Sfoglia per Autore
Synthesis and biological investigation of peptidomimetic SARS‐CoV‐2 main protease inhibitors bearing quinoline‐based heterocycles at P3
2025-01-01 Rossi, Sara; Deidda, Graziano; Fiaschi, Lia; Ibba, Roberta; Pieroni, Mariachiara; Dichiara, Maria; Carullo, Gabriele; Butini, Stefania; Ramunno, Anna; Brogi, Simone; Lolicato, Marco; Arrigoni, Cristina; Cabella, Noemi; Bavagnoli, Laura; Maga, Giovanni; Varasi, Ilenia; Biba, Camilla; Vicenti, Ilaria; Gemma, Sandra; Crespan, Emmanuele; Zazzi, Maurizio; Campiani, Giuseppe
Discovery of p-Trifluoromethylbenzohydrazide Derivatives as Potent Antiviral Agents against Monkeypox Virus
2025-01-01 Rossi, Sara; Pozzetti, Luca; Carullo, Gabriele; Dichiara, Maria; Butini, Stefania; Radi, Marco; Ramunno, Anna; Terrosi, Chiara; Barra, Giovanni; Berisio, Rita; Gemma, Sandra; Cusi, Maria Grazia; Campiani, Giuseppe
Development of selective sigma-1 receptor ligands with antiallodynic activity: A focus on piperidine and piperazine scaffolds
2025-01-01 Cosentino, Giuseppe; Dichiara, Maria; Ambrosio, Francesca Alessandra; Leotta, Claudia Giovanna; Costa, Giosuè; Procopio, Francesca; Costanzo, Giuliana; Raffa, Alessandro; Artacho-Cordón, Antonia; Ruiz-Cantero, M. Carmen; Pasquinucci, Lorella; Marrazzo, Agostino; Pitari, Giovanni Mario; Cobos, Enrique J.; Alcaro, Stefano; Amata, Emanuele
Uncovering a Mutation-Independent Therapeutic Strategy against Inherited Retinal Diseases: Development of Class I HDAC/LSD1 Hybrid Inhibitors
2025-01-01 Carullo, Gabriele; Piano, Ilaria; Salamone, Giulia; Corsi, Francesca; Orsini, Noemi; Dichiara, Maria; Cursaro, Ilaria; Fontana, Anna; Galante, Alessia; Contri, Chiara; Guadagno, Ludovica; Caroli, Jonatan; Mattevi, Andrea; Vincenzi, Fabrizio; Varani, Katia; Brogi, Simone; Gemma, Sandra; Butini, Stefania; Gargini, Claudia; Strettoi, Enrica; Campiani, Giuseppe
Unlocking the potential of biostimulants in sustainable agriculture: Effect of wood distillate on the nutritional profiling of apples
2024-01-01 Fedeli, Riccardo; Dichiara, Maria; Carullo, Gabriele; Tudino, Valeria; Gemma, Sandra; Butini, Stefania; Campiani, Giuseppe; Loppi, Stefano
Exploring Structural Requirements for Sigma-1 Receptor Linear Ligands: Experimental and Computational Approaches
2024-01-01 Lombardo, Lisa; Mirabile, Salvatore; Gitto, Rosaria; Cosentino, Giuseppe; Alcaro, Stefano; Dichiara, Maria; Marrazzo, Agostino; Amata, Emanuele; Ortuso, Francesco; De Luca, Laura
Biostimulants for Sustainable Food Production: Effects of Wood Distillate to Fortify Chickpea Flour for Development of Functional Bakery Products
