Sfoglia per Autore
Structural and antigen-binding surface definition of an anti-CD93 monoclonal antibody for the treatment of degenerative vascular eye diseases
2025-01-01 Raucci, Luisa; Perrone, Cosimo Damiano; Barbera, Stefano; de Boer, Laurens Julius; Tosi, Gian Marco; Brunetti, Jlenia; Bracci, Luisa; Pozzi, Cecilia; Galvagni, Federico; Orlandini, Maurizio
Morita−Baylis−Hillman Adduct Chemistry as a Tool for the Design of Lysine-Targeted Covalent Ligands
2025-01-01 Paolino, Marco; Tassone, Giusy; Governa, Paolo; Saletti, Mario; Lami, Matteo; Carletti, Riccardo; Sacchetta, Filippo; Pozzi, Cecilia; Orlandini, Maurizio; Manetti, Fabrizio; Olivucci, Massimo; Cappelli, Andrea
Design of 2-Aminobenzothiazole Derivatives Targeting Trypanosomatid PTR1 by a Multidisciplinary Fragment Hybridization Approach
2025-01-01 Panecka-Hofman, Joanna; Linciano, Pasquale; Pöhner, Ina; Dyguda-Kazimierowicz, Edyta; Jedwabny, Wiktoria; Landi, Giacomo; Santarem, Nuno; Witt, Gesa; Ellinger, Bernhard; Kuzikov, Maria; Luciani, Rosaria; Ferrari, Stefania; Aiello, Daniele; Mangani, Stefano; Pozzi, Cecilia; Cordeiro-da-Silva, Anabela; Gul, Sheraz; Costi, Maria Paola; Wade, Rebecca C.
Identification of pyrazolo-piperidinone derivatives targeting YAP-TEAD interface 3 as anticancer agents through integrated virtual screening and mass spectrometry proteomics
2025-01-01 Scalvini, Laura; Tagliazucchi, Lorenzo; Elisi, Gian Marco; Zappaterra, Dana; Moschella, Maria Gaetana; Fantini, Sebastian; Aiello, Daniele; Guerrini, Remo; Albanese, Valentina; Pacifico, Salvatore; Lopresti, Ludovica; Malpezzi, Giulia; Saporito, Giulia; Ferrari, Stefania; Lamesta, Michele; Losi, Lorena; Pozzi, Cecilia; Mangani, Stefano; Marverti, Gaetano; Venturelli, Alberto; Ponterini, Glauco; D'Arca, Domenico; Mor, Marco; Costi, Maria Paola
Metal ion binding to human Glutaminyl Cyclase: a structural perspective
2024-01-01 Tassone, Giusy; Pozzi, Cecilia; Mangani, Stefano
The discovery of aryl-2-nitroethyl triamino pyrimidines as anti-Trypanosoma brucei agents
2024-01-01 Linciano, Pasquale; Pozzi, Cecilia; Tassone, Giusy; Landi, Giacomo; Mangani, Stefano; Santucci, Matteo; Luciani, Rosaria; Ferrari, Stefania; Santarem, Nuno; Tagliazucchi, Lorenzo; Cordeiro-da-Silva, Anabela; Tonelli, Michele; Tondi, Donatella; Bertarini, Laura; Gul, Sheraz; Witt, Gesa; B Moraes, Carolina; Costantino, Luca; Paola Costi, Maria
Exploiting the bile acid binding protein as transporter of a Cholic Acid/Mirin bioconjugate for potential applications in liver cancer therapy
2024-01-01 Tassone, Giusy; Maramai, Samuele; Paolino, Marco; Lamponi, Stefania; Poggialini, Federica; Dreassi, Elena; Petricci, Elena; Alcaro, Stefano; Pozzi, Cecilia; Romeo, Isabella
Identification of Innovative Folate Inhibitors Leveraging the Amino Dihydrotriazine Motif from Cycloguanil for Their Potential as Anti-Trypanosoma brucei Agents
2024-01-01 Francesconi, Valeria; Rizzo, Marco; Pozzi, Cecilia; Tagliazucchi, Lorenzo; Konchie Simo, Claude U.; Saporito, Giulia; Landi, Giacomo; Mangani, Stefano; Carbone, Anna; Schenone, Silvia; Santarém, Nuno; Tavares, Joana; Cordeiro-da-Silva, Anabela; Costi, Maria Paola; Tonelli, Michele
