Sfoglia per Autore
Deciphering the landscape of allosteric glutaminase 1 inhibitors as anticancer agents
2025-01-01 Vagaggini, C.; D'Ursi, P.; Poggialini, F.; Fossa, P.; Francesconi, V.; Trombetti, G.; Orro, A.; Dreassi, E.; Schenone, S.; Tonelli, M.; Carbone, A.
Insects as Source of Nutraceuticals with Antioxidant, Antihypertensive, and Antidiabetic Properties: Focus on the Species Approved in Europe up to 2024
2025-01-01 Brai, A.; Pasqualini, C.; Poggialini, F.; Vagaggini, C.; Dreassi, E.
Harnessing prebiotic formamide chemistry: a novel platform for antiviral exploration
2025-01-01 Martina, M. G.; Vagaggini, C.; Dreassi, E.; De Angelis, M.; Nencioni, L.; Dragoni, F.; Giammarino, F.; Boccuto, A.; Zazzi, M.; Vicenti, I.; Radi, M.
Investigating the potential of the SI306 Src inhibitor and its liposomal formulation in the non-small cell lung cancer treatment
2025-01-01 Poggialini, F.; Rango, E.; Vagaggini, C.; Diana, S.; Brai, A.; Grossi, G.; Frosini, M.; Musumeci, F.; Carbone, A.; Botta, M.; Dreassi, E.; Schenone, S.
Discovery of reversible monoacylglycerol lipase (MAGL) inhibitors based on ortho-hydroxyanilide scaffold
2025-01-01 Bononi, G.; Gado, F.; Masoni, S.; Scalabrini, D.; Vedova, L. D.; Di Stefano, M.; Piazza, L.; Poles, C.; Lonzi, C.; Landucci, E.; Vagaggini, C.; Poggialini, F.; Brai, A.; Caligiuri, I.; Rizzolio, F.; Mohamed, K. A.; Bertini, S.; De Lorenzi, E.; Dreassi, E.; Macchia, M.; Minutolo, F.; Laprairie, R. B.; Granchi, C.; Tuccinardi, T.
Optimization of 2,3-dihydrophthalazine-1,4-dione PARP inhibitor scaffold for nanomolar potency and specificity towards human PARP10
2025-01-01 Alaviuhkola, J.; Nizi, M. G.; Vagaggini, C.; Sarnari, C.; Lippok, B.; Maksimainen, M. M.; Bosetti, C.; Dhakar, S. S.; Manfroni, G.; Massari, S.; Dreassi, E.; Korn, P.; Tabarrini, O.; Lehtio, L.
Light-mediated activation/deactivation control and in vitro ADME-Tox profiling of a donepezil-like Dual AChE/MAO-B Inhibitor
2025-01-01 Poggialini, Federica; Governa, Paolo; Vagaggini, Chiara; Maramai, Samuele; Lamponi, Stefania; Mugnaini, Claudia; Brizzi, Antonella; Purgatorio, Rosa; De Candia, Modesto; Catto, Marco; Dreassi, Elena; Manetti, Fabrizio; Corelli, Federico; Altomare, Cosimo Damiano; Cappelli, Andrea; Paolino, Marco
Fluoromethylcarnitine, a novel inhibitor of trimethylamine levels in trimethylaminuria and trimethylamine N-oxide related disorders
2025-01-01 Cini, Elena; Vinciarelli, Giorgia; Siciliano, Sofia; Del Castello, Giorgio; Dreassi, Elena; Poggialini, Federica; Vagaggini, Chiara; Taddei, Maurizio; Battistuzzi, Gianfranco; Castagnetti, Andrea; Viciani, Elisa; Salvini, Laura; Sidoti, Antonina; Alibrandi, Simona; Giannini, Giuseppe
Evaluation of anti-tumoral activity in 3D cell model of a Src inhibitor prodrug for glioblastoma treatment
2025-01-01 Clementi, L.; Poggialini, F.; Musumeci, F.; Taglienti, J.; Cornacchia, E.; Vagaggini, C.; Carbone, A.; Grossi, G.; Dreassi, E.; Angelucci, A.; Schenone, S.
Exploitation of the Nutraceutical Potential of the Infesting Seaweed Chaetomorpha linum as a Yellow Mealworms’ Feed: Focus on Nutrients and Antioxidant Activity
2025-01-01 Brai, A.; Brogi, E.; Tarchi, F.; Poggialini, F.; Vagaggini, C.; Simoni, S.; Francardi, V.; Dreassi, E
Inhibition of Pseudomonas aeruginosa Carbonic Anhydrases, Exploring Ciprofloxacin Functionalization Toward New Antibacterial Agents: An In-Depth Multidisciplinary Study
2024-01-01 Marinacci, B.; D'Agostino, I.; Angeli, A.; Carradori, S.; Melfi, F.; Grande, R.; Corsiani, M.; Ferraroni, M.; Agamennone, M.; Tondo, A. R.; Zara, S.; Puca, V.; Pellegrini, B.; Vagaggini, C.; Dreassi, E.; Patrauchan, M. A.; Capasso, C.; Nicolotti, O.; Carta, F.; Supuran, C. T.
