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Antimalarial agents against both sexual and asexual parasites stages: structure-activity relationships and biological studies of the Malaria Box compound 1-[5-(4-bromo-2-chlorophenyl)furan-2-yl]- N -[(piperidin-4-yl)methyl]methanamine (MMV019918) and analogues
2018-01-01 Vallone, Alessandra; D'Alessandro, Sarah; Brogi, Simone; Brindisi, Margherita; Chemi, Giulia; Alfano, Gloria; Lamponi, Stefania; Lee, Soon Goo; Jez, Joseph M.; Koolen, Karin J. M.; Dechering, Koen J.; Saponara, Simona; Fusi, Fabio; Gorelli, Beatrice; Taramelli, Donatella; Parapini, Silvia; Caldelari, Reto; Campiani, Giuseppe; Gemma, Sandra; Butini, Stefania
Activation of the Wnt pathway by small peptides: rational design, synthesis and biological evaluation
2017-01-01 Brogi, Simone; Maramai, Samuele; Brindisi, Margherita; Chemi, Giulia; Porcari, Valentina; Corallo, Claudio; Gennari, Luigi; Novellino, Ettore; Ramunno, Anna; Butini, Stefania; Campiani, Giuseppe; Gemma, Sandra
Identification of novel fluorescent probes preventing PrP(Sc) replication in prion diseases
2017-01-01 Zaccagnini, Ludovica; Brogi, Simone; Brindisi, Margherita; Gemma, Sandra; Chemi, Giulia; Legname, Giuseppe; Campiani, Giuseppe; Butini, Stefania
First dual AK/GSK-3β inhibitors endowed with antioxidant properties as multifunctional, potential neuroprotective agents
2017-01-01 Brogi, Simone; Ramunno, Anna; Savi, Lida; Chemi, Giulia; Alfano, Gloria; Pecorelli, Alessandra; Pambianchi, Erika; Galatello, Paola; Compagnoni, Giulia; Focher, Federico; Biamonti, Giuseppe; Valacchi, Giuseppe; Butini, Stefania; Gemma, Sandra; Campiani, Giuseppe; Brindisi, Margherita
Computational tool for fast in silico evaluation of hERG K+ channel affinity
2017-01-01 Chemi, Giulia; Gemma, Sandra; Campiani, Giuseppe; Brogi, Simone; Butini, Stefania; Brindisi, Margherita
Structural characterization of Giardia duodenalis thioredoxin reductase (gTrxR) and computational analysis of its interaction with NBDHEX
2017-01-01 Brogi, Simone; Fiorillo, Annarita; Chemi, Giulia; Butini, Stefania; Lalle, Marco; Ilari, Andrea; Gemma, Sandra; Campiani, Giuseppe
Titolo | Data di pubblicazione | Autore(i) | File | Abstract |
---|---|---|---|---|
Antimalarial agents against both sexual and asexual parasites stages: structure-activity relationships and biological studies of the Malaria Box compound 1-[5-(4-bromo-2-chlorophenyl)furan-2-yl]- N -[(piperidin-4-yl)methyl]methanamine (MMV019918) and analogues | 1-gen-2018 | Vallone, Alessandra; D'Alessandro, Sarah; Brogi, Simone; Brindisi, Margherita; Chemi, Giulia; Alfano, Gloria; Lamponi, Stefania; Lee, Soon Goo; Jez, Joseph M.; Koolen, Karin J. M.; Dechering, Koen J.; Saponara, Simona; Fusi, Fabio; Gorelli, Beatrice; Taramelli, Donatella; Parapini, Silvia; Caldelari, Reto; Campiani, Giuseppe; Gemma, Sandra; Butini, Stefania | - | |
Activation of the Wnt pathway by small peptides: rational design, synthesis and biological evaluation | 1-gen-2017 | Brogi, Simone; Maramai, Samuele; Brindisi, Margherita; Chemi, Giulia; Porcari, Valentina; Corallo, Claudio; Gennari, Luigi; Novellino, Ettore; Ramunno, Anna; Butini, Stefania; Campiani, Giuseppe; Gemma, Sandra | - | |
Identification of novel fluorescent probes preventing PrP(Sc) replication in prion diseases | 1-gen-2017 | Zaccagnini, Ludovica; Brogi, Simone; Brindisi, Margherita; Gemma, Sandra; Chemi, Giulia; Legname, Giuseppe; Campiani, Giuseppe; Butini, Stefania | - | |
First dual AK/GSK-3β inhibitors endowed with antioxidant properties as multifunctional, potential neuroprotective agents | 1-gen-2017 | Brogi, Simone; Ramunno, Anna; Savi, Lida; Chemi, Giulia; Alfano, Gloria; Pecorelli, Alessandra; Pambianchi, Erika; Galatello, Paola; Compagnoni, Giulia; Focher, Federico; Biamonti, Giuseppe; Valacchi, Giuseppe; Butini, Stefania; Gemma, Sandra; Campiani, Giuseppe; Brindisi, Margherita | - | |
Computational tool for fast in silico evaluation of hERG K+ channel affinity | 1-gen-2017 | Chemi, Giulia; Gemma, Sandra; Campiani, Giuseppe; Brogi, Simone; Butini, Stefania; Brindisi, Margherita | - | |
Structural characterization of Giardia duodenalis thioredoxin reductase (gTrxR) and computational analysis of its interaction with NBDHEX | 1-gen-2017 | Brogi, Simone; Fiorillo, Annarita; Chemi, Giulia; Butini, Stefania; Lalle, Marco; Ilari, Andrea; Gemma, Sandra; Campiani, Giuseppe | - |
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