Sfoglia per Autore
Development of Epigenetic Modifiers with Therapeutic Potential in FMS-Related Tyrosine Kinase 3/Internal Tandem Duplication (FLT3/ITD) Acute Myeloid Leukemia and Other Blood Malignancies
2024-01-01 Carullo, Gabriele; Rossi, Sara; Giudice, Valentina; Pezzotta, Alex; Chianese, Ugo; Scala, Pasqualina; Carbone, Sabrina; Fontana, Anna; Panzeca, Giovanna; Pasquini, Silvia; Contri, Chiara; Gemma, Sandra; Ramunno, Anna; Saponara, Simona; Galvani, Francesca; Lodola, Alessio; Mor, Marco; Benedetti, Rosaria; Selleri, Carmine; Varani, Katia; Butini, Stefania; Altucci, Lucia; Vincenzi, Fabrizio; Pistocchi, Anna; Campiani, Giuseppe
Screening of the antioxidant and vasorelaxant activity of wine waste ultrasonic extracts, and HRMS targeted and semi-targeted profiling of glycosylated polyphenols vs free polyphenols
2024-01-01 Medana, Claudio; Spizzirri, Umile Gianfranco; Schiavo, Valentina; Fusi, Fabio; Panti, Alice; Saponara, Simona; Marcolongo, Paola; Affricano, Alex; Asteggiano, Alberto; Aiello, Francesca; Restuccia, Donatella
A novel combinatory treatment against a CDDP-resistant non-small cell lung cancer based on a Ruthenium(II)-cyclopentadienyl compound
2024-01-01 Salaroglio, Iris C.; Stefanova, Denitsa; Teixeira, Ricardo G.; Oliveira, Nuno F. B.; Ahmed, Amer; Fusi, Fabio; Tzankova, Virginia; Yordanov, Yordan; Machuqueiro, Miguel; Saponara, Simona; Valente, Andreia; Riganti, Chiara
The Enigma of Norbormide, a Rattus-Selective Toxicant
2024-01-01 Fusi, Fabio; Saponara, Simona; Brimble, Margaret A.; Rennison, David; Hopkins, Brian; Bova, Sergio
Traceability and authentication in agri-food production: A multivariate approach to the characterization of the Italian food excellence elephant garlic (Allium ampeloprasum L.), a vasoactive nutraceutical
2024-01-01 Carullo, G.; Borghini, F.; Fusi, F.; Saponara, S.; Fontana, A.; Pozzetti, L.; Fedeli, R.; Panti, A.; Gorelli, B.; Aquino, G.; Basilicata, M. G.; Pepe, G.; Campiglia, P.; Biagiotti, S.; Gemma, S.; Butini, S.; Pianezze, S.; Loppi, S.; Cavaglioni, A.; Perini, M.; Campiani, G.
Targeting Relevant HDACs to Support the Survival of Cone Photoreceptors in Inherited Retinal Diseases: Identification of a Potent Pharmacological Tool with In Vitro and In Vivo Efficacy
2024-01-01 Carullo, Gabriele; Orsini, Noemi; Piano, Ilaria; Pozzetti, Luca; Papa, Alessandro; Fontana, Anna; Napoli, Debora; Corsi, Francesca; Marco, Beatrice Di; Galante, Alessia; Marotta, Ludovica; Panzeca, Giovanna; O'Brien, Justine; Sanchez, Alicia Gomez; Doherty, Harry; Mahon, Niamh; Clarke, Leni; Contri, Chiara; Pasquini, Silvia; Gorelli, Beatrice; Saponara, Simona; Valoti, Massimo; Vincenzi, Fabrizio; Varani, Katia; Ramunno, Anna; Brogi, Simone; Butini, Stefania; Gemma, Sandra; Kennedy, Breandán N.; Gargini, Claudia; Strettoi, Enrica; Campiani, Giuseppe
Spirotetrahydroisoquinoline-Based Histone Deacetylase Inhibitors as New Antifibrotic Agents: Biological Evaluation in Human Fibroblasts from Bronchoalveolar Lavages of Idiopathic Pulmonary Fibrosis Patients
