Sfoglia per Rivista ACS MEDICINAL CHEMISTRY LETTERS
Exploring oxidovanadium(IV) complexes as YopH inhibitors: mechanism of action and modeling studies
2015-01-01 Martins, Priscila G. A; Mori, Mattia; Chiaradia Delatorre, Louise D; Menegatti, Angela C. O; Mascarello, Alessandra; Botta, Bruno; Benítez, Julio; Gambino, Dinorah; Terenzi, Hernán
Exploring the implication of DDX3X in DENV infection: discovery of the first-in-class DDX3X fluorescent inhibitor
2020-01-01 Brai, Annalaura; Boccuto, Adele; Monti, Martina; Marchi, Serena; Vicenti, Ilaria; Saladini, Francesco; Trivisani, CLAUDIA IMMACOLATA; Pollutri, Alessandro; Trombetta, CLAUDIA MARIA; Montomoli, Emanuele; Riva, Valentina; Garbelli, Anna; Maria Nola, Emanuele; Zazzi, Maurizio; Maga, Giovanni; Dreassi, Elena; Botta, Maurizio
From Taxuspine X to structurally simplified Taxanes with remarkable P-Glycoprotein inhibitory activity
2010-01-01 Castagnolo, Daniele; Contemori, Lorenzo; Maccari, Giorgio; Avramova, S. I.; Neri, Alessandro; Sgaragli, Gian Pietro; Botta, Maurizio
Improving the Potency of N-Aryl-2,5-dimethylpyrroles against Multidrug-Resistant and Intracellular Mycobacteria
2020-01-01 Touitou, M.; Manetti, F.; Ribeiro, C. M.; Pavan, F. R.; Scalacci, N.; Zrebna, K.; Begum, N.; Semenya, D.; Gupta, A.; Bhakta, S.; Mchugh, T. D.; Senderowitz, H.; Kyriazi, M.; Castagnolo, D.
In Memory of Maurizio Botta: His Vision of Medicinal Chemistry
2020-01-01 Botta, Lorenzo; Mori, Mattia
Ligand promiscuity between the efflux pumps human p-glycoprotein and s. aureus NorA
2012-01-01 Brincat, Jp; Broccatelli, F; Sabatini, S; Frosini, Maria; Neri, Annalisa; Kaatz, Gw; Cruciani, G; Carosati, E.
Multifunctional Cholinesterase and Amyloid Beta Fibrillization Modulators. Synthesis and Biological Investigation
2013-01-01 Butini, Stefania; Brindisi, Margherita; Brogi, Simone; Maramai, Samuele; Egeria, Guarino; Alessandro, Panico; Ashima, Saxena; Ved, Chauhan; Raffaella, Colombo; Laura, Verga; Ersilia De, Lorenzi; Manuela, Bartolini; Vincenza, Andrisano; Ettore, Novellino; Campiani, Giuseppe; Gemma, Sandra
New frontiers in kinases: special issue
2014-01-01 Botta, Maurizio
Novel Macrocyclic Amidinoureas: Potent Non-Azole Antifungals Active against Wild-Type and Resistant Candida Species
2013-01-01 Sanguinetti, M.; Sanfilippo, S.; Castagnolo, Daniele; Sanglard, D.; Posteraro, B.; Donzellini, G.; Botta, Maurizio
Novel N-Substituted Benzomorphan-Based Compounds: From MOR-Agonist/DOR-Antagonist to Biased/Unbiased MOR Agonists
2020-01-01 Pasquinucci, Lorella; Parenti, Carmela; Ruiz-Cantero M., Carmen; Georgoussi, Zafiroula; Pallaki, Paschalina; Cobos J., Enrique; Amata, Emanuele; Marrazzo, Agostino; Prezzavento, Orazio; Arena, Emanuela; Dichiara, Maria; Salerno, Loredana; Turnaturi, Rita
Pharmacophore-based virtual screening for identification of negative modulators of GLI1 as potential anticancer agents
2020-01-01 Manetti, Fabrizio; Stecca, Barbara; Santini, Roberta; Maresca, Luisa; Giannini, Giuseppe; Taddei, Maurizio; Petricci, Elena
Plasmin-Binding Tripeptide-Decorated Liposomes Loading Pyrazolo[3,4- d]pyrimidines for Targeting Hepatocellular Carcinoma
2018-01-01 Calandro, Pierpaolo; Iovenitti, Giulia; Zamperini, Claudio; Candita, Francesca; Dreassi, Elena; Chiariello, Mario; Angelucci, Adriano; Schenone, Silvia; Botta, Maurizio; Mancini, Arianna
Probing the binding site of abl tyrosine kinase using in situ click chemistry
2013-01-01 Peruzzotti, C.; Borrelli, S.; Ventura, M.; Pantano, R.; Fumagalli, G.; Christodoulou, M. S.; Monticelli, D.; Luzzani, M.; Fallacara, A. L.; Tintori, Cristina; Botta, Maurizio; Passarella, D.
