Sfoglia per Autore
Benzenesulfonamide decorated dihydropyrimidin(thi)ones: carbonic anhydrase profiling and antiproliferative activity
2024-01-01 Aslan, Hakan; Renzi, Gioele; Angeli, Andrea; D'Agostino, Ilaria; Ronca, Roberto; Massardi, Maria Luisa; Tavani, Camilla; Carradori, Simone; Ferraroni, Marta; Governa, Paolo; Manetti, Fabrizio; Carta, Fabrizio; Supuran, Claudiu T.
Deletion of 82–85 N-Terminal Residues in SARS-CoV-2 Nsp1 Restricts Virus Replication
2024-01-01 Gori Savellini, Gianni; Anichini, Gabriele; Manetti, Fabrizio; Trivisani, Claudia Immacolata; Cusi, Maria Grazia
Consensus screening for a challenging target: the quest for P-glycoprotein inhibitors
2024-01-01 Governa, Paolo; Biagi, Marco; Manetti, Fabrizio; Forli, Stefano
Early investigation of a novel SI306 theranostic prodrug for glioblastoma treatment
2024-01-01 Vagaggini, Chiara; Petroni, Debora; D'Agostino, Ilaria; Poggialini, Federica; Cavallini, Chiara; Cianciusi, Annarita; Salis, Annalisa; D'Antona, Lucia; Francesconi, Valeria; Manetti, Fabrizio; Damonte, Gianluca; Musumeci, Francesca; Menichetti, Luca; Dreassi, Elena; Carbone, Anna; Schenone, Silvia
Applying molecular hybridization to design a new class of pyrazolo[3,4-d]pyrimidines as Src inhibitors active in hepatocellular carcinoma
2024-01-01 Di Maria, Salvatore; Passannanti, Raffaele; Poggialini, Federica; Vagaggini, Chiara; Serafinelli, Alessia; Bianchi, Elena; Governa, Paolo; Botta, Lorenzo; Maga, Giovanni; Crespan, Emmanuele; Manetti, Fabrizio; Dreassi, Elena; Musumeci, Francesca; Carbone, Anna; Schenone, Silvia
Cooperative chemoenzymatic and biocatalytic cascades to access chiral sulfur compounds bearing C(sp3)–S stereocentres
2024-01-01 Zhao, Fei; Mattana, Ariane; Alam, Ruqaiya; Montgomery, Sarah L.; Pandya, Akash; Manetti, Fabrizio; Dominguez, Beatriz; Castagnolo, Daniele
Zingiberene, a non-zinc-binding class I HDAC inhibitor: a novel strategy for the management of neuropathic pain
2023-01-01 Borgonetti, Vittoria; Governa, Paolo; Manetti, Fabrizio; Galeotti, Nicoletta
Targeting GLI1 and GLI2 with small molecule inhibitors to suppress GLI-dependent transcription and tumor growth
2023-01-01 Maresca, Luisa; Crivaro, Enrica; Migliorini, Francesca; Anichini, Giulia; Giammona, Alessandro; Pepe, Sara; Poggialini, Federica; Vagaggini, Chiara; Giannini, Giuseppe; Sestini, Serena; Borgognoni, Lorenzo; Lapucci, Andrea; Dreassi, Elena; Taddei, Maurizio; Manetti, Fabrizio; Petricci, Elena; Stecca, Barbara
Effect of in vitro simulated digestion on the anti-Helicobacter Pylori activity of different Propolis extracts
2023-01-01 Governa, Paolo; Romagnoli, Giulia; Albanese, Paola; Rossi, Federico; Manetti, Fabrizio; Biagi, Marco
CanB, a druggable cellular target in mycobacterium tuberculosis
2023-01-01 Degiacomi, G; Gianibbi, B; Recchia, D; Stelitano, G; Truglio, Gi; Marra, P; Stamilla, A; Makarov, V; Chiarelli, Lr; Manetti, F; Pasca, Mr
Helichrysum stoechas (L.) Moench reduces body weight gain and modulates mood disorders via inhibition of silent information regulator 1 (SIRT1) by arzanol
2023-01-01 Borgonetti, Vittoria; Caroli, Clarissa; Governa, Paolo; Virginia, Brighenti; Pollastro, Federica; Franchini, Silvia; Manetti, Fabrizio; Les, Francisco; López, Victor; Pellati, Federica; Galeotti, Nicoletta
Antiviral activity of cannabidiolic acid and its methyl ester against SARS-CoV-2
2023-01-01 Tamburello, Martina; Salamone, Stefano; Anceschi, Lisa; Governa, Paolo; Brighenti, Virginia; Morellini, Alice; Rossini, Giada; Manetti, Fabrizio; Gallinella, Giorgio; Pollastro, Federica; Pellati, Federica
Cannabidiol-rich non-psychotropic Cannabis sativa L. oils attenuate peripheral neuropathy symptoms by regulation of CB2-mediated microglial neuroinflammation
2023-01-01 Borgonetti, Vittoria; Anceschi, Lisa; Brighenti, Virginia; Corsi, Lorenzo; Governa, Paolo; Manetti, Fabrizio; Pellati, Federica; Galeotti, Nicoletta
