Sfoglia per Autore
Natural products as payloads for antibody-drug conjugates: Cyclopamine linked to cetuximab for hedgehog pathway inhibition
2026-01-01 Ricciardella, Giovanni; Migliorini, Francesca; Maresca, Luisa; Cini, Elena; Ievoli, Giovanni; Petricci, Elena; Taddei, Maurizio; Zambardino, Demetra; Stecca, Barbara; Montalbano, Alberto; Crivaro, Enrica
An integrated NMR approach for evaluating linker-payload conjugation with monoclonal antibodies
2026-01-01 Ghini, Veronica; Siciliano, Sofia; Querci, Leonardo; Angiolini, Lorenzo; Truglio, Giuseppina Ivana; Cini, Elena; Piccioli, Mario; Petricci, Elena; Turano, Paola
Plantacare 2000: A Biosurfactant for an Eco‐Friendly Palladium Catalyzed Cyanation of Aromatic Bromides
2025-01-01 Zurzolo, Simone; Ermini, Elena; Locatelli, Erica; Petricci, Elena; Truglio, Giuseppina I.; Vaccaro, Luigi; Valentini, Federica; Taddei, Maurizio
ProTide-enabled antibody-drug conjugates: A novel platform for the targeted delivery of phosphorylated drugs
2025-01-01 Siciliano, Sofia; Bernardi, Clizia; Finetti, Federica; Guerrini, Asia; Monti, Maria Chiara; Morretta, Elva; Petricci, Elena; Poggialini, Federica; Romagnoli, Giulia; Taddei, Maurizio; Trabalzini, Lorenza; Vinciarelli, Giorgia; Zambardino, Demetra; Cini, Elena
A Comprehensive In Vitro and In Silico Approach for Targeting 4-Hydroxyphenyl Pyruvate Dioxygenase: Towards New Therapeutics for Alkaptonuria
2025-01-01 Bernardini, G.; Trezza, A.; Petricci, E.; Romagnoli, G.; Zambardino, D.; Manetti, F.; Braconi, D.; Geminiani, M.; Santucci, A.
Machine Learning for Predicting the Drug-to-Antibody Ratio (DAR) in the Synthesis of Antibody–Drug Conjugates (ADCs)
2025-01-01 Angiolini, Lorenzo; Manetti, Fabrizio; Spiga, Ottavia; Tafi, Andrea; Visibelli, Anna; Petricci, Elena
Exploiting the bile acid binding protein as transporter of a Cholic Acid/Mirin bioconjugate for potential applications in liver cancer therapy
2024-01-01 Tassone, Giusy; Maramai, Samuele; Paolino, Marco; Lamponi, Stefania; Poggialini, Federica; Dreassi, Elena; Petricci, Elena; Alcaro, Stefano; Pozzi, Cecilia; Romeo, Isabella
A nanoencapsulated oral formulation of fenretinide promotes local and metastatic breast cancer dormancy in HER2/neu transgenic mice
2024-01-01 De Angelis, M. L.; Francescangeli, F.; Aricò, E.; Verachi, P.; Zucchetti, M.; Matteo, C.; Petricci, E.; Pilozzi, E.; Orienti, I.; Boe, A.; Eramo, A.; Rossi, R.; Corati, T.; Macchia, D.; Pacca, A. M.; Zeuner, A.; Baiocchi, M.
Switching mechanistic pathways by micellar catalysis: A highly selective rhodium catalyst for the hydroaminomethylation of olefins with anilines in water
2023-01-01 Migliorini, F.; Monciatti, E.; Romagnoli, G.; Parisi, M. L.; Taubert, J.; Vogt, M.; Langer, R.; Petricci, E.