Dimerization of the C-type lectin-like receptor CD93 promotes its binding to Multimerin-2 in endothelial cells
2023-01-01 Barbera, Stefano; Raucci, Luisa; Tassone, Giusy; Tinti, Laura; Prischi, Filippo; Santucci, Annalisa; Mongiat, Maurizio; Tosi, Gian Marco; Galvagni, Federico; Dimberg, Anna; Pozzi, Cecilia; Orlandini, Maurizio
Antitarget, Anti-SARS-CoV-2 Leads, Drugs, and the Drug Discovery-Genetics Alliance Perspective
2023-01-01 Pozzi, Cecilia; Vanet, Anne; Francesconi, Valeria; Tagliazucchi, Lorenzo; Tassone, Giusy; Venturelli, Alberto; Spyrakis, Francesca; Mazzorana, Marco; P Costi, Maria; Tonelli, Michele
Structural characterization of human heat shock protein 90 N-Terminal domain and its variants K112R and K112A in complex with a potent 1,2,3-Triazole-based inhibitor
2022-01-01 Tassone, Giusy; Mazzorana, Marco; Mangani, Stefano; Petricci, Elena; Cini, Elena; Giannini, Giuseppe; Pozzi, Cecilia; Maramai, Samuele
Exploiting ELIOT for Scaffold-Repurposing Opportunities: TRIM33 a Possible Novel E3 Ligase to Expand the Toolbox for PROTAC Design
2022-01-01 Palomba, Tommaso; Tassone, Giusy; Vacca, Carmine; Bartalucci, Matteo; Valeri, Aurora; Pozzi, Cecilia; Cross, Simon; Siragusa, Lydia; Desantis, Jenny
Optimization of 1,2,4-Triazole-3-thiones toward Broad-Spectrum Metallo-β-lactamase Inhibitors Showing Potent Synergistic Activity on VIM- and NDM-1-Producing Clinical Isolates
2022-01-01 Legru, Alice; Verdirosa, Federica; Vo-Hoang, Yen; Tassone, Giusy; Vascon, Filippo; Thomas, Caitlyn A; Sannio, Filomena; Corsica, Giuseppina; Benvenuti, Manuela; Feller, Georges; Coulon, Rémi; Marcoccia, Francesca; Devente, Savannah Rowane; Bouajila, Ezeddine; Piveteau, Catherine; Leroux, Florence; Deprez-Poulain, Rebecca; Deprez, Benoît; Licznar-Fajardo, Patricia; Crowder, Michael W; Cendron, Laura; Pozzi, Cecilia; Mangani, Stefano; Docquier, Jean-Denis; Hernandez, Jean-François; Gavara, Laurent
1,2,4-Triazole-3-Thione analogues with a 2-Ethylbenzoic acid at position 4 as VIM-type metallo-β-Lactamase inhibitors
2022-01-01 Verdirosa, Federica; Gavara, Laurent; Sevaille, Laurent; Tassone, Giusy; Corsica, Giuseppina; Legru, Alice; Feller, Georges; Chelini, Giulia; Mercuri, Paola Sandra; Tanfoni, Silvia; Sannio, Filomena; Benvenuti, Manuela; Cerboni, Giulia; De Luca, Filomena; Bouajila, Ezeddine; Vo Hoang, Yen; Licznar-Fajardo, Patricia; Galleni, Moreno; Pozzi, Cecilia; Mangani, Stefano; Docquier, Jean-Denis; Hernandez, Jean-François
Structural Basis of Parasitic HSP90 ATPase Inhibition by Small Molecules
2022-01-01 Tassone, Giusy; Mazzorana, Marco; Pozzi, Cecilia
Xanthopsin-like systems via site-specific click-functionalization of a retinoic acid binding protein
2022-01-01 Tassone, G.; Paolino, M.; Pozzi, C.; Reale, A.; Salvini, L.; Giorgi, G.; Orlandini, M.; Galvagni, F.; Mangani, S.; Yang, X.; Carlotti, B.; Ortica, F.; Latterini, L.; Olivucci, M.; Cappelli, A.
