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Mostrati risultati da 1 a 20 di 47
Titolo Data di pubblicazione Autore(i) File Abstract
Consensus screening for a challenging target: the quest for P-glycoprotein inhibitors 1-gen-2024 Governa, Paolo; Biagi, Marco; Manetti, Fabrizio; Forli, Stefano -
Enhanced mapping of small-molecule binding sites in cells 1-gen-2024 Wozniak, Jacob M; Li, Weichao; Governa, Paolo; Chen, Li-Yun; Jadhav, Appaso; Dongre, Ashok; Forli, Stefano; Parker, Christopher G -
Helichrysum stoechas (L.) Moench reduces body weight gain and modulates mood disorders via inhibition of silent information regulator 1 (SIRT1) by arzanol 1-gen-2023 Borgonetti, Vittoria; Caroli, Clarissa; Governa, Paolo; Virginia, Brighenti; Pollastro, Federica; Franchini, Silvia; Manetti, Fabrizio; Les, Francisco; López, Victor; Pellati, Federica; Galeotti, Nicoletta -
Zingiberene, a non-zinc-binding class I HDAC inhibitor: A novel strategy for the management of neuropathic pain 1-gen-2023 Borgonetti, Vittoria; Governa, Paolo; Manetti, Fabrizio; Galeotti, Nicoletta -
A Novel Perilla frutescens (L.) Britton Cell-Derived Phytocomplex Regulates Keratinocytes Inflammatory Cascade and Barrier Function and Preserves Vaginal Mucosal Integrity In Vivo 1-gen-2023 Pressi, Giovanna; Rigillo, Giovanna; Governa, Paolo; Borgonetti, Vittoria; Baini, Giulia; Rizzi, Raffaella; Guarnerio, Chiara; Bertaiola, Oriana; Frigo, Marco; Merlin, Matilde; Paltrinieri, Stefania; Zambonin, Roberto; Pandolfo, Stefano; Biagi, Marco -
Effect of in vitro simulated digestion on the anti-Helicobacter Pylori activity of different Propolis extracts 1-gen-2023 Governa, Paolo; Romagnoli, Giulia; Albanese, Paola; Rossi, Federico; Manetti, Fabrizio; Biagi, Marco -
Cannabidiol-rich non-psychotropic Cannabis sativa L. oils attenuate peripheral neuropathy symptoms by regulation of CB2-mediated microglial neuroinflammation 1-gen-2023 Borgonetti, Vittoria; Anceschi, Lisa; Brighenti, Virginia; Corsi, Lorenzo; Governa, Paolo; Manetti, Fabrizio; Pellati, Federica; Galeotti, Nicoletta -
Antiviral Activity of Cannabidiolic Acid and Its Methyl Ester against SARS-CoV-2 1-gen-2023 Tamburello, Martina; Salamone, Stefano; Anceschi, Lisa; Governa, Paolo; Brighenti, Virginia; Morellini, Alice; Rossini, Giada; Manetti, Fabrizio; Gallinella, Giorgio; Pollastro, Federica; Pellati, Federica -
In Vitro Cell Culture of Rhus coriaria L.: A Standardized Phytocomplex Rich of Gallic Acid Derivatives with Antioxidant and Skin Repair Activity 1-gen-2022 Pressi, G.; Bertaiola, O.; Guarnerio, C.; Barbieri, E.; Rigillo, G.; Governa, P.; Biagi, M.; Guzzo, F.; Semenzato, A. -
Quinolines and Oxazino-quinoline Derivatives as Small Molecule GLI1 Inhibitors Identified by Virtual Screening 1-gen-2022 Manetti, Fabrizio; Maresca, Luisa; Crivaro, Enrica; Pepe, Sara; Cini, Elena; Singh, Snigdha; Governa, Paolo; Maramai, Samuele; Giannini, Giuseppe; Stecca, Barbara; Petricci, Elena -
Recent research results have converted gp120 binders to a therapeutic option for the treatment of HIV-1 infection. A medicinal chemistry point of view 1-gen-2022 Governa, Paolo; Manetti, Fabrizio -
Investigation on the neuroprotective effect of a cannabidiol-enriched non-psychotropic Cannabis sativa L. extract in an in vitro model of excitotoxicity 1-gen-2022 Borgonetti, Vittoria; Biagi, Marco; Galeotti, Nicoletta; Manetti, Fabrizio; Governa, Paolo -
Non-psychotropic Cannabis sativa L. phytocomplex modulates microglial inflammatory response through CB2 receptors-, endocannabinoids-, and NF-κB-mediated signaling 1-gen-2022 Borgonetti, V.; Benatti, C.; Governa, P.; Isoldi, G.; Pellati, F.; Alboni, S.; Tascedda, F.; Montopoli, M.; Galeotti, N.; Manetti, F.; Miraldi, E.; Biagi, M.; Rigillo, G. -
The Veterinary Anti-Parasitic Selamectin Is a Novel Inhibitor of the Mycobacterium tuberculosis DprE1 Enzyme 1-gen-2022 Ezquerra-Aznárez, José Manuel; Degiacomi, Giulia; Gašparovič, Henrich; Stelitano, Giovanni; Sammartino, Josè Camilla; Korduláková, Jana; Governa, Paolo; Manetti, Fabrizio; Pasca, Maria Rosalia; Chiarelli, Laurent Roberto; Ramón-García, Santiago -
Survey on the Recent Advances in 4-Hydroxyphenylpyruvate Dioxygenase (HPPD) Inhibition by Diketone and Triketone Derivatives and Congeneric Compounds: Structural Analysis of HPPD/Inhibitor Complexes and Structure-Activity Relationship Considerations 1-gen-2022 Governa, Paolo; Bernardini, Giulia; Braconi, Daniela; Manetti, Fabrizio; Santucci, Annalisa; Petricci, Elena -
Effects of in vitro simulated digestion on the antioxidant activity of different Camellia sinensis (L.) Kuntze leaves extracts 1-gen-2022 Governa, Paolo; Manetti, Fabrizio; Miraldi, Elisabetta; Biagi, Marco -
Identification and development of active principles from plant sources 1-gen-2021 Governa, Paolo -
FFAR1/GPR40: One target, different binding sites, many agonists, no drugs, but a continuous and unprofitable tug-of-war between ligand lipophilicity, activity, and toxicity 1-gen-2021 Governa, Paolo; Caroleo, Maria Cristina; Carullo, Gabriele; Aiello, Francesca; Cione, Erika; Manetti, Fabrizio -
Pinocembrin and its linolenoyl ester derivative induce wound healing activity in HaCaT cell line potentially involving a GPR120/FFA4 mediated pathway 1-gen-2021 Mazzotta, Sarah; Governa, Paolo; Borgonetti, Vittoria; Marcolongo, Paola; Nanni, Claudio; Gamberucci, Alessandra; Manetti, Fabrizio; Pessina, Federica; Carullo, Gabriele; Brizzi, Antonella; Aiello, Francesca -
Cannabidiol Isolated From Cannabis sativa L. Protects Intestinal Barrier From In Vitro Inflammation and Oxidative Stress 1-gen-2021 Cocetta, Veronica; Governa, Paolo; Borgonetti, Vittoria; Tinazzi, Mattia; Peron, Gregorio; Catanzaro, Daniela; Berretta, Massimiliano; Biagi, Marco; Manetti, Fabrizio; Dall'Acqua, Stefano; Montopoli, Monica -
Mostrati risultati da 1 a 20 di 47
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