Sfoglia per Autore
Early investigation of a novel SI306 theranostic prodrug for glioblastoma treatment
2024-01-01 Vagaggini, Chiara; Petroni, Debora; D'Agostino, Ilaria; Poggialini, Federica; Cavallini, Chiara; Cianciusi, Annarita; Salis, Annalisa; D'Antona, Lucia; Francesconi, Valeria; Manetti, Fabrizio; Damonte, Gianluca; Musumeci, Francesca; Menichetti, Luca; Dreassi, Elena; Carbone, Anna; Schenone, Silvia
Optimization of potent, broad-spectrum, and specific anti-influenza compounds targeting RNA polymerase PA-PB1 heterodimerization
2024-01-01 Bonomini, Anna; Felicetti, Tommaso; Pacetti, Martina; Bertagnin, Chiara; Coletti, Alice; Giammarino, Federica; De Angelis, Marta; Poggialini, Federica; Macchiarulo, Antonio; Sabatini, Stefano; Mercorelli, Beatrice; Nencioni, Lucia; Vicenti, Ilaria; Dreassi, Elena; Cecchetti, Violetta; Tabarrini, Oriana; Loregian, Arianna; Massari, Serena
An update on antibacterial AlkylGuanidino Ureas: Design of new derivatives, synergism with colistin and data analysis of the whole library
2024-01-01 Ardino, C.; Sannio, F.; Poli, G.; Galati, S.; Dreassi, E.; Botta, L.; Docquier, J. D.; D'Agostino, I.
Serendipitous identification of azine anticancer agents using a privileged scaffold morphing strategy
2024-01-01 Cesarini, Silvia; Vicenti, Ilaria; Poggialini, Federica; Filippi, Silvia; Mancin, Eleonora; Fiaschi, Lia; De Marchi, Elisa; Giammarino, Federica; Vagaggini, Chiara; Bizzarri, Bruno Mattia; Saladino, Raffaele; Dreassi, Elena; Zazzi, Maurizio; Botta, Lorenzo
Design, synthesis, ADME and biological evaluation of benzylpiperidine and benzylpiperazine derivatives as novel reversible monoacylglycerol lipase (MAGL) inhibitors
2024-01-01 Di Stefano, M.; Masoni, S.; Bononi, G.; Poli, G.; Galati, S.; Gado, F.; Manzi, S.; Vagaggini, C.; Brai, A.; Caligiuri, I.; Asif, K.; Rizzolio, F.; Macchia, M.; Chicca, A.; Sodi, A.; Di Bussolo, V.; Minutolo, F.; Meier, P.; Gertsch, J.; Granchi, C.; Dreassi, E.; Tuccinardi, T.
Identification of Novel Non-Nucleoside Inhibitors of Zika Virus NS5 Protein Targeting MTase Activity
2024-01-01 Fiorucci, D.; Meaccini, M.; Poli, G.; Stincarelli, M. A.; Vagaggini, C.; Giannecchini, S.; Sutto-Ortiz, P.; Canard, B.; Decroly, E.; Dreassi, E.; Brai, A.; Botta, M.
Targeting GLI1 and GLI2 with small molecule inhibitors to suppress GLI-dependent transcription and tumor growth
2023-01-01 Maresca, Luisa; Crivaro, Enrica; Migliorini, Francesca; Anichini, Giulia; Giammona, Alessandro; Pepe, Sara; Poggialini, Federica; Vagaggini, Chiara; Giannini, Giuseppe; Sestini, Serena; Borgognoni, Lorenzo; Lapucci, Andrea; Dreassi, Elena; Taddei, Maurizio; Manetti, Fabrizio; Petricci, Elena; Stecca, Barbara
Efficient use of agricultural waste to naturally fortify Tenebrio molitor mealworms and evaluation of their nutraceutical properties
2023-01-01 Brai, A.; Poggialini, F.; Trivisani, C. I.; Vagaggini, C.; Tarchi, F.; Francardi, V.; Dreassi, E.
Tyrosine kinase inhibitor Si409 has in vitro and in vivo anti-tumor activity against diffuse large B-cell lymphoma
2023-01-01 Rango, E.; Di Maria, S.; Zamperini, C.; Poggialini, F.; Crespan, E.; Perini, C.; Sabetta, S.; Saponara, S.; Fusi, F.; Maga, G.; Angelucci, A.; Gaudio, E.; Berton, F.; Schenone, S.; Botta, L.; Dreassi, E.; Botta, M.
