Sfoglia per Autore
4-Hydroxyphenylpyruvate Dioxygenase and Its Inhibition in Plants and Animals: Small Molecules as Herbicides and Agents for the Treatment of Human Inherited Diseases
2017-01-01 Santucci, Annalisa; Bernardini, Giulia; Braconi, Daniela; Petricci, Elena; Manetti, Fabrizio
Gli1 inhibitors and uses thereof
2017-01-01 Giannini, Giuseppe; Taddei, Maurizio; Manetti, Fabrizio; Petricci, Elena; Stecca, Barbara
Synthesis and SAR evaluation of novel thioridazine derivatives active against drug-resistant tuberculosis
2017-01-01 Scalacci, Nicolò; Brown, Alistair K.; Pavan, Fernando R.; Ribeiro, Camila M.; Manetti, Fabrizio; Bhakta, Sanjib; Maitra, Arundhati; Smith, Darren L.; Petricci, Elena; Castagnolo, Daniele
Smoothened-antagonists reverse homogentisic acid-induced alterations of Hedgehog signaling and primary cilium length in alkaptonuria
2017-01-01 Gambassi, Silvia; Geminiani, Michela; Thorpe, Stephen D.; Bernardini, Giulia; Millucci, Lia; Braconi, Daniela; Orlandini, Maurizio; Thompson, Clare L.; Petricci, Elena; Manetti, Fabrizio; Taddei, Maurizio; Knight, Martin M.; Santucci, Annalisa
Design and synthesis of 1-((1,5-bis(4-chlorophenyl)-2-methyl-1H-pyrrol-3-yl)methyl)-4-methylpiperazine (BM212) and N-Adamantan-2-yl-N'-((E)-3,7-dimethyl-octa-2,6-dienyl)-ethane-1,2-diamine (SQ109) pyrrole hybrid derivatives: discovery of potent anti-tubercular agents effective against multi-drug resistant mycobacteria
2016-01-01 Sanjib, Bhakta; Nicolò, Scalacci; Arundhati, Maitra; Alistair K., Brown; Saiprasad, Dasugari; Dimitrios, Evangelopoulos; Timothy D., Mchugh; Parisa N., Mortazavi; Alexander, Twist; Petricci, Elena; Manetti, Fabrizio; Daniele, Castagnolo
Ruthenium-catalysed C-alkylation of 1,3-dicarbonyl compounds with primary alcohols and synthesis of 3-keto-quinolines
2016-01-01 Cini, Elena; Petricci, Elena; Truglio, GIUSEPPINA IVANA; Vecchio, Marialaura; Taddei, Maurizio
Microwave Assisted Hydrogenation of Pyridinecarboxylates: a Convenient Access to Valuable Scaffolds for Diversity Oriented Synthesis
2016-01-01 Ferrini, Serena; Cini, Elena; Petricci, Elena; Taddei, Maurizio
Design, synthesis and biological characterization of a new class of osteogenic (1H)-quinolone derivatives
2016-01-01 Manetti, Fabrizio; Petricci, Elena; Gabrielli, Annalisa; Mann, Andrè; Faure, Hélène; Gorojankina, Tatiana; Brasseur, Laurent; Hoch, Lucile; Ruat, Martial; Taddei, Maurizio
Novel acylguanidine derivatives targeting smoothened induce antiproliferative and pro-apoptotic effects in chronic myeloid leukemia cells
2016-01-01 Chiarenza, Alessandra; Manetti, Fabrizio; Petricci, Elena; Ruat, Martial; Naldini, Antonella; Taddei, Maurizio; Carraro, Fabio
Evaluation of WO2014207069 A1: Multitarget Hedgehog pathway inhibitors and uses thereof
2016-01-01 Manetti, Fabrizio; Petricci, Elena
Hedgehog associated to microparticles inhibits adipocyte differentiation via a non-canonical pathway
2016-01-01 Fleury, Audrey; Hoch, Lucile; Martinez, M. Carmen; Faure, Hélène; Taddei, Maurizio; Petricci, Elena; Manetti, Fabrizio; Girard, Nicolas; Mann, André; Jacques, Caroline; Larghero, Jérome; Ruat, Martial; Andriantsitohaina, Ramaroson; Le Lay, Soazig
Overcoming resistence to imatinib by targeting hedgehog signaling
2015-01-01 Chiarenza, Alessandra; Manetti, Fabrizio; Petricci, Elena; Taddei, Maurizio; Naldini, Antonella; Carraro, Fabio
Synthesis of 1,2,3-substituted pyrroles from propargylamines via a one-pot tandem enyne cross metathesis-cyclization reaction
2015-01-01 Chachignon, Helene; Scalacci, Nicolo; Petricci, Elena; Castagnolo, Daniele
MRT-92 inhibits Hedgehog signaling by blocking overlapping binding sites in the transmembrane domain of the Smoothened receptor
2015-01-01 Hoch, L; Faure, H; Roudaut, H; Schoenfelder, A; Mann, A; Girard, N; Bihannic, L; Ayrault, O; Petricci, Elena; Taddei, Maurizio; Rognan, D; Ruat, M. 2.