Effects of in vitro simulated digestion on the antioxidant activity of different Camellia sinensis (L.) Kuntze leaves extracts
2022-01-01 Governa, Paolo; Manetti, Fabrizio; Miraldi, Elisabetta; Biagi, Marco
Conformational insights into the C-terminal mutations of human rhodopsin in retinitis pigmentosa
2022-01-01 Picarazzi, Francesca; Manetti, Fabrizio; Marigo, Valeria; Mori, Mattia
Quinolines and Oxazino-quinoline derivatives as small molecule GLI1 inhibitors identified by virtual screening
2022-01-01 Manetti, Fabrizio; Maresca, Luisa; Crivaro, Enrica; Pepe, Sara; Cini, Elena; Singh, Snigdha; Governa, Paolo; Maramai, Samuele; Giannini, Giuseppe; Stecca, Barbara; Petricci, Elena
Investigation on the neuroprotective effect of a cannabidiol-enriched non-psychotropic Cannabis sativa L. extract in an in vitro model of excitotoxicity
2022-01-01 Borgonetti, Vittoria; Biagi, Marco; Galeotti, Nicoletta; Manetti, Fabrizio; Governa, Paolo
Synthesis and biological activity evaluation of 3-(hetero) arylideneindolin-2-ones as potential c-Src inhibitors
2022-01-01 Princiotto, Salvatore; Musso, Loana; Manetti, Fabrizio; Marcellini, Valentina; Maga, Giovanni; Crespan, Emmanuele; Perini, Cecilia; Zaffaroni, Nadia; Beretta, Giovanni Luca; Dallavalle, Sabrina
Structural rigidification of N-Aryl-pyrroles into indoles active against Intracellular and drug-resistant mycobacteria
2022-01-01 Semenya, Dorothy; Touitou, Meir; Ribeiro, Camila Maringolo; Pavan, Fernando Rogerio; Pisano, Luca; Singh, Vinayak; Chibale, Kelly; Bano, Georg; Toscani, Anita; Manetti, Fabrizio; Gianibbi, Beatrice; Castagnolo, Daniele
Recent research results have converted gp120 binders to a therapeutic option for the treatment of HIV-1 infection. A medicinal chemistry point of view
2022-01-01 Governa, Paolo; Manetti, Fabrizio
Titolo | Data di pubblicazione | Autore(i) | File | Abstract |
---|---|---|---|---|
Benzenesulfonamide decorated dihydropyrimidin(thi)ones: carbonic anhydrase profiling and antiproliferative activity | 1-gen-2024 | Aslan, Hakan; Renzi, Gioele; Angeli, Andrea; D'Agostino, Ilaria; Ronca, Roberto; Massardi, Maria Luisa; Tavani, Camilla; Carradori, Simone; Ferraroni, Marta; Governa, Paolo; Manetti, Fabrizio; Carta, Fabrizio; Supuran, Claudiu T. | - | |
Deletion of 82–85 N-Terminal Residues in SARS-CoV-2 Nsp1 Restricts Virus Replication | 1-gen-2024 | Gori Savellini, Gianni; Anichini, Gabriele; Manetti, Fabrizio; Trivisani, Claudia Immacolata; Cusi, Maria Grazia | - | |
Consensus screening for a challenging target: the quest for P-glycoprotein inhibitors | 1-gen-2024 | Governa, Paolo; Biagi, Marco; Manetti, Fabrizio; Forli, Stefano | - | |
Early investigation of a novel SI306 theranostic prodrug for glioblastoma treatment | 1-gen-2024 | Vagaggini, Chiara; Petroni, Debora; D'Agostino, Ilaria; Poggialini, Federica; Cavallini, Chiara; Cianciusi, Annarita; Salis, Annalisa; D'Antona, Lucia; Francesconi, Valeria; Manetti, Fabrizio; Damonte, Gianluca; Musumeci, Francesca; Menichetti, Luca; Dreassi, Elena; Carbone, Anna; Schenone, Silvia | - | |
Applying molecular hybridization to design a new class of pyrazolo[3,4-d]pyrimidines as Src inhibitors active in hepatocellular carcinoma | 1-gen-2024 | Di Maria, Salvatore; Passannanti, Raffaele; Poggialini, Federica; Vagaggini, Chiara; Serafinelli, Alessia; Bianchi, Elena; Governa, Paolo; Botta, Lorenzo; Maga, Giovanni; Crespan, Emmanuele; Manetti, Fabrizio; Dreassi, Elena; Musumeci, Francesca; Carbone, Anna; Schenone, Silvia | - | |
Cooperative chemoenzymatic and biocatalytic cascades to access chiral sulfur compounds bearing C(sp3)–S stereocentres | 1-gen-2024 | Zhao, Fei; Mattana, Ariane; Alam, Ruqaiya; Montgomery, Sarah L.; Pandya, Akash; Manetti, Fabrizio; Dominguez, Beatriz; Castagnolo, Daniele | - | |
Zingiberene, a non-zinc-binding class I HDAC inhibitor: a novel strategy for the management of neuropathic pain | 1-gen-2023 | Borgonetti, Vittoria; Governa, Paolo; Manetti, Fabrizio; Galeotti, Nicoletta | - | |
