Sfoglia per Autore
Targeting class I histone deacetylases triggers antitumor responses in colorectal cancer in vitro and in vivo
2026-01-01 Carullo, Gabriele; Falbo, Federica; Tudino, Valeria; Song, Jiazhao; Fava, Marianna; Fontana, Anna; Koch, Adrian; Heiß, Anita; Erlenbach-Wuensch, Katharina; Panzeca, Giovanna; Brogi, Simone; Bichicchi, Alessia; Saponara, Simona; Fusi, Fabio; Vincenzi, Fabrizio; Varani, Katia; Cappello, Martina; Pasquini, Silvia; Ramunno, Anna; Pepe, Giacomo; Butini, Stefania; Aiello, Francesca; Gemma, Sandra; Schneider-Stock, Regine; Campiani, Giuseppe
The insulin-releasing agent quercetin-3-oleate stimulates CaV1.2 channels similarly to quercetin, though with a reduced vasorelaxant activity
2025-01-01 Fusi, Fabio; Saponara, Simona; Carullo, Gabriele; Panti, Alice; Bichicchi, Alessia; Pifferi, Alice; Gianibbi, Beatrice; Spiga, Ottavia; Falbo, Federica; Spizzirri, Umile Gianfranco; Campiani, Giuseppe; Aiello, Francesca
New Vanillyl-capped HDAC inhibitors exhibit anti-tumor efficacy in neuroblastoma and glioblastoma cells
2025-01-01 Cursaro, Ilaria; Frattaruolo, Luca; Scalvini, Laura; Contri, Chiara; Bichicchi, Alessia; Tardiolo, Nicola; Tudino, Valeria; Rossi, Sara; Manti, Eugenia Nicol; Cappello, Martina; Papulino, Chiara; Maellaro, Emilia; Marcolongo, Paola; Benedetti, Rosaria; Altucci, Lucia; Varani, Katia; Mor, Marco; Frosini, Maria; Vincenzi, Fabrizio; Cappello, Anna Rita; Lodola, Alessio; Saponara, Simona; Butini, Stefania; Carullo, Gabriele; Gemma, Sandra; Campiani, Giuseppe
New dimension of ciprofloxacin hybrids: Synthesis, characterization and anticancer evaluation of newly C3-modified ciprofloxacin derivatives
2025-01-01 Koszelewski, Dominik; Ostaszewski, Ryszard; Zaremba, Arleta; Riganti, Chiara; Kopecka, Joanna; Contino, Marialessandra; Pajeva, Ilza; Tsakovska, Ivanka; Saponara, Simona; Ahmed, Amer; Stefanova, Denitsa; Tzankova, Virginia; Yordanov, Yordan
Spirotetrahydroisoquinoline-Based Histone Deacetylase Inhibitors as New Antifibrotic Agents: Biological Evaluation in Human Fibroblasts from Bronchoalveolar Lavages of Idiopathic Pulmonary Fibrosis Patients
2025-01-01 Fontana, Anna; Bergantini, Laura; Carullo, Gabriele; Scalvini, Laura; D'Alessandro, Miriana; Papulino, Chiara; Cameli, Paolo; Gangi, Sara; Vincenzi, Fabrizio; Varani, Katia; Contri, Chiara; Pasquini, Silvia; Pistocchi, Anna; Pezzotta, Alex; Carbone, Sabrina; Saponara, Simona; Gemma, Sandra; Altucci, Lucia; Benedetti, Rosaria; Lodola, Alessio; Mor, Marco; Bargagli, Elena; Butini, Stefania; Campiani, Giuseppe
Screening of the antioxidant and vasorelaxant activity of wine waste ultrasonic extracts, and HRMS targeted and semi-targeted profiling of glycosylated polyphenols vs free polyphenols