Multitarget, selective compound design yields potent inhibitors of a Kinetoplastid Pteridine Reductase 1
2022-01-01 Pöhner, Ina; Quotadamo, Antonio; Panecka-Hofman, Joanna; Luciani, Rosaria; Santucci, Matteo; Linciano, Pasquale; Landi, Giacomo; Di Pisa, Flavio; Dello Iacono, Lucia; Pozzi, Cecilia; Mangani, Stefano; Gul, Sheraz; Witt, Gesa; Ellinger, Bernhard; Kuzikov, Maria; Santarem, Nuno; Cordeiro-da-Silva, Anabela; Costi, Maria P; Venturelli, Alberto; Wade, Rebecca C
Destabilizers of the thymidylate synthase homodimer accelerate its proteasomal degradation and inhibit cancer growth
2022-01-01 Costantino, Luca; Ferrari, Stefania; Santucci, Matteo; Salo-Ahen, Outi Mh; Carosati, Emanuele; Franchini, Silvia; Lauriola, Angela; Pozzi, Cecilia; Trande, Matteo; Gozzi, Gaia; Saxena, Puneet; Cannazza, Giuseppe; Losi, Lorena; Cardinale, Daniela; Venturelli, Alberto; Quotadamo, Antonio; Linciano, Pasquale; Tagliazucchi, Lorenzo; Moschella, Maria Gaetana; Guerrini, Remo; Pacifico, Salvatore; Luciani, Rosaria; Genovese, Filippo; Henrich, Stefan; Alboni, Silvia; Santarem, Nuno; Da Silva Cordeiro, Anabela; Giovannetti, Elisa; Peters, Godefridus J; Pinton, Paolo; Rimessi, Alessandro; Cruciani, Gabriele; Stroud, Robert M; Wade, Rebecca C; Mangani, Stefano; Marverti, Gaetano; D'Arca, Domenico; Ponterini, Glauco; Costi, Maria Paola
Iron Binding in the Ferroxidase Site of Human Mitochondrial Ferritin
2021-01-01 Ciambellotti, Silvia; Pratesi, Alessandro; Tassone, Giusy; Turano, Paola; Mangani, Stefano; Pozzi, Cecilia
1,2,4-Triazole-3-thione compounds with a 4-ethyl alkyl/aryl sulfide substituent are broad-spectrum metallo-β-lactamase inhibitors with re-sensitization activity
2021-01-01 Legru, Alice; Verdirosa, Federica; Hernandez, Jean-François; Tassone, Giusy; Sannio, Filomena; Benvenuti, Manuela; Conde, Pierre-Alexis; Bossis, Guillaume; Thomas, Caitlyn A; Crowder, Michael W; Dillenberger, Melissa; Becker, Katja; Pozzi, Cecilia; Mangani, Stefano; Docquier, Jean-Denis; Gavara, Laurent
| Titolo | Data di pubblicazione | Autore(i) | File | Abstract |
|---|---|---|---|---|
| Structural and antigen-binding surface definition of an anti-CD93 monoclonal antibody for the treatment of degenerative vascular eye diseases | 1-gen-2025 | Raucci, Luisa; Perrone, Cosimo Damiano; Barbera, Stefano; de Boer, Laurens Julius; Tosi, Gian Marco; Brunetti, Jlenia; Bracci, Luisa; Pozzi, Cecilia; Galvagni, Federico; Orlandini, Maurizio | - | |
| Morita−Baylis−Hillman Adduct Chemistry as a Tool for the Design of Lysine-Targeted Covalent Ligands | 1-gen-2025 | Paolino, Marco; Tassone, Giusy; Governa, Paolo; Saletti, Mario; Lami, Matteo; Carletti, Riccardo; Sacchetta, Filippo; Pozzi, Cecilia; Orlandini, Maurizio; Manetti, Fabrizio; Olivucci, Massimo; Cappelli, Andrea | - | |
| Design of 2-Aminobenzothiazole Derivatives Targeting Trypanosomatid PTR1 by a Multidisciplinary Fragment Hybridization Approach | 1-gen-2025 | Panecka-Hofman, Joanna; Linciano, Pasquale; Pöhner, Ina; Dyguda-Kazimierowicz, Edyta; Jedwabny, Wiktoria; Landi, Giacomo; Santarem, Nuno; Witt, Gesa; Ellinger, Bernhard; Kuzikov, Maria; Luciani, Rosaria; Ferrari, Stefania; Aiello, Daniele; Mangani, Stefano; Pozzi, Cecilia; Cordeiro-da-Silva, Anabela; Gul, Sheraz; Costi, Maria Paola; Wade, Rebecca C. | - | |