Targeting GLI1 and GLI2 with small molecule inhibitors to suppress GLI-dependent transcription and tumor growth
2023-01-01 Maresca, Luisa; Crivaro, Enrica; Migliorini, Francesca; Anichini, Giulia; Giammona, Alessandro; Pepe, Sara; Poggialini, Federica; Vagaggini, Chiara; Giannini, Giuseppe; Sestini, Serena; Borgognoni, Lorenzo; Lapucci, Andrea; Dreassi, Elena; Taddei, Maurizio; Manetti, Fabrizio; Petricci, Elena; Stecca, Barbara
Micellar Catalysis for a Sustainable Hydroaminomethylation Process in Water
2023-01-01 Monciatti, Elisabetta; Migliorini, Francesca; Romagnoli, Giulia; Vogt, Matthias; Langer, Robert; Parisi, MARIA LAURA; Petricci, Elena
Survey on the recent advances in 4-Hydroxyphenylpyruvate Dioxygenase (HPPD) inhibition by diketone and triketone derivatives and congeneric compounds: structural analysis of HPPD/inhibitor complexes and structure-activity relationship considerations
2022-01-01 Governa, Paolo; Bernardini, Giulia; Braconi, Daniela; Manetti, Fabrizio; Santucci, Annalisa; Petricci, Elena
Antibacterial alkylguanidino ureas: Molecular simplification approach, searching for membrane-based MoA
2022-01-01 D'Agostino, I.; Ardino, C.; Poli, G.; Sannio, F.; Lucidi, M.; Poggialini, F.; Visaggio, D.; Rango, E.; Filippi, S.; Petricci, E.; Visca, P.; Botta, L.; Docquier, J. -D.; Dreassi, E.
Quinolines and Oxazino-quinoline derivatives as small molecule GLI1 inhibitors identified by virtual screening
2022-01-01 Manetti, Fabrizio; Maresca, Luisa; Crivaro, Enrica; Pepe, Sara; Cini, Elena; Singh, Snigdha; Governa, Paolo; Maramai, Samuele; Giannini, Giuseppe; Stecca, Barbara; Petricci, Elena
A pH-responsive crosslinker platform for antibody-drug conjugate (ADC) targeting delivery
2022-01-01 Migliorini, Francesca; Cini, Elena; Dreassi, Elena; Finetti, Federica; Ievoli, Giovanni; Macrì, Giulia; Petricci, Elena; Rango, Enrico; Trabalzini, Lorenza; Taddei, Maurizio
Structural characterization of human heat shock protein 90 N-Terminal domain and its variants K112R and K112A in complex with a potent 1,2,3-Triazole-based inhibitor
2022-01-01 Tassone, Giusy; Mazzorana, Marco; Mangani, Stefano; Petricci, Elena; Cini, Elena; Giannini, Giuseppe; Pozzi, Cecilia; Maramai, Samuele
Requirements for MRN endonuclease processing of topoisomerase II-mediated DNA damage in mammalian cells
2022-01-01 Sun, Yilun; Soans, Eroica; Mishina, Margarita; Petricci, Elena; Pommier, Yves; Nitiss, Karin C.; Nitiss, John L.
An Intramolecular Hydroaminomethylation-Based Approach to Pyrrolizidine Alkaloids under Microwave-Assisted Heating
2022-01-01 Petricci, Elena; Zurzolo, Simone; Matassini, Camilla; Maramai, Samuele; Cardona, Francesca; Goti, Andrea; Taddei, Maurizio
Antibody drug conjugates with hydroxamic acid cargos for histone deacetylase (HDAC) inhibition
2021-01-01 Cianferotti, C.; Faltoni, V.; Cini, E.; Ermini, E.; Migliorini, F.; Petricci, E.; Taddei, M.; Salvini, L.; Battistuzzi, G.; Milazzo, F. M.; Anastasi, A. M.; Chiapparino, C.; De Santis, R.; Giannini, G.