2024-01-01 Fedeli, Riccardo; Spizzirri, Umile Gianfranco; Aquino, Giovanna; Basilicata, Manuela Giovanna; Pepe, Giacomo; Campiglia, Pietro; Celletti, Silvia; Tudino, Valeria; Dichiara, Maria; Gemma, Sandra; Butini, Stefania; Carullo, Gabriele; Aiello, Francesca; Restuccia, Donatella; Campiani, Giuseppe; Loppi, Stefano
Designing drugs optimized for both blood–brain barrier permeation and intra-cerebral partition
2024-01-01 Dichiara, Maria; Cosentino, Giuseppe; Giordano, Giorgia; Pasquinucci, Lorella; Marrazzo, Agostino; Costanzo, Giuliana; Amata, Emanuele
Design, Synthesis, and Cytotoxic Assessment of New Haloperidol Analogues as Potential Anticancer Compounds Targeting Sigma Receptors
2024-01-01 Zampieri, Daniele; Romano, Maurizio; Fortuna, Sara; Amata, Emanuele; Dichiara, Maria; Cosentino, Giuseppe; Marrazzo, Agostino; Mamolo, Maria Grazia
A novel potent class I HDAC inhibitor reverses the STAT4/p66Shc apoptotic defect in B cells from chronic lymphocytic leukemia patients
2024-01-01 Rossi, Sara; Tatangelo, Vanessa; Dichiara, Maria; Butini, Stefania; Gemma, Sandra; Brogi, Simone; Pasquini, Silvia; Cappello, Martina; Vincenzi, Fabrizio; Varani, Katia; Lopresti, Ludovica; Malchiodi, Margherita; Carrara, Chiara; Gozzetti, Alessandro; Bocchia, Monica; Marotta, Giuseppe; Patrussi, Laura; Carullo, Gabriele; Baldari, Cosima T.; Campiani, Giuseppe
Structure–Property Optimization of a Series of Imidazopyridines for Visceral Leishmaniasis
2023-01-01 Dichiara, Maria; Simpson, Quillon J.; Quotadamo, Antonio; Jalani, Hitesh B.; Huang, Anson X.; Millard, Caroline C.; Klug, Dana M.; Tse, Edwin G.; Todd, Matthew H.; Silva, Daniel Gedder; da Silva Emery, Flavio; Carlson, J. Eric; Zheng, Shao-Liang; Vleminckx, Margot; Matheeussen, An; Caljon, Guy; Pollastri, Michael P.; Sjö, Peter; Perry, Benjamin; Ferrins, Lori
Open Source Antibiotics: Simple Diarylimidazoles Are Potent against Methicillin-Resistant Staphylococcus aureus
2023-01-01 Klug, Dana M.; Tse, Edwin G.; Silva, Daniel G.; Cao, Yafeng; Charman, Susan A.; Chauhan, Jyoti; Crighton, Elly; Dichiara, Maria; Drake, Chris; Drewry, David; da Silva Emery, Flavio; Ferrins, Lori; Graves, Lee; Hopkins, Emily; Kresina, Thomas A. C.; Lorente-Macías, Álvaro; Perry, Benjamin; Phipps, Richard; Quiroga, Bruno; Quotadamo, Antonio; Sabatino, Giada N.; Sama, Anthony; Schätzlein, Andreas; Simpson, Quillon J.; Steele, Jonathan; Shanu-Wilson, Julia; Sjö, Peter; Stapleton, Paul; Swain, Christopher J.; Vaideanu, Alexandra; Xie, Huanxu; Zuercher, William; Todd, Matthew H.
