Sfoglia per Autore
Consensus screening for a challenging target: the quest for P-glycoprotein inhibitors
2024-01-01 Governa, Paolo; Biagi, Marco; Manetti, Fabrizio; Forli, Stefano
Enhanced mapping of small-molecule binding sites in cells
2024-01-01 Wozniak, Jacob M; Li, Weichao; Governa, Paolo; Chen, Li-Yun; Jadhav, Appaso; Dongre, Ashok; Forli, Stefano; Parker, Christopher G
Helichrysum stoechas (L.) Moench reduces body weight gain and modulates mood disorders via inhibition of silent information regulator 1 (SIRT1) by arzanol
2023-01-01 Borgonetti, Vittoria; Caroli, Clarissa; Governa, Paolo; Virginia, Brighenti; Pollastro, Federica; Franchini, Silvia; Manetti, Fabrizio; Les, Francisco; López, Victor; Pellati, Federica; Galeotti, Nicoletta
Zingiberene, a non-zinc-binding class I HDAC inhibitor: A novel strategy for the management of neuropathic pain
2023-01-01 Borgonetti, Vittoria; Governa, Paolo; Manetti, Fabrizio; Galeotti, Nicoletta
A Novel Perilla frutescens (L.) Britton Cell-Derived Phytocomplex Regulates Keratinocytes Inflammatory Cascade and Barrier Function and Preserves Vaginal Mucosal Integrity In Vivo
2023-01-01 Pressi, Giovanna; Rigillo, Giovanna; Governa, Paolo; Borgonetti, Vittoria; Baini, Giulia; Rizzi, Raffaella; Guarnerio, Chiara; Bertaiola, Oriana; Frigo, Marco; Merlin, Matilde; Paltrinieri, Stefania; Zambonin, Roberto; Pandolfo, Stefano; Biagi, Marco
Effect of in vitro simulated digestion on the anti-Helicobacter Pylori activity of different Propolis extracts
2023-01-01 Governa, Paolo; Romagnoli, Giulia; Albanese, Paola; Rossi, Federico; Manetti, Fabrizio; Biagi, Marco
Cannabidiol-rich non-psychotropic Cannabis sativa L. oils attenuate peripheral neuropathy symptoms by regulation of CB2-mediated microglial neuroinflammation
2023-01-01 Borgonetti, Vittoria; Anceschi, Lisa; Brighenti, Virginia; Corsi, Lorenzo; Governa, Paolo; Manetti, Fabrizio; Pellati, Federica; Galeotti, Nicoletta
Antiviral Activity of Cannabidiolic Acid and Its Methyl Ester against SARS-CoV-2
2023-01-01 Tamburello, Martina; Salamone, Stefano; Anceschi, Lisa; Governa, Paolo; Brighenti, Virginia; Morellini, Alice; Rossini, Giada; Manetti, Fabrizio; Gallinella, Giorgio; Pollastro, Federica; Pellati, Federica
In Vitro Cell Culture of Rhus coriaria L.: A Standardized Phytocomplex Rich of Gallic Acid Derivatives with Antioxidant and Skin Repair Activity
2022-01-01 Pressi, G.; Bertaiola, O.; Guarnerio, C.; Barbieri, E.; Rigillo, G.; Governa, P.; Biagi, M.; Guzzo, F.; Semenzato, A.
Quinolines and Oxazino-quinoline Derivatives as Small Molecule GLI1 Inhibitors Identified by Virtual Screening
2022-01-01 Manetti, Fabrizio; Maresca, Luisa; Crivaro, Enrica; Pepe, Sara; Cini, Elena; Singh, Snigdha; Governa, Paolo; Maramai, Samuele; Giannini, Giuseppe; Stecca, Barbara; Petricci, Elena
Recent research results have converted gp120 binders to a therapeutic option for the treatment of HIV-1 infection. A medicinal chemistry point of view
2022-01-01 Governa, Paolo; Manetti, Fabrizio
Investigation on the neuroprotective effect of a cannabidiol-enriched non-psychotropic Cannabis sativa L. extract in an in vitro model of excitotoxicity
2022-01-01 Borgonetti, Vittoria; Biagi, Marco; Galeotti, Nicoletta; Manetti, Fabrizio; Governa, Paolo
Non-psychotropic Cannabis sativa L. phytocomplex modulates microglial inflammatory response through CB2 receptors-, endocannabinoids-, and NF-κB-mediated signaling
2022-01-01 Borgonetti, V.; Benatti, C.; Governa, P.; Isoldi, G.; Pellati, F.; Alboni, S.; Tascedda, F.; Montopoli, M.; Galeotti, N.; Manetti, F.; Miraldi, E.; Biagi, M.; Rigillo, G.
