BROGI, SIMONE

BROGI, SIMONE  

Dipartimento di Biotecnologie, Chimica e Farmacia  

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Risultati 1 - 20 di 58 (tempo di esecuzione: 0.0 secondi).
Titolo Data di pubblicazione Autore(i) File Abstract
3D-QSAR using pharmacophore-based alignment and virtual screening for discovery of novel MCF-7 cell line inhibitors 1-gen-2013 Brogi, Simone; Panagiota, Papazafiri; Vassilios, Roussis; Tafi, Andrea -
A stereoselective approach to peptidomimetic BACE1 inhibitors 1-gen-2013 Butini, Stefania; Emanuele, Gabellieri; Brindisi, Margherita; Giovani, Simone; Maramai, Samuele; Kshirsagar, Giridhar; Egeria, Guarino; Brogi, Simone; Valeria La, Pietra; Mariateresa, Giustiniano; Luciana, Marinelli; Ettore, Novellino; Campiani, Giuseppe; Cappelli, Andrea; Gemma, Sandra -
Activation of the Wnt pathway by small peptides: rational design, synthesis and biological evaluation 1-gen-2017 Brogi, Simone; Maramai, Samuele; Brindisi, Margherita; Chemi, Giulia; Porcari, Valentina; Corallo, Claudio; Gennari, Luigi; Novellino, Ettore; Ramunno, Anna; Butini, Stefania; Campiani, Giuseppe; Gemma, Sandra -
Allosteric Modulation of Ionotropic Glutamate Receptors: An Outlook on New Therapeutic Approaches To Treat Central Nervous System Disorders 1-gen-2019 Brogi, Simone; Campiani, Giuseppe; Brindisi, Margherita; Butini, Stefania -
Antimalarial agents against both sexual and asexual parasites stages: structure-activity relationships and biological studies of the Malaria Box compound 1-[5-(4-bromo-2-chlorophenyl)furan-2-yl]- N -[(piperidin-4-yl)methyl]methanamine (MMV019918) and analogues 1-gen-2018 Vallone, Alessandra; D'Alessandro, Sarah; Brogi, Simone; Brindisi, Margherita; Chemi, Giulia; Alfano, Gloria; Lamponi, Stefania; Lee, Soon Goo; Jez, Joseph M.; Koolen, Karin J. M.; Dechering, Koen J.; Saponara, Simona; Fusi, Fabio; Gorelli, Beatrice; Taramelli, Donatella; Parapini, Silvia; Caldelari, Reto; Campiani, Giuseppe; Gemma, Sandra; Butini, Stefania -
Bridged bicyclic 2,3-dioxabicyclo[3.3.1]nonanes as antiplasmodial agents: Synthesis, structure-activity relationships and studies on their biomimetic reaction with Fe(II) 1-gen-2019 D'Alessandro, S.; Alfano, G.; Di Cerbo, L.; Brogi, S.; Chemi, G.; Relitti, N.; Brindisi, M.; Lamponi, S.; Novellino, E.; Campiani, G.; Gemma, S.; Basilico, N.; Taramelli, D.; Baratto, M. C.; Pogni, R.; Butini, S. -
Characterization of COR627 and COR628, two novel positive allosteric modulators of the GABA B receptor 1-gen-2012 Castelli, M. P.; Casu, A.; Casti, P.; Lobina, C.; Carai, M. A. M.; Colombo, G.; Solinas, M.; Giunta, D.; Mugnaini, Claudia; Pasquini, Serena; Tafi, Andrea; Brogi, Simone; Gessa, G. L.; Corelli, Federico -
Cinnamic acids derived compounds with antileishmanial activity target Leishmania amazonensis arginase 1-gen-2019 da Silva, Edson Roberto; Brogi, Simone; Grillo, Alessandro; Campiani, Giuseppe; Gemma, Sandra; Vieira, Paulo Cezar; Maquiaveli, Claudia do Carmo -
Computational tool for fast in silico evaluation of hERG K+ channel affinity 1-gen-2017 Chemi, Giulia; Gemma, Sandra; Campiani, Giuseppe; Brogi, Simone; Butini, Stefania; Brindisi, Margherita -
Computer-driven development of an in silico tool for finding selective histone deacetylase 1 inhibitors 1-gen-2020 Sirous, H.; Campiani, G.; Brogi, S.; Calderone, V.; Chemi, G. -