2024-01-01 Medana, Claudio; Spizzirri, Umile Gianfranco; Schiavo, Valentina; Fusi, Fabio; Panti, Alice; Saponara, Simona; Marcolongo, Paola; Affricano, Alex; Asteggiano, Alberto; Aiello, Francesca; Restuccia, Donatella
Targeting Relevant HDACs to Support the Survival of Cone Photoreceptors in Inherited Retinal Diseases: Identification of a Potent Pharmacological Tool with In Vitro and In Vivo Efficacy
2024-01-01 Carullo, Gabriele; Orsini, Noemi; Piano, Ilaria; Pozzetti, Luca; Papa, Alessandro; Fontana, Anna; Napoli, Debora; Corsi, Francesca; Marco, Beatrice Di; Galante, Alessia; Marotta, Ludovica; Panzeca, Giovanna; O'Brien, Justine; Sanchez, Alicia Gomez; Doherty, Harry; Mahon, Niamh; Clarke, Leni; Contri, Chiara; Pasquini, Silvia; Gorelli, Beatrice; Saponara, Simona; Valoti, Massimo; Vincenzi, Fabrizio; Varani, Katia; Ramunno, Anna; Brogi, Simone; Butini, Stefania; Gemma, Sandra; Kennedy, Breandán N.; Gargini, Claudia; Strettoi, Enrica; Campiani, Giuseppe
The Enigma of Norbormide, a Rattus-Selective Toxicant
2024-01-01 Fusi, Fabio; Saponara, Simona; Brimble, Margaret A.; Rennison, David; Hopkins, Brian; Bova, Sergio
Development of Epigenetic Modifiers with Therapeutic Potential in FMS-Related Tyrosine Kinase 3/Internal Tandem Duplication (FLT3/ITD) Acute Myeloid Leukemia and Other Blood Malignancies
2024-01-01 Carullo, Gabriele; Rossi, Sara; Giudice, Valentina; Pezzotta, Alex; Chianese, Ugo; Scala, Pasqualina; Carbone, Sabrina; Fontana, Anna; Panzeca, Giovanna; Pasquini, Silvia; Contri, Chiara; Gemma, Sandra; Ramunno, Anna; Saponara, Simona; Galvani, Francesca; Lodola, Alessio; Mor, Marco; Benedetti, Rosaria; Selleri, Carmine; Varani, Katia; Butini, Stefania; Altucci, Lucia; Vincenzi, Fabrizio; Pistocchi, Anna; Campiani, Giuseppe
A novel combinatory treatment against a CDDP-resistant non-small cell lung cancer based on a Ruthenium(II)-cyclopentadienyl compound
2024-01-01 Salaroglio, Iris C.; Stefanova, Denitsa; Teixeira, Ricardo G.; Oliveira, Nuno F. B.; Ahmed, Amer; Fusi, Fabio; Tzankova, Virginia; Yordanov, Yordan; Machuqueiro, Miguel; Saponara, Simona; Valente, Andreia; Riganti, Chiara
Traceability and authentication in agri-food production: A multivariate approach to the characterization of the Italian food excellence elephant garlic (Allium ampeloprasum L.), a vasoactive nutraceutical
2024-01-01 Carullo, G.; Borghini, F.; Fusi, F.; Saponara, S.; Fontana, A.; Pozzetti, L.; Fedeli, R.; Panti, A.; Gorelli, B.; Aquino, G.; Basilicata, M. G.; Pepe, G.; Campiglia, P.; Biagiotti, S.; Gemma, S.; Butini, S.; Pianezze, S.; Loppi, S.; Cavaglioni, A.; Perini, M.; Campiani, G.