Triazolo[3,4- b]benzothiazole scaffold as versatile nicotinamide mimic allowing nanomolar inhibition of different PARP enzymes
2023-01-01 Murthy, S.; Nizi, M. G.; Maksimainen, M. M.; Massari, S.; Alaviuhkola, J.; Lippok, B. E.; Vagaggini, C.; Sowa, S. T.; Galera-Prat, A.; Ashok, Y.; Venkannagari, H.; Prunskaite-Hyyrylainen, R.; Dreassi, E.; Luscher, B.; Korn, P.; Tabarrini, O.; Lehtio, L.
Progress towards adjuvant development: focus on antiviral therapy
2023-01-01 Brai, A.; Poggialini, F.; Pasqualini, C.; Trivisani, C. I.; Vagaggini, C.; Dreassi, E.
The impact of counterions in biological activity: case study of antibacterial alkylguanidino ureas
2023-01-01 Ardino, C.; Sannio, F.; Pasero, C.; Botta, L.; Dreassi, E.; Docquier, J. D.; D'Agostino, I.
Tenebrio molitor as a Simple and Cheap Preclinical Pharmacokinetic and Toxicity Model
2023-01-01 Brai, Annalaura; Poggialini, Federica; Vagaggini, Chiara; Pasqualini, Claudia; Simoni, Sauro; Francardi, Valeria; Dreassi, Elena
Discovery and Optimization of a Novel Macrocyclic Amidinourea Series Active as Acidic Mammalian Chitinase Inhibitors
2023-01-01 Balestri, Lorenzo Jacopo Ilic; Trivisani, Claudia Immacolata; Orofino, Francesco; Fiorucci, Diego; Truglio, Giuseppina Ivana; D'Agostino, Ilaria; Poggialini, Federica; Botta, Lorenzo; Docquier, Jean-Denis; Dreassi, Elena
THE REPLACEMENT OF FLOUR-BASED FEED WITH PELLETS REDUCES DUSTINESS AND IMPROVES TENEBRIO MOLITOR BREEDERS’ SAFETY
2023-01-01 Brai, A.; Tarchi, F.; Pasqualini, C.; Poggialini, F.; Vagaggini, C.; Frosinini, R.; Simoni, S.; Francardi, V.; Dreassi, E.
Brevundimonas aurantiaca M3d10, isolated from the olive fly, produces hydroxylated astaxanthin
2023-01-01 Centini, Marisanna; Martinez-Sañudo, Isabel; Biagi, Marco; Dreassi, Elena; Mazzon, Luca; Marri, Laura
Biological Evaluation and In Vitro Characterization of ADME Profile of In-House Pyrazolo[3,4-d]pyrimidines as Dual Tyrosine Kinase Inhibitors Active against Glioblastoma Multiforme
2023-01-01 Poggialini, Federica; Vagaggini, Chiara; Brai, Annalaura; Pasqualini, Claudia; Crespan, Emmanuele; Maga, Giovanni; Perini, Cecilia; Cabella, Noemi; Botta, Lorenzo; Musumeci, Francesca; Frosini, Maria; Schenone, Silvia; Dreassi, Elena
Exploiting fall foliage by-products to optimize Tenebrio molitor nutraceutical value
2023-01-01 Brai, A.; Provenzani, M. P.; Pasqualini, C.; Poggialini, F.; Vagaggini, C.; Tarchi, F.; Frosinini, R.; Francardi, V.; Simoni, S.; Dreassi, E.
Sweet cherry extract as permeation enhancer of tyrosine kinase inhibitors: a promising prospective for future oral anticancer therapies
2023-01-01 Poggialini, F.; Vagaggini, C.; Brai, A.; Pasqualini, C.; Carbone, A.; Musumeci, F.; Schenone, S.; Dreassi, E.
