Sfoglia per Autore
Antibody drug conjugates (ADCs) charged with HDAC inhibitor for targeted epigenetic modulation
2018-01-01 Cini, Elena; Faltoni, Valentina; Petricci, Elena; Taddei, Maurizio; Salvini, Laura; Giannini, Giuseppe; Vesci, Loredana; Milazzo, Ferdinando Maria; Anastasi, Anna Maria; Battistuzzi, Gianfranco; De Santis, Rita
Continuous-Flow Palladium-Catalyzed Synthesis of Cyclohexanones from Phenols using Sodium Formate as a Safe Hydrogen Source
2018-01-01 Valentini, Federica; Santillo, Niccolò; Petrucci, Chiara; Lanari, Daniela; Petricci, Elena; Taddei, Maurizio; Vaccaro, Luigi
Stereoselective Synthesis of Sofosbuvir through Nucleoside Phosphorylation Controlled by Kinetic Resolution
2018-01-01 Cini, Elena; Barreca, Giuseppe; Carcone, Luca; Manetti, Fabrizio; Rasparini, Marcello; Taddei, Maurizio
Iron-Catalyzed Reductive Amination of Aldehydes in Isopropyl Alcohol/Water Media as Hydrogen Sources
2018-01-01 Petricci, Elena; Santillo, Niccolò; Castagnolo, Daniele; Cini, Elena; Taddei, Maurizio
N-ACYLTHIOUREA AND N-ACYLUREA INHIBITORS OF THE HEDGEHOG PROTEIN SIGNALLING PATHWAY
2017-01-01 Martial, Ruat; Hélène, Faure; Elisabeth, Traiffort; Angèle, Schoenfelder; André, Mann; Taddei, Maurizio; Antonio, Solinas; Manetti, Fabrizio
Histone Deacetylase Inhibitors-based antibody drug conjugates (ADCs) and use in therapy
2017-01-01 Vesci, Loredana; De Santis, Rita; Maria Milazzo, Ferdinando; Giannini, Giuseppe; Taddei, Maurizio; Faltoni, Valentina; Petricci, Elena
Gli1 inhibitors and uses thereof
2017-01-01 Giannini, Giuseppe; Taddei, Maurizio; Manetti, Fabrizio; Petricci, Elena; Stecca, Barbara
Synthesis of small molecules active on tumor relevant cellular signaling pathways
2017-01-01 Gabrielli, Annalisa; Taddei, Maurizio
Pd/C catalysis under microwave dielectric heating
2017-01-01 Cini, Elena; Petricci, Elena; Taddei, Maurizio
Smoothened-antagonists reverse homogentisic acid-induced alterations of Hedgehog signaling and primary cilium length in alkaptonuria
2017-01-01 Gambassi, Silvia; Geminiani, Michela; Thorpe, Stephen D.; Bernardini, Giulia; Millucci, Lia; Braconi, Daniela; Orlandini, Maurizio; Thompson, Clare L.; Petricci, Elena; Manetti, Fabrizio; Taddei, Maurizio; Knight, Martin M.; Santucci, Annalisa
Benzodiazepine scaffold as drug-like molecular simplification of FR235222: A chemical tool for exploring HDAC inhibition
2017-01-01 Randino, Rosario; Moronese, Ilaria; Cini, Elena; Bizzarro, Valentina; Persico, Marco; Grimaldi, Manuela; Scrima, Mario; D’Ursi, Anna Maria; Novellino, Ettore; Sobarzo Sánchez, Eduardo; Rastrelli, Luca; Fattorusso, Caterina; Petrella, Antonello; Rodriquez, Manuela; Taddei, Maurizio
Nucleoside phosphoramidates useful for the treatment of viral infections and preparation thereof
2016-01-01 Barreca, Giuseppe; Rasparini, Marcello; Poggiali, Andrea; Carcone, Luca; Tufaro, Roberto Rocco; Marras, Giovanni; Taddei, Maurizio; Cini, Elena
Acyl guanidine derivatives modulating the hedgehog protein signaling pathway
2016-01-01 Martial, Ruat; Hélène, Faure; Elisabeth, Traiffort; Hermine, Roudaut; André, Mann; Angèle, Schoenfelder; Taddei, Maurizio; Manetti, Fabrizio; Antonio, Solinas
N-Acylthiourees et N-acylurees inhibiteurs de la voie de signalisation des proteines Hedgehog
2016-01-01 Martial, Ruat; Hélène, Faure; Elisabeth, Traiffort; Angèle, Schoenfelder; André, Mann; Taddei, Maurizio; Antonio, Solinas; Manetti, Fabrizio
Novel acylguanidine derivatives targeting smoothened induce antiproliferative and pro-apoptotic effects in chronic myeloid leukemia cells
