GIOVANI, SIMONE
GIOVANI, SIMONE
A stereoselective approach to peptidomimetic BACE1 inhibitors
2013-01-01 Butini, Stefania; Emanuele, Gabellieri; Brindisi, Margherita; Giovani, Simone; Maramai, Samuele; Kshirsagar, Giridhar; Egeria, Guarino; Brogi, Simone; Valeria La, Pietra; Mariateresa, Giustiniano; Luciana, Marinelli; Ettore, Novellino; Campiani, Giuseppe; Cappelli, Andrea; Gemma, Sandra
From (+)-epigallocatechin gallate to a simplified synthetic analogue as a cytoadherence inhibitor for P. falciparum
2014-01-01 Gemma, Sandra; Brogi, Simone; Pradeep R., Patil; Giovani, Simone; Lamponi, Stefania; Cappelli, Andrea; Ettore, Novellino; Alan, Brown; Matthew K., Higgins; Khairul, Mustafa; Tadge, Szestak; Alister G., Craig; Campiani, Giuseppe; Butini, Stefania; Brindisi, Margherita
In silico study of subtilisin-like protease 1 (SUB1) from different Plasmodium species in complex with peptidyl-difluorostatones and characterization of potent pan-SUB1 inhibitors
2016-01-01 Brogi, Simone; Giovani, Simone; Brindisi, Margherita; Gemma, Sandra; Novellino, Ettore; Campiani, Giuseppe; Blackman, Michael J; Butini, Stefania
Plasmodium falciparum subtilisin-like protease 1: discovery of potent difluorostatone-based inhibitors
2015-01-01 Giovani, Simone; Penzo, Maria; Butini, Stefania; Brindisi, Margherita; Gemma, Sandra; Novellino, Ettore; Campiani, Giuseppe; Blackman, Michael J.; Brogi, Simone
Quinolylhydrazones as novel inhibitors of Plasmodium falciparum serine protease PfSUB1
2012-01-01 Gemma, Sandra; Giovani, Simone; Brindisi, Margherita; Tripaldi, Pierangela; Brogi, Simone; Savini, Luisa; Fiorini, Isabella; Ettore, Novellino; Butini, Stefania; Campiani, Giuseppe; Maria, Penzo; Michael J., Blackman
Rational design of the first difluorostatone-based PfSUB1 inhibitors
2014-01-01 Giovani, Simone; Maria, Penzo; Brogi, Simone; Brindisi, Margherita; Gemma, Sandra; Ettore, Novellino; Savini, Luisa; Michael J., Blackman; Campiani, Giuseppe; Butini, Stefania
Targeting clinically-relevant metallo-β-lactamases: from high-throughput docking to broad-spectrum inhibitors
2016-01-01 Brindisi, Margherita; Brogi, Simone; Giovani, Simone; Gemma, Sandra; Lamponi, Stefania; DE LUCA, Filomena; Novellino, Ettore; Campiani, Giuseppe; Docquier, JEAN DENIS; Butini, Stefania
Titolo | Data di pubblicazione | Autore(i) | File | Abstract |
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A stereoselective approach to peptidomimetic BACE1 inhibitors | 1-gen-2013 | Butini, Stefania; Emanuele, Gabellieri; Brindisi, Margherita; Giovani, Simone; Maramai, Samuele; Kshirsagar, Giridhar; Egeria, Guarino; Brogi, Simone; Valeria La, Pietra; Mariateresa, Giustiniano; Luciana, Marinelli; Ettore, Novellino; Campiani, Giuseppe; Cappelli, Andrea; Gemma, Sandra | - | |
From (+)-epigallocatechin gallate to a simplified synthetic analogue as a cytoadherence inhibitor for P. falciparum | 1-gen-2014 | Gemma, Sandra; Brogi, Simone; Pradeep R., Patil; Giovani, Simone; Lamponi, Stefania; Cappelli, Andrea; Ettore, Novellino; Alan, Brown; Matthew K., Higgins; Khairul, Mustafa; Tadge, Szestak; Alister G., Craig; Campiani, Giuseppe; Butini, Stefania; Brindisi, Margherita | - | |
In silico study of subtilisin-like protease 1 (SUB1) from different Plasmodium species in complex with peptidyl-difluorostatones and characterization of potent pan-SUB1 inhibitors | 1-gen-2016 | Brogi, Simone; Giovani, Simone; Brindisi, Margherita; Gemma, Sandra; Novellino, Ettore; Campiani, Giuseppe; Blackman, Michael J; Butini, Stefania | - | |
Plasmodium falciparum subtilisin-like protease 1: discovery of potent difluorostatone-based inhibitors | 1-gen-2015 | Giovani, Simone; Penzo, Maria; Butini, Stefania; Brindisi, Margherita; Gemma, Sandra; Novellino, Ettore; Campiani, Giuseppe; Blackman, Michael J.; Brogi, Simone | - | |
Quinolylhydrazones as novel inhibitors of Plasmodium falciparum serine protease PfSUB1 | 1-gen-2012 | Gemma, Sandra; Giovani, Simone; Brindisi, Margherita; Tripaldi, Pierangela; Brogi, Simone; Savini, Luisa; Fiorini, Isabella; Ettore, Novellino; Butini, Stefania; Campiani, Giuseppe; Maria, Penzo; Michael J., Blackman | - | |
Rational design of the first difluorostatone-based PfSUB1 inhibitors | 1-gen-2014 | Giovani, Simone; Maria, Penzo; Brogi, Simone; Brindisi, Margherita; Gemma, Sandra; Ettore, Novellino; Savini, Luisa; Michael J., Blackman; Campiani, Giuseppe; Butini, Stefania | - | |
Targeting clinically-relevant metallo-β-lactamases: from high-throughput docking to broad-spectrum inhibitors | 1-gen-2016 | Brindisi, Margherita; Brogi, Simone; Giovani, Simone; Gemma, Sandra; Lamponi, Stefania; DE LUCA, Filomena; Novellino, Ettore; Campiani, Giuseppe; Docquier, JEAN DENIS; Butini, Stefania | - |