2024-01-01 Fontana, Anna; Bergantini, Laura; Carullo, Gabriele; Scalvini, Laura; D'Alessandro, Miriana; Papulino, Chiara; Cameli, Paolo; Gangi, Sara; Vincenzi, Fabrizio; Varani, Katia; Contri, Chiara; Pasquini, Silvia; Pistocchi, Anna; Pezzotta, Alex; Carbone, Sabrina; Saponara, Simona; Gemma, Sandra; Altucci, Lucia; Benedetti, Rosaria; Lodola, Alessio; Mor, Marco; Bargagli, Elena; Butini, Stefania; Campiani, Giuseppe
Wine Lees as Source of Antioxidant Molecules: Green Extraction Procedure and Biological Activity
2023-01-01 Luca Michele, De; Restuccia, Donatella; Gianfranco Spizzirri, Umile; Crupi, Pasquale; Ioele, Giuseppina; Gorelli, Beatrice; Lisa Clodoveo, Maria; Saponara, Simona; Aiello, Francesca
Development of potent and selective FAAH inhibitors with improved drug-like properties as potential tools to treat neuroinflammatory conditions
2023-01-01 Papa, Alessandro; Pasquini, Silvia; Galvani, Francesca; Cammarota, Mariarosaria; Contri, Chiara; Carullo, Gabriele; Gemma, Sandra; Ramunno, Anna; Lamponi, Stefania; Gorelli, Beatrice; Saponara, Simona; Varani, Katia; Mor, Marco; Campiani, Giuseppe; Boscia, Francesca; Vincenzi, Fabrizio; Lodola, Alessio; Butini, Stefania
Artificial intelligence-driven identification of morin analogues acting as CaV1.2 channel blockers: synthesis and biological evaluation
2023-01-01 Carullo, G.; Falbo, F.; Ahmed, A.; Trezza, A.; Gianibbi, B.; Nicolotti, O.; Campiani, G.; Aiello, F.; Saponara, S.; Fusi, F.
Tyrosine kinase inhibitor Si409 has in vitro and in vivo anti-tumor activity against diffuse large B-cell lymphoma
2023-01-01 Rango, E.; Di Maria, S.; Zamperini, C.; Poggialini, F.; Crespan, E.; Perini, C.; Sabetta, S.; Saponara, S.; Fusi, F.; Maga, G.; Angelucci, A.; Gaudio, E.; Berton, F.; Schenone, S.; Botta, L.; Dreassi, E.; Botta, M.
Nutritionally enriched tomatoes (Solanum lycopersicum L.) grown with wood distillate: chemical and biological characterization for quality assessment
2023-01-01 Fedeli, Riccardo; Marotta, Ludovica; Frattaruolo, Luca; Panti, Alice; Carullo, Gabriele; Fusi, Fabio; Saponara, Simona; Gemma, Sandra; Butini, Stefania; Cappello, Anna Rita; Vannini, Andrea; Campiani, Giuseppe; Loppi, Stefano
Vietnamese Dalbergia tonkinensis: A Promising Source of Mono- and Bifunctional Vasodilators
2022-01-01 Cuong, Nguyen Manh; Son, Ninh The; Nhan, Ngu Truong; Fukuyama, Yoshiyasu; Ahmed, Amer; Saponara, Simona; Trezza, Alfonso; Gianibbi, Beatrice; Vigni, Ginevra; Spiga, Ottavia; Fusi, Fabio
Nitrobenzoxadiazole derivatives of the rat selective toxicant norbormide as fluorescent probes for live cell imaging
2022-01-01 Wang, Z. L.; Li, F. F.; Quach, R.; Ferrarese, A.; Forgiarini, A.; Ferrari, M.; D'Amore, C.; Bova, S.; Orso, G.; Fusi, F.; Saponara, S.; Hopkins, B.; Brimble, M. A.; Rennison, D.
Sdox, a H2S releasing anthracycline, with a safer profile than doxorubicin toward vasculature
2022-01-01 Durante, M.; Frosini, M.; Chiaino, E.; Fusi, F.; Gamberucci, A.; Gorelli, B.; Chegaev, K.; Riganti, C.; Saponara, S.
Functional, electrophysiology, and molecular dynamics analysis of quercetin-induced contraction of rat vascular musculature
2022-01-01 Trezza, A.; Spiga, O.; Mugnai, P.; Saponara, S.; Sgaragli, G.; Fusi, F.
Off-label use of hydroxychloroquine in COVID-19: analysis of reports of suspected adverse reactions from the Italian National Network of Pharmacovigilance
2022-01-01 Fallani, E.; Cevenini, F.; Lazzerini, P. E.; Verdini, A.; Saponara, S.
