Sfoglia per Autore
Dissecting the Interaction Domains of SARS-CoV-2 Nucleocapsid Protein and Human RNA Helicase DDX3X and Search for Potential Inhibitors
2026-01-01 Lodola, Camilla; Pallotta, Maria Michela; Manetti, Fabrizio; Governa, Paolo; Crespan, Emmanuele; Maga, Giovanni; Secchi, Massimiliano
Sulfur Oxidation Unlocks Ene‐Reductase Catalysis for Stereoselective C(sp3)–S(VI) Bond Formation in β‐Sulfone‐carboxylic Acid Esters
2026-01-01 Mattana, Ariane; Rodríguez‐fernández, Laura; Zhao, Fei; Wu, Jingyue; Otun, Christopher W. O.; Manetti, Fabrizio; Montgomery, Sarah L.; Gotor‐fernández, Vicente; Barry, Sarah M.; Dominguez, Beatriz; Castagnolo, Daniele
A Comprehensive In Vitro and In Silico Approach for Targeting 4-Hydroxyphenyl Pyruvate Dioxygenase: Towards New Therapeutics for Alkaptonuria
2025-01-01 Bernardini, G.; Trezza, A.; Petricci, E.; Romagnoli, G.; Zambardino, D.; Manetti, F.; Braconi, D.; Geminiani, M.; Santucci, A.
Morita−Baylis−Hillman Adduct Chemistry as a Tool for the Design of Lysine-Targeted Covalent Ligands
2025-01-01 Paolino, Marco; Tassone, Giusy; Governa, Paolo; Saletti, Mario; Lami, Matteo; Carletti, Riccardo; Sacchetta, Filippo; Pozzi, Cecilia; Orlandini, Maurizio; Manetti, Fabrizio; Olivucci, Massimo; Cappelli, Andrea
Machine Learning for Predicting the Drug-to-Antibody Ratio (DAR) in the Synthesis of Antibody–Drug Conjugates (ADCs)
2025-01-01 Angiolini, Lorenzo; Manetti, Fabrizio; Spiga, Ottavia; Tafi, Andrea; Visibelli, Anna; Petricci, Elena
Light-mediated activation/deactivation control and in vitro ADME-Tox profiling of a donepezil-like Dual AChE/MAO-B Inhibitor
2025-01-01 Poggialini, Federica; Governa, Paolo; Vagaggini, Chiara; Maramai, Samuele; Lamponi, Stefania; Mugnaini, Claudia; Brizzi, Antonella; Purgatorio, Rosa; De Candia, Modesto; Catto, Marco; Dreassi, Elena; Manetti, Fabrizio; Corelli, Federico; Altomare, Cosimo Damiano; Cappelli, Andrea; Paolino, Marco
Deletion of 82–85 N-Terminal Residues in SARS-CoV-2 Nsp1 Restricts Virus Replication
2024-01-01 Gori Savellini, Gianni; Anichini, Gabriele; Manetti, Fabrizio; Trivisani, Claudia Immacolata; Cusi, Maria Grazia
Cooperative chemoenzymatic and biocatalytic cascades to access chiral sulfur compounds bearing C(sp3)–S stereocentres
2024-01-01 Zhao, Fei; Mattana, Ariane; Alam, Ruqaiya; Montgomery, Sarah L.; Pandya, Akash; Manetti, Fabrizio; Dominguez, Beatriz; Castagnolo, Daniele
Applying molecular hybridization to design a new class of pyrazolo[3,4-d]pyrimidines as Src inhibitors active in hepatocellular carcinoma
2024-01-01 Di Maria, Salvatore; Passannanti, Raffaele; Poggialini, Federica; Vagaggini, Chiara; Serafinelli, Alessia; Bianchi, Elena; Governa, Paolo; Botta, Lorenzo; Maga, Giovanni; Crespan, Emmanuele; Manetti, Fabrizio; Dreassi, Elena; Musumeci, Francesca; Carbone, Anna; Schenone, Silvia
Early investigation of a novel SI306 theranostic prodrug for glioblastoma treatment
2024-01-01 Vagaggini, Chiara; Petroni, Debora; D'Agostino, Ilaria; Poggialini, Federica; Cavallini, Chiara; Cianciusi, Annarita; Salis, Annalisa; D'Antona, Lucia; Francesconi, Valeria; Manetti, Fabrizio; Damonte, Gianluca; Musumeci, Francesca; Menichetti, Luca; Dreassi, Elena; Carbone, Anna; Schenone, Silvia
Consensus screening for a challenging target: the quest for P-glycoprotein inhibitors
2024-01-01 Governa, Paolo; Biagi, Marco; Manetti, Fabrizio; Forli, Stefano
Benzenesulfonamide decorated dihydropyrimidin(thi)ones: carbonic anhydrase profiling and antiproliferative activity
2024-01-01 Aslan, Hakan; Renzi, Gioele; Angeli, Andrea; D'Agostino, Ilaria; Ronca, Roberto; Massardi, Maria Luisa; Tavani, Camilla; Carradori, Simone; Ferraroni, Marta; Governa, Paolo; Manetti, Fabrizio; Carta, Fabrizio; Supuran, Claudiu T.
