Sfoglia per Autore
Esc peptides as novel potentiators of defective cystic fibrosis transmembrane conductance regulator: an unprecedented property of antimicrobial peptides
2022-01-01 Ferrera, L.; Cappiello, F.; Loffredo, M. R.; Puglisi, E.; Casciaro, B.; Botta, B.; Galietta, L. J. V.; Mori, M.; Mangoni, M. L.
Discovery of spirooxadiazoline oxindoles with dual-stage antimalarial activity
2022-01-01 Lopes, E. A.; Mestre, R.; Fontinha, D.; Legac, J.; Pei, J. V.; Sanches-Vaz, M.; Mori, M.; Lehane, A. M.; Rosenthal, P. J.; Prudencio, M.; Santos, M. M. M.
A selective competitive inhibitor of aldehyde dehydrogenase 1A3 hinders cancer cell growth, invasiveness and stemness in vitro
2021-01-01 Gelardi, E. L. M.; Colombo, G.; Picarazzi, F.; Ferraris, D. M.; Mangione, A.; Petrarolo, G.; Aronica, E.; Rizzi, M.; Mori, M.; La Motta, C.; Garavaglia, S.
Active Components from Cassia abbreviata Prevent HIV-1 Entry by Distinct Mechanisms of Action
2021-01-01 Zheng, Yue; Yang, Xian-Wen; Schols, Dominique; Mori, Mattia; Botta, Bruno; Chevigné, Andy; Mulinge, Martin; Steinmetz, André; Schmit, Jean-Claude; Seguin-Devaux, Carole
Design and Synthesis of Piperazine-Based Compounds Conjugated to Humanized Ferritin as Delivery System of siRNA in Cancer Cells
2021-01-01 Pediconi, N.; Ghirga, F.; Del Plato, C.; Peruzzi, G.; Athanassopoulos, C. M.; Mori, M.; Crestoni, M. E.; Corinti, D.; Ugozzoli, F.; Massera, C.; Arcovito, A.; Botta, B.; Boffi, A.; Quaglio, D.; Baiocco, P.
Sofosbuvir selects for drug-resistant amino acid variants in the zika virus RNA-dependent RNA-polymerase complex in vitro
2021-01-01 Boccuto, A.; Dragoni, F.; Picarazzi, F.; Lai, A.; Ventura, C. D.; Veo, C.; Giammarino, F.; Saladini, F.; Zehender, G.; Zazzi, M.; Mori, M.; Vicenti, I.
Identification of effective anticancer g-quadruplex-targeting chemotypes through the exploration of a high diversity library of natural compounds
2021-01-01 Platella, C.; Ghirga, F.; Zizza, P.; Pompili, L.; Marzano, S.; Pagano, B.; Quaglio, D.; Vergine, V.; Cammarone, S.; Botta, B.; Biroccio, A.; Mori, M.; Montesarchio, D.
Design and Synthesis of New Withaferin A Inspired Hedgehog Pathway Inhibitors
2021-01-01 Bonandi, E.; Mori, M.; Infante, P.; Basili, I.; Di Marcotullio, L.; Calcaterra, A.; Catti, F.; Botta, B.; Passarella, D.
Hepatic miR-144 Drives Fumarase Activity Preventing NRF2 Activation During Obesity
2021-01-01 Azzimato, V.; Chen, P.; Barreby, E.; Morgantini, C.; Levi, L.; Vankova, A.; Jager, J.; Sulen, A.; Diotallevi, M.; Shen, J. X.; Miller, A.; Ellis, E.; Ryden, M.; Naslund, E.; Thorell, A.; Lauschke, V. M.; Channon, K. M.; Crabtree, M. J.; Haschemi, A.; Craige, S. M.; Mori, M.; Spallotta, F.; Aouadi, M.
Glabrescione B delivery by self-assembling micelles efficiently inhibits tumor growth in preclinical models of Hedgehog-dependent medulloblastoma
2021-01-01 Infante, P.; Malfanti, A.; Quaglio, D.; Balducci, S.; De Martin, S.; Bufalieri, F.; Mastrotto, F.; Basili, I.; Garofalo, M.; Lospinoso Severini, L.; Mori, M.; Manni, I.; Moretti, M.; Nicoletti, C.; Piaggio, G.; Caliceti, P.; Botta, B.; Ghirga, F.; Salmaso, S.; Di Marcotullio, L.
INHIBITORS OF ANTIBIOTIC RESISTANCE MEDIATED BY ARN T
2020-01-01 Imperi, Francesco; Ascenzioni, Fiorentina; Mori, Mattia; Ghirga, Francesca; Quaglio, Deborah; Corradi, Silvia; LO SCIUTO, Alessandra; Botta, Bruno; Calcaterra, Andrea; Stefanelli, Roberta
Dual smo/braf inhibition by flavonolignans from silybum marianum†
2020-01-01 Diukendjieva, A.; Zaharieva, M. M.; Mori, M.; Alov, P.; Tsakovska, I.; Pencheva, T.; Najdenski, H.; Kren, V.; Felici, C.; Bufalieri, F.; Di Marcotullio, L.; Botta, B.; Botta, M.; Pajeva, I.
Evaluation of sofosbuvir activity and resistance profile against West Nile virus in vitro.
2020-01-01 Dragoni, F; Boccuto, A; Picarazzi, F; Giannini, A; Giammarino, F; Saladini, F; Mori, M; Mastrangelo, E; Zazzi, M; Vicenti, I.
Targeting the RdRp of Emerging RNA Viruses: The Structure-Based Drug Design Challenge
2020-01-01 Picarazzi, F.; Vicenti, I.; Saladini, F.; Zazzi, M.; Mori, M.
What makes thienoguanosine an outstanding fluorescent DNA probe?
2020-01-01 Mely, Y.; Kuchlyan, J.; Martinez-Fernandez, L.; Mori, M.; Gavvala, K.; Ciaco, S.; Boudier, C.; Richert, L.; Didier, P.; Tor, Y.; Improta, R.
In Memory of Maurizio Botta: His Vision of Medicinal Chemistry
2020-01-01 Botta, Lorenzo; Mori, Mattia
Discovery of small molecule inhibitors of Leishmania braziliensis Hsp90 chaperone
2020-01-01 Batista, F. A. H.; Ramos, S. L.; Tassone, G.; Leitao, A.; Montanari, C. A.; Botta, M.; Mori, M.; Borges, J. C.
Structural Elucidation and Antimicrobial Characterization of Novel Diterpenoids from Fabiana densa var. ramulosa
2020-01-01 Quaglio, D.; Corradi, S.; Erazo, S.; Vergine, V.; Berardozzi, S.; Sciubba, F.; Cappiello, F.; Crestoni, M. E.; Ascenzioni, F.; Imperi, F.; Delle Monache, F.; Mori, M.; Loffredo, M. R.; Ghirga, F.; Casciaro, B.; Botta, B.; Mangoni, M. L.
Experimental and Computational Druggability Exploration of the 14-3-3ζ/SOS1pS1161PPI Interface
2020-01-01 Ballone, A.; Picarazzi, F.; Prosser, C.; Davis, J.; Ottmann, C.; Mori, M.
Ent-Beyerane Diterpenes as a Key Platform for the Development of ArnT-Mediated Colistin Resistance Inhibitors
2020-01-01 Quaglio, D.; Mangoni, M. L.; Stefanelli, R