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Titolo Data di pubblicazione Autore(i) File Abstract
4-Hydroxyphenylpyruvate Dioxygenase and Its Inhibition in Plants and Animals: Small Molecules as Herbicides and Agents for the Treatment of Human Inherited Diseases 1-gen-2017 Santucci, Annalisa; Bernardini, Giulia; Braconi, Daniela; Petricci, Elena; Manetti, Fabrizio -
Gli1 inhibitors and uses thereof 1-gen-2017 Giannini, Giuseppe; Taddei, Maurizio; Manetti, Fabrizio; Petricci, Elena; Stecca, Barbara -
Synthesis and SAR evaluation of novel thioridazine derivatives active against drug-resistant tuberculosis 1-gen-2017 Scalacci, Nicolò; Brown, Alistair K.; Pavan, Fernando R.; Ribeiro, Camila M.; Manetti, Fabrizio; Bhakta, Sanjib; Maitra, Arundhati; Smith, Darren L.; Petricci, Elena; Castagnolo, Daniele -
Smoothened-antagonists reverse homogentisic acid-induced alterations of Hedgehog signaling and primary cilium length in alkaptonuria 1-gen-2017 Gambassi, Silvia; Geminiani, Michela; Thorpe, Stephen D.; Bernardini, Giulia; Millucci, Lia; Braconi, Daniela; Orlandini, Maurizio; Thompson, Clare L.; Petricci, Elena; Manetti, Fabrizio; Taddei, Maurizio; Knight, Martin M.; Santucci, Annalisa -
Design and synthesis of 1-((1,5-bis(4-chlorophenyl)-2-methyl-1H-pyrrol-3-yl)methyl)-4-methylpiperazine (BM212) and N-Adamantan-2-yl-N'-((E)-3,7-dimethyl-octa-2,6-dienyl)-ethane-1,2-diamine (SQ109) pyrrole hybrid derivatives: discovery of potent anti-tubercular agents effective against multi-drug resistant mycobacteria 1-gen-2016 Sanjib, Bhakta; Nicolò, Scalacci; Arundhati, Maitra; Alistair K., Brown; Saiprasad, Dasugari; Dimitrios, Evangelopoulos; Timothy D., Mchugh; Parisa N., Mortazavi; Alexander, Twist; Petricci, Elena; Manetti, Fabrizio; Daniele, Castagnolo -
Ruthenium-catalysed C-alkylation of 1,3-dicarbonyl compounds with primary alcohols and synthesis of 3-keto-quinolines 1-gen-2016 Cini, Elena; Petricci, Elena; Truglio, GIUSEPPINA IVANA; Vecchio, Marialaura; Taddei, Maurizio -
Microwave Assisted Hydrogenation of Pyridinecarboxylates: a Convenient Access to Valuable Scaffolds for Diversity Oriented Synthesis 1-gen-2016 Ferrini, Serena; Cini, Elena; Petricci, Elena; Taddei, Maurizio -
Design, synthesis and biological characterization of a new class of osteogenic (1H)-quinolone derivatives 1-gen-2016 Manetti, Fabrizio; Petricci, Elena; Gabrielli, Annalisa; Mann, Andrè; Faure, Hélène; Gorojankina, Tatiana; Brasseur, Laurent; Hoch, Lucile; Ruat, Martial; Taddei, Maurizio -
Novel acylguanidine derivatives targeting smoothened induce antiproliferative and pro-apoptotic effects in chronic myeloid leukemia cells 1-gen-2016 Chiarenza, Alessandra; Manetti, Fabrizio; Petricci, Elena; Ruat, Martial; Naldini, Antonella; Taddei, Maurizio; Carraro, Fabio -
Evaluation of WO2014207069 A1: Multitarget Hedgehog pathway inhibitors and uses thereof 1-gen-2016 Manetti, Fabrizio; Petricci, Elena -
Hedgehog associated to microparticles inhibits adipocyte differentiation via a non-canonical pathway 1-gen-2016 Fleury, Audrey; Hoch, Lucile; Martinez, M. Carmen; Faure, Hélène; Taddei, Maurizio; Petricci, Elena; Manetti, Fabrizio; Girard, Nicolas; Mann, André; Jacques, Caroline; Larghero, Jérome; Ruat, Martial; Andriantsitohaina, Ramaroson; Le Lay, Soazig -
Overcoming resistence to imatinib by targeting hedgehog signaling 1-gen-2015 Chiarenza, Alessandra; Manetti, Fabrizio; Petricci, Elena; Taddei, Maurizio; Naldini, Antonella; Carraro, Fabio -
Synthesis of 1,​2,​3-​substituted pyrroles from propargylamines via a one-​pot tandem enyne cross metathesis-​cyclization reaction 1-gen-2015 Chachignon, Helene; Scalacci, Nicolo; Petricci, Elena; Castagnolo, Daniele -
MRT-92 inhibits Hedgehog signaling by blocking overlapping binding sites in the transmembrane domain of the Smoothened receptor 1-gen-2015 Hoch, L; Faure, H; Roudaut, H; Schoenfelder, A; Mann, A; Girard, N; Bihannic, L; Ayrault, O; Petricci, Elena; Taddei, Maurizio; Rognan, D; Ruat, M. 2. -
Targeting the Hedgehog Signaling Pathway with Small Molecules from Natural Sources 1-gen-2015 Petricci, Elena; Manetti, Fabrizio -
A highly stereo-controlled protocol to prepare pipecolic acids based on Heck and cyclohydrocarbonylation reactions 1-gen-2015 Arena, Giada; Cini, Elena; Petricci, Elena; Randino, E.; Taddei, Maurizio -
Domino Hydrogenation-Reductive Amination of Phenols, a Simple Process To Access Substituted Cyclohexylamines 1-gen-2015 Jumde, VARSHA RAVINDRA; Petricci, Elena; Petrucci, C; Santillo, Niccolo'; Taddei, Maurizio; Vaccaro, L. 2. -
Structure–Activity Relationships and Mechanism of Action of Small Molecule Smoothened Modulators Discovered by High-Throughput Screening and Rational Design 1-gen-2014 Manetti, Fabrizio; Taddei, Maurizio; Petricci, Elena -
SYNTHESIS AND BIOLOGICAL EVALUATION OF SMALL MOLECULES DERIVATIVES OF THE NATURAL HISTONE DEACETYLASE INHIBITOR FR235222 1-gen-2014 Randino, Rosario; Cini, Elena; Anna Maria, D�Ursi; Petricci, Elena; Rodriquez, Manuela -
TRYPTOPHAN-BASED LINEAR DIPEPTIDESAND 1,4-DIKETOPIPERAZINES AS SIMPLIFIED SCAFFOLD OF THE NATURAL CYCLOTETRAPEPTIDE FR235222 1-gen-2014 Rodriquez, Manuela; Cini, Elena; Petricci, Elena; Anna Maria, D’Ursi; Carmela, Saturnino; Randino, Rosario -
Mostrati risultati da 41 a 60 di 96
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