Zingiberene, a non-zinc-binding class I HDAC inhibitor: a novel strategy for the management of neuropathic pain
2023-01-01 Borgonetti, Vittoria; Governa, Paolo; Manetti, Fabrizio; Galeotti, Nicoletta
Antiviral activity of cannabidiolic acid and its methyl ester against SARS-CoV-2
2023-01-01 Tamburello, Martina; Salamone, Stefano; Anceschi, Lisa; Governa, Paolo; Brighenti, Virginia; Morellini, Alice; Rossini, Giada; Manetti, Fabrizio; Gallinella, Giorgio; Pollastro, Federica; Pellati, Federica
CanB, a druggable cellular target in mycobacterium tuberculosis
2023-01-01 Degiacomi, G; Gianibbi, B; Recchia, D; Stelitano, G; Truglio, Gi; Marra, P; Stamilla, A; Makarov, V; Chiarelli, Lr; Manetti, F; Pasca, Mr
Targeting GLI1 and GLI2 with small molecule inhibitors to suppress GLI-dependent transcription and tumor growth
2023-01-01 Maresca, Luisa; Crivaro, Enrica; Migliorini, Francesca; Anichini, Giulia; Giammona, Alessandro; Pepe, Sara; Poggialini, Federica; Vagaggini, Chiara; Giannini, Giuseppe; Sestini, Serena; Borgognoni, Lorenzo; Lapucci, Andrea; Dreassi, Elena; Taddei, Maurizio; Manetti, Fabrizio; Petricci, Elena; Stecca, Barbara
Effect of in vitro simulated digestion on the anti-Helicobacter Pylori activity of different Propolis extracts
2023-01-01 Governa, Paolo; Romagnoli, Giulia; Albanese, Paola; Rossi, Federico; Manetti, Fabrizio; Biagi, Marco
Cannabidiol-rich non-psychotropic Cannabis sativa L. oils attenuate peripheral neuropathy symptoms by regulation of CB2-mediated microglial neuroinflammation
2023-01-01 Borgonetti, Vittoria; Anceschi, Lisa; Brighenti, Virginia; Corsi, Lorenzo; Governa, Paolo; Manetti, Fabrizio; Pellati, Federica; Galeotti, Nicoletta
Helichrysum stoechas (L.) Moench reduces body weight gain and modulates mood disorders via inhibition of silent information regulator 1 (SIRT1) by arzanol
2023-01-01 Borgonetti, Vittoria; Caroli, Clarissa; Governa, Paolo; Virginia, Brighenti; Pollastro, Federica; Franchini, Silvia; Manetti, Fabrizio; Les, Francisco; López, Victor; Pellati, Federica; Galeotti, Nicoletta
Effects of in vitro simulated digestion on the antioxidant activity of different Camellia sinensis (L.) Kuntze leaves extracts
2022-01-01 Governa, Paolo; Manetti, Fabrizio; Miraldi, Elisabetta; Biagi, Marco
| Titolo | Data di pubblicazione | Autore(i) | File | Abstract |
|---|---|---|---|---|
| Dissecting the Interaction Domains of SARS-CoV-2 Nucleocapsid Protein and Human RNA Helicase DDX3X and Search for Potential Inhibitors | 1-gen-2026 | Lodola, Camilla; Pallotta, Maria Michela; Manetti, Fabrizio; Governa, Paolo; Crespan, Emmanuele; Maga, Giovanni; Secchi, Massimiliano | - | |
| Sulfur Oxidation Unlocks Ene‐Reductase Catalysis for Stereoselective C(sp3)–S(VI) Bond Formation in β‐Sulfone‐carboxylic Acid Esters | 1-gen-2026 | Mattana, Ariane; Rodríguez‐fernández, Laura; Zhao, Fei; Wu, Jingyue; Otun, Christopher W. O.; Manetti, Fabrizio; Montgomery, Sarah L.; Gotor‐fernández, Vicente; Barry, Sarah M.; Dominguez, Beatriz; Castagnolo, Daniele | - | |