PERTRAS observational study: clinical and economic analysis of trastuzumab plus neoadjuvant pertuzumab in women with HER-2 positive breast cancer. [Studio osservazionale PERTRAS: analisi clinica ed economica di trastuzumab più pertuzumab neoadiuvante in donne con carcinoma mammario HER-2 positivo]
2024-01-01 Ciacci, Benedetta; Gianluca Lacerenza, Leonardo; Bengala, Carmelo; Bindi, Michele; Petrucci, Elisa; Barbaro, Sara; Falcone, Emilia; Tricca, Marcella; Meini, Barbara; Messuti, Luciana; Pastina, Ilaria; Sposato, Bruno; Serafini, Andrea; Saponara, Simona
Tyrosine kinase inhibitor Si409 has in vitro and in vivo anti-tumor activity against diffuse large B-cell lymphoma
2023-01-01 Rango, E.; Di Maria, S.; Zamperini, C.; Poggialini, F.; Crespan, E.; Perini, C.; Sabetta, S.; Saponara, S.; Fusi, F.; Maga, G.; Angelucci, A.; Gaudio, E.; Berton, F.; Schenone, S.; Botta, L.; Dreassi, E.; Botta, M.
Artificial intelligence-driven identification of morin analogues acting as CaV1.2 channel blockers: synthesis and biological evaluation
2023-01-01 Carullo, G.; Falbo, F.; Ahmed, A.; Trezza, A.; Gianibbi, B.; Nicolotti, O.; Campiani, G.; Aiello, F.; Saponara, S.; Fusi, F.
Wine Lees as Source of Antioxidant Molecules: Green Extraction Procedure and Biological Activity
2023-01-01 De Luca, Michele; Restuccia, Donatella; Spizzirri, Umile Gianfranco; Crupi, Pasquale; Ioele, Giuseppina; Gorelli, Beatrice; Clodoveo, Maria Lisa; Saponara, Simona; Aiello, Francesca
Nutritionally enriched tomatoes (Solanum lycopersicum L.) grown with wood distillate: chemical and biological characterization for quality assessment
2023-01-01 Fedeli, Riccardo; Marotta, Ludovica; Frattaruolo, Luca; Panti, Alice; Carullo, Gabriele; Fusi, Fabio; Saponara, Simona; Gemma, Sandra; Butini, Stefania; Cappello, Anna Rita; Vannini, Andrea; Campiani, Giuseppe; Loppi, Stefano
Development of potent and selective FAAH inhibitors with improved drug-like properties as potential tools to treat neuroinflammatory conditions
2023-01-01 Papa, Alessandro; Pasquini, Silvia; Galvani, Francesca; Cammarota, Mariarosaria; Contri, Chiara; Carullo, Gabriele; Gemma, Sandra; Ramunno, Anna; Lamponi, Stefania; Gorelli, Beatrice; Saponara, Simona; Varani, Katia; Mor, Marco; Campiani, Giuseppe; Boscia, Francesca; Vincenzi, Fabrizio; Lodola, Alessio; Butini, Stefania
Vietnamese Dalbergia tonkinensis: A Promising Source of Mono- and Bifunctional Vasodilators
2022-01-01 Cuong, Nguyen Manh; Son, Ninh The; Nhan, Ngu Truong; Fukuyama, Yoshiyasu; Ahmed, Amer; Saponara, Simona; Trezza, Alfonso; Gianibbi, Beatrice; Vigni, Ginevra; Spiga, Ottavia; Fusi, Fabio
Sdox, a H2S releasing anthracycline, with a safer profile than doxorubicin toward vasculature
2022-01-01 Durante, M.; Frosini, M.; Chiaino, E.; Fusi, F.; Gamberucci, A.; Gorelli, B.; Chegaev, K.; Riganti, C.; Saponara, S.