The Veterinary Anti-Parasitic Selamectin Is a Novel Inhibitor of the Mycobacterium tuberculosis DprE1 Enzyme
2022-01-01 Ezquerra-Aznárez, José Manuel; Degiacomi, Giulia; Gašparovič, Henrich; Stelitano, Giovanni; Sammartino, Josè Camilla; Korduláková, Jana; Governa, Paolo; Manetti, Fabrizio; Pasca, Maria Rosalia; Chiarelli, Laurent Roberto; Ramón-García, Santiago
Survey on the Recent Advances in 4-Hydroxyphenylpyruvate Dioxygenase (HPPD) Inhibition by Diketone and Triketone Derivatives and Congeneric Compounds: Structural Analysis of HPPD/Inhibitor Complexes and Structure-Activity Relationship Considerations
2022-01-01 Governa, Paolo; Bernardini, Giulia; Braconi, Daniela; Manetti, Fabrizio; Santucci, Annalisa; Petricci, Elena
Effects of in vitro simulated digestion on the antioxidant activity of different Camellia sinensis (L.) Kuntze leaves extracts
2022-01-01 Governa, Paolo; Manetti, Fabrizio; Miraldi, Elisabetta; Biagi, Marco
Identification and development of active principles from plant sources
2021-01-01 Governa, Paolo
FFAR1/GPR40: One target, different binding sites, many agonists, no drugs, but a continuous and unprofitable tug-of-war between ligand lipophilicity, activity, and toxicity
2021-01-01 Governa, Paolo; Caroleo, Maria Cristina; Carullo, Gabriele; Aiello, Francesca; Cione, Erika; Manetti, Fabrizio
Pinocembrin and its linolenoyl ester derivative induce wound healing activity in HaCaT cell line potentially involving a GPR120/FFA4 mediated pathway
2021-01-01 Mazzotta, Sarah; Governa, Paolo; Borgonetti, Vittoria; Marcolongo, Paola; Nanni, Claudio; Gamberucci, Alessandra; Manetti, Fabrizio; Pessina, Federica; Carullo, Gabriele; Brizzi, Antonella; Aiello, Francesca
Cannabidiol Isolated From Cannabis sativa L. Protects Intestinal Barrier From In Vitro Inflammation and Oxidative Stress
2021-01-01 Cocetta, Veronica; Governa, Paolo; Borgonetti, Vittoria; Tinazzi, Mattia; Peron, Gregorio; Catanzaro, Daniela; Berretta, Massimiliano; Biagi, Marco; Manetti, Fabrizio; Dall'Acqua, Stefano; Montopoli, Monica
Titolo | Data di pubblicazione | Autore(i) | File | Abstract |
---|---|---|---|---|
Consensus screening for a challenging target: the quest for P-glycoprotein inhibitors | 1-gen-2024 | Governa, Paolo; Biagi, Marco; Manetti, Fabrizio; Forli, Stefano | - | |
Enhanced mapping of small-molecule binding sites in cells | 1-gen-2024 | Wozniak, Jacob M; Li, Weichao; Governa, Paolo; Chen, Li-Yun; Jadhav, Appaso; Dongre, Ashok; Forli, Stefano; Parker, Christopher G | - | |
Helichrysum stoechas (L.) Moench reduces body weight gain and modulates mood disorders via inhibition of silent information regulator 1 (SIRT1) by arzanol | 1-gen-2023 | Borgonetti, Vittoria; Caroli, Clarissa; Governa, Paolo; Virginia, Brighenti; Pollastro, Federica; Franchini, Silvia; Manetti, Fabrizio; Les, Francisco; López, Victor; Pellati, Federica; Galeotti, Nicoletta | - | |
Zingiberene, a non-zinc-binding class I HDAC inhibitor: A novel strategy for the management of neuropathic pain | 1-gen-2023 | Borgonetti, Vittoria; Governa, Paolo; Manetti, Fabrizio; Galeotti, Nicoletta | - | |
A Novel Perilla frutescens (L.) Britton Cell-Derived Phytocomplex Regulates Keratinocytes Inflammatory Cascade and Barrier Function and Preserves Vaginal Mucosal Integrity In Vivo | 1-gen-2023 | Pressi, Giovanna; Rigillo, Giovanna; Governa, Paolo; Borgonetti, Vittoria; Baini, Giulia; Rizzi, Raffaella; Guarnerio, Chiara; Bertaiola, Oriana; Frigo, Marco; Merlin, Matilde; Paltrinieri, Stefania; Zambonin, Roberto; Pandolfo, Stefano; Biagi, Marco | - | |
Effect of in vitro simulated digestion on the anti-Helicobacter Pylori activity of different Propolis extracts | 1-gen-2023 | Governa, Paolo; Romagnoli, Giulia; Albanese, Paola; Rossi, Federico; Manetti, Fabrizio; Biagi, Marco | - | |
Cannabidiol-rich non-psychotropic Cannabis sativa L. oils attenuate peripheral neuropathy symptoms by regulation of CB2-mediated microglial neuroinflammation | 1-gen-2023 | Borgonetti, Vittoria; Anceschi, Lisa; Brighenti, Virginia; Corsi, Lorenzo; Governa, Paolo; Manetti, Fabrizio; Pellati, Federica; Galeotti, Nicoletta | - | |