| A Comprehensive In Vitro and In Silico Approach for Targeting 4-Hydroxyphenyl Pyruvate Dioxygenase: Towards New Therapeutics for Alkaptonuria | 1-gen-2025 | Bernardini, G.; Trezza, A.; Petricci, E.; Romagnoli, G.; Zambardino, D.; Manetti, F.; Braconi, D.; Geminiani, M.; Santucci, A. | - | |
| Morita−Baylis−Hillman Adduct Chemistry as a Tool for the Design of Lysine-Targeted Covalent Ligands | 1-gen-2025 | Paolino, Marco; Tassone, Giusy; Governa, Paolo; Saletti, Mario; Lami, Matteo; Carletti, Riccardo; Sacchetta, Filippo; Pozzi, Cecilia; Orlandini, Maurizio; Manetti, Fabrizio; Olivucci, Massimo; Cappelli, Andrea | - | |
| Machine Learning for Predicting the Drug-to-Antibody Ratio (DAR) in the Synthesis of Antibody–Drug Conjugates (ADCs) | 1-gen-2025 | Angiolini, Lorenzo; Manetti, Fabrizio; Spiga, Ottavia; Tafi, Andrea; Visibelli, Anna; Petricci, Elena | - | |
| Light-mediated activation/deactivation control and in vitro ADME-Tox profiling of a donepezil-like Dual AChE/MAO-B Inhibitor | 1-gen-2025 | Poggialini, Federica; Governa, Paolo; Vagaggini, Chiara; Maramai, Samuele; Lamponi, Stefania; Mugnaini, Claudia; Brizzi, Antonella; Purgatorio, Rosa; De Candia, Modesto; Catto, Marco; Dreassi, Elena; Manetti, Fabrizio; Corelli, Federico; Altomare, Cosimo Damiano; Cappelli, Andrea; Paolino, Marco | - | |
| Deletion of 82–85 N-Terminal Residues in SARS-CoV-2 Nsp1 Restricts Virus Replication | 1-gen-2024 | Gori Savellini, Gianni; Anichini, Gabriele; Manetti, Fabrizio; Trivisani, Claudia Immacolata; Cusi, Maria Grazia | - | |
| Cooperative chemoenzymatic and biocatalytic cascades to access chiral sulfur compounds bearing C(sp3)–S stereocentres | 1-gen-2024 | Zhao, Fei; Mattana, Ariane; Alam, Ruqaiya; Montgomery, Sarah L.; Pandya, Akash; Manetti, Fabrizio; Dominguez, Beatriz; Castagnolo, Daniele | - | |
| Applying molecular hybridization to design a new class of pyrazolo[3,4-d]pyrimidines as Src inhibitors active in hepatocellular carcinoma | 1-gen-2024 | Di Maria, Salvatore; Passannanti, Raffaele; Poggialini, Federica; Vagaggini, Chiara; Serafinelli, Alessia; Bianchi, Elena; Governa, Paolo; Botta, Lorenzo; Maga, Giovanni; Crespan, Emmanuele; Manetti, Fabrizio; Dreassi, Elena; Musumeci, Francesca; Carbone, Anna; Schenone, Silvia | - | |
| Early investigation of a novel SI306 theranostic prodrug for glioblastoma treatment | 1-gen-2024 | Vagaggini, Chiara; Petroni, Debora; D'Agostino, Ilaria; Poggialini, Federica; Cavallini, Chiara; Cianciusi, Annarita; Salis, Annalisa; D'Antona, Lucia; Francesconi, Valeria; Manetti, Fabrizio; Damonte, Gianluca; Musumeci, Francesca; Menichetti, Luca; Dreassi, Elena; Carbone, Anna; Schenone, Silvia | - | |