Development and validation of derivatization-based LC-MS/MS method for quantification of short-chain fatty acids in human, rat, and mouse plasma
2023-01-01 Vagaggini, Chiara; Brai, Annalaura; Bonente, Denise; Lombardi, Jessica; Poggialini, Federica; Pasqualini, Claudia; Barone, Virginia; Nicoletti, Claudio; Bertelli, Eugenio; Dreassi, Elena
| Titolo | Data di pubblicazione | Autore(i) | File | Abstract |
|---|---|---|---|---|
| Early investigation of a novel SI306 theranostic prodrug for glioblastoma treatment | 1-gen-2024 | Vagaggini, Chiara; Petroni, Debora; D'Agostino, Ilaria; Poggialini, Federica; Cavallini, Chiara; Cianciusi, Annarita; Salis, Annalisa; D'Antona, Lucia; Francesconi, Valeria; Manetti, Fabrizio; Damonte, Gianluca; Musumeci, Francesca; Menichetti, Luca; Dreassi, Elena; Carbone, Anna; Schenone, Silvia | - | |
| Optimization of potent, broad-spectrum, and specific anti-influenza compounds targeting RNA polymerase PA-PB1 heterodimerization | 1-gen-2024 | Bonomini, Anna; Felicetti, Tommaso; Pacetti, Martina; Bertagnin, Chiara; Coletti, Alice; Giammarino, Federica; De Angelis, Marta; Poggialini, Federica; Macchiarulo, Antonio; Sabatini, Stefano; Mercorelli, Beatrice; Nencioni, Lucia; Vicenti, Ilaria; Dreassi, Elena; Cecchetti, Violetta; Tabarrini, Oriana; Loregian, Arianna; Massari, Serena | - | |
| An update on antibacterial AlkylGuanidino Ureas: Design of new derivatives, synergism with colistin and data analysis of the whole library | 1-gen-2024 | Ardino, C.; Sannio, F.; Poli, G.; Galati, S.; Dreassi, E.; Botta, L.; Docquier, J. D.; D'Agostino, I. | - | |
| Serendipitous identification of azine anticancer agents using a privileged scaffold morphing strategy | 1-gen-2024 | Cesarini, Silvia; Vicenti, Ilaria; Poggialini, Federica; Filippi, Silvia; Mancin, Eleonora; Fiaschi, Lia; De Marchi, Elisa; Giammarino, Federica; Vagaggini, Chiara; Bizzarri, Bruno Mattia; Saladino, Raffaele; Dreassi, Elena; Zazzi, Maurizio; Botta, Lorenzo | - | |
| Design, synthesis, ADME and biological evaluation of benzylpiperidine and benzylpiperazine derivatives as novel reversible monoacylglycerol lipase (MAGL) inhibitors | 1-gen-2024 | Di Stefano, M.; Masoni, S.; Bononi, G.; Poli, G.; Galati, S.; Gado, F.; Manzi, S.; Vagaggini, C.; Brai, A.; Caligiuri, I.; Asif, K.; Rizzolio, F.; Macchia, M.; Chicca, A.; Sodi, A.; Di Bussolo, V.; Minutolo, F.; Meier, P.; Gertsch, J.; Granchi, C.; Dreassi, E.; Tuccinardi, T. | - | |
| Identification of Novel Non-Nucleoside Inhibitors of Zika Virus NS5 Protein Targeting MTase Activity | 1-gen-2024 | Fiorucci, D.; Meaccini, M.; Poli, G.; Stincarelli, M. A.; Vagaggini, C.; Giannecchini, S.; Sutto-Ortiz, P.; Canard, B.; Decroly, E.; Dreassi, E.; Brai, A.; Botta, M. | - | |
| Targeting GLI1 and GLI2 with small molecule inhibitors to suppress GLI-dependent transcription and tumor growth | 1-gen-2023 | Maresca, Luisa; Crivaro, Enrica; Migliorini, Francesca; Anichini, Giulia; Giammona, Alessandro; Pepe, Sara; Poggialini, Federica; Vagaggini, Chiara; Giannini, Giuseppe; Sestini, Serena; Borgognoni, Lorenzo; Lapucci, Andrea; Dreassi, Elena; Taddei, Maurizio; Manetti, Fabrizio; Petricci, Elena; Stecca, Barbara | - | |
| Efficient use of agricultural waste to naturally fortify Tenebrio molitor mealworms and evaluation of their nutraceutical properties | 1-gen-2023 | Brai, A.; Poggialini, F.; Trivisani, C. I.; Vagaggini, C.; Tarchi, F.; Francardi, V.; Dreassi, E. | - | |