New Insights into the Opioid Analgesic Profile of cis-(−)-N-Normetazocine-derived Ligands
2023-01-01 Costanzo, Giuliana; Turnaturi, Rita; Parenti, Carmela; Spoto, Salvatore; Piana, Silvia; Dichiara, Maria; Zagni, Chiara; Galambos, Anna Rita; Essmat, Nariman; Marrazzo, Agostino; Amata, Emanuele; Al-Khrasani, Mahmoud; Pasquinucci, Lorella
Discovery and computational studies of piperidine/piperazine-based compounds endowed with sigma receptor affinity
2023-01-01 De Luca, Laura; Lombardo, Lisa; Mirabile, Salvatore; Marrazzo, Agostino; Dichiara, Maria; Cosentino, Giuseppe; Amata, Emanuele; Gitto, Rosaria
Discovery of first novel sigma/HDACi dual-ligands with a potent in vitro antiproliferative activity
2023-01-01 Barbaraci, Carla; di Giacomo, Viviana; Maruca, Annalisa; Patamia, Vincenzo; Rocca, Roberta; Dichiara, Maria; Di Rienzo, Annalisa; Cacciatore, Ivana; Cataldi, Amelia; Balaha, Marwa; Rapino, Monica; Zagni, Chiara; Zampieri, Daniele; Pasquinucci, Lorella; Parenti, Carmela; Amata, Emanuele; Rescifina, Antonio; Alcaro, Stefano; Marrazzo, Agostino
Cytotoxicity profiles and neuroprotective properties of the novel ifenprodil analogues as sigma ligands
2023-01-01 Zampieri, Daniele; Calabretti, Antonella; Romano, Maurizio; Fortuna, Sara; Collina, Simona; Amata, Emanuele; Dichiara, Maria; Marrazzo, Agostino; Mamolo Maria, Grazia.
Dual Piperidine-Based Histamine H3 and Sigma-1 Receptor Ligands in the Treatment of Nociceptive and Neuropathic Pain
2023-01-01 Szczepańska, Katarzyna; Karcz, Tadeusz; Dichiara, Maria; Mogilski, Szczepan; Kalinowska-Tłuścik, Justyna; Pilarski, Bogusław; Leniak, Arkadiusz; Pietruś, Wojciech; Podlewska, Sabina; Popiołek-Barczyk, Katarzyna; Humphrys, Laura J.; Ruiz-Cantero, M. Carmen; Reiner-Link, David; Leitzbach, Luisa; Łażewska, Dorota; Pockes, Steffen; Górka, Michał; Zmysłowski, Adam; Calmels, Thierry; Cobos, Enrique J.; Marrazzo, Agostino; Stark, Holger; Bojarski, Andrzej J.; Amata, Emanuele; Kieć-Kononowicz, Katarzyna
Discovery of AD258 as a Sigma Receptor Ligand with Potent Antiallodynic Activity
2023-01-01 Dichiara, Maria; Ambrosio, Francesca Alessandra; Lee, Sang Min; Ruiz-Cantero, M. Carmen; Lombino, Jessica; Coricello, Adriana; Costa, Giosuè; Shah, Dhara; Costanzo, Giuliana; Pasquinucci, Lorella; Son, Kyung No; Cosentino, Giuseppe; González-Cano, Rafael; Marrazzo, Agostino; Aakalu, Vinay Kumar; Cobos, Enrique J.; Alcaro, Stefano; Amata, Emanuele
Synthesis, computational insights, and evaluation of novel sigma receptors ligands
2023-01-01 Dichiara, Maria; Ambrosio, Francesca Alessandra; Barbaraci, Carla; Gonzalez-Cano, Rafael; Costa, Giosuè.; Parenti, Carmela; Marrazzo, Agostino; Pasquinucci, Lorella; Cobos Enrique, J.; Alcaro, Stefano; Amata, Emanuele
Structural and molecular insight into Piperazine and Piperidine derivatives as Histamine H3 and Sigma-1 receptor antagonists with promising antinociceptive properties