Functional, electrophysiology, and molecular dynamics analysis of quercetin-induced contraction of rat vascular musculature
2022-01-01 Trezza, A.; Spiga, O.; Mugnai, P.; Saponara, S.; Sgaragli, G.; Fusi, F.
| Titolo | Data di pubblicazione | Autore(i) | File | Abstract |
|---|---|---|---|---|
| Targeting class I histone deacetylases triggers antitumor responses in colorectal cancer in vitro and in vivo | 1-gen-2026 | Carullo, Gabriele; Falbo, Federica; Tudino, Valeria; Song, Jiazhao; Fava, Marianna; Fontana, Anna; Koch, Adrian; Heiß, Anita; Erlenbach-Wuensch, Katharina; Panzeca, Giovanna; Brogi, Simone; Bichicchi, Alessia; Saponara, Simona; Fusi, Fabio; Vincenzi, Fabrizio; Varani, Katia; Cappello, Martina; Pasquini, Silvia; Ramunno, Anna; Pepe, Giacomo; Butini, Stefania; Aiello, Francesca; Gemma, Sandra; Schneider-Stock, Regine; Campiani, Giuseppe | - | |
| The insulin-releasing agent quercetin-3-oleate stimulates CaV1.2 channels similarly to quercetin, though with a reduced vasorelaxant activity | 1-gen-2025 | Fusi, Fabio; Saponara, Simona; Carullo, Gabriele; Panti, Alice; Bichicchi, Alessia; Pifferi, Alice; Gianibbi, Beatrice; Spiga, Ottavia; Falbo, Federica; Spizzirri, Umile Gianfranco; Campiani, Giuseppe; Aiello, Francesca | - | |
| New Vanillyl-capped HDAC inhibitors exhibit anti-tumor efficacy in neuroblastoma and glioblastoma cells | 1-gen-2025 | Cursaro, Ilaria; Frattaruolo, Luca; Scalvini, Laura; Contri, Chiara; Bichicchi, Alessia; Tardiolo, Nicola; Tudino, Valeria; Rossi, Sara; Manti, Eugenia Nicol; Cappello, Martina; Papulino, Chiara; Maellaro, Emilia; Marcolongo, Paola; Benedetti, Rosaria; Altucci, Lucia; Varani, Katia; Mor, Marco; Frosini, Maria; Vincenzi, Fabrizio; Cappello, Anna Rita; Lodola, Alessio; Saponara, Simona; Butini, Stefania; Carullo, Gabriele; Gemma, Sandra; Campiani, Giuseppe | - | |
| New dimension of ciprofloxacin hybrids: Synthesis, characterization and anticancer evaluation of newly C3-modified ciprofloxacin derivatives | 1-gen-2025 | Koszelewski, Dominik; Ostaszewski, Ryszard; Zaremba, Arleta; Riganti, Chiara; Kopecka, Joanna; Contino, Marialessandra; Pajeva, Ilza; Tsakovska, Ivanka; Saponara, Simona; Ahmed, Amer; Stefanova, Denitsa; Tzankova, Virginia; Yordanov, Yordan | - | |
| Spirotetrahydroisoquinoline-Based Histone Deacetylase Inhibitors as New Antifibrotic Agents: Biological Evaluation in Human Fibroblasts from Bronchoalveolar Lavages of Idiopathic Pulmonary Fibrosis Patients | 1-gen-2025 | Fontana, Anna; Bergantini, Laura; Carullo, Gabriele; Scalvini, Laura; D'Alessandro, Miriana; Papulino, Chiara; Cameli, Paolo; Gangi, Sara; Vincenzi, Fabrizio; Varani, Katia; Contri, Chiara; Pasquini, Silvia; Pistocchi, Anna; Pezzotta, Alex; Carbone, Sabrina; Saponara, Simona; Gemma, Sandra; Altucci, Lucia; Benedetti, Rosaria; Lodola, Alessio; Mor, Marco; Bargagli, Elena; Butini, Stefania; Campiani, Giuseppe | - | |