Antiviral Activity of Cannabidiolic Acid and Its Methyl Ester against SARS-CoV-2 | 1-gen-2023 | Tamburello, Martina; Salamone, Stefano; Anceschi, Lisa; Governa, Paolo; Brighenti, Virginia; Morellini, Alice; Rossini, Giada; Manetti, Fabrizio; Gallinella, Giorgio; Pollastro, Federica; Pellati, Federica | - | |
In Vitro Cell Culture of Rhus coriaria L.: A Standardized Phytocomplex Rich of Gallic Acid Derivatives with Antioxidant and Skin Repair Activity | 1-gen-2022 | Pressi, G.; Bertaiola, O.; Guarnerio, C.; Barbieri, E.; Rigillo, G.; Governa, P.; Biagi, M.; Guzzo, F.; Semenzato, A. | - | |
Quinolines and Oxazino-quinoline Derivatives as Small Molecule GLI1 Inhibitors Identified by Virtual Screening | 1-gen-2022 | Manetti, Fabrizio; Maresca, Luisa; Crivaro, Enrica; Pepe, Sara; Cini, Elena; Singh, Snigdha; Governa, Paolo; Maramai, Samuele; Giannini, Giuseppe; Stecca, Barbara; Petricci, Elena | - | |
Recent research results have converted gp120 binders to a therapeutic option for the treatment of HIV-1 infection. A medicinal chemistry point of view | 1-gen-2022 | Governa, Paolo; Manetti, Fabrizio | - | |
Investigation on the neuroprotective effect of a cannabidiol-enriched non-psychotropic Cannabis sativa L. extract in an in vitro model of excitotoxicity | 1-gen-2022 | Borgonetti, Vittoria; Biagi, Marco; Galeotti, Nicoletta; Manetti, Fabrizio; Governa, Paolo | - | |
Non-psychotropic Cannabis sativa L. phytocomplex modulates microglial inflammatory response through CB2 receptors-, endocannabinoids-, and NF-κB-mediated signaling | 1-gen-2022 | Borgonetti, V.; Benatti, C.; Governa, P.; Isoldi, G.; Pellati, F.; Alboni, S.; Tascedda, F.; Montopoli, M.; Galeotti, N.; Manetti, F.; Miraldi, E.; Biagi, M.; Rigillo, G. | - | |
The Veterinary Anti-Parasitic Selamectin Is a Novel Inhibitor of the Mycobacterium tuberculosis DprE1 Enzyme | 1-gen-2022 | Ezquerra-Aznárez, José Manuel; Degiacomi, Giulia; Gašparovič, Henrich; Stelitano, Giovanni; Sammartino, Josè Camilla; Korduláková, Jana; Governa, Paolo; Manetti, Fabrizio; Pasca, Maria Rosalia; Chiarelli, Laurent Roberto; Ramón-García, Santiago | - | |
Survey on the Recent Advances in 4-Hydroxyphenylpyruvate Dioxygenase (HPPD) Inhibition by Diketone and Triketone Derivatives and Congeneric Compounds: Structural Analysis of HPPD/Inhibitor Complexes and Structure-Activity Relationship Considerations | 1-gen-2022 | Governa, Paolo; Bernardini, Giulia; Braconi, Daniela; Manetti, Fabrizio; Santucci, Annalisa; Petricci, Elena | - | |
Effects of in vitro simulated digestion on the antioxidant activity of different Camellia sinensis (L.) Kuntze leaves extracts | 1-gen-2022 | Governa, Paolo; Manetti, Fabrizio; Miraldi, Elisabetta; Biagi, Marco | - | |
Identification and development of active principles from plant sources | 1-gen-2021 | Governa, Paolo | - | |
FFAR1/GPR40: One target, different binding sites, many agonists, no drugs, but a continuous and unprofitable tug-of-war between ligand lipophilicity, activity, and toxicity | 1-gen-2021 | Governa, Paolo; Caroleo, Maria Cristina; Carullo, Gabriele; Aiello, Francesca; Cione, Erika; Manetti, Fabrizio | - | |
Pinocembrin and its linolenoyl ester derivative induce wound healing activity in HaCaT cell line potentially involving a GPR120/FFA4 mediated pathway | 1-gen-2021 | Mazzotta, Sarah; Governa, Paolo; Borgonetti, Vittoria; Marcolongo, Paola; Nanni, Claudio; Gamberucci, Alessandra; Manetti, Fabrizio; Pessina, Federica; Carullo, Gabriele; Brizzi, Antonella; Aiello, Francesca | - | |
Cannabidiol Isolated From Cannabis sativa L. Protects Intestinal Barrier From In Vitro Inflammation and Oxidative Stress | 1-gen-2021 | Cocetta, Veronica; Governa, Paolo; Borgonetti, Vittoria; Tinazzi, Mattia; Peron, Gregorio; Catanzaro, Daniela; Berretta, Massimiliano; Biagi, Marco; Manetti, Fabrizio; Dall'Acqua, Stefano; Montopoli, Monica | - |
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