Targeting GLI1 and GLI2 with small molecule inhibitors to suppress GLI-dependent transcription and tumor growth | 1-gen-2023 | Maresca, Luisa; Crivaro, Enrica; Migliorini, Francesca; Anichini, Giulia; Giammona, Alessandro; Pepe, Sara; Poggialini, Federica; Vagaggini, Chiara; Giannini, Giuseppe; Sestini, Serena; Borgognoni, Lorenzo; Lapucci, Andrea; Dreassi, Elena; Taddei, Maurizio; Manetti, Fabrizio; Petricci, Elena; Stecca, Barbara | - | |
Effect of in vitro simulated digestion on the anti-Helicobacter Pylori activity of different Propolis extracts | 1-gen-2023 | Governa, Paolo; Romagnoli, Giulia; Albanese, Paola; Rossi, Federico; Manetti, Fabrizio; Biagi, Marco | - | |
CanB, a druggable cellular target in mycobacterium tuberculosis | 1-gen-2023 | Degiacomi, G; Gianibbi, B; Recchia, D; Stelitano, G; Truglio, Gi; Marra, P; Stamilla, A; Makarov, V; Chiarelli, Lr; Manetti, F; Pasca, Mr | - | |
Helichrysum stoechas (L.) Moench reduces body weight gain and modulates mood disorders via inhibition of silent information regulator 1 (SIRT1) by arzanol | 1-gen-2023 | Borgonetti, Vittoria; Caroli, Clarissa; Governa, Paolo; Virginia, Brighenti; Pollastro, Federica; Franchini, Silvia; Manetti, Fabrizio; Les, Francisco; López, Victor; Pellati, Federica; Galeotti, Nicoletta | - | |
Antiviral activity of cannabidiolic acid and its methyl ester against SARS-CoV-2 | 1-gen-2023 | Tamburello, Martina; Salamone, Stefano; Anceschi, Lisa; Governa, Paolo; Brighenti, Virginia; Morellini, Alice; Rossini, Giada; Manetti, Fabrizio; Gallinella, Giorgio; Pollastro, Federica; Pellati, Federica | - | |
Cannabidiol-rich non-psychotropic Cannabis sativa L. oils attenuate peripheral neuropathy symptoms by regulation of CB2-mediated microglial neuroinflammation | 1-gen-2023 | Borgonetti, Vittoria; Anceschi, Lisa; Brighenti, Virginia; Corsi, Lorenzo; Governa, Paolo; Manetti, Fabrizio; Pellati, Federica; Galeotti, Nicoletta | - | |
Effects of in vitro simulated digestion on the antioxidant activity of different Camellia sinensis (L.) Kuntze leaves extracts | 1-gen-2022 | Governa, Paolo; Manetti, Fabrizio; Miraldi, Elisabetta; Biagi, Marco | - | |
Conformational insights into the C-terminal mutations of human rhodopsin in retinitis pigmentosa | 1-gen-2022 | Picarazzi, Francesca; Manetti, Fabrizio; Marigo, Valeria; Mori, Mattia | - | |
Quinolines and Oxazino-quinoline derivatives as small molecule GLI1 inhibitors identified by virtual screening | 1-gen-2022 | Manetti, Fabrizio; Maresca, Luisa; Crivaro, Enrica; Pepe, Sara; Cini, Elena; Singh, Snigdha; Governa, Paolo; Maramai, Samuele; Giannini, Giuseppe; Stecca, Barbara; Petricci, Elena | - | |
Investigation on the neuroprotective effect of a cannabidiol-enriched non-psychotropic Cannabis sativa L. extract in an in vitro model of excitotoxicity | 1-gen-2022 | Borgonetti, Vittoria; Biagi, Marco; Galeotti, Nicoletta; Manetti, Fabrizio; Governa, Paolo | - | |
Synthesis and biological activity evaluation of 3-(hetero) arylideneindolin-2-ones as potential c-Src inhibitors | 1-gen-2022 | Princiotto, Salvatore; Musso, Loana; Manetti, Fabrizio; Marcellini, Valentina; Maga, Giovanni; Crespan, Emmanuele; Perini, Cecilia; Zaffaroni, Nadia; Beretta, Giovanni Luca; Dallavalle, Sabrina | - | |
Structural rigidification of N-Aryl-pyrroles into indoles active against Intracellular and drug-resistant mycobacteria | 1-gen-2022 | Semenya, Dorothy; Touitou, Meir; Ribeiro, Camila Maringolo; Pavan, Fernando Rogerio; Pisano, Luca; Singh, Vinayak; Chibale, Kelly; Bano, Georg; Toscani, Anita; Manetti, Fabrizio; Gianibbi, Beatrice; Castagnolo, Daniele | - | |
Recent research results have converted gp120 binders to a therapeutic option for the treatment of HIV-1 infection. A medicinal chemistry point of view | 1-gen-2022 | Governa, Paolo; Manetti, Fabrizio | - |
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