A Comprehensive Evaluation of Sdox, a Promising H2S-Releasing Doxorubicin for the Treatment of Chemoresistant Tumors
2022-01-01 Alov, Petko; Al Sharif, Merilin; Aluani, Denitsa; Chegaev, Konstantin; Dinic, Jelena; Divac Rankov, Aleksandra; Fernandes, Miguel X; Fusi, Fabio; García-Sosa, Alfonso T; Juvonen, Risto; Kondeva-Burdina, Magdalena; Padrón, José M; Pajeva, Ilza; Pencheva, Tania; Puerta, Adrián; Raunio, Hannu; Riganti, Chiara; Tsakovska, Ivanka; Tzankova, Virginia; Yordanov, Yordan; Saponara, Simona
Novel Labdane Diterpenes-Based Synthetic Derivatives: Identification of a Bifunctional Vasodilator That Inhibits CaV1.2 and Stimulates KCa1.1 Channels
2022-01-01 Carullo, Gabriele; Saponara, Simona; Ahmed, Amer; Gorelli, Beatrice; Mazzotta, Sarah; Trezza, Alfonso; Gianibbi, Beatrice; Campiani, Giuseppe; Fusi, Fabio; Aiello, Francesca
Azetidin-2-one-based small molecules as dual hHDAC6/HDAC8 inhibitors: Investigation of their mechanism of action and impact of dual inhibition profile on cell viability
2022-01-01 Federico, S.; Khan, T.; Fontana, A.; Brogi, S.; Benedetti, R.; Sarno, F.; Carullo, G.; Pezzotta, A.; Saraswati, A. P.; Passaro, E.; Pozzetti, L.; Papa, A.; Relitti, N.; Gemma, S.; Butini, S.; Pistocchi, A.; Ramunno, A.; Vincenzi, F.; Varani, K.; Tatangelo, V.; Patrussi, L.; Baldari, C. T.; Saponara, S.; Gorelli, B.; Lamponi, S.; Valoti, M.; Saccoccia, F.; Giannaccari, M.; Ruberti, G.; Herp, D.; Jung, M.; Altucci, L.; Campiani, G.
Titolo | Data di pubblicazione | Autore(i) | File | Abstract |
---|---|---|---|---|
Development of Epigenetic Modifiers with Therapeutic Potential in FMS-Related Tyrosine Kinase 3/Internal Tandem Duplication (FLT3/ITD) Acute Myeloid Leukemia and Other Blood Malignancies | 1-gen-2024 | Carullo, Gabriele; Rossi, Sara; Giudice, Valentina; Pezzotta, Alex; Chianese, Ugo; Scala, Pasqualina; Carbone, Sabrina; Fontana, Anna; Panzeca, Giovanna; Pasquini, Silvia; Contri, Chiara; Gemma, Sandra; Ramunno, Anna; Saponara, Simona; Galvani, Francesca; Lodola, Alessio; Mor, Marco; Benedetti, Rosaria; Selleri, Carmine; Varani, Katia; Butini, Stefania; Altucci, Lucia; Vincenzi, Fabrizio; Pistocchi, Anna; Campiani, Giuseppe | - | |
Screening of the antioxidant and vasorelaxant activity of wine waste ultrasonic extracts, and HRMS targeted and semi-targeted profiling of glycosylated polyphenols vs free polyphenols | 1-gen-2024 | Medana, Claudio; Spizzirri, Umile Gianfranco; Schiavo, Valentina; Fusi, Fabio; Panti, Alice; Saponara, Simona; Marcolongo, Paola; Affricano, Alex; Asteggiano, Alberto; Aiello, Francesca; Restuccia, Donatella | - | |
A novel combinatory treatment against a CDDP-resistant non-small cell lung cancer based on a Ruthenium(II)-cyclopentadienyl compound | 1-gen-2024 | Salaroglio, Iris C.; Stefanova, Denitsa; Teixeira, Ricardo G.; Oliveira, Nuno F. B.; Ahmed, Amer; Fusi, Fabio; Tzankova, Virginia; Yordanov, Yordan; Machuqueiro, Miguel; Saponara, Simona; Valente, Andreia; Riganti, Chiara | - | |
The Enigma of Norbormide, a Rattus-Selective Toxicant | 1-gen-2024 | Fusi, Fabio; Saponara, Simona; Brimble, Margaret A.; Rennison, David; Hopkins, Brian; Bova, Sergio | - | |