| Screening of the antioxidant and vasorelaxant activity of wine waste ultrasonic extracts, and HRMS targeted and semi-targeted profiling of glycosylated polyphenols vs free polyphenols | 1-gen-2024 | Medana, Claudio; Spizzirri, Umile Gianfranco; Schiavo, Valentina; Fusi, Fabio; Panti, Alice; Saponara, Simona; Marcolongo, Paola; Affricano, Alex; Asteggiano, Alberto; Aiello, Francesca; Restuccia, Donatella | - | |
| Targeting Relevant HDACs to Support the Survival of Cone Photoreceptors in Inherited Retinal Diseases: Identification of a Potent Pharmacological Tool with In Vitro and In Vivo Efficacy | 1-gen-2024 | Carullo, Gabriele; Orsini, Noemi; Piano, Ilaria; Pozzetti, Luca; Papa, Alessandro; Fontana, Anna; Napoli, Debora; Corsi, Francesca; Marco, Beatrice Di; Galante, Alessia; Marotta, Ludovica; Panzeca, Giovanna; O'Brien, Justine; Sanchez, Alicia Gomez; Doherty, Harry; Mahon, Niamh; Clarke, Leni; Contri, Chiara; Pasquini, Silvia; Gorelli, Beatrice; Saponara, Simona; Valoti, Massimo; Vincenzi, Fabrizio; Varani, Katia; Ramunno, Anna; Brogi, Simone; Butini, Stefania; Gemma, Sandra; Kennedy, Breandán N.; Gargini, Claudia; Strettoi, Enrica; Campiani, Giuseppe | - | |
| The Enigma of Norbormide, a Rattus-Selective Toxicant | 1-gen-2024 | Fusi, Fabio; Saponara, Simona; Brimble, Margaret A.; Rennison, David; Hopkins, Brian; Bova, Sergio | - | |
| Development of Epigenetic Modifiers with Therapeutic Potential in FMS-Related Tyrosine Kinase 3/Internal Tandem Duplication (FLT3/ITD) Acute Myeloid Leukemia and Other Blood Malignancies | 1-gen-2024 | Carullo, Gabriele; Rossi, Sara; Giudice, Valentina; Pezzotta, Alex; Chianese, Ugo; Scala, Pasqualina; Carbone, Sabrina; Fontana, Anna; Panzeca, Giovanna; Pasquini, Silvia; Contri, Chiara; Gemma, Sandra; Ramunno, Anna; Saponara, Simona; Galvani, Francesca; Lodola, Alessio; Mor, Marco; Benedetti, Rosaria; Selleri, Carmine; Varani, Katia; Butini, Stefania; Altucci, Lucia; Vincenzi, Fabrizio; Pistocchi, Anna; Campiani, Giuseppe | - | |
| A novel combinatory treatment against a CDDP-resistant non-small cell lung cancer based on a Ruthenium(II)-cyclopentadienyl compound | 1-gen-2024 | Salaroglio, Iris C.; Stefanova, Denitsa; Teixeira, Ricardo G.; Oliveira, Nuno F. B.; Ahmed, Amer; Fusi, Fabio; Tzankova, Virginia; Yordanov, Yordan; Machuqueiro, Miguel; Saponara, Simona; Valente, Andreia; Riganti, Chiara | - | |
| Traceability and authentication in agri-food production: A multivariate approach to the characterization of the Italian food excellence elephant garlic (Allium ampeloprasum L.), a vasoactive nutraceutical | 1-gen-2024 | Carullo, G.; Borghini, F.; Fusi, F.; Saponara, S.; Fontana, A.; Pozzetti, L.; Fedeli, R.; Panti, A.; Gorelli, B.; Aquino, G.; Basilicata, M. G.; Pepe, G.; Campiglia, P.; Biagiotti, S.; Gemma, S.; Butini, S.; Pianezze, S.; Loppi, S.; Cavaglioni, A.; Perini, M.; Campiani, G. | - | |
