Sfoglia per Rivista ACS INFECTIOUS DISEASES
ANT2681: SAR Studies Leading to the Identification of a Metallo-β-lactamase Inhibitor with Potential for Clinical Use in Combination with Meropenem for the Treatment of Infections Caused by NDM-Producing Enterobacteriaceae
2020-01-01 Davies, D. T.; Leiris, S.; Sprynski, N.; Castandet, J.; Lozano, C.; Bousquet, J.; Zalacain, M.; Vasa, S.; Dasari, P. K.; Pattipati, R.; Vempala, N.; Gujjewar, S.; Godi, S.; Jallala, R.; Sathyap, R. R.; Darshanoju, N. A.; Ravu, V. R.; Juventhala, R. R.; Pottabathini, N.; Sharma, S.; Pothukanuri, S.; Holden, K.; Warn, P.; Marcoccia, F.; Benvenuti, M.; Pozzi, C.; Mangani, S.; Docquier, J. D.; Lemonnier, M.; Everett, M.
Chemical Optimization of Selective Pseudomonas aeruginosa LasB Elastase Inhibitors and Their Impact on LasB-Mediated Activation of IL-1β in Cellular and Animal Infection Models
2023-01-01 Everett, Martin J; Davies, David T; Leiris, Simon; Sprynski, Nicolas; Llanos, Agustina; Castandet, Jérôme M; Lozano, Clarisse; Larock, Christopher N; Larock, Doris L; Corsica, Giuseppina; Docquier, Jean-Denis; Pallin, Thomas D; Cridland, Andrew; Blench, Toby; Zalacain, Magdalena; Lemonnier, Marc
Optimization of Potent and Specific Trypanothione Reductase Inhibitors: A Structure-Based Drug Discovery Approach
2022-01-01 Battista, Theo; Federico, Stefano; Brogi, Simone; Pozzetti, Luca; Khan, Tuhina; Butini, Stefania; Ramunno, Anna; Fiorentino, Eleonora; Orsini, Stefania; Di Muccio, Trentina; Fiorillo, Annarita; Exertier, Cécile; Di Risola, Daniel; Colotti, Gianni; Gemma, Sandra; Ilari, Andrea; Campiani, Giuseppe
SAR Studies Leading to the Identification of a Novel Series of Metallo-β-lactamase Inhibitors for the Treatment of Carbapenem-Resistant Enterobacteriaceae Infections That Display Efficacy in an Animal Infection Model
2019-01-01 Leiris, Simon; Coelho, Alicia; Castandet, Jérôme; Bayet, Maëlle; Lozano, Clarisse; Bougnon, Juliette; Bousquet, Justine; Everett, Martin; Lemonnier, Marc; Sprynski, Nicolas; Zalacain, Magdalena; Pallin, Thomas David; Cramp, Michael C.; Jennings, Neil; Raphy, Gilles; Jones, Mark W.; Pattipati, Ramesh; Shankar, Battu; Sivasubrahmanyam, Relangi; Soodhagani, Ashok K.; Juventhala, Ramakrishna R.; Pottabathini, Narender; Pothukanuri, Srinivasu; Benvenuti, Manuela; Pozzi, Cecilia; Mangani, Stefano; De Luca, Filomena; Cerboni, Giulia; Docquier, Jean-Denis; Davies, David T.
Screening and Phenotypical Characterization of Schistosoma mansoni Histone Deacetylase 8 (SmHDAC8) Inhibitors as Multistage Antischistosomal Agents
2020-01-01 Saccoccia, F.; Brindisi, M.; Gimmelli, R.; Relitti, N.; Guidi, A.; Saraswati, A. P.; Cavella, C.; Brogi, S.; Chemi, G.; Butini, S.; Papoff, G.; Senger, J.; Herp, D.; Jung, M.; Campiani, G.; Gemma, S.; Ruberti, G.
