TASSONE, GIUSY

TASSONE, GIUSY  

Dipartimento di Biotecnologie, Chimica e Farmacia  

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Risultati 1 - 20 di 32 (tempo di esecuzione: 0.0 secondi).
Titolo Data di pubblicazione Autore(i) File Abstract
1,2,4-Triazole-3-Thione Analogues with a 2-Ethylbenzoic Acid at Position 4 as VIM-type Metallo-β-Lactamase Inhibitors 1-gen-2022 Verdirosa, Federica; Gavara, Laurent; Sevaille, Laurent; Tassone, Giusy; Corsica, Giuseppina; Legru, Alice; Feller, Georges; Chelini, Giulia; Mercuri, Paola Sandra; Tanfoni, Silvia; Sannio, Filomena; Benvenuti, Manuela; Cerboni, Giulia; De Luca, Filomena; Bouajila, Ezeddine; Vo Hoang, Yen; Licznar-Fajardo, Patricia; Galleni, Moreno; Pozzi, Cecilia; Mangani, Stefano; Docquier, Jean-Denis; Hernandez, Jean-François -
1,2,4-Triazole-3-thione compounds with a 4-ethyl alkyl/aryl sulfide substituent are broad-spectrum metallo-β-lactamase inhibitors with re-sensitization activity 1-gen-2021 Legru, Alice; Verdirosa, Federica; Hernandez, Jean-François; Tassone, Giusy; Sannio, Filomena; Benvenuti, Manuela; Conde, Pierre-Alexis; Bossis, Guillaume; Thomas, Caitlyn A; Crowder, Michael W; Dillenberger, Melissa; Becker, Katja; Pozzi, Cecilia; Mangani, Stefano; Docquier, Jean-Denis; Gavara, Laurent -
Amino-thiadiazole as innovative inhibitors of human glutaminyl cyclase for the treatment of Alzheimer disease 1-gen-2018 Pozzi, Cecilia; Tassone, Giusy; Linciano, Pasquale; Costi, MARIA PAOLA; Mangani, Stefano -
Amino-thiadiazole as innovative inhibitors of human glutaminyl cyclase, a validated target towards Alzheimer disease 1-gen-2018 Pozzi, Cecilia; Tassone, Giusy; Linciano, Pasquale; Benvenuti, Manuela; Costi, MARIA PAOLA; Mangani, Stefano -
Chemically stable inhibitors of 14-3-3 protein–protein interactions derived from BV02 1-gen-2019 Iralde-Lorente, Leire; Cau, Ylenia; Clementi, Letizia; Franci, Lorenzo; Tassone, Giusy; Valensin, Daniela; Mori, Mattia; Angelucci, Adriano; Chiariello, Mario; Botta, Maurizio -
Dimerization of the C-type lectin-like receptor CD93 promotes its binding to Multimerin-2 in endothelial cells 1-gen-2023 Barbera, Stefano; Raucci, Luisa; Tassone, Giusy; Tinti, Laura; Prischi, Filippo; Santucci, Annalisa; Mongiat, Maurizio; Tosi, Gian Marco; Galvagni, Federico; Dimberg, Anna; Pozzi, Cecilia; Orlandini, Maurizio -
Discovery of ANT3310, a Novel Broad-Spectrum Serine β-Lactamase Inhibitor of the Diazabicyclooctane Class, Which Strongly Potentiates Meropenem Activity against Carbapenem-Resistant Enterobacterales and Acinetobacter baumannii 1-gen-2020 Davies, D. T.; Leiris, S.; Zalacain, M.; Sprynski, N.; Castandet, J.; Bousquet, J.; Lozano, C.; Llanos, A.; Alibaud, L.; Vasa, S.; Pattipati, R.; Valige, R.; Kummari, B.; Pothukanuri, S.; De Piano, C.; Morrissey, I.; Holden, K.; Warn, P.; Marcoccia, F.; Benvenuti, M.; Pozzi, C.; Tassone, G.; Mangani, S.; Docquier, J. D.; Pallin, D.; Elliot, R.; Lemonnier, M.; Everett, M. -
Discovery of small molecule inhibitors of Leishmania braziliensis Hsp90 chaperone 1-gen-2020 Batista, F. A. H.; Ramos, S. L.; Tassone, G.; Leitao, A.; Montanari, C. A.; Botta, M.; Mori, M.; Borges, J. C. -
Dynamic interplay between copper toxicity and mitochondrial dysfunction in alzheimer’s disease 1-gen-2021 Tassone, G.; Kola, A.; Valensin, D.; Pozzi, C. -