A molecular spectroscopy approach for the investigation of early phase ochronotic pigment development in Alkaptonuria
2021-01-01 Bernini, A.; Petricci, E.; Atrei, A.; Baratto, M. C.; Manetti, F.; Santucci, A.
| Titolo | Data di pubblicazione | Autore(i) | File | Abstract |
|---|---|---|---|---|
| Natural products as payloads for antibody-drug conjugates: Cyclopamine linked to cetuximab for hedgehog pathway inhibition | 1-gen-2026 | Ricciardella, Giovanni; Migliorini, Francesca; Maresca, Luisa; Cini, Elena; Ievoli, Giovanni; Petricci, Elena; Taddei, Maurizio; Zambardino, Demetra; Stecca, Barbara; Montalbano, Alberto; Crivaro, Enrica | - | |
| An integrated NMR approach for evaluating linker-payload conjugation with monoclonal antibodies | 1-gen-2026 | Ghini, Veronica; Siciliano, Sofia; Querci, Leonardo; Angiolini, Lorenzo; Truglio, Giuseppina Ivana; Cini, Elena; Piccioli, Mario; Petricci, Elena; Turano, Paola | - | |
| Plantacare 2000: A Biosurfactant for an Eco‐Friendly Palladium Catalyzed Cyanation of Aromatic Bromides | 1-gen-2025 | Zurzolo, Simone; Ermini, Elena; Locatelli, Erica; Petricci, Elena; Truglio, Giuseppina I.; Vaccaro, Luigi; Valentini, Federica; Taddei, Maurizio | - | |
| ProTide-enabled antibody-drug conjugates: A novel platform for the targeted delivery of phosphorylated drugs | 1-gen-2025 | Siciliano, Sofia; Bernardi, Clizia; Finetti, Federica; Guerrini, Asia; Monti, Maria Chiara; Morretta, Elva; Petricci, Elena; Poggialini, Federica; Romagnoli, Giulia; Taddei, Maurizio; Trabalzini, Lorenza; Vinciarelli, Giorgia; Zambardino, Demetra; Cini, Elena | - | |
| A Comprehensive In Vitro and In Silico Approach for Targeting 4-Hydroxyphenyl Pyruvate Dioxygenase: Towards New Therapeutics for Alkaptonuria | 1-gen-2025 | Bernardini, G.; Trezza, A.; Petricci, E.; Romagnoli, G.; Zambardino, D.; Manetti, F.; Braconi, D.; Geminiani, M.; Santucci, A. | - | |
| Machine Learning for Predicting the Drug-to-Antibody Ratio (DAR) in the Synthesis of Antibody–Drug Conjugates (ADCs) | 1-gen-2025 | Angiolini, Lorenzo; Manetti, Fabrizio; Spiga, Ottavia; Tafi, Andrea; Visibelli, Anna; Petricci, Elena | - | |
| Exploiting the bile acid binding protein as transporter of a Cholic Acid/Mirin bioconjugate for potential applications in liver cancer therapy | 1-gen-2024 | Tassone, Giusy; Maramai, Samuele; Paolino, Marco; Lamponi, Stefania; Poggialini, Federica; Dreassi, Elena; Petricci, Elena; Alcaro, Stefano; Pozzi, Cecilia; Romeo, Isabella | - | |
| A nanoencapsulated oral formulation of fenretinide promotes local and metastatic breast cancer dormancy in HER2/neu transgenic mice | 1-gen-2024 | De Angelis, M. L.; Francescangeli, F.; Aricò, E.; Verachi, P.; Zucchetti, M.; Matteo, C.; Petricci, E.; Pilozzi, E.; Orienti, I.; Boe, A.; Eramo, A.; Rossi, R.; Corati, T.; Macchia, D.; Pacca, A. M.; Zeuner, A.; Baiocchi, M. | - | |
| Switching mechanistic pathways by micellar catalysis: A highly selective rhodium catalyst for the hydroaminomethylation of olefins with anilines in water | 1-gen-2023 | Migliorini, F.; Monciatti, E.; Romagnoli, G.; Parisi, M. L.; Taubert, J.; Vogt, M.; Langer, R.; Petricci, E. | - | |