| Identification of pyrazolo-piperidinone derivatives targeting YAP-TEAD interface 3 as anticancer agents through integrated virtual screening and mass spectrometry proteomics | 1-gen-2025 | Scalvini, Laura; Tagliazucchi, Lorenzo; Elisi, Gian Marco; Zappaterra, Dana; Moschella, Maria Gaetana; Fantini, Sebastian; Aiello, Daniele; Guerrini, Remo; Albanese, Valentina; Pacifico, Salvatore; Lopresti, Ludovica; Malpezzi, Giulia; Saporito, Giulia; Ferrari, Stefania; Lamesta, Michele; Losi, Lorena; Pozzi, Cecilia; Mangani, Stefano; Marverti, Gaetano; Venturelli, Alberto; Ponterini, Glauco; D'Arca, Domenico; Mor, Marco; Costi, Maria Paola | - | |
| Metal ion binding to human Glutaminyl Cyclase: a structural perspective | 1-gen-2024 | Tassone, Giusy; Pozzi, Cecilia; Mangani, Stefano | - | |
| The discovery of aryl-2-nitroethyl triamino pyrimidines as anti-Trypanosoma brucei agents | 1-gen-2024 | Linciano, Pasquale; Pozzi, Cecilia; Tassone, Giusy; Landi, Giacomo; Mangani, Stefano; Santucci, Matteo; Luciani, Rosaria; Ferrari, Stefania; Santarem, Nuno; Tagliazucchi, Lorenzo; Cordeiro-da-Silva, Anabela; Tonelli, Michele; Tondi, Donatella; Bertarini, Laura; Gul, Sheraz; Witt, Gesa; B Moraes, Carolina; Costantino, Luca; Paola Costi, Maria | - | |
| Exploiting the bile acid binding protein as transporter of a Cholic Acid/Mirin bioconjugate for potential applications in liver cancer therapy | 1-gen-2024 | Tassone, Giusy; Maramai, Samuele; Paolino, Marco; Lamponi, Stefania; Poggialini, Federica; Dreassi, Elena; Petricci, Elena; Alcaro, Stefano; Pozzi, Cecilia; Romeo, Isabella | - | |
| Identification of Innovative Folate Inhibitors Leveraging the Amino Dihydrotriazine Motif from Cycloguanil for Their Potential as Anti-Trypanosoma brucei Agents | 1-gen-2024 | Francesconi, Valeria; Rizzo, Marco; Pozzi, Cecilia; Tagliazucchi, Lorenzo; Konchie Simo, Claude U.; Saporito, Giulia; Landi, Giacomo; Mangani, Stefano; Carbone, Anna; Schenone, Silvia; Santarém, Nuno; Tavares, Joana; Cordeiro-da-Silva, Anabela; Costi, Maria Paola; Tonelli, Michele | - | |
| Dimerization of the C-type lectin-like receptor CD93 promotes its binding to Multimerin-2 in endothelial cells | 1-gen-2023 | Barbera, Stefano; Raucci, Luisa; Tassone, Giusy; Tinti, Laura; Prischi, Filippo; Santucci, Annalisa; Mongiat, Maurizio; Tosi, Gian Marco; Galvagni, Federico; Dimberg, Anna; Pozzi, Cecilia; Orlandini, Maurizio | - | |
| Antitarget, Anti-SARS-CoV-2 Leads, Drugs, and the Drug Discovery-Genetics Alliance Perspective | 1-gen-2023 | Pozzi, Cecilia; Vanet, Anne; Francesconi, Valeria; Tagliazucchi, Lorenzo; Tassone, Giusy; Venturelli, Alberto; Spyrakis, Francesca; Mazzorana, Marco; P Costi, Maria; Tonelli, Michele | - | |
| Structural characterization of human heat shock protein 90 N-Terminal domain and its variants K112R and K112A in complex with a potent 1,2,3-Triazole-based inhibitor | 1-gen-2022 | Tassone, Giusy; Mazzorana, Marco; Mangani, Stefano; Petricci, Elena; Cini, Elena; Giannini, Giuseppe; Pozzi, Cecilia; Maramai, Samuele | - | |
| Exploiting ELIOT for Scaffold-Repurposing Opportunities: TRIM33 a Possible Novel E3 Ligase to Expand the Toolbox for PROTAC Design | 1-gen-2022 | Palomba, Tommaso; Tassone, Giusy; Vacca, Carmine; Bartalucci, Matteo; Valeri, Aurora; Pozzi, Cecilia; Cross, Simon; Siragusa, Lydia; Desantis, Jenny | - | |