Pyrazolo[3,4-d]pyrimidine Prodrugs: Strategic Optimization of the Aqueous Solubility of Dual Src/Abl Inhibitors
2013-01-01 Vignaroli, Giulia; Zamperini, Claudio; Dreassi, Elena; Radi, Marco; Angelucci, A.; Sanità, P.; Crespan, Emmanuele; Kissova, M.; Maga, Giovanni; Schenone, S.; Musumeci, F.; Botta, Maurizio
Quinolines and Oxazino-quinoline derivatives as small molecule GLI1 inhibitors identified by virtual screening
2022-01-01 Manetti, Fabrizio; Maresca, Luisa; Crivaro, Enrica; Pepe, Sara; Cini, Elena; Singh, Snigdha; Governa, Paolo; Maramai, Samuele; Giannini, Giuseppe; Stecca, Barbara; Petricci, Elena
Screen of Unfocused Libraries Identified Compounds with Direct or Synergistic Antibacterial Activity
2020-01-01 Mugnaini, C.; Sannio, F.; Brizzi, A.; Del Prete, R.; Simone, T.; Ferraro, T.; De Luca, F.; Corelli, F.; Docquier, J. D.
Separation of betti reaction product enantiomers: Absolute configuration and inhibition of botulinum neurotoxin A
2011-01-01 Cardellina, J. H.; Vieira, R. C.; Eccard, V.; Skerry, J.; Montgomery, V.; Campbell, Y.; Roxas-Duncan, V.; Leister, W.; Leclair, C. A.; Maloney, D. J.; Padula, D.; Pescitelli, G.; Khavrutskii, I.; Hu, X.; Wallqvist, A.; Smith, L. A.
Sigma Receptor Ligands Carrying a Nitric Oxide Donor Nitrate Moiety: Synthesis, In Silico, and Biological Evaluation
2020-01-01 Amata, Emanuele; Dichiara, Maria; Gentile, Davide; Marrazzo, Agostino; Turnaturi, Rita; Arena, Emanuela; La Mantia, Alfonsina; Tomasello R., Barbara; Acquaviva, Rosaria; Di Giacomo, Claudia; Rescifina, Antonio; Prezzavento, Orazio
Spiroindoline-Capped Selective HDAC6 Inhibitors: Design, Synthesis, Structural Analysis, and Biological Evaluation
2020-01-01 Saraswati, A Prasanth; Relitti, Nicola; Brindisi, Margherita; Osko, Jeremy D; Chemi, Giulia; Federico, Stefano; Grillo, Alessandro; Brogi, Simone; Mccabe, Niamh H; Turkington, Richard C; Ibrahim, Ola; O'Sullivan, Jeffrey; Lamponi, Stefania; Ghanim, Magda; Kelly, Vincent P; Zisterer, Daniela; Amet, Rebecca; Hannon Barroeta, Patricia; Vanni, Francesca; Ulivieri, Cristina; Herp, Daniel; Sarno, Federica; Di Costanzo, Antonella; Saccoccia, Fulvio; Ruberti, Giovina; Jung, Manfred; Altucci, Lucia; Gemma, Sandra; Butini, Stefania; Christianson, David W; Campiani, Giuseppe
Structural Elucidation and Antimicrobial Characterization of Novel Diterpenoids from Fabiana densa var. ramulosa
2020-01-01 Quaglio, D.; Corradi, S.; Erazo, S.; Vergine, V.; Berardozzi, S.; Sciubba, F.; Cappiello, F.; Crestoni, M. E.; Ascenzioni, F.; Imperi, F.; Delle Monache, F.; Mori, M.; Loffredo, M. R.; Ghirga, F.; Casciaro, B.; Botta, B.; Mangoni, M. L.