| Targeting GLI1 and GLI2 with small molecule inhibitors to suppress GLI-dependent transcription and tumor growth | 1-gen-2023 | Maresca, Luisa; Crivaro, Enrica; Migliorini, Francesca; Anichini, Giulia; Giammona, Alessandro; Pepe, Sara; Poggialini, Federica; Vagaggini, Chiara; Giannini, Giuseppe; Sestini, Serena; Borgognoni, Lorenzo; Lapucci, Andrea; Dreassi, Elena; Taddei, Maurizio; Manetti, Fabrizio; Petricci, Elena; Stecca, Barbara | - | |
| Micellar Catalysis for a Sustainable Hydroaminomethylation Process in Water | 1-gen-2023 | Monciatti, Elisabetta; Migliorini, Francesca; Romagnoli, Giulia; Vogt, Matthias; Langer, Robert; Parisi, MARIA LAURA; Petricci, Elena | - | |
| Survey on the recent advances in 4-Hydroxyphenylpyruvate Dioxygenase (HPPD) inhibition by diketone and triketone derivatives and congeneric compounds: structural analysis of HPPD/inhibitor complexes and structure-activity relationship considerations | 1-gen-2022 | Governa, Paolo; Bernardini, Giulia; Braconi, Daniela; Manetti, Fabrizio; Santucci, Annalisa; Petricci, Elena | - | |
| Antibacterial alkylguanidino ureas: Molecular simplification approach, searching for membrane-based MoA | 1-gen-2022 | D'Agostino, I.; Ardino, C.; Poli, G.; Sannio, F.; Lucidi, M.; Poggialini, F.; Visaggio, D.; Rango, E.; Filippi, S.; Petricci, E.; Visca, P.; Botta, L.; Docquier, J. -D.; Dreassi, E. | - | |
| Quinolines and Oxazino-quinoline derivatives as small molecule GLI1 inhibitors identified by virtual screening | 1-gen-2022 | Manetti, Fabrizio; Maresca, Luisa; Crivaro, Enrica; Pepe, Sara; Cini, Elena; Singh, Snigdha; Governa, Paolo; Maramai, Samuele; Giannini, Giuseppe; Stecca, Barbara; Petricci, Elena | - | |
| A pH-responsive crosslinker platform for antibody-drug conjugate (ADC) targeting delivery | 1-gen-2022 | Migliorini, Francesca; Cini, Elena; Dreassi, Elena; Finetti, Federica; Ievoli, Giovanni; Macrì, Giulia; Petricci, Elena; Rango, Enrico; Trabalzini, Lorenza; Taddei, Maurizio | - | |
| Structural characterization of human heat shock protein 90 N-Terminal domain and its variants K112R and K112A in complex with a potent 1,2,3-Triazole-based inhibitor | 1-gen-2022 | Tassone, Giusy; Mazzorana, Marco; Mangani, Stefano; Petricci, Elena; Cini, Elena; Giannini, Giuseppe; Pozzi, Cecilia; Maramai, Samuele | - | |
| Requirements for MRN endonuclease processing of topoisomerase II-mediated DNA damage in mammalian cells | 1-gen-2022 | Sun, Yilun; Soans, Eroica; Mishina, Margarita; Petricci, Elena; Pommier, Yves; Nitiss, Karin C.; Nitiss, John L. | - | |
| An Intramolecular Hydroaminomethylation-Based Approach to Pyrrolizidine Alkaloids under Microwave-Assisted Heating | 1-gen-2022 | Petricci, Elena; Zurzolo, Simone; Matassini, Camilla; Maramai, Samuele; Cardona, Francesca; Goti, Andrea; Taddei, Maurizio | - | |
| Antibody drug conjugates with hydroxamic acid cargos for histone deacetylase (HDAC) inhibition | 1-gen-2021 | Cianferotti, C.; Faltoni, V.; Cini, E.; Ermini, E.; Migliorini, F.; Petricci, E.; Taddei, M.; Salvini, L.; Battistuzzi, G.; Milazzo, F. M.; Anastasi, A. M.; Chiapparino, C.; De Santis, R.; Giannini, G. | - | |
| A molecular spectroscopy approach for the investigation of early phase ochronotic pigment development in Alkaptonuria | 1-gen-2021 | Bernini, A.; Petricci, E.; Atrei, A.; Baratto, M. C.; Manetti, F.; Santucci, A. | - |
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