Crystal structures of Schistosoma mansoni histone deacetylase 8 reveal a novel binding site for allosteric inhibitors 1-gen-2022 Saccoccia, Fulvio; Pozzetti, Luca; Gimmelli, Roberto; Butini, Stefania; Guidi, Alessandra; Papoff, Giuliana; Giannaccari, Marialaura; Brogi, Simone; Scognamiglio, Viviana; Gemma, Sandra; Ruberti, Giovina; Campiani, Giuseppe -
Design, Synthesis, and Pharmacological Characterization of Indole-3-ylacetamides, Indole-3-yloxoacetamides, and Indole-3-ylcarboxamides: Potent and Selective CB2 Cannabinoid Receptor Inverse Agonists 1-gen-2012 Pasquini, Serena; Mugnaini, Claudia; Ligresti, A.; Tafi, Andrea; Brogi, Simone; Falciani, C.; Pedani, Valentina; Pesco, N.; Guida, F.; Luongo, L.; Varani, K.; Borea, P. A.; Maione, S.; Di Marzo, V.; Corelli, Federico -
Development of a practical and scalable route for the preparation of the deacetoxytubuvaline (dTuv) fragment of pretubulysin and analogs 1-gen-2016 Brindisi, Margherita; Maramai, Samuele; Grillo, Alessandro; Brogi, Simone; Butini, Stefania; Ettore, Novellino; Campiani, Giuseppe; Gemma, Sandra -
Development of HuperTacrines as non-toxic, cholinesterase inhibitors for the potential treatment of Alzheimer's disease 1-gen-2015 Chioua, Mourad; Pérez, Marta; Bautista Aguilera, Oscar M; Yañez, Matilde; López, Manuela G; Romero, Alejandro; Cacabelos, Ramón; de la Bellacasa, Raimon Puig; Brogi, Simone; Butini, Stefania; Borrell, José I; Marco Contelles, Jose -
Development of Potent Inhibitors of Fatty Acid Amide Hydrolase Useful for the Treatment of Neuropathic Pain 1-gen-2018 Brindisi, Margherita; Borrelli, Giuseppe; Brogi, Simone; Grillo, Alessandro; Maramai, Samuele; Paolino, Marco; Benedusi, Mascia; Pecorelli, Alessandra; Valacchi, Giuseppe; Di Cesare Mannelli, Lorenzo; Ghelardini, Carla; Allarà, Marco; Ligresti, Alessia; Minetti, Patrizia; Campiani, Giuseppe; Butini, Stefania; di Marzo, Vincenzo; Gemma, Sandra -
Dietary polyphenols rutin, taxifolin and quercetin related compounds target: Leishmania amazonensis arginase 1-gen-2019 Da Silva, E. R.; Brogi, S.; Lucon-Junior, J. F.; Campiani, G.; Gemma, S.; Maquiaveli, C. D. C. -
Discovery of GPCR ligands for probing signal transduction pathways 1-gen-2014 Brogi, Simone; Tafi, Andrea; Désaubry, Laurent; Nebigil, Canan -
Disease modifying anti-Alzheimer’s drugs: inhibitors of human cholinesterases interfering with β-amyloid aggregation 1-gen-2014 Brogi, Simone; Butini, Stefania; Maramai, Samuele; Raffaella, Colombo; Laura, Verga; Cristina, Lanni; Ersilia De, Lorenzi; Lamponi, Stefania; Andreassi, Marco; Manuela, Bartolini; Vincenza, Andrisano; Ettore, Novellino; Campiani, Giuseppe; Brindisi, Margherita; Gemma, Sandra -
Dopamine D3 receptor antagonists as potential therapeutics for the treatment of neurological diseases 1-gen-2016 Maramai, Samuele; Gemma, Sandra; Brogi, Simone; Campiani, Giuseppe; Butini, Stefania; Stark, Holger; Brindisi, Margherita -
Exploring clotrimazole-based pharmacophore: 3D-QSAR studies and synthesis of novel antiplasmodial agents 1-gen-2015 Brogi, Simone; Brindisi, Margherita; Joshi, BHUPENDRA PRASAD; SANNA COCCONE, Salvatore; Parapini, Silvia; Basilico, Nicoletta; Novellino, Ettore; Campiani, Giuseppe; Gemma, Sandra; Butini, Stefania -