Novel multitarget directed ligands inspired by riluzole: A serendipitous synthesis of substituted benzo[b][1,4]thiazepines potentially useful as neuroprotective agents
2024-01-01 Maramai, S.; Saletti, M.; Paolino, M.; Giuliani, G.; Cazzola, J.; Spaiardi, P.; Talpo, F.; Frosini, M.; Pifferi, A.; Ballarotto, M.; Carotti, A.; Poggialini, F.; Vagaggini, C.; Dreassi, E.; Giorgi, G.; Dondio, G.; Cappelli, A.; Rosario Biella, G.; Anzini, M.
A Drug Discovery Approach to a Reveal Novel Antioxidant Natural Source: The Case of Chestnut Burr Biomass
2024-01-01 Trezza, Alfonso; Geminiani, Michela; Cutrera, Giuseppe; Dreassi, Elena; Frusciante, Luisa; Lamponi, Stefania; Spiga, Ottavia; Santucci, Annalisa
Exploiting the bile acid binding protein as transporter of a Cholic Acid/Mirin bioconjugate for potential applications in liver cancer therapy
2024-01-01 Tassone, Giusy; Maramai, Samuele; Paolino, Marco; Lamponi, Stefania; Poggialini, Federica; Dreassi, Elena; Petricci, Elena; Alcaro, Stefano; Pozzi, Cecilia; Romeo, Isabella
Applying molecular hybridization to design a new class of pyrazolo[3,4-d]pyrimidines as Src inhibitors active in hepatocellular carcinoma
2024-01-01 Di Maria, Salvatore; Passannanti, Raffaele; Poggialini, Federica; Vagaggini, Chiara; Serafinelli, Alessia; Bianchi, Elena; Governa, Paolo; Botta, Lorenzo; Maga, Giovanni; Crespan, Emmanuele; Manetti, Fabrizio; Dreassi, Elena; Musumeci, Francesca; Carbone, Anna; Schenone, Silvia
Phytochemical Composition, Anti-Inflammatory Property, and Anti-Atopic Effect of Chaetomorpha linum Extract
2024-01-01 Frusciante, Luisa; Geminiani, Michela; Trezza, Alfonso; Olmastroni, Tommaso; Mastroeni, Pierfrancesco; Salvini, Laura; Lamponi, Stefania; Bernini, Andrea; Grasso, Daniela; Dreassi, Elena; Spiga, Ottavia; Santucci, Annalisa
Upcycling Milk Industry Byproducts into Tenebrio molitor Larvae: Investigation on Fat, Protein, and Sugar Composition
2024-01-01 Brai, Annalaura; Neri, Cassia; Tarchi, Franca; Poggialini, Federica; Vagaggini, Chiara; Frosinini, Riccardo; Simoni, Sauro; Francardi, Valeria; Dreassi, Elena
Optimization of potent, broad-spectrum, and specific anti-influenza compounds targeting RNA polymerase PA-PB1 heterodimerization
2024-01-01 Bonomini, Anna; Felicetti, Tommaso; Pacetti, Martina; Bertagnin, Chiara; Coletti, Alice; Giammarino, Federica; De Angelis, Marta; Poggialini, Federica; Macchiarulo, Antonio; Sabatini, Stefano; Mercorelli, Beatrice; Nencioni, Lucia; Vicenti, Ilaria; Dreassi, Elena; Cecchetti, Violetta; Tabarrini, Oriana; Loregian, Arianna; Massari, Serena
An update on antibacterial AlkylGuanidino Ureas: Design of new derivatives, synergism with colistin and data analysis of the whole library
2024-01-01 Ardino, C.; Sannio, F.; Poli, G.; Galati, S.; Dreassi, E.; Botta, L.; Docquier, J. D.; D'Agostino, I.