| Titolo | Data di pubblicazione | Autore(i) | File | Abstract |
|---|---|---|---|---|
| Exploring oxidovanadium(IV) complexes as YopH inhibitors: mechanism of action and modeling studies | 1-gen-2015 | Martins, Priscila G. A; Mori, Mattia; Chiaradia Delatorre, Louise D; Menegatti, Angela C. O; Mascarello, Alessandra; Botta, Bruno; Benítez, Julio; Gambino, Dinorah; Terenzi, Hernán | - | |
| Exploring the implication of DDX3X in DENV infection: discovery of the first-in-class DDX3X fluorescent inhibitor | 1-gen-2020 | Brai, Annalaura; Boccuto, Adele; Monti, Martina; Marchi, Serena; Vicenti, Ilaria; Saladini, Francesco; Trivisani, CLAUDIA IMMACOLATA; Pollutri, Alessandro; Trombetta, CLAUDIA MARIA; Montomoli, Emanuele; Riva, Valentina; Garbelli, Anna; Maria Nola, Emanuele; Zazzi, Maurizio; Maga, Giovanni; Dreassi, Elena; Botta, Maurizio | - | |
| From Taxuspine X to structurally simplified Taxanes with remarkable P-Glycoprotein inhibitory activity | 1-gen-2010 | Castagnolo, Daniele; Contemori, Lorenzo; Maccari, Giorgio; Avramova, S. I.; Neri, Alessandro; Sgaragli, Gian Pietro; Botta, Maurizio | - | |
| Improving the Potency of N-Aryl-2,5-dimethylpyrroles against Multidrug-Resistant and Intracellular Mycobacteria | 1-gen-2020 | Touitou, M.; Manetti, F.; Ribeiro, C. M.; Pavan, F. R.; Scalacci, N.; Zrebna, K.; Begum, N.; Semenya, D.; Gupta, A.; Bhakta, S.; Mchugh, T. D.; Senderowitz, H.; Kyriazi, M.; Castagnolo, D. | - | |
| In Memory of Maurizio Botta: His Vision of Medicinal Chemistry | 1-gen-2020 | Botta, Lorenzo; Mori, Mattia | - | |
| Ligand promiscuity between the efflux pumps human p-glycoprotein and s. aureus NorA | 1-gen-2012 | Brincat, Jp; Broccatelli, F; Sabatini, S; Frosini, Maria; Neri, Annalisa; Kaatz, Gw; Cruciani, G; Carosati, E. | - | |
| Multifunctional Cholinesterase and Amyloid Beta Fibrillization Modulators. Synthesis and Biological Investigation | 1-gen-2013 | Butini, Stefania; Brindisi, Margherita; Brogi, Simone; Maramai, Samuele; Egeria, Guarino; Alessandro, Panico; Ashima, Saxena; Ved, Chauhan; Raffaella, Colombo; Laura, Verga; Ersilia De, Lorenzi; Manuela, Bartolini; Vincenza, Andrisano; Ettore, Novellino; Campiani, Giuseppe; Gemma, Sandra | - | |
| New frontiers in kinases: special issue | 1-gen-2014 | Botta, Maurizio | - | |
| Novel Macrocyclic Amidinoureas: Potent Non-Azole Antifungals Active against Wild-Type and Resistant Candida Species | 1-gen-2013 | Sanguinetti, M.; Sanfilippo, S.; Castagnolo, Daniele; Sanglard, D.; Posteraro, B.; Donzellini, G.; Botta, Maurizio | - | |
| Novel N-Substituted Benzomorphan-Based Compounds: From MOR-Agonist/DOR-Antagonist to Biased/Unbiased MOR Agonists | 1-gen-2020 | Pasquinucci, Lorella; Parenti, Carmela; Ruiz-Cantero M., Carmen; Georgoussi, Zafiroula; Pallaki, Paschalina; Cobos J., Enrique; Amata, Emanuele; Marrazzo, Agostino; Prezzavento, Orazio; Arena, Emanuela; Dichiara, Maria; Salerno, Loredana; Turnaturi, Rita | - | |
| Pharmacophore-based virtual screening for identification of negative modulators of GLI1 as potential anticancer agents | 1-gen-2020 | Manetti, Fabrizio; Stecca, Barbara; Santini, Roberta; Maresca, Luisa; Giannini, Giuseppe; Taddei, Maurizio; Petricci, Elena | - | |