| PERTRAS observational study: clinical and economic analysis of trastuzumab plus neoadjuvant pertuzumab in women with HER-2 positive breast cancer. [Studio osservazionale PERTRAS: analisi clinica ed economica di trastuzumab più pertuzumab neoadiuvante in donne con carcinoma mammario HER-2 positivo] | 1-gen-2024 | Ciacci, Benedetta; Gianluca Lacerenza, Leonardo; Bengala, Carmelo; Bindi, Michele; Petrucci, Elisa; Barbaro, Sara; Falcone, Emilia; Tricca, Marcella; Meini, Barbara; Messuti, Luciana; Pastina, Ilaria; Sposato, Bruno; Serafini, Andrea; Saponara, Simona | - | |
| Tyrosine kinase inhibitor Si409 has in vitro and in vivo anti-tumor activity against diffuse large B-cell lymphoma | 1-gen-2023 | Rango, E.; Di Maria, S.; Zamperini, C.; Poggialini, F.; Crespan, E.; Perini, C.; Sabetta, S.; Saponara, S.; Fusi, F.; Maga, G.; Angelucci, A.; Gaudio, E.; Berton, F.; Schenone, S.; Botta, L.; Dreassi, E.; Botta, M. | - | |
| Artificial intelligence-driven identification of morin analogues acting as CaV1.2 channel blockers: synthesis and biological evaluation | 1-gen-2023 | Carullo, G.; Falbo, F.; Ahmed, A.; Trezza, A.; Gianibbi, B.; Nicolotti, O.; Campiani, G.; Aiello, F.; Saponara, S.; Fusi, F. | - | |
| Wine Lees as Source of Antioxidant Molecules: Green Extraction Procedure and Biological Activity | 1-gen-2023 | De Luca, Michele; Restuccia, Donatella; Spizzirri, Umile Gianfranco; Crupi, Pasquale; Ioele, Giuseppina; Gorelli, Beatrice; Clodoveo, Maria Lisa; Saponara, Simona; Aiello, Francesca | - | |
| Nutritionally enriched tomatoes (Solanum lycopersicum L.) grown with wood distillate: chemical and biological characterization for quality assessment | 1-gen-2023 | Fedeli, Riccardo; Marotta, Ludovica; Frattaruolo, Luca; Panti, Alice; Carullo, Gabriele; Fusi, Fabio; Saponara, Simona; Gemma, Sandra; Butini, Stefania; Cappello, Anna Rita; Vannini, Andrea; Campiani, Giuseppe; Loppi, Stefano | - | |
| Development of potent and selective FAAH inhibitors with improved drug-like properties as potential tools to treat neuroinflammatory conditions | 1-gen-2023 | Papa, Alessandro; Pasquini, Silvia; Galvani, Francesca; Cammarota, Mariarosaria; Contri, Chiara; Carullo, Gabriele; Gemma, Sandra; Ramunno, Anna; Lamponi, Stefania; Gorelli, Beatrice; Saponara, Simona; Varani, Katia; Mor, Marco; Campiani, Giuseppe; Boscia, Francesca; Vincenzi, Fabrizio; Lodola, Alessio; Butini, Stefania | - | |
| Vietnamese Dalbergia tonkinensis: A Promising Source of Mono- and Bifunctional Vasodilators | 1-gen-2022 | Cuong, Nguyen Manh; Son, Ninh The; Nhan, Ngu Truong; Fukuyama, Yoshiyasu; Ahmed, Amer; Saponara, Simona; Trezza, Alfonso; Gianibbi, Beatrice; Vigni, Ginevra; Spiga, Ottavia; Fusi, Fabio | - | |
| Sdox, a H2S releasing anthracycline, with a safer profile than doxorubicin toward vasculature | 1-gen-2022 | Durante, M.; Frosini, M.; Chiaino, E.; Fusi, F.; Gamberucci, A.; Gorelli, B.; Chegaev, K.; Riganti, C.; Saponara, S. | - | |
| Functional, electrophysiology, and molecular dynamics analysis of quercetin-induced contraction of rat vascular musculature | 1-gen-2022 | Trezza, A.; Spiga, O.; Mugnai, P.; Saponara, S.; Sgaragli, G.; Fusi, F. | - |
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