Exploiting fall foliage by-products to optimize Tenebrio molitor nutraceutical value
2024-01-01 Brai, A.; Provenzani, M. P.; Pasqualini, C.; Poggialini, F.; Vagaggini, C.; Tarchi, F.; Frosinini, R.; Francardi, V.; Simoni, S.; Dreassi, E.
| Titolo | Data di pubblicazione | Autore(i) | File | Abstract |
|---|---|---|---|---|
| Deciphering the landscape of allosteric glutaminase 1 inhibitors as anticancer agents | 1-gen-2025 | Vagaggini, C.; D'Ursi, P.; Poggialini, F.; Fossa, P.; Francesconi, V.; Trombetti, G.; Orro, A.; Dreassi, E.; Schenone, S.; Tonelli, M.; Carbone, A. | - | |
| Insects as Source of Nutraceuticals with Antioxidant, Antihypertensive, and Antidiabetic Properties: Focus on the Species Approved in Europe up to 2024 | 1-gen-2025 | Brai, A.; Pasqualini, C.; Poggialini, F.; Vagaggini, C.; Dreassi, E. | - | |
| Harnessing prebiotic formamide chemistry: a novel platform for antiviral exploration | 1-gen-2025 | Martina, M. G.; Vagaggini, C.; Dreassi, E.; De Angelis, M.; Nencioni, L.; Dragoni, F.; Giammarino, F.; Boccuto, A.; Zazzi, M.; Vicenti, I.; Radi, M. | - | |
| Investigating the potential of the SI306 Src inhibitor and its liposomal formulation in the non-small cell lung cancer treatment | 1-gen-2025 | Poggialini, F.; Rango, E.; Vagaggini, C.; Diana, S.; Brai, A.; Grossi, G.; Frosini, M.; Musumeci, F.; Carbone, A.; Botta, M.; Dreassi, E.; Schenone, S. | - | |
| Discovery of reversible monoacylglycerol lipase (MAGL) inhibitors based on ortho-hydroxyanilide scaffold | 1-gen-2025 | Bononi, G.; Gado, F.; Masoni, S.; Scalabrini, D.; Vedova, L. D.; Di Stefano, M.; Piazza, L.; Poles, C.; Lonzi, C.; Landucci, E.; Vagaggini, C.; Poggialini, F.; Brai, A.; Caligiuri, I.; Rizzolio, F.; Mohamed, K. A.; Bertini, S.; De Lorenzi, E.; Dreassi, E.; Macchia, M.; Minutolo, F.; Laprairie, R. B.; Granchi, C.; Tuccinardi, T. | - | |
| Optimization of 2,3-dihydrophthalazine-1,4-dione PARP inhibitor scaffold for nanomolar potency and specificity towards human PARP10 | 1-gen-2025 | Alaviuhkola, J.; Nizi, M. G.; Vagaggini, C.; Sarnari, C.; Lippok, B.; Maksimainen, M. M.; Bosetti, C.; Dhakar, S. S.; Manfroni, G.; Massari, S.; Dreassi, E.; Korn, P.; Tabarrini, O.; Lehtio, L. | - | |
| Light-mediated activation/deactivation control and in vitro ADME-Tox profiling of a donepezil-like Dual AChE/MAO-B Inhibitor | 1-gen-2025 | Poggialini, Federica; Governa, Paolo; Vagaggini, Chiara; Maramai, Samuele; Lamponi, Stefania; Mugnaini, Claudia; Brizzi, Antonella; Purgatorio, Rosa; De Candia, Modesto; Catto, Marco; Dreassi, Elena; Manetti, Fabrizio; Corelli, Federico; Altomare, Cosimo Damiano; Cappelli, Andrea; Paolino, Marco | - | |
| Fluoromethylcarnitine, a novel inhibitor of trimethylamine levels in trimethylaminuria and trimethylamine N-oxide related disorders | 1-gen-2025 | Cini, Elena; Vinciarelli, Giorgia; Siciliano, Sofia; Del Castello, Giorgio; Dreassi, Elena; Poggialini, Federica; Vagaggini, Chiara; Taddei, Maurizio; Battistuzzi, Gianfranco; Castagnetti, Andrea; Viciani, Elisa; Salvini, Laura; Sidoti, Antonina; Alibrandi, Simona; Giannini, Giuseppe | - | |
| Evaluation of anti-tumoral activity in 3D cell model of a Src inhibitor prodrug for glioblastoma treatment | 1-gen-2025 | Clementi, L.; Poggialini, F.; Musumeci, F.; Taglienti, J.; Cornacchia, E.; Vagaggini, C.; Carbone, A.; Grossi, G.; Dreassi, E.; Angelucci, A.; Schenone, S. | - | |
| Exploitation of the Nutraceutical Potential of the Infesting Seaweed Chaetomorpha linum as a Yellow Mealworms’ Feed: Focus on Nutrients and Antioxidant Activity | 1-gen-2025 | Brai, A.; Brogi, E.; Tarchi, F.; Poggialini, F.; Vagaggini, C.; Simoni, S.; Francardi, V.; Dreassi, E | - | |