| Plasmin-Binding Tripeptide-Decorated Liposomes Loading Pyrazolo[3,4- d]pyrimidines for Targeting Hepatocellular Carcinoma | 1-gen-2018 | Calandro, Pierpaolo; Iovenitti, Giulia; Zamperini, Claudio; Candita, Francesca; Dreassi, Elena; Chiariello, Mario; Angelucci, Adriano; Schenone, Silvia; Botta, Maurizio; Mancini, Arianna | - | |
| Probing the binding site of abl tyrosine kinase using in situ click chemistry | 1-gen-2013 | Peruzzotti, C.; Borrelli, S.; Ventura, M.; Pantano, R.; Fumagalli, G.; Christodoulou, M. S.; Monticelli, D.; Luzzani, M.; Fallacara, A. L.; Tintori, Cristina; Botta, Maurizio; Passarella, D. | - | |
| Pyrazolo[3,4-d]pyrimidine Prodrugs: Strategic Optimization of the Aqueous Solubility of Dual Src/Abl Inhibitors | 1-gen-2013 | Vignaroli, Giulia; Zamperini, Claudio; Dreassi, Elena; Radi, Marco; Angelucci, A.; Sanità, P.; Crespan, Emmanuele; Kissova, M.; Maga, Giovanni; Schenone, S.; Musumeci, F.; Botta, Maurizio | - | |
| Quinolines and Oxazino-quinoline derivatives as small molecule GLI1 inhibitors identified by virtual screening | 1-gen-2022 | Manetti, Fabrizio; Maresca, Luisa; Crivaro, Enrica; Pepe, Sara; Cini, Elena; Singh, Snigdha; Governa, Paolo; Maramai, Samuele; Giannini, Giuseppe; Stecca, Barbara; Petricci, Elena | - | |
| Screen of Unfocused Libraries Identified Compounds with Direct or Synergistic Antibacterial Activity | 1-gen-2020 | Mugnaini, C.; Sannio, F.; Brizzi, A.; Del Prete, R.; Simone, T.; Ferraro, T.; De Luca, F.; Corelli, F.; Docquier, J. D. | - | |
| Separation of betti reaction product enantiomers: Absolute configuration and inhibition of botulinum neurotoxin A | 1-gen-2011 | Cardellina, J. H.; Vieira, R. C.; Eccard, V.; Skerry, J.; Montgomery, V.; Campbell, Y.; Roxas-Duncan, V.; Leister, W.; Leclair, C. A.; Maloney, D. J.; Padula, D.; Pescitelli, G.; Khavrutskii, I.; Hu, X.; Wallqvist, A.; Smith, L. A. | - | |
| Sigma Receptor Ligands Carrying a Nitric Oxide Donor Nitrate Moiety: Synthesis, In Silico, and Biological Evaluation | 1-gen-2020 | Amata, Emanuele; Dichiara, Maria; Gentile, Davide; Marrazzo, Agostino; Turnaturi, Rita; Arena, Emanuela; La Mantia, Alfonsina; Tomasello R., Barbara; Acquaviva, Rosaria; Di Giacomo, Claudia; Rescifina, Antonio; Prezzavento, Orazio | - | |
| Spiroindoline-Capped Selective HDAC6 Inhibitors: Design, Synthesis, Structural Analysis, and Biological Evaluation | 1-gen-2020 | Saraswati, A Prasanth; Relitti, Nicola; Brindisi, Margherita; Osko, Jeremy D; Chemi, Giulia; Federico, Stefano; Grillo, Alessandro; Brogi, Simone; Mccabe, Niamh H; Turkington, Richard C; Ibrahim, Ola; O'Sullivan, Jeffrey; Lamponi, Stefania; Ghanim, Magda; Kelly, Vincent P; Zisterer, Daniela; Amet, Rebecca; Hannon Barroeta, Patricia; Vanni, Francesca; Ulivieri, Cristina; Herp, Daniel; Sarno, Federica; Di Costanzo, Antonella; Saccoccia, Fulvio; Ruberti, Giovina; Jung, Manfred; Altucci, Lucia; Gemma, Sandra; Butini, Stefania; Christianson, David W; Campiani, Giuseppe | - | |
| Structural Elucidation and Antimicrobial Characterization of Novel Diterpenoids from Fabiana densa var. ramulosa | 1-gen-2020 | Quaglio, D.; Corradi, S.; Erazo, S.; Vergine, V.; Berardozzi, S.; Sciubba, F.; Cappiello, F.; Crestoni, M. E.; Ascenzioni, F.; Imperi, F.; Delle Monache, F.; Mori, M.; Loffredo, M. R.; Ghirga, F.; Casciaro, B.; Botta, B.; Mangoni, M. L. | - |
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