2016-01-01 Chiarenza, Alessandra; Manetti, Fabrizio; Petricci, Elena; Ruat, Martial; Naldini, Antonella; Taddei, Maurizio; Carraro, Fabio
Microwave Assisted Hydrogenation of Pyridinecarboxylates: a Convenient Access to Valuable Scaffolds for Diversity Oriented Synthesis
2016-01-01 Ferrini, Serena; Cini, Elena; Petricci, Elena; Taddei, Maurizio
Convergent Synthesis of the Renin Inhibitor Aliskiren Based on C5–C6 Disconnection and CO2H–NH2Equivalence
2016-01-01 Cini, Elena; Banfi, Luca; Barreca, Giuseppe; Carcone, Luca; Malpezzi, Luciana; Manetti, Fabrizio; Marras, Giovanni; Rasparini, Marcello; Riva, Renata; Roseblade, Stephen; Russo, Adele; Taddei, Maurizio; Vitale, Romina; Zanotti Gerosa, Antonio
Ruthenium-catalysed C-alkylation of 1,3-dicarbonyl compounds with primary alcohols and synthesis of 3-keto-quinolines
2016-01-01 Cini, Elena; Petricci, Elena; Truglio, GIUSEPPINA IVANA; Vecchio, Marialaura; Taddei, Maurizio
Design, synthesis and biological characterization of a new class of osteogenic (1H)-quinolone derivatives
2016-01-01 Manetti, Fabrizio; Petricci, Elena; Gabrielli, Annalisa; Mann, Andrè; Faure, Hélène; Gorojankina, Tatiana; Brasseur, Laurent; Hoch, Lucile; Ruat, Martial; Taddei, Maurizio
Hedgehog associated to microparticles inhibits adipocyte differentiation via a non-canonical pathway
2016-01-01 Fleury, Audrey; Hoch, Lucile; Martinez, M. Carmen; Faure, Hélène; Taddei, Maurizio; Petricci, Elena; Manetti, Fabrizio; Girard, Nicolas; Mann, André; Jacques, Caroline; Larghero, Jérome; Ruat, Martial; Andriantsitohaina, Ramaroson; Le Lay, Soazig
Titolo | Data di pubblicazione | Autore(i) | File | Abstract |
---|---|---|---|---|
Antibody drug conjugates (ADCs) charged with HDAC inhibitor for targeted epigenetic modulation | 1-gen-2018 | Cini, Elena; Faltoni, Valentina; Petricci, Elena; Taddei, Maurizio; Salvini, Laura; Giannini, Giuseppe; Vesci, Loredana; Milazzo, Ferdinando Maria; Anastasi, Anna Maria; Battistuzzi, Gianfranco; De Santis, Rita | - | |
Continuous-Flow Palladium-Catalyzed Synthesis of Cyclohexanones from Phenols using Sodium Formate as a Safe Hydrogen Source | 1-gen-2018 | Valentini, Federica; Santillo, Niccolò; Petrucci, Chiara; Lanari, Daniela; Petricci, Elena; Taddei, Maurizio; Vaccaro, Luigi | - | |
Stereoselective Synthesis of Sofosbuvir through Nucleoside Phosphorylation Controlled by Kinetic Resolution | 1-gen-2018 | Cini, Elena; Barreca, Giuseppe; Carcone, Luca; Manetti, Fabrizio; Rasparini, Marcello; Taddei, Maurizio | - | |
Iron-Catalyzed Reductive Amination of Aldehydes in Isopropyl Alcohol/Water Media as Hydrogen Sources | 1-gen-2018 | Petricci, Elena; Santillo, Niccolò; Castagnolo, Daniele; Cini, Elena; Taddei, Maurizio | - | |
N-ACYLTHIOUREA AND N-ACYLUREA INHIBITORS OF THE HEDGEHOG PROTEIN SIGNALLING PATHWAY | 1-gen-2017 | Martial, Ruat; Hélène, Faure; Elisabeth, Traiffort; Angèle, Schoenfelder; André, Mann; Taddei, Maurizio; Antonio, Solinas; Manetti, Fabrizio | - | |
Histone Deacetylase Inhibitors-based antibody drug conjugates (ADCs) and use in therapy | 1-gen-2017 | Vesci, Loredana; De Santis, Rita; Maria Milazzo, Ferdinando; Giannini, Giuseppe; Taddei, Maurizio; Faltoni, Valentina; Petricci, Elena | - | |
Gli1 inhibitors and uses thereof | 1-gen-2017 | Giannini, Giuseppe; Taddei, Maurizio; Manetti, Fabrizio; Petricci, Elena; Stecca, Barbara | - | |
Synthesis of small molecules active on tumor relevant cellular signaling pathways | 1-gen-2017 | Gabrielli, Annalisa; Taddei, Maurizio | - | |