| Inhibition of Pseudomonas aeruginosa Carbonic Anhydrases, Exploring Ciprofloxacin Functionalization Toward New Antibacterial Agents: An In-Depth Multidisciplinary Study | 1-gen-2024 | Marinacci, B.; D'Agostino, I.; Angeli, A.; Carradori, S.; Melfi, F.; Grande, R.; Corsiani, M.; Ferraroni, M.; Agamennone, M.; Tondo, A. R.; Zara, S.; Puca, V.; Pellegrini, B.; Vagaggini, C.; Dreassi, E.; Patrauchan, M. A.; Capasso, C.; Nicolotti, O.; Carta, F.; Supuran, C. T. | - | |
| Novel multitarget directed ligands inspired by riluzole: A serendipitous synthesis of substituted benzo[b][1,4]thiazepines potentially useful as neuroprotective agents | 1-gen-2024 | Maramai, S.; Saletti, M.; Paolino, M.; Giuliani, G.; Cazzola, J.; Spaiardi, P.; Talpo, F.; Frosini, M.; Pifferi, A.; Ballarotto, M.; Carotti, A.; Poggialini, F.; Vagaggini, C.; Dreassi, E.; Giorgi, G.; Dondio, G.; Cappelli, A.; Rosario Biella, G.; Anzini, M. | - | |
| A Drug Discovery Approach to a Reveal Novel Antioxidant Natural Source: The Case of Chestnut Burr Biomass | 1-gen-2024 | Trezza, Alfonso; Geminiani, Michela; Cutrera, Giuseppe; Dreassi, Elena; Frusciante, Luisa; Lamponi, Stefania; Spiga, Ottavia; Santucci, Annalisa | - | |
| Exploiting the bile acid binding protein as transporter of a Cholic Acid/Mirin bioconjugate for potential applications in liver cancer therapy | 1-gen-2024 | Tassone, Giusy; Maramai, Samuele; Paolino, Marco; Lamponi, Stefania; Poggialini, Federica; Dreassi, Elena; Petricci, Elena; Alcaro, Stefano; Pozzi, Cecilia; Romeo, Isabella | - | |
| Applying molecular hybridization to design a new class of pyrazolo[3,4-d]pyrimidines as Src inhibitors active in hepatocellular carcinoma | 1-gen-2024 | Di Maria, Salvatore; Passannanti, Raffaele; Poggialini, Federica; Vagaggini, Chiara; Serafinelli, Alessia; Bianchi, Elena; Governa, Paolo; Botta, Lorenzo; Maga, Giovanni; Crespan, Emmanuele; Manetti, Fabrizio; Dreassi, Elena; Musumeci, Francesca; Carbone, Anna; Schenone, Silvia | - | |
| Phytochemical Composition, Anti-Inflammatory Property, and Anti-Atopic Effect of Chaetomorpha linum Extract | 1-gen-2024 | Frusciante, Luisa; Geminiani, Michela; Trezza, Alfonso; Olmastroni, Tommaso; Mastroeni, Pierfrancesco; Salvini, Laura; Lamponi, Stefania; Bernini, Andrea; Grasso, Daniela; Dreassi, Elena; Spiga, Ottavia; Santucci, Annalisa | - | |
| Upcycling Milk Industry Byproducts into Tenebrio molitor Larvae: Investigation on Fat, Protein, and Sugar Composition | 1-gen-2024 | Brai, Annalaura; Neri, Cassia; Tarchi, Franca; Poggialini, Federica; Vagaggini, Chiara; Frosinini, Riccardo; Simoni, Sauro; Francardi, Valeria; Dreassi, Elena | - | |
| Optimization of potent, broad-spectrum, and specific anti-influenza compounds targeting RNA polymerase PA-PB1 heterodimerization | 1-gen-2024 | Bonomini, Anna; Felicetti, Tommaso; Pacetti, Martina; Bertagnin, Chiara; Coletti, Alice; Giammarino, Federica; De Angelis, Marta; Poggialini, Federica; Macchiarulo, Antonio; Sabatini, Stefano; Mercorelli, Beatrice; Nencioni, Lucia; Vicenti, Ilaria; Dreassi, Elena; Cecchetti, Violetta; Tabarrini, Oriana; Loregian, Arianna; Massari, Serena | - | |
| An update on antibacterial AlkylGuanidino Ureas: Design of new derivatives, synergism with colistin and data analysis of the whole library | 1-gen-2024 | Ardino, C.; Sannio, F.; Poli, G.; Galati, S.; Dreassi, E.; Botta, L.; Docquier, J. D.; D'Agostino, I. | - | |
| Exploiting fall foliage by-products to optimize Tenebrio molitor nutraceutical value | 1-gen-2024 | Brai, A.; Provenzani, M. P.; Pasqualini, C.; Poggialini, F.; Vagaggini, C.; Tarchi, F.; Frosinini, R.; Francardi, V.; Simoni, S.; Dreassi, E. | - |
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