2022-01-01 Szczepańska, Katarzyna; Podlewska, Sabina; Dichiara, Maria; Gentile, Davide; Patamia, Vincenzo; Rosier, Niklas; Mönnich, Denise; Ruiz Cantero M., Carmen; Karcz, Tadeusz; Łażewska, Dorota; Siwek, Agata; Pockes, Steffen; Cobos J., Enrique; Marrazzo, Agostino; Stark, Holger; Rescifina, Antonio; Bojarski J., Andrzej; Amata, Emanuele; Kieć-Kononowicz, Katarkyna
| Titolo | Data di pubblicazione | Autore(i) | File | Abstract |
|---|---|---|---|---|
| Synthesis and biological investigation of peptidomimetic SARS‐CoV‐2 main protease inhibitors bearing quinoline‐based heterocycles at P3 | 1-gen-2025 | Rossi, Sara; Deidda, Graziano; Fiaschi, Lia; Ibba, Roberta; Pieroni, Mariachiara; Dichiara, Maria; Carullo, Gabriele; Butini, Stefania; Ramunno, Anna; Brogi, Simone; Lolicato, Marco; Arrigoni, Cristina; Cabella, Noemi; Bavagnoli, Laura; Maga, Giovanni; Varasi, Ilenia; Biba, Camilla; Vicenti, Ilaria; Gemma, Sandra; Crespan, Emmanuele; Zazzi, Maurizio; Campiani, Giuseppe | - | |
| Discovery of p-Trifluoromethylbenzohydrazide Derivatives as Potent Antiviral Agents against Monkeypox Virus | 1-gen-2025 | Rossi, Sara; Pozzetti, Luca; Carullo, Gabriele; Dichiara, Maria; Butini, Stefania; Radi, Marco; Ramunno, Anna; Terrosi, Chiara; Barra, Giovanni; Berisio, Rita; Gemma, Sandra; Cusi, Maria Grazia; Campiani, Giuseppe | - | |
| Development of selective sigma-1 receptor ligands with antiallodynic activity: A focus on piperidine and piperazine scaffolds | 1-gen-2025 | Cosentino, Giuseppe; Dichiara, Maria; Ambrosio, Francesca Alessandra; Leotta, Claudia Giovanna; Costa, Giosuè; Procopio, Francesca; Costanzo, Giuliana; Raffa, Alessandro; Artacho-Cordón, Antonia; Ruiz-Cantero, M. Carmen; Pasquinucci, Lorella; Marrazzo, Agostino; Pitari, Giovanni Mario; Cobos, Enrique J.; Alcaro, Stefano; Amata, Emanuele | - | |
| Uncovering a Mutation-Independent Therapeutic Strategy against Inherited Retinal Diseases: Development of Class I HDAC/LSD1 Hybrid Inhibitors | 1-gen-2025 | Carullo, Gabriele; Piano, Ilaria; Salamone, Giulia; Corsi, Francesca; Orsini, Noemi; Dichiara, Maria; Cursaro, Ilaria; Fontana, Anna; Galante, Alessia; Contri, Chiara; Guadagno, Ludovica; Caroli, Jonatan; Mattevi, Andrea; Vincenzi, Fabrizio; Varani, Katia; Brogi, Simone; Gemma, Sandra; Butini, Stefania; Gargini, Claudia; Strettoi, Enrica; Campiani, Giuseppe | - | |
| Unlocking the potential of biostimulants in sustainable agriculture: Effect of wood distillate on the nutritional profiling of apples | 1-gen-2024 | Fedeli, Riccardo; Dichiara, Maria; Carullo, Gabriele; Tudino, Valeria; Gemma, Sandra; Butini, Stefania; Campiani, Giuseppe; Loppi, Stefano | - | |
| Exploring Structural Requirements for Sigma-1 Receptor Linear Ligands: Experimental and Computational Approaches | 1-gen-2024 | Lombardo, Lisa; Mirabile, Salvatore; Gitto, Rosaria; Cosentino, Giuseppe; Alcaro, Stefano; Dichiara, Maria; Marrazzo, Agostino; Amata, Emanuele; Ortuso, Francesco; De Luca, Laura | - | |