Targeting the Hedgehog Signaling Pathway with Small Molecules from Natural Sources
2015-01-01 Petricci, Elena; Manetti, Fabrizio
A highly stereo-controlled protocol to prepare pipecolic acids based on Heck and cyclohydrocarbonylation reactions
2015-01-01 Arena, Giada; Cini, Elena; Petricci, Elena; Randino, E.; Taddei, Maurizio
Domino Hydrogenation-Reductive Amination of Phenols, a Simple Process To Access Substituted Cyclohexylamines
2015-01-01 Jumde, VARSHA RAVINDRA; Petricci, Elena; Petrucci, C; Santillo, Niccolo'; Taddei, Maurizio; Vaccaro, L. 2.
Structure–Activity Relationships and Mechanism of Action of Small Molecule Smoothened Modulators Discovered by High-Throughput Screening and Rational Design
2014-01-01 Manetti, Fabrizio; Taddei, Maurizio; Petricci, Elena
SYNTHESIS AND BIOLOGICAL EVALUATION OF SMALL MOLECULES DERIVATIVES OF THE NATURAL HISTONE DEACETYLASE INHIBITOR FR235222
2014-01-01 Randino, Rosario; Cini, Elena; Anna Maria, D�Ursi; Petricci, Elena; Rodriquez, Manuela
TRYPTOPHAN-BASED LINEAR DIPEPTIDESAND 1,4-DIKETOPIPERAZINES AS SIMPLIFIED SCAFFOLD OF THE NATURAL CYCLOTETRAPEPTIDE FR235222
2014-01-01 Rodriquez, Manuela; Cini, Elena; Petricci, Elena; Anna Maria, D’Ursi; Carmela, Saturnino; Randino, Rosario
Titolo | Data di pubblicazione | Autore(i) | File | Abstract |
---|---|---|---|---|
4-Hydroxyphenylpyruvate Dioxygenase and Its Inhibition in Plants and Animals: Small Molecules as Herbicides and Agents for the Treatment of Human Inherited Diseases | 1-gen-2017 | Santucci, Annalisa; Bernardini, Giulia; Braconi, Daniela; Petricci, Elena; Manetti, Fabrizio | - | |
Gli1 inhibitors and uses thereof | 1-gen-2017 | Giannini, Giuseppe; Taddei, Maurizio; Manetti, Fabrizio; Petricci, Elena; Stecca, Barbara | - | |
Synthesis and SAR evaluation of novel thioridazine derivatives active against drug-resistant tuberculosis | 1-gen-2017 | Scalacci, Nicolò; Brown, Alistair K.; Pavan, Fernando R.; Ribeiro, Camila M.; Manetti, Fabrizio; Bhakta, Sanjib; Maitra, Arundhati; Smith, Darren L.; Petricci, Elena; Castagnolo, Daniele | - | |
Smoothened-antagonists reverse homogentisic acid-induced alterations of Hedgehog signaling and primary cilium length in alkaptonuria | 1-gen-2017 | Gambassi, Silvia; Geminiani, Michela; Thorpe, Stephen D.; Bernardini, Giulia; Millucci, Lia; Braconi, Daniela; Orlandini, Maurizio; Thompson, Clare L.; Petricci, Elena; Manetti, Fabrizio; Taddei, Maurizio; Knight, Martin M.; Santucci, Annalisa | - | |
Design and synthesis of 1-((1,5-bis(4-chlorophenyl)-2-methyl-1H-pyrrol-3-yl)methyl)-4-methylpiperazine (BM212) and N-Adamantan-2-yl-N'-((E)-3,7-dimethyl-octa-2,6-dienyl)-ethane-1,2-diamine (SQ109) pyrrole hybrid derivatives: discovery of potent anti-tubercular agents effective against multi-drug resistant mycobacteria | 1-gen-2016 | Sanjib, Bhakta; Nicolò, Scalacci; Arundhati, Maitra; Alistair K., Brown; Saiprasad, Dasugari; Dimitrios, Evangelopoulos; Timothy D., Mchugh; Parisa N., Mortazavi; Alexander, Twist; Petricci, Elena; Manetti, Fabrizio; Daniele, Castagnolo | - | |
Ruthenium-catalysed C-alkylation of 1,3-dicarbonyl compounds with primary alcohols and synthesis of 3-keto-quinolines | 1-gen-2016 | Cini, Elena; Petricci, Elena; Truglio, GIUSEPPINA IVANA; Vecchio, Marialaura; Taddei, Maurizio | - | |
Microwave Assisted Hydrogenation of Pyridinecarboxylates: a Convenient Access to Valuable Scaffolds for Diversity Oriented Synthesis | 1-gen-2016 | Ferrini, Serena; Cini, Elena; Petricci, Elena; Taddei, Maurizio | - | |