| Optimization of 1,2,4-Triazole-3-thiones toward Broad-Spectrum Metallo-β-lactamase Inhibitors Showing Potent Synergistic Activity on VIM- and NDM-1-Producing Clinical Isolates | 1-gen-2022 | Legru, Alice; Verdirosa, Federica; Vo-Hoang, Yen; Tassone, Giusy; Vascon, Filippo; Thomas, Caitlyn A; Sannio, Filomena; Corsica, Giuseppina; Benvenuti, Manuela; Feller, Georges; Coulon, Rémi; Marcoccia, Francesca; Devente, Savannah Rowane; Bouajila, Ezeddine; Piveteau, Catherine; Leroux, Florence; Deprez-Poulain, Rebecca; Deprez, Benoît; Licznar-Fajardo, Patricia; Crowder, Michael W; Cendron, Laura; Pozzi, Cecilia; Mangani, Stefano; Docquier, Jean-Denis; Hernandez, Jean-François; Gavara, Laurent | - | |
| 1,2,4-Triazole-3-Thione analogues with a 2-Ethylbenzoic acid at position 4 as VIM-type metallo-β-Lactamase inhibitors | 1-gen-2022 | Verdirosa, Federica; Gavara, Laurent; Sevaille, Laurent; Tassone, Giusy; Corsica, Giuseppina; Legru, Alice; Feller, Georges; Chelini, Giulia; Mercuri, Paola Sandra; Tanfoni, Silvia; Sannio, Filomena; Benvenuti, Manuela; Cerboni, Giulia; De Luca, Filomena; Bouajila, Ezeddine; Vo Hoang, Yen; Licznar-Fajardo, Patricia; Galleni, Moreno; Pozzi, Cecilia; Mangani, Stefano; Docquier, Jean-Denis; Hernandez, Jean-François | - | |
| Structural Basis of Parasitic HSP90 ATPase Inhibition by Small Molecules | 1-gen-2022 | Tassone, Giusy; Mazzorana, Marco; Pozzi, Cecilia | - | |
| Xanthopsin-like systems via site-specific click-functionalization of a retinoic acid binding protein | 1-gen-2022 | Tassone, G.; Paolino, M.; Pozzi, C.; Reale, A.; Salvini, L.; Giorgi, G.; Orlandini, M.; Galvagni, F.; Mangani, S.; Yang, X.; Carlotti, B.; Ortica, F.; Latterini, L.; Olivucci, M.; Cappelli, A. | - | |
| Multitarget, selective compound design yields potent inhibitors of a Kinetoplastid Pteridine Reductase 1 | 1-gen-2022 | Pöhner, Ina; Quotadamo, Antonio; Panecka-Hofman, Joanna; Luciani, Rosaria; Santucci, Matteo; Linciano, Pasquale; Landi, Giacomo; Di Pisa, Flavio; Dello Iacono, Lucia; Pozzi, Cecilia; Mangani, Stefano; Gul, Sheraz; Witt, Gesa; Ellinger, Bernhard; Kuzikov, Maria; Santarem, Nuno; Cordeiro-da-Silva, Anabela; Costi, Maria P; Venturelli, Alberto; Wade, Rebecca C | - | |
| Destabilizers of the thymidylate synthase homodimer accelerate its proteasomal degradation and inhibit cancer growth | 1-gen-2022 | Costantino, Luca; Ferrari, Stefania; Santucci, Matteo; Salo-Ahen, Outi Mh; Carosati, Emanuele; Franchini, Silvia; Lauriola, Angela; Pozzi, Cecilia; Trande, Matteo; Gozzi, Gaia; Saxena, Puneet; Cannazza, Giuseppe; Losi, Lorena; Cardinale, Daniela; Venturelli, Alberto; Quotadamo, Antonio; Linciano, Pasquale; Tagliazucchi, Lorenzo; Moschella, Maria Gaetana; Guerrini, Remo; Pacifico, Salvatore; Luciani, Rosaria; Genovese, Filippo; Henrich, Stefan; Alboni, Silvia; Santarem, Nuno; Da Silva Cordeiro, Anabela; Giovannetti, Elisa; Peters, Godefridus J; Pinton, Paolo; Rimessi, Alessandro; Cruciani, Gabriele; Stroud, Robert M; Wade, Rebecca C; Mangani, Stefano; Marverti, Gaetano; D'Arca, Domenico; Ponterini, Glauco; Costi, Maria Paola | - | |
| Iron Binding in the Ferroxidase Site of Human Mitochondrial Ferritin | 1-gen-2021 | Ciambellotti, Silvia; Pratesi, Alessandro; Tassone, Giusy; Turano, Paola; Mangani, Stefano; Pozzi, Cecilia | - | |
| 1,2,4-Triazole-3-thione compounds with a 4-ethyl alkyl/aryl sulfide substituent are broad-spectrum metallo-β-lactamase inhibitors with re-sensitization activity | 1-gen-2021 | Legru, Alice; Verdirosa, Federica; Hernandez, Jean-François; Tassone, Giusy; Sannio, Filomena; Benvenuti, Manuela; Conde, Pierre-Alexis; Bossis, Guillaume; Thomas, Caitlyn A; Crowder, Michael W; Dillenberger, Melissa; Becker, Katja; Pozzi, Cecilia; Mangani, Stefano; Docquier, Jean-Denis; Gavara, Laurent | - |
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