| Biostimulants for Sustainable Food Production: Effects of Wood Distillate to Fortify Chickpea Flour for Development of Functional Bakery Products | 1-gen-2024 | Fedeli, Riccardo; Spizzirri, Umile Gianfranco; Aquino, Giovanna; Basilicata, Manuela Giovanna; Pepe, Giacomo; Campiglia, Pietro; Celletti, Silvia; Tudino, Valeria; Dichiara, Maria; Gemma, Sandra; Butini, Stefania; Carullo, Gabriele; Aiello, Francesca; Restuccia, Donatella; Campiani, Giuseppe; Loppi, Stefano | - | |
| Designing drugs optimized for both blood–brain barrier permeation and intra-cerebral partition | 1-gen-2024 | Dichiara, Maria; Cosentino, Giuseppe; Giordano, Giorgia; Pasquinucci, Lorella; Marrazzo, Agostino; Costanzo, Giuliana; Amata, Emanuele | - | |
| Design, Synthesis, and Cytotoxic Assessment of New Haloperidol Analogues as Potential Anticancer Compounds Targeting Sigma Receptors | 1-gen-2024 | Zampieri, Daniele; Romano, Maurizio; Fortuna, Sara; Amata, Emanuele; Dichiara, Maria; Cosentino, Giuseppe; Marrazzo, Agostino; Mamolo, Maria Grazia | - | |
| A novel potent class I HDAC inhibitor reverses the STAT4/p66Shc apoptotic defect in B cells from chronic lymphocytic leukemia patients | 1-gen-2024 | Rossi, Sara; Tatangelo, Vanessa; Dichiara, Maria; Butini, Stefania; Gemma, Sandra; Brogi, Simone; Pasquini, Silvia; Cappello, Martina; Vincenzi, Fabrizio; Varani, Katia; Lopresti, Ludovica; Malchiodi, Margherita; Carrara, Chiara; Gozzetti, Alessandro; Bocchia, Monica; Marotta, Giuseppe; Patrussi, Laura; Carullo, Gabriele; Baldari, Cosima T.; Campiani, Giuseppe | - | |
| Structure–Property Optimization of a Series of Imidazopyridines for Visceral Leishmaniasis | 1-gen-2023 | Dichiara, Maria; Simpson, Quillon J.; Quotadamo, Antonio; Jalani, Hitesh B.; Huang, Anson X.; Millard, Caroline C.; Klug, Dana M.; Tse, Edwin G.; Todd, Matthew H.; Silva, Daniel Gedder; da Silva Emery, Flavio; Carlson, J. Eric; Zheng, Shao-Liang; Vleminckx, Margot; Matheeussen, An; Caljon, Guy; Pollastri, Michael P.; Sjö, Peter; Perry, Benjamin; Ferrins, Lori | - | |
| Open Source Antibiotics: Simple Diarylimidazoles Are Potent against Methicillin-Resistant Staphylococcus aureus | 1-gen-2023 | Klug, Dana M.; Tse, Edwin G.; Silva, Daniel G.; Cao, Yafeng; Charman, Susan A.; Chauhan, Jyoti; Crighton, Elly; Dichiara, Maria; Drake, Chris; Drewry, David; da Silva Emery, Flavio; Ferrins, Lori; Graves, Lee; Hopkins, Emily; Kresina, Thomas A. C.; Lorente-Macías, Álvaro; Perry, Benjamin; Phipps, Richard; Quiroga, Bruno; Quotadamo, Antonio; Sabatino, Giada N.; Sama, Anthony; Schätzlein, Andreas; Simpson, Quillon J.; Steele, Jonathan; Shanu-Wilson, Julia; Sjö, Peter; Stapleton, Paul; Swain, Christopher J.; Vaideanu, Alexandra; Xie, Huanxu; Zuercher, William; Todd, Matthew H. | - | |
| New Insights into the Opioid Analgesic Profile of cis-(−)-N-Normetazocine-derived Ligands | 1-gen-2023 | Costanzo, Giuliana; Turnaturi, Rita; Parenti, Carmela; Spoto, Salvatore; Piana, Silvia; Dichiara, Maria; Zagni, Chiara; Galambos, Anna Rita; Essmat, Nariman; Marrazzo, Agostino; Amata, Emanuele; Al-Khrasani, Mahmoud; Pasquinucci, Lorella | - | |