Traceability and authentication in agri-food production: A multivariate approach to the characterization of the Italian food excellence elephant garlic (Allium ampeloprasum L.), a vasoactive nutraceutical | 1-gen-2024 | Carullo, G.; Borghini, F.; Fusi, F.; Saponara, S.; Fontana, A.; Pozzetti, L.; Fedeli, R.; Panti, A.; Gorelli, B.; Aquino, G.; Basilicata, M. G.; Pepe, G.; Campiglia, P.; Biagiotti, S.; Gemma, S.; Butini, S.; Pianezze, S.; Loppi, S.; Cavaglioni, A.; Perini, M.; Campiani, G. | - | |
Targeting Relevant HDACs to Support the Survival of Cone Photoreceptors in Inherited Retinal Diseases: Identification of a Potent Pharmacological Tool with In Vitro and In Vivo Efficacy | 1-gen-2024 | Carullo, Gabriele; Orsini, Noemi; Piano, Ilaria; Pozzetti, Luca; Papa, Alessandro; Fontana, Anna; Napoli, Debora; Corsi, Francesca; Marco, Beatrice Di; Galante, Alessia; Marotta, Ludovica; Panzeca, Giovanna; O'Brien, Justine; Sanchez, Alicia Gomez; Doherty, Harry; Mahon, Niamh; Clarke, Leni; Contri, Chiara; Pasquini, Silvia; Gorelli, Beatrice; Saponara, Simona; Valoti, Massimo; Vincenzi, Fabrizio; Varani, Katia; Ramunno, Anna; Brogi, Simone; Butini, Stefania; Gemma, Sandra; Kennedy, Breandán N.; Gargini, Claudia; Strettoi, Enrica; Campiani, Giuseppe | - | |
Spirotetrahydroisoquinoline-Based Histone Deacetylase Inhibitors as New Antifibrotic Agents: Biological Evaluation in Human Fibroblasts from Bronchoalveolar Lavages of Idiopathic Pulmonary Fibrosis Patients | 1-gen-2024 | Fontana, Anna; Bergantini, Laura; Carullo, Gabriele; Scalvini, Laura; D'Alessandro, Miriana; Papulino, Chiara; Cameli, Paolo; Gangi, Sara; Vincenzi, Fabrizio; Varani, Katia; Contri, Chiara; Pasquini, Silvia; Pistocchi, Anna; Pezzotta, Alex; Carbone, Sabrina; Saponara, Simona; Gemma, Sandra; Altucci, Lucia; Benedetti, Rosaria; Lodola, Alessio; Mor, Marco; Bargagli, Elena; Butini, Stefania; Campiani, Giuseppe | - | |
Wine Lees as Source of Antioxidant Molecules: Green Extraction Procedure and Biological Activity | 1-gen-2023 | Luca Michele, De; Restuccia, Donatella; Gianfranco Spizzirri, Umile; Crupi, Pasquale; Ioele, Giuseppina; Gorelli, Beatrice; Lisa Clodoveo, Maria; Saponara, Simona; Aiello, Francesca | - | |
Development of potent and selective FAAH inhibitors with improved drug-like properties as potential tools to treat neuroinflammatory conditions | 1-gen-2023 | Papa, Alessandro; Pasquini, Silvia; Galvani, Francesca; Cammarota, Mariarosaria; Contri, Chiara; Carullo, Gabriele; Gemma, Sandra; Ramunno, Anna; Lamponi, Stefania; Gorelli, Beatrice; Saponara, Simona; Varani, Katia; Mor, Marco; Campiani, Giuseppe; Boscia, Francesca; Vincenzi, Fabrizio; Lodola, Alessio; Butini, Stefania | - | |
Artificial intelligence-driven identification of morin analogues acting as CaV1.2 channel blockers: synthesis and biological evaluation | 1-gen-2023 | Carullo, G.; Falbo, F.; Ahmed, A.; Trezza, A.; Gianibbi, B.; Nicolotti, O.; Campiani, G.; Aiello, F.; Saponara, S.; Fusi, F. | - | |
Tyrosine kinase inhibitor Si409 has in vitro and in vivo anti-tumor activity against diffuse large B-cell lymphoma | 1-gen-2023 | Rango, E.; Di Maria, S.; Zamperini, C.; Poggialini, F.; Crespan, E.; Perini, C.; Sabetta, S.; Saponara, S.; Fusi, F.; Maga, G.; Angelucci, A.; Gaudio, E.; Berton, F.; Schenone, S.; Botta, L.; Dreassi, E.; Botta, M. | - | |
