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Titolo Data di pubblicazione Autore(i) File Abstract
Synthetic bioactive olivetol-related amides: the influence of the phenolic group in cannabinoid receptor activity 1-gen-2020 Brizzi, Antonella; Aiello, Francesca; Boccella, Serena; Grazia Cascio, Maria; De Petrocellis, Luciano; Frosini, Maria; Gado, Francesca; Ligresti, Alessia; Luongo, Livio; Marini, Pietro; Mugnaini, Claudia; Pessina, Federica; Corelli, Federico; Maione, Sabatino; Manera, Clementina; Pertwee, Roger G.; Di Marzo, Vincenzo -
Cytotoxic Effects of Cannabinoids on Human HT-29 Colorectal Adenocarcinoma Cells: Different Mechanisms of THC, CBD, and CB83 1-gen-2020 Cerretani, Daniela; Collodel, Giulia; Brizzi, Antonella; Fiaschi, ANNA IDA; Menchiari, Andrea; Moretti, Elena; Moltoni, Laura; Micheli, Lucia -
Anti-addictive properties of COR659 – Additional pharmacological evidence and comparison with a series of novel analogues 1-gen-2019 Maccioni, Paola; Colombo, Giancarlo; Lorrai, Irene; Fara, Federica; Carai, Mauro A. M.; Gessa, Gian Luigi; Brizzi, Antonella; Mugnaini, Claudia; Corelli, Federico -
Old strategies and new perspectives in modulating the endocannabinoid system 1-gen-2019 Brizzi, Antonella; Pessina, Federica -
3-Amino-alkylated indoles: Unexplored green products acting as anti-inflammatory agents 1-gen-2019 Mazzotta, S.; Frattaruolo, L.; Brindisi, M.; Ulivieri, C.; Vanni, F.; Brizzi, A.; Carullo, G.; Cappello, A. R.; Aiello, F. -
Synthesis of novel 2-(1-adamantanylcarboxamido)thiophene derivatives. Selective cannabinoid type 2 (CB2) receptor agonists as potential agents for the treatment of skin inflammatory disease 1-gen-2019 Mugnaini, Claudia; Rabbito, Alessandro; Brizzi, Antonella; Palombi, Nastasja; Petrosino, Stefania; Verde, Roberta; Di Marzo, Vincenzo; Ligresti, Alessia; Corelli, Federico -
Quercetin/oleic acid-based G-protein-coupled receptor 40 ligands as new insulin secretion modulators 1-gen-2017 Badolato, Mariateresa; Carullo, Gabriele; Perri, Mariarita; Cione, Erika; Manetti, Fabrizio; Di Gioia, Maria Luisa; Brizzi, Antonella; Caroleo, Maria Cristina; Aiello, Francesca -
Suppressing effect of COR659 on alcohol, sucrose, and chocolate self-administration in rats: Involvement of the GABAB and cannabinoid CB1 receptors 1-gen-2017 Maccioni, Paola; Colombo, Giancarlo; Lorrai, Irene; Zaru, Alessandro; Carai, Mauro A. M.; Gessa, Gian Luigi; Brizzi, Antonella; Mugnaini, Claudia; Corelli, Federico -
Design and Synthesis of New Transient Receptor Potential Vanilloid Type-1 (TRPV1) Channel Modulators: Identification, Molecular Modeling Analysis, and Pharmacological Characterization of the N-(4-Hydroxy-3-methoxybenzyl)-4-(thiophen-2-yl)butanamide, a Small Molecule Endowed with Agonist TRPV1 Activity and Protective Effects against Oxidative Stress 1-gen-2016 Aiello, F.; Badolato, M.; Pessina, Federica; Sticozzi, C.; Maestrini, Vanessa; Aldinucci, C.; Luongo, L.; Guida, F.; Ligresti, A.; Artese, A.; Allarà, M.; Costa, G.; Frosini, Maria; Schiano Morello, A.; De Petrocellis, L.; Valacchi, G.; Alcaro, S.; Maione, S.; Di Marzo, V.; Corelli, Federico; Brizzi, Antonella -
Investigations on the 4-Quinolone-3-carboxylic Acid Motif. 7. Synthesis and Pharmacological Evaluation of 4-Quinolone-3-carboxamides and 4-Hydroxy-2-quinolone-3-carboxamides as High Affinity Cannabinoid Receptor 2 (CB2R) Ligands with Improved Aqueous Solubility 1-gen-2016 Mugnaini, Claudia; Brizzi, Antonella; Ligresti, Alessia; Allarà, Marco; Lamponi, Stefania; Vacondio, Federica; Silva, Claudia; Mor, Marco; Di Marzo, Vincenzo; Corelli, Federico -
TRPV1-FAAH-COX: The Couples Game in Pain Treatment 1-gen-2016 Aiello, Francesca; Carullo, Gabriele; Badolato, Mariateresa; Brizzi, Antonella -
Ligandi TRPV1 1-gen-2014 Brizzi, Antonella; Corelli, Federico; Aiello, Francesca -
Structure-affinity relationships and pharmacological characterization of new alkyl-resorcinol cannabinoid receptor ligands: Identification of a dual cannabinoid receptor/TRPA1 channel agonist 1-gen-2014 Brizzi, Antonella; Aiello, Francesca; Marini, Pietro; Cascio, Maria Grazia; Corelli, Federico; Brizzi, Vittorio; De Petrocellis, Luciano; Ligresti, Alessia; Luongo, Livio; Lamponi, Stefania; Maione, Sabatino; Pertwee, Roger G.; Di Marzo, Vincenzo -
Active manganese dioxide promoted cyclization of ortho-(1H-pyrrol-1-yl)aryl and heteroaryl carboxylic acids to 5H-pyrrolo[1,2-a][3,1]benzoxazin-5-one derivatives 1-gen-2013 Fedora, Grande; Brizzi, Antonella; Garofalo, Antonio; Francesca, Aiello -
New fluoroquinolones active against fluoroquinolones-resistant Mycobacterium tuberculosis strains. 1-gen-2013 Guerrini, Valentina; De Rosa, M.; Pasquini, S.; Mugnaini, Claudia; Brizzi, Antonella; Cuppone, ANNA MARIA; Pozzi, Gianni; Corelli, Federico -
Investigations on the 4-Quinolone-3-carboxylic Acid Motif. 6. Synthesis and Pharmacological Evaluation of 7-Substituted 4-Quinolone-3-carboxamide Derivatives as High Affinity Ligands for Cannabinoid Receptors 1-gen-2012 Pasquini, Serena; DE ROSA, Maria; Ligresti, A.; Mugnaini, Claudia; Brizzi, Antonella; Caradonna, N. P.; Cascio, M. G.; Bolognini, D.; Pertwee, R. G.; Di Marzo, V.; Corelli, Federico -
Regioselective functionalization of quinolin-4(1H)-ones via sequential palladium-catalyzed reactions 1-gen-2011 Mugnaini, Claudia; Falciani, Chiara; DE ROSA, Maria; Brizzi, Antonella; Pasquini, Serena; Corelli, Federico -
1-Aryl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide: An effective scaffold for the design of either CB1 and CB2 receptor ligands 1-gen-2011 Piscitelli, F; Ligresti, A; LA REGINA, G; Gatti, V; Brizzi, Antonella; Pasquini, Serena; Allarà, M; CARAI M. A., M; Novellino, E; Colombo, G; DI MARZO, V; Corelli, Federico; Silvestri, R. -
Resorcinol-sn-Glycerol Derivatives: Novel 2-Arachidonoylglycerol (2-AG) Mimetics Endowed with High Affinity and Selectivity for Cannabinoid Type 1 (CB1) Receptor 1-gen-2011 Brizzi, Antonella; Cascio, M. G.; Frosini, Maria; Ligresti, A; Aiello, F; Biotti, I; Brizzi, Vittorio; Pertwee, R. G.; Corelli, Federico; DI MARZO, V. -
Development and characterization of immobilized cannabinoid receptor (CB1/CB2) open tubular column for on-line screening. 1-gen-2011 Moaddel, R; Rosenberg, A; Spelman, K; Frazier, J; Frazier, C; Nocerino, S; Brizzi, Antonella; Mugnaini, Claudia; Wainer, I. W. -
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