Pd/C catalysis under microwave dielectric heating | 1-gen-2017 | Cini, Elena; Petricci, Elena; Taddei, Maurizio | - | |
Smoothened-antagonists reverse homogentisic acid-induced alterations of Hedgehog signaling and primary cilium length in alkaptonuria | 1-gen-2017 | Gambassi, Silvia; Geminiani, Michela; Thorpe, Stephen D.; Bernardini, Giulia; Millucci, Lia; Braconi, Daniela; Orlandini, Maurizio; Thompson, Clare L.; Petricci, Elena; Manetti, Fabrizio; Taddei, Maurizio; Knight, Martin M.; Santucci, Annalisa | - | |
Benzodiazepine scaffold as drug-like molecular simplification of FR235222: A chemical tool for exploring HDAC inhibition | 1-gen-2017 | Randino, Rosario; Moronese, Ilaria; Cini, Elena; Bizzarro, Valentina; Persico, Marco; Grimaldi, Manuela; Scrima, Mario; D’Ursi, Anna Maria; Novellino, Ettore; Sobarzo Sánchez, Eduardo; Rastrelli, Luca; Fattorusso, Caterina; Petrella, Antonello; Rodriquez, Manuela; Taddei, Maurizio | - | |
Nucleoside phosphoramidates useful for the treatment of viral infections and preparation thereof | 1-gen-2016 | Barreca, Giuseppe; Rasparini, Marcello; Poggiali, Andrea; Carcone, Luca; Tufaro, Roberto Rocco; Marras, Giovanni; Taddei, Maurizio; Cini, Elena | - | |
Acyl guanidine derivatives modulating the hedgehog protein signaling pathway | 1-gen-2016 | Martial, Ruat; Hélène, Faure; Elisabeth, Traiffort; Hermine, Roudaut; André, Mann; Angèle, Schoenfelder; Taddei, Maurizio; Manetti, Fabrizio; Antonio, Solinas | - | |
N-Acylthiourees et N-acylurees inhibiteurs de la voie de signalisation des proteines Hedgehog | 1-gen-2016 | Martial, Ruat; Hélène, Faure; Elisabeth, Traiffort; Angèle, Schoenfelder; André, Mann; Taddei, Maurizio; Antonio, Solinas; Manetti, Fabrizio | - | |
Novel acylguanidine derivatives targeting smoothened induce antiproliferative and pro-apoptotic effects in chronic myeloid leukemia cells | 1-gen-2016 | Chiarenza, Alessandra; Manetti, Fabrizio; Petricci, Elena; Ruat, Martial; Naldini, Antonella; Taddei, Maurizio; Carraro, Fabio | - | |
Microwave Assisted Hydrogenation of Pyridinecarboxylates: a Convenient Access to Valuable Scaffolds for Diversity Oriented Synthesis | 1-gen-2016 | Ferrini, Serena; Cini, Elena; Petricci, Elena; Taddei, Maurizio | - | |
Convergent Synthesis of the Renin Inhibitor Aliskiren Based on C5–C6 Disconnection and CO2H–NH2Equivalence | 1-gen-2016 | Cini, Elena; Banfi, Luca; Barreca, Giuseppe; Carcone, Luca; Malpezzi, Luciana; Manetti, Fabrizio; Marras, Giovanni; Rasparini, Marcello; Riva, Renata; Roseblade, Stephen; Russo, Adele; Taddei, Maurizio; Vitale, Romina; Zanotti Gerosa, Antonio | - | |
Ruthenium-catalysed C-alkylation of 1,3-dicarbonyl compounds with primary alcohols and synthesis of 3-keto-quinolines | 1-gen-2016 | Cini, Elena; Petricci, Elena; Truglio, GIUSEPPINA IVANA; Vecchio, Marialaura; Taddei, Maurizio | - | |
Design, synthesis and biological characterization of a new class of osteogenic (1H)-quinolone derivatives | 1-gen-2016 | Manetti, Fabrizio; Petricci, Elena; Gabrielli, Annalisa; Mann, Andrè; Faure, Hélène; Gorojankina, Tatiana; Brasseur, Laurent; Hoch, Lucile; Ruat, Martial; Taddei, Maurizio | - | |
Hedgehog associated to microparticles inhibits adipocyte differentiation via a non-canonical pathway | 1-gen-2016 | Fleury, Audrey; Hoch, Lucile; Martinez, M. Carmen; Faure, Hélène; Taddei, Maurizio; Petricci, Elena; Manetti, Fabrizio; Girard, Nicolas; Mann, André; Jacques, Caroline; Larghero, Jérome; Ruat, Martial; Andriantsitohaina, Ramaroson; Le Lay, Soazig | - |
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