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Mostrati risultati da 21 a 40 di 194
Titolo Data di pubblicazione Autore(i) File Abstract
Suppressing effect of CMPPE, a new positive allosteric modulator of the GABAB receptor, on alcohol self-administration and reinstatement of alcohol seeking in rats 1-gen-2019 Maccioni, Paola; Fara, Federica; Lorrai, Irene; Acciaro, Carla; Mugnaini, Claudia; Corelli, Federico; Colombo, Giancarlo -
Operant, oral alcohol self-administration: Sex differences in Sardinian alcohol-preferring rats 1-gen-2019 Lorrai, Irene; Contini, Andrea; Luigi Gessa, Gian; Mugnaini, Claudia; Corelli, Federico; Colombo, Giancarlo; Maccioni, Paola -
Anti-addictive properties of COR659 – Additional pharmacological evidence and comparison with a series of novel analogues 1-gen-2019 Maccioni, Paola; Colombo, Giancarlo; Lorrai, Irene; Fara, Federica; Carai, Mauro A. M.; Gessa, Gian Luigi; Brizzi, Antonella; Mugnaini, Claudia; Corelli, Federico -
Suppressing effect of COR659 on alcohol, sucrose, and chocolate self-administration in rats: Involvement of the GABAB and cannabinoid CB1 receptors 1-gen-2017 Maccioni, Paola; Colombo, Giancarlo; Lorrai, Irene; Zaru, Alessandro; Carai, Mauro A. M.; Gessa, Gian Luigi; Brizzi, Antonella; Mugnaini, Claudia; Corelli, Federico -
USO DI DERIVATI DELL’ACIDO 2-AMMINOTIOFEN-3- CARBOSSILICO PER IL TRATTAMENTO DELLE DIPENDENZE DA CIBO 1-gen-2016 Colombo, Giancarlo; Carai, Mauro; Gessa Gian, Luigi; Mugnaini, Claudia; Corelli, Federico; Maccioni, Paola -
Reducing effect of saikosaponin A, an active ingredient of Bupleurum falcatum, on alcohol self-administration in rats: Possible involvement of the GABAB receptor 1-gen-2016 Maccioni, Paola; Lorrai, Irene; Carai, Mauro A. M.; Riva, Antonella; Morazzoni, Paolo; Mugnaini, Claudia; Corelli, Federico; Gessa, Gian Luigi; Colombo, Giancarlo -
The allosteric modulation of the GABAB receptor: a medicinal chemistry perspective 1-gen-2016 Mugnaini, Claudia; Corelli, Federico -
Total Synthesis of δ-Sanshool and Analogues Thereof 1-gen-2016 Mugnaini, Claudia; Corelli, Federico -
Chemistry of GABAB receptor ligands: focus on agonists and antagonists 1-gen-2016 Corelli, Federico; Mugnaini, Claudia -
Human Tuberculosis. III. Current and Prospective Approaches in Anti-Tubercular Therapy 1-gen-2016 Sgaragli, Giampietro; Frosini, Maria; Saponara, Simona; Corelli, Federico -
Design and Synthesis of New Transient Receptor Potential Vanilloid Type-1 (TRPV1) Channel Modulators: Identification, Molecular Modeling Analysis, and Pharmacological Characterization of the N-(4-Hydroxy-3-methoxybenzyl)-4-(thiophen-2-yl)butanamide, a Small Molecule Endowed with Agonist TRPV1 Activity and Protective Effects against Oxidative Stress 1-gen-2016 Aiello, F.; Badolato, M.; Pessina, Federica; Sticozzi, C.; Maestrini, Vanessa; Aldinucci, C.; Luongo, L.; Guida, F.; Ligresti, A.; Artese, A.; Allarà, M.; Costa, G.; Frosini, Maria; Schiano Morello, A.; De Petrocellis, L.; Valacchi, G.; Alcaro, S.; Maione, S.; Di Marzo, V.; Corelli, Federico; Brizzi, Antonella -
Investigations on the 4-Quinolone-3-carboxylic Acid Motif. 7. Synthesis and Pharmacological Evaluation of 4-Quinolone-3-carboxamides and 4-Hydroxy-2-quinolone-3-carboxamides as High Affinity Cannabinoid Receptor 2 (CB2R) Ligands with Improved Aqueous Solubility 1-gen-2016 Mugnaini, Claudia; Brizzi, Antonella; Ligresti, Alessia; Allarà, Marco; Lamponi, Stefania; Vacondio, Federica; Silva, Claudia; Mor, Marco; Di Marzo, Vincenzo; Corelli, Federico -
Anxiety-like behaviors at the end of the nocturnal period in sP rats with a “history” of unpredictable, limited access to alcohol. 1-gen-2015 Colombo, G.; Lobina, C.; Maccioni, P.; Carai, M. A. M.; Lorrai, I.; Zaru, A.; Contini, A.; Mugnaini, Claudia; Corelli, Federico; Gessa, G. -
Inhibition of alcohol self-administration by positive allosteric modulators of the GABA(B) receptor in rats: lack of tolerance and potentiation of baclofen 1-gen-2015 Maccioni, P.; Vargiolu, D.; Thomas, A.; Malherbe, P.; Mugnaini, Claudia; Corelli, Federico; Leite Morris, K.; Gessa, G. L.; Colombo, G. -
Ligandi TRPV1 1-gen-2014 Brizzi, Antonella; Corelli, Federico; Aiello, Francesca -
NUOVA TERAPIA PER IL TRATTAMENTO DELL'IPERURICEMIA NELLA SINDROME DI LESCH-NYHAN 1-gen-2014 Micheli, Vanna; Iacomelli, Gabriella; Corelli, Federico; Mugnaini, Claudia; Baldini, Eva -
Synthesis, 1 structural properties, and pharmacological evaluation of 2-(acylamino)thiophene-3-carboxamides and analogues thereof 1-gen-2014 Mugnaini, Claudia; Pedani, Valentina; Giunta, D.; Sechi, B.; Solinas, M.; Casti, A.; Castelli, M. P.; Giorgi, Gianluca; Corelli, Federico -
Hsp90 Inhibitors, part 2: combining ligand-based and structure-based approches for virtual screening application 1-gen-2014 Caroli, A.; Ballante, F.; Wickersham, R. B.; Corelli, Federico; Ragno, R. -
Structure-affinity relationships and pharmacological characterization of new alkyl-resorcinol cannabinoid receptor ligands: Identification of a dual cannabinoid receptor/TRPA1 channel agonist 1-gen-2014 Brizzi, Antonella; Aiello, Francesca; Marini, Pietro; Cascio, Maria Grazia; Corelli, Federico; Brizzi, Vittorio; De Petrocellis, Luciano; Ligresti, Alessia; Luongo, Livio; Lamponi, Stefania; Maione, Sabatino; Pertwee, Roger G.; Di Marzo, Vincenzo -
New fluoroquinolones active against fluoroquinolones-resistant Mycobacterium tuberculosis strains. 1-gen-2013 Guerrini, Valentina; De Rosa, M.; Pasquini, S.; Mugnaini, Claudia; Brizzi, Antonella; Cuppone, ANNA MARIA; Pozzi, Gianni; Corelli, Federico -
Mostrati risultati da 21 a 40 di 194
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