Nutritionally enriched tomatoes (Solanum lycopersicum L.) grown with wood distillate: chemical and biological characterization for quality assessment | 1-gen-2023 | Fedeli, Riccardo; Marotta, Ludovica; Frattaruolo, Luca; Panti, Alice; Carullo, Gabriele; Fusi, Fabio; Saponara, Simona; Gemma, Sandra; Butini, Stefania; Cappello, Anna Rita; Vannini, Andrea; Campiani, Giuseppe; Loppi, Stefano | - | |
Vietnamese Dalbergia tonkinensis: A Promising Source of Mono- and Bifunctional Vasodilators | 1-gen-2022 | Cuong, Nguyen Manh; Son, Ninh The; Nhan, Ngu Truong; Fukuyama, Yoshiyasu; Ahmed, Amer; Saponara, Simona; Trezza, Alfonso; Gianibbi, Beatrice; Vigni, Ginevra; Spiga, Ottavia; Fusi, Fabio | - | |
Nitrobenzoxadiazole derivatives of the rat selective toxicant norbormide as fluorescent probes for live cell imaging | 1-gen-2022 | Wang, Z. L.; Li, F. F.; Quach, R.; Ferrarese, A.; Forgiarini, A.; Ferrari, M.; D'Amore, C.; Bova, S.; Orso, G.; Fusi, F.; Saponara, S.; Hopkins, B.; Brimble, M. A.; Rennison, D. | - | |
Sdox, a H2S releasing anthracycline, with a safer profile than doxorubicin toward vasculature | 1-gen-2022 | Durante, M.; Frosini, M.; Chiaino, E.; Fusi, F.; Gamberucci, A.; Gorelli, B.; Chegaev, K.; Riganti, C.; Saponara, S. | - | |
Functional, electrophysiology, and molecular dynamics analysis of quercetin-induced contraction of rat vascular musculature | 1-gen-2022 | Trezza, A.; Spiga, O.; Mugnai, P.; Saponara, S.; Sgaragli, G.; Fusi, F. | - | |
Off-label use of hydroxychloroquine in COVID-19: analysis of reports of suspected adverse reactions from the Italian National Network of Pharmacovigilance | 1-gen-2022 | Fallani, E.; Cevenini, F.; Lazzerini, P. E.; Verdini, A.; Saponara, S. | - | |
A Comprehensive Evaluation of Sdox, a Promising H2S-Releasing Doxorubicin for the Treatment of Chemoresistant Tumors | 1-gen-2022 | Alov, Petko; Al Sharif, Merilin; Aluani, Denitsa; Chegaev, Konstantin; Dinic, Jelena; Divac Rankov, Aleksandra; Fernandes, Miguel X; Fusi, Fabio; García-Sosa, Alfonso T; Juvonen, Risto; Kondeva-Burdina, Magdalena; Padrón, José M; Pajeva, Ilza; Pencheva, Tania; Puerta, Adrián; Raunio, Hannu; Riganti, Chiara; Tsakovska, Ivanka; Tzankova, Virginia; Yordanov, Yordan; Saponara, Simona | - | |
Novel Labdane Diterpenes-Based Synthetic Derivatives: Identification of a Bifunctional Vasodilator That Inhibits CaV1.2 and Stimulates KCa1.1 Channels | 1-gen-2022 | Carullo, Gabriele; Saponara, Simona; Ahmed, Amer; Gorelli, Beatrice; Mazzotta, Sarah; Trezza, Alfonso; Gianibbi, Beatrice; Campiani, Giuseppe; Fusi, Fabio; Aiello, Francesca | - | |
Azetidin-2-one-based small molecules as dual hHDAC6/HDAC8 inhibitors: Investigation of their mechanism of action and impact of dual inhibition profile on cell viability | 1-gen-2022 | Federico, S.; Khan, T.; Fontana, A.; Brogi, S.; Benedetti, R.; Sarno, F.; Carullo, G.; Pezzotta, A.; Saraswati, A. P.; Passaro, E.; Pozzetti, L.; Papa, A.; Relitti, N.; Gemma, S.; Butini, S.; Pistocchi, A.; Ramunno, A.; Vincenzi, F.; Varani, K.; Tatangelo, V.; Patrussi, L.; Baldari, C. T.; Saponara, S.; Gorelli, B.; Lamponi, S.; Valoti, M.; Saccoccia, F.; Giannaccari, M.; Ruberti, G.; Herp, D.; Jung, M.; Altucci, L.; Campiani, G. | - |
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