| Tyrosine kinase inhibitor Si409 has in vitro and in vivo anti-tumor activity against diffuse large B-cell lymphoma | 1-gen-2023 | Rango, E.; Di Maria, S.; Zamperini, C.; Poggialini, F.; Crespan, E.; Perini, C.; Sabetta, S.; Saponara, S.; Fusi, F.; Maga, G.; Angelucci, A.; Gaudio, E.; Berton, F.; Schenone, S.; Botta, L.; Dreassi, E.; Botta, M. | - | |
| Triazolo[3,4- b]benzothiazole scaffold as versatile nicotinamide mimic allowing nanomolar inhibition of different PARP enzymes | 1-gen-2023 | Murthy, S.; Nizi, M. G.; Maksimainen, M. M.; Massari, S.; Alaviuhkola, J.; Lippok, B. E.; Vagaggini, C.; Sowa, S. T.; Galera-Prat, A.; Ashok, Y.; Venkannagari, H.; Prunskaite-Hyyrylainen, R.; Dreassi, E.; Luscher, B.; Korn, P.; Tabarrini, O.; Lehtio, L. | - | |
| Progress towards adjuvant development: focus on antiviral therapy | 1-gen-2023 | Brai, A.; Poggialini, F.; Pasqualini, C.; Trivisani, C. I.; Vagaggini, C.; Dreassi, E. | - | |
| The impact of counterions in biological activity: case study of antibacterial alkylguanidino ureas | 1-gen-2023 | Ardino, C.; Sannio, F.; Pasero, C.; Botta, L.; Dreassi, E.; Docquier, J. D.; D'Agostino, I. | - | |
| Tenebrio molitor as a Simple and Cheap Preclinical Pharmacokinetic and Toxicity Model | 1-gen-2023 | Brai, Annalaura; Poggialini, Federica; Vagaggini, Chiara; Pasqualini, Claudia; Simoni, Sauro; Francardi, Valeria; Dreassi, Elena | - | |
| Discovery and Optimization of a Novel Macrocyclic Amidinourea Series Active as Acidic Mammalian Chitinase Inhibitors | 1-gen-2023 | Balestri, Lorenzo Jacopo Ilic; Trivisani, Claudia Immacolata; Orofino, Francesco; Fiorucci, Diego; Truglio, Giuseppina Ivana; D'Agostino, Ilaria; Poggialini, Federica; Botta, Lorenzo; Docquier, Jean-Denis; Dreassi, Elena | - | |
| THE REPLACEMENT OF FLOUR-BASED FEED WITH PELLETS REDUCES DUSTINESS AND IMPROVES TENEBRIO MOLITOR BREEDERS’ SAFETY | 1-gen-2023 | Brai, A.; Tarchi, F.; Pasqualini, C.; Poggialini, F.; Vagaggini, C.; Frosinini, R.; Simoni, S.; Francardi, V.; Dreassi, E. | - | |
| Brevundimonas aurantiaca M3d10, isolated from the olive fly, produces hydroxylated astaxanthin | 1-gen-2023 | Centini, Marisanna; Martinez-Sañudo, Isabel; Biagi, Marco; Dreassi, Elena; Mazzon, Luca; Marri, Laura | - | |
| Biological Evaluation and In Vitro Characterization of ADME Profile of In-House Pyrazolo[3,4-d]pyrimidines as Dual Tyrosine Kinase Inhibitors Active against Glioblastoma Multiforme | 1-gen-2023 | Poggialini, Federica; Vagaggini, Chiara; Brai, Annalaura; Pasqualini, Claudia; Crespan, Emmanuele; Maga, Giovanni; Perini, Cecilia; Cabella, Noemi; Botta, Lorenzo; Musumeci, Francesca; Frosini, Maria; Schenone, Silvia; Dreassi, Elena | - | |
| Exploiting fall foliage by-products to optimize Tenebrio molitor nutraceutical value | 1-gen-2023 | Brai, A.; Provenzani, M. P.; Pasqualini, C.; Poggialini, F.; Vagaggini, C.; Tarchi, F.; Frosinini, R.; Francardi, V.; Simoni, S.; Dreassi, E. | - | |
| Sweet cherry extract as permeation enhancer of tyrosine kinase inhibitors: a promising prospective for future oral anticancer therapies | 1-gen-2023 | Poggialini, F.; Vagaggini, C.; Brai, A.; Pasqualini, C.; Carbone, A.; Musumeci, F.; Schenone, S.; Dreassi, E. | - | |
| Development and validation of derivatization-based LC-MS/MS method for quantification of short-chain fatty acids in human, rat, and mouse plasma | 1-gen-2023 | Vagaggini, Chiara; Brai, Annalaura; Bonente, Denise; Lombardi, Jessica; Poggialini, Federica; Pasqualini, Claudia; Barone, Virginia; Nicoletti, Claudio; Bertelli, Eugenio; Dreassi, Elena | - |
Legenda icone
- file ad accesso aperto
- file disponibili sulla rete interna
- file disponibili agli utenti autorizzati
- file disponibili solo agli amministratori
- file sotto embargo
- nessun file disponibile