| Discovery and computational studies of piperidine/piperazine-based compounds endowed with sigma receptor affinity | 1-gen-2023 | De Luca, Laura; Lombardo, Lisa; Mirabile, Salvatore; Marrazzo, Agostino; Dichiara, Maria; Cosentino, Giuseppe; Amata, Emanuele; Gitto, Rosaria | - | |
| Discovery of first novel sigma/HDACi dual-ligands with a potent in vitro antiproliferative activity | 1-gen-2023 | Barbaraci, Carla; di Giacomo, Viviana; Maruca, Annalisa; Patamia, Vincenzo; Rocca, Roberta; Dichiara, Maria; Di Rienzo, Annalisa; Cacciatore, Ivana; Cataldi, Amelia; Balaha, Marwa; Rapino, Monica; Zagni, Chiara; Zampieri, Daniele; Pasquinucci, Lorella; Parenti, Carmela; Amata, Emanuele; Rescifina, Antonio; Alcaro, Stefano; Marrazzo, Agostino | - | |
| Cytotoxicity profiles and neuroprotective properties of the novel ifenprodil analogues as sigma ligands | 1-gen-2023 | Zampieri, Daniele; Calabretti, Antonella; Romano, Maurizio; Fortuna, Sara; Collina, Simona; Amata, Emanuele; Dichiara, Maria; Marrazzo, Agostino; Mamolo Maria, Grazia. | - | |
| Dual Piperidine-Based Histamine H3 and Sigma-1 Receptor Ligands in the Treatment of Nociceptive and Neuropathic Pain | 1-gen-2023 | Szczepańska, Katarzyna; Karcz, Tadeusz; Dichiara, Maria; Mogilski, Szczepan; Kalinowska-Tłuścik, Justyna; Pilarski, Bogusław; Leniak, Arkadiusz; Pietruś, Wojciech; Podlewska, Sabina; Popiołek-Barczyk, Katarzyna; Humphrys, Laura J.; Ruiz-Cantero, M. Carmen; Reiner-Link, David; Leitzbach, Luisa; Łażewska, Dorota; Pockes, Steffen; Górka, Michał; Zmysłowski, Adam; Calmels, Thierry; Cobos, Enrique J.; Marrazzo, Agostino; Stark, Holger; Bojarski, Andrzej J.; Amata, Emanuele; Kieć-Kononowicz, Katarzyna | - | |
| Discovery of AD258 as a Sigma Receptor Ligand with Potent Antiallodynic Activity | 1-gen-2023 | Dichiara, Maria; Ambrosio, Francesca Alessandra; Lee, Sang Min; Ruiz-Cantero, M. Carmen; Lombino, Jessica; Coricello, Adriana; Costa, Giosuè; Shah, Dhara; Costanzo, Giuliana; Pasquinucci, Lorella; Son, Kyung No; Cosentino, Giuseppe; González-Cano, Rafael; Marrazzo, Agostino; Aakalu, Vinay Kumar; Cobos, Enrique J.; Alcaro, Stefano; Amata, Emanuele | - | |
| Synthesis, computational insights, and evaluation of novel sigma receptors ligands | 1-gen-2023 | Dichiara, Maria; Ambrosio, Francesca Alessandra; Barbaraci, Carla; Gonzalez-Cano, Rafael; Costa, Giosuè.; Parenti, Carmela; Marrazzo, Agostino; Pasquinucci, Lorella; Cobos Enrique, J.; Alcaro, Stefano; Amata, Emanuele | - | |
| Structural and molecular insight into Piperazine and Piperidine derivatives as Histamine H3 and Sigma-1 receptor antagonists with promising antinociceptive properties | 1-gen-2022 | Szczepańska, Katarzyna; Podlewska, Sabina; Dichiara, Maria; Gentile, Davide; Patamia, Vincenzo; Rosier, Niklas; Mönnich, Denise; Ruiz Cantero M., Carmen; Karcz, Tadeusz; Łażewska, Dorota; Siwek, Agata; Pockes, Steffen; Cobos J., Enrique; Marrazzo, Agostino; Stark, Holger; Rescifina, Antonio; Bojarski J., Andrzej; Amata, Emanuele; Kieć-Kononowicz, Katarkyna | - |
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