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Titolo Data di pubblicazione Autore(i) File Abstract
Antibody drug conjugates (ADCs) charged with HDAC inhibitor for targeted epigenetic modulation 1-gen-2018 Cini, Elena; Faltoni, Valentina; Petricci, Elena; Taddei, Maurizio; Salvini, Laura; Giannini, Giuseppe; Vesci, Loredana; Milazzo, Ferdinando Maria; Anastasi, Anna Maria; Battistuzzi, Gianfranco; De Santis, Rita -
Continuous-Flow Palladium-Catalyzed Synthesis of Cyclohexanones from Phenols using Sodium Formate as a Safe Hydrogen Source 1-gen-2018 Valentini, Federica; Santillo, Niccolò; Petrucci, Chiara; Lanari, Daniela; Petricci, Elena; Taddei, Maurizio; Vaccaro, Luigi -
Stereoselective Synthesis of Sofosbuvir through Nucleoside Phosphorylation Controlled by Kinetic Resolution 1-gen-2018 Cini, Elena; Barreca, Giuseppe; Carcone, Luca; Manetti, Fabrizio; Rasparini, Marcello; Taddei, Maurizio -
Iron-Catalyzed Reductive Amination of Aldehydes in Isopropyl Alcohol/Water Media as Hydrogen Sources 1-gen-2018 Petricci, Elena; Santillo, Niccolò; Castagnolo, Daniele; Cini, Elena; Taddei, Maurizio -
N-ACYLTHIOUREA AND N-ACYLUREA INHIBITORS OF THE HEDGEHOG PROTEIN SIGNALLING PATHWAY 1-gen-2017 Martial, Ruat; Hélène, Faure; Elisabeth, Traiffort; Angèle, Schoenfelder; André, Mann; Taddei, Maurizio; Antonio, Solinas; Manetti, Fabrizio -
Histone Deacetylase Inhibitors-based antibody drug conjugates (ADCs) and use in therapy 1-gen-2017 Vesci, Loredana; De Santis, Rita; Maria Milazzo, Ferdinando; Giannini, Giuseppe; Taddei, Maurizio; Faltoni, Valentina; Petricci, Elena -
Gli1 inhibitors and uses thereof 1-gen-2017 Giannini, Giuseppe; Taddei, Maurizio; Manetti, Fabrizio; Petricci, Elena; Stecca, Barbara -
Synthesis of small molecules active on tumor relevant cellular signaling pathways 1-gen-2017 Gabrielli, Annalisa; Taddei, Maurizio -
Pd/C catalysis under microwave dielectric heating 1-gen-2017 Cini, Elena; Petricci, Elena; Taddei, Maurizio -
Smoothened-antagonists reverse homogentisic acid-induced alterations of Hedgehog signaling and primary cilium length in alkaptonuria 1-gen-2017 Gambassi, Silvia; Geminiani, Michela; Thorpe, Stephen D.; Bernardini, Giulia; Millucci, Lia; Braconi, Daniela; Orlandini, Maurizio; Thompson, Clare L.; Petricci, Elena; Manetti, Fabrizio; Taddei, Maurizio; Knight, Martin M.; Santucci, Annalisa -
Benzodiazepine scaffold as drug-like molecular simplification of FR235222: A chemical tool for exploring HDAC inhibition 1-gen-2017 Randino, Rosario; Moronese, Ilaria; Cini, Elena; Bizzarro, Valentina; Persico, Marco; Grimaldi, Manuela; Scrima, Mario; D’Ursi, Anna Maria; Novellino, Ettore; Sobarzo Sánchez, Eduardo; Rastrelli, Luca; Fattorusso, Caterina; Petrella, Antonello; Rodriquez, Manuela; Taddei, Maurizio -
Nucleoside phosphoramidates useful for the treatment of viral infections and preparation thereof 1-gen-2016 Barreca, Giuseppe; Rasparini, Marcello; Poggiali, Andrea; Carcone, Luca; Tufaro, Roberto Rocco; Marras, Giovanni; Taddei, Maurizio; Cini, Elena -
Acyl guanidine derivatives modulating the hedgehog protein signaling pathway 1-gen-2016 Martial, Ruat; Hélène, Faure; Elisabeth, Traiffort; Hermine, Roudaut; André, Mann; Angèle, Schoenfelder; Taddei, Maurizio; Manetti, Fabrizio; Antonio, Solinas -
N-Acylthiourees et N-acylurees inhibiteurs de la voie de signalisation des proteines Hedgehog 1-gen-2016 Martial, Ruat; Hélène, Faure; Elisabeth, Traiffort; Angèle, Schoenfelder; André, Mann; Taddei, Maurizio; Antonio, Solinas; Manetti, Fabrizio -
Novel acylguanidine derivatives targeting smoothened induce antiproliferative and pro-apoptotic effects in chronic myeloid leukemia cells 1-gen-2016 Chiarenza, Alessandra; Manetti, Fabrizio; Petricci, Elena; Ruat, Martial; Naldini, Antonella; Taddei, Maurizio; Carraro, Fabio -
Microwave Assisted Hydrogenation of Pyridinecarboxylates: a Convenient Access to Valuable Scaffolds for Diversity Oriented Synthesis 1-gen-2016 Ferrini, Serena; Cini, Elena; Petricci, Elena; Taddei, Maurizio -
Convergent Synthesis of the Renin Inhibitor Aliskiren Based on C5–C6 Disconnection and CO2H–NH2Equivalence 1-gen-2016 Cini, Elena; Banfi, Luca; Barreca, Giuseppe; Carcone, Luca; Malpezzi, Luciana; Manetti, Fabrizio; Marras, Giovanni; Rasparini, Marcello; Riva, Renata; Roseblade, Stephen; Russo, Adele; Taddei, Maurizio; Vitale, Romina; Zanotti Gerosa, Antonio -
Ruthenium-catalysed C-alkylation of 1,3-dicarbonyl compounds with primary alcohols and synthesis of 3-keto-quinolines 1-gen-2016 Cini, Elena; Petricci, Elena; Truglio, GIUSEPPINA IVANA; Vecchio, Marialaura; Taddei, Maurizio -
Design, synthesis and biological characterization of a new class of osteogenic (1H)-quinolone derivatives 1-gen-2016 Manetti, Fabrizio; Petricci, Elena; Gabrielli, Annalisa; Mann, Andrè; Faure, Hélène; Gorojankina, Tatiana; Brasseur, Laurent; Hoch, Lucile; Ruat, Martial; Taddei, Maurizio -
Hedgehog associated to microparticles inhibits adipocyte differentiation via a non-canonical pathway 1-gen-2016 Fleury, Audrey; Hoch, Lucile; Martinez, M. Carmen; Faure, Hélène; Taddei, Maurizio; Petricci, Elena; Manetti, Fabrizio; Girard, Nicolas; Mann, André; Jacques, Caroline; Larghero, Jérome; Ruat, Martial; Andriantsitohaina, Ramaroson; Le Lay, Soazig -
Mostrati risultati da 21 a 40 di 278
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