Evidence of Pyrimethamine and Cycloguanil Analogues as Dual Inhibitors of Trypanosoma brucei Pteridine Reductase and Dihydrofolate Reductase 1-gen-2021 Tassone, Giusy; Landi, Giacomo; Linciano, Pasquale; Francesconi, Valeria; Tonelli, Michele; Tagliazucchi, Lorenzo; Costi, Maria Paola; Mangani, Stefano; Pozzi, Cecilia -
Exploiting ELIOT for Scaffold-Repurposing Opportunities: TRIM33 a Possible Novel E3 Ligase to Expand the Toolbox for PROTAC Design 1-gen-2022 Palomba, Tommaso; Tassone, Giusy; Vacca, Carmine; Bartalucci, Matteo; Valeri, Aurora; Pozzi, Cecilia; Cross, Simon; Siragusa, Lydia; Desantis, Jenny -
High-resolution crystal structure of Trypanosoma brucei pteridine reductase 1 in complex with an innovative tricyclic-based inhibitor 1-gen-2020 Landi, Giacomo; Linciano, Pasquale; Tassone, Giusy; Costi, Maria Paola; Mangani, Stefano; Pozzi, Cecilia -
Identification of Phosphate-Containing Compounds as New Inhibitors of 14-3-3/c-Abl Protein-Protein Interaction 1-gen-2020 Iralde-Lorente, Leire; Tassone, Giusy; Clementi, Letizia; Franci, Lorenzo; Munier, Claire C; Cau, Ylenia; Mori, Mattia; Chiariello, Mario; Angelucci, Adriano; Perry, Matthew W D; Pozzi, Cecilia; Mangani, Stefano; Botta, Maurizio -
Iron Binding in the Ferroxidase Site of Human Mitochondrial Ferritin 1-gen-2021 Ciambellotti, Silvia; Pratesi, Alessandro; Tassone, Giusy; Turano, Paola; Mangani, Stefano; Pozzi, Cecilia -
Mechanistic Aspects of the Asymmetric Transfer Hydrogenation in the Manufacture of Noradrenaline 1-gen-2022 Scorzelli, F.; Tassone, G.; Padula, D.; Zacche, M. -
Optimization of 1,2,4-Triazole-3-thiones toward Broad-Spectrum Metallo-β-lactamase Inhibitors Showing Potent Synergistic Activity on VIM- and NDM-1-Producing Clinical Isolates 1-gen-2022 Legru, Alice; Verdirosa, Federica; Vo-Hoang, Yen; Tassone, Giusy; Vascon, Filippo; Thomas, Caitlyn A; Sannio, Filomena; Corsica, Giuseppina; Benvenuti, Manuela; Feller, Georges; Coulon, Rémi; Marcoccia, Francesca; Devente, Savannah Rowane; Bouajila, Ezeddine; Piveteau, Catherine; Leroux, Florence; Deprez-Poulain, Rebecca; Deprez, Benoît; Licznar-Fajardo, Patricia; Crowder, Michael W; Cendron, Laura; Pozzi, Cecilia; Mangani, Stefano; Docquier, Jean-Denis; Hernandez, Jean-François; Gavara, Laurent -
Probing the role of Arg97 in Heat shock protein 90 N-terminal domain from the parasite Leishmania braziliensis through site-directed mutagenesis on the human counterpart 1-gen-2018 Tassone, Giusy; Mangani, Stefano; Botta, Maurizio; Pozzi, Cecilia -
Probing the role of Arg97 in the parasite Leishmania braziliensis Hsp90 through site directed mutagenesis on the human counterpart 1-gen-2018 Tassone, Giusy; Pozzi, Cecilia; Mangani, Stefano; Botta, Maurizio -
Probing the role of Arg97 in the parasite Leishmania braziliensis Hsp90 through site directed mutagenesis on the human counterpart 1-gen-2018 Tassone, Giusy; Pozzi, Cecilia; Mangani, Stefano; Botta, Maurizio -
Structural Bases for the Synergistic Inhibition of Human Thymidylate Synthase and Ovarian Cancer Cell Growth by Drug Combinations 1-gen-2021 Pozzi, Cecilia; Santucci, Matteo; Marverti, Gaetano; D'Arca, Domenico; Tagliazucchi, Lorenzo; Ferrari, Stefania; Gozzi, Gaia; Losi, Lorena; Tassone, Giusy; Mangani, Stefano; Ponterini, Glauco; Costi, Maria Paola -