towards the engineering of a photon-only two-stroke rotary molecular motor | 1-gen-2022 | Filatov Gulak, Michael; Paolino, Marco; Pierron, Robin; Cappelli, Andrea; Giorgi, Gianluca; Léonard, Jérémie; Huix-Rotllant, Miquel; Ferré, Nicolas; Yang, Xuchun; Kaliakin, Danil; Blanco-González, Alejandro; Olivucci, Massimo | - | |
Milk kefir enriched with inulin-grafted seed extract from white wine pomace: chemical characterisation, antioxidant profile and in vitro gastrointestinal digestion | 1-gen-2022 | Carullo, G.; Spizzirri, U. G.; Montopoli, M.; Cocetta, V.; Armentano, B.; Tinazzi, M.; Sciubba, F.; Giorgi, G.; Enrica Di Cocco, M.; Bohn, T.; Aiello, F.; Restuccia, D. | - | |
An easy access to furan fused polyheterocyclic systems | 1-gen-2022 | Benzi, Alice; Bianchi, Lara; Giorgi, Gianluca; Maccagno, Massimo; Petrillo, Giovanni; Spinelli, Domenico; Tavani, Cinzia | - | |
Selective Fatty Acid Amide Hydrolase Inhibitors as Potential Novel Antiepileptic Agents | 1-gen-2021 | Grillo, Alessandro; Fezza, Filomena; Chemi, Giulia; Colangeli, Roberto; Brogi, Simone; Fazio, Domenico; Federico, Stefano; Papa, Alessandro; Relitti, Nicola; Di Maio, Roberto; Giorgi, Gianluca; Lamponi, Stefania; Valoti, Massimo; Gorelli, Beatrice; Saponara, Simona; Benedusi, Mascia; Pecorelli, Alessandra; Minetti, Patrizia; Valacchi, Giuseppe; Butini, Stefania; Campiani, Giuseppe; Gemma, Sandra; Maccarrone, Mauro; Di Giovanni, Giuseppe | - | |
On the Transition from a Biomimetic Molecular Switch to a Rotary Molecular Motor | 1-gen-2021 | Paolino, Marco; Giovannini, Tommaso; Manathunga, Madushanka; Latterini, Loredana; Zampini, Giulia; Pierron, Robin; Léonard, Jérémie; Fusi, Stefania; Giorgi, Gianluca; Giuliani, Germano; Cappelli, Andrea; Cappelli, Chiara; Olivucci, Massimo | - | |
In memory of Giovanni Sindona | 1-gen-2021 | Giorgi, G.; Napoli, A. | - | |
Laccase-Catalyzed 1,4-Dioxane-Mediated synthesis of Belladine N-Oxides with anti-influenza a virus activity | 1-gen-2021 | Zippilli, Claudio; Botta, Lorenzo; Mattia Bizzarri, Bruno; Nencioni, Lucia; De Angelis, Marta; Protto, Virginia; Giorgi, Gianluca; Baratto, MARIA CAMILLA; Pogni, Rebecca; Saladino, Raffaele | - | |
In search for novel liver X receptors modulators by extending the structure–activity relationships of cholenamide derivatives | 1-gen-2021 | Pontini, L.; Palazzoli, P.; Maggioni, D.; Damiano, G.; Giorgi, G.; Russo, V.; Marinozzi, M. | - | |
Design, synthesis, and physicochemical and pharmacological profiling of 7‐Hydroxy-5-oxopyrazolo[4,3‐b]pyridine-6-carboxamide derivatives with antiosteoarthritic activity in vivo | 1-gen-2020 | Mugnaini, Claudia; Kostrzewa, Magdalena; Bryk, Marta; Mokhtar Mahmoud, Ali; Brizzi, Antonella; Lamponi, Stefania; Giorgi, Gianluca; Ferlenghi, Francesca; Vacondio, Federica; Maccioni, Paola; Colombo, Giancarlo; Mor, Marco; Starowicz, Katarzyna; Di Marzo, Vincenzo; Ligresti, Alessia; Corelli, Federico | - | |
2-Aryl-3-Vinyl Substituted Imidazo[1,2-a]pyridines and fluorescent electrocyclization derivatives therefrom | 1-gen-2020 | Benzi, A.; Bianchi, L.; Giorgi, G.; Maccagno, M.; Petrillo, G.; Tavani, C. | - |
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