| Consensus screening for a challenging target: the quest for P-glycoprotein inhibitors | 1-gen-2024 | Governa, Paolo; Biagi, Marco; Manetti, Fabrizio; Forli, Stefano | - | |
| Benzenesulfonamide decorated dihydropyrimidin(thi)ones: carbonic anhydrase profiling and antiproliferative activity | 1-gen-2024 | Aslan, Hakan; Renzi, Gioele; Angeli, Andrea; D'Agostino, Ilaria; Ronca, Roberto; Massardi, Maria Luisa; Tavani, Camilla; Carradori, Simone; Ferraroni, Marta; Governa, Paolo; Manetti, Fabrizio; Carta, Fabrizio; Supuran, Claudiu T. | - | |
| Zingiberene, a non-zinc-binding class I HDAC inhibitor: a novel strategy for the management of neuropathic pain | 1-gen-2023 | Borgonetti, Vittoria; Governa, Paolo; Manetti, Fabrizio; Galeotti, Nicoletta | - | |
| Antiviral activity of cannabidiolic acid and its methyl ester against SARS-CoV-2 | 1-gen-2023 | Tamburello, Martina; Salamone, Stefano; Anceschi, Lisa; Governa, Paolo; Brighenti, Virginia; Morellini, Alice; Rossini, Giada; Manetti, Fabrizio; Gallinella, Giorgio; Pollastro, Federica; Pellati, Federica | - | |
| CanB, a druggable cellular target in mycobacterium tuberculosis | 1-gen-2023 | Degiacomi, G; Gianibbi, B; Recchia, D; Stelitano, G; Truglio, Gi; Marra, P; Stamilla, A; Makarov, V; Chiarelli, Lr; Manetti, F; Pasca, Mr | - | |
| Targeting GLI1 and GLI2 with small molecule inhibitors to suppress GLI-dependent transcription and tumor growth | 1-gen-2023 | Maresca, Luisa; Crivaro, Enrica; Migliorini, Francesca; Anichini, Giulia; Giammona, Alessandro; Pepe, Sara; Poggialini, Federica; Vagaggini, Chiara; Giannini, Giuseppe; Sestini, Serena; Borgognoni, Lorenzo; Lapucci, Andrea; Dreassi, Elena; Taddei, Maurizio; Manetti, Fabrizio; Petricci, Elena; Stecca, Barbara | - | |
| Effect of in vitro simulated digestion on the anti-Helicobacter Pylori activity of different Propolis extracts | 1-gen-2023 | Governa, Paolo; Romagnoli, Giulia; Albanese, Paola; Rossi, Federico; Manetti, Fabrizio; Biagi, Marco | - | |
| Cannabidiol-rich non-psychotropic Cannabis sativa L. oils attenuate peripheral neuropathy symptoms by regulation of CB2-mediated microglial neuroinflammation | 1-gen-2023 | Borgonetti, Vittoria; Anceschi, Lisa; Brighenti, Virginia; Corsi, Lorenzo; Governa, Paolo; Manetti, Fabrizio; Pellati, Federica; Galeotti, Nicoletta | - | |
| Helichrysum stoechas (L.) Moench reduces body weight gain and modulates mood disorders via inhibition of silent information regulator 1 (SIRT1) by arzanol | 1-gen-2023 | Borgonetti, Vittoria; Caroli, Clarissa; Governa, Paolo; Virginia, Brighenti; Pollastro, Federica; Franchini, Silvia; Manetti, Fabrizio; Les, Francisco; López, Victor; Pellati, Federica; Galeotti, Nicoletta | - | |
| Effects of in vitro simulated digestion on the antioxidant activity of different Camellia sinensis (L.) Kuntze leaves extracts | 1-gen-2022 | Governa, Paolo; Manetti, Fabrizio; Miraldi, Elisabetta; Biagi, Marco | - |
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