Serinol-Based Benzoic Acid Esters as New Scaffolds for the Development of Adenovirus Infection Inhibitors: Design, Synthesis, and in Vitro Biological Evaluation
2021-01-01 Mazzotta, S.; Berastegui-Cabrera, J.; Carullo, G.; Vega-Holm, M.; Carretero-Ledesma, M.; Mendolia, L.; Aiello, F.; Iglesias-Guerra, F.; Pachon, J.; Vega-Perez, J. M.; Sanchez-Cespedes, J.
Structural Insights into the Development of Cycloguanil Derivatives as Trypanosoma brucei Pteridine-Reductase-1 Inhibitors
2019-01-01 Landi, Giacomo; Linciano, Pasquale; Borsari, Chiara; Bertolacini, Claudia P; Moraes, Carolina B; Cordeiro-da-Silva, Anabela; Gul, Sheraz; Witt, Gesa; Kuzikov, Maria; Costi, Maria Paola; Pozzi, Cecilia; Mangani, Stefano
(Thia)calixarenephosphonic Acids as Potent Inhibitors of the Nucleic Acid Chaperone Activity of the HIV-1 Nucleocapsid Protein with a New Binding Mode and Multitarget Antiviral Activity
2020-01-01 Humbert, N; Kovalenko, L; Saladini, F; Giannini, A; Pires, M; Botzanowski, T; Cherenok, S; Boudier, C; Sharma, Kk; Real, E; Zaporozhets, Oa; Cianférani, S; Seguin-Devaux, C; Poggialini, F; Botta, M; Zazzi, M; Kalchenko, Vi; Mori, M; Mély, Y.
Zidovudine-β-Lactam Pronucleoside Strategy for Selective Delivery into Gram-Negative Bacteria Triggered by β-Lactamases
2023-01-01 Rosales-Hurtado, Miyanou; Sannio, Filomena; Lari, Lindita; Verdirosa, Federica; Feller, Georges; Carretero, Elodie; Vo-Hoang, Yen; Licznar-Fajardo, Patricia; Docquier, Jean-Denis; Gavara, Laurent
| Titolo | Data di pubblicazione | Autore(i) | File | Abstract |
|---|---|---|---|---|
| ANT2681: SAR Studies Leading to the Identification of a Metallo-β-lactamase Inhibitor with Potential for Clinical Use in Combination with Meropenem for the Treatment of Infections Caused by NDM-Producing Enterobacteriaceae | 1-gen-2020 | Davies, D. T.; Leiris, S.; Sprynski, N.; Castandet, J.; Lozano, C.; Bousquet, J.; Zalacain, M.; Vasa, S.; Dasari, P. K.; Pattipati, R.; Vempala, N.; Gujjewar, S.; Godi, S.; Jallala, R.; Sathyap, R. R.; Darshanoju, N. A.; Ravu, V. R.; Juventhala, R. R.; Pottabathini, N.; Sharma, S.; Pothukanuri, S.; Holden, K.; Warn, P.; Marcoccia, F.; Benvenuti, M.; Pozzi, C.; Mangani, S.; Docquier, J. D.; Lemonnier, M.; Everett, M. | - | |
| Chemical Optimization of Selective Pseudomonas aeruginosa LasB Elastase Inhibitors and Their Impact on LasB-Mediated Activation of IL-1β in Cellular and Animal Infection Models | 1-gen-2023 | Everett, Martin J; Davies, David T; Leiris, Simon; Sprynski, Nicolas; Llanos, Agustina; Castandet, Jérôme M; Lozano, Clarisse; Larock, Christopher N; Larock, Doris L; Corsica, Giuseppina; Docquier, Jean-Denis; Pallin, Thomas D; Cridland, Andrew; Blench, Toby; Zalacain, Magdalena; Lemonnier, Marc | - | |
| Optimization of Potent and Specific Trypanothione Reductase Inhibitors: A Structure-Based Drug Discovery Approach | 1-gen-2022 | Battista, Theo; Federico, Stefano; Brogi, Simone; Pozzetti, Luca; Khan, Tuhina; Butini, Stefania; Ramunno, Anna; Fiorentino, Eleonora; Orsini, Stefania; Di Muccio, Trentina; Fiorillo, Annarita; Exertier, Cécile; Di Risola, Daniel; Colotti, Gianni; Gemma, Sandra; Ilari, Andrea; Campiani, Giuseppe | - | |
| SAR Studies Leading to the Identification of a Novel Series of Metallo-β-lactamase Inhibitors for the Treatment of Carbapenem-Resistant Enterobacteriaceae Infections That Display Efficacy in an Animal Infection Model | 1-gen-2019 | Leiris, Simon; Coelho, Alicia; Castandet, Jérôme; Bayet, Maëlle; Lozano, Clarisse; Bougnon, Juliette; Bousquet, Justine; Everett, Martin; Lemonnier, Marc; Sprynski, Nicolas; Zalacain, Magdalena; Pallin, Thomas David; Cramp, Michael C.; Jennings, Neil; Raphy, Gilles; Jones, Mark W.; Pattipati, Ramesh; Shankar, Battu; Sivasubrahmanyam, Relangi; Soodhagani, Ashok K.; Juventhala, Ramakrishna R.; Pottabathini, Narender; Pothukanuri, Srinivasu; Benvenuti, Manuela; Pozzi, Cecilia; Mangani, Stefano; De Luca, Filomena; Cerboni, Giulia; Docquier, Jean-Denis; Davies, David T. | - | |
| Screening and Phenotypical Characterization of Schistosoma mansoni Histone Deacetylase 8 (SmHDAC8) Inhibitors as Multistage Antischistosomal Agents | 1-gen-2020 | Saccoccia, F.; Brindisi, M.; Gimmelli, R.; Relitti, N.; Guidi, A.; Saraswati, A. P.; Cavella, C.; Brogi, S.; Chemi, G.; Butini, S.; Papoff, G.; Senger, J.; Herp, D.; Jung, M.; Campiani, G.; Gemma, S.; Ruberti, G. | - | |
| Serinol-Based Benzoic Acid Esters as New Scaffolds for the Development of Adenovirus Infection Inhibitors: Design, Synthesis, and in Vitro Biological Evaluation | 1-gen-2021 | Mazzotta, S.; Berastegui-Cabrera, J.; Carullo, G.; Vega-Holm, M.; Carretero-Ledesma, M.; Mendolia, L.; Aiello, F.; Iglesias-Guerra, F.; Pachon, J.; Vega-Perez, J. M.; Sanchez-Cespedes, J. | - | |
| Structural Insights into the Development of Cycloguanil Derivatives as Trypanosoma brucei Pteridine-Reductase-1 Inhibitors | 1-gen-2019 | Landi, Giacomo; Linciano, Pasquale; Borsari, Chiara; Bertolacini, Claudia P; Moraes, Carolina B; Cordeiro-da-Silva, Anabela; Gul, Sheraz; Witt, Gesa; Kuzikov, Maria; Costi, Maria Paola; Pozzi, Cecilia; Mangani, Stefano | - | |
| (Thia)calixarenephosphonic Acids as Potent Inhibitors of the Nucleic Acid Chaperone Activity of the HIV-1 Nucleocapsid Protein with a New Binding Mode and Multitarget Antiviral Activity | 1-gen-2020 | Humbert, N; Kovalenko, L; Saladini, F; Giannini, A; Pires, M; Botzanowski, T; Cherenok, S; Boudier, C; Sharma, Kk; Real, E; Zaporozhets, Oa; Cianférani, S; Seguin-Devaux, C; Poggialini, F; Botta, M; Zazzi, M; Kalchenko, Vi; Mori, M; Mély, Y. | - | |
| Zidovudine-β-Lactam Pronucleoside Strategy for Selective Delivery into Gram-Negative Bacteria Triggered by β-Lactamases | 1-gen-2023 | Rosales-Hurtado, Miyanou; Sannio, Filomena; Lari, Lindita; Verdirosa, Federica; Feller, Georges; Carretero, Elodie; Vo-Hoang, Yen; Licznar-Fajardo, Patricia; Docquier, Jean-Denis; Gavara, Laurent | - |
Legenda icone
- file ad accesso aperto
- file disponibili sulla rete interna
- file disponibili agli utenti autorizzati
- file disponibili solo agli amministratori
- file sotto embargo
- nessun file disponibile