Design, synthesis and biological characterization of a new class of osteogenic (1H)-quinolone derivatives | 1-gen-2016 | Manetti, Fabrizio; Petricci, Elena; Gabrielli, Annalisa; Mann, Andrè; Faure, Hélène; Gorojankina, Tatiana; Brasseur, Laurent; Hoch, Lucile; Ruat, Martial; Taddei, Maurizio | - | |
Novel acylguanidine derivatives targeting smoothened induce antiproliferative and pro-apoptotic effects in chronic myeloid leukemia cells | 1-gen-2016 | Chiarenza, Alessandra; Manetti, Fabrizio; Petricci, Elena; Ruat, Martial; Naldini, Antonella; Taddei, Maurizio; Carraro, Fabio | - | |
Evaluation of WO2014207069 A1: Multitarget Hedgehog pathway inhibitors and uses thereof | 1-gen-2016 | Manetti, Fabrizio; Petricci, Elena | - | |
Hedgehog associated to microparticles inhibits adipocyte differentiation via a non-canonical pathway | 1-gen-2016 | Fleury, Audrey; Hoch, Lucile; Martinez, M. Carmen; Faure, Hélène; Taddei, Maurizio; Petricci, Elena; Manetti, Fabrizio; Girard, Nicolas; Mann, André; Jacques, Caroline; Larghero, Jérome; Ruat, Martial; Andriantsitohaina, Ramaroson; Le Lay, Soazig | - | |
Overcoming resistence to imatinib by targeting hedgehog signaling | 1-gen-2015 | Chiarenza, Alessandra; Manetti, Fabrizio; Petricci, Elena; Taddei, Maurizio; Naldini, Antonella; Carraro, Fabio | - | |
Synthesis of 1,2,3-substituted pyrroles from propargylamines via a one-pot tandem enyne cross metathesis-cyclization reaction | 1-gen-2015 | Chachignon, Helene; Scalacci, Nicolo; Petricci, Elena; Castagnolo, Daniele | - | |
MRT-92 inhibits Hedgehog signaling by blocking overlapping binding sites in the transmembrane domain of the Smoothened receptor | 1-gen-2015 | Hoch, L; Faure, H; Roudaut, H; Schoenfelder, A; Mann, A; Girard, N; Bihannic, L; Ayrault, O; Petricci, Elena; Taddei, Maurizio; Rognan, D; Ruat, M. 2. | - | |
Targeting the Hedgehog Signaling Pathway with Small Molecules from Natural Sources | 1-gen-2015 | Petricci, Elena; Manetti, Fabrizio | - | |
A highly stereo-controlled protocol to prepare pipecolic acids based on Heck and cyclohydrocarbonylation reactions | 1-gen-2015 | Arena, Giada; Cini, Elena; Petricci, Elena; Randino, E.; Taddei, Maurizio | - | |
Domino Hydrogenation-Reductive Amination of Phenols, a Simple Process To Access Substituted Cyclohexylamines | 1-gen-2015 | Jumde, VARSHA RAVINDRA; Petricci, Elena; Petrucci, C; Santillo, Niccolo'; Taddei, Maurizio; Vaccaro, L. 2. | - | |
Structure–Activity Relationships and Mechanism of Action of Small Molecule Smoothened Modulators Discovered by High-Throughput Screening and Rational Design | 1-gen-2014 | Manetti, Fabrizio; Taddei, Maurizio; Petricci, Elena | - | |
SYNTHESIS AND BIOLOGICAL EVALUATION OF SMALL MOLECULES DERIVATIVES OF THE NATURAL HISTONE DEACETYLASE INHIBITOR FR235222 | 1-gen-2014 | Randino, Rosario; Cini, Elena; Anna Maria, D�Ursi; Petricci, Elena; Rodriquez, Manuela | - | |
TRYPTOPHAN-BASED LINEAR DIPEPTIDESAND 1,4-DIKETOPIPERAZINES AS SIMPLIFIED SCAFFOLD OF THE NATURAL CYCLOTETRAPEPTIDE FR235222 | 1-gen-2014 | Rodriquez, Manuela; Cini, Elena; Petricci, Elena; Anna Maria, D’Ursi; Carmela, Saturnino; Randino, Rosario | - |
Legenda icone
- file ad accesso aperto
- file disponibili sulla rete interna
- file disponibili agli utenti autorizzati
- file disponibili solo agli amministratori
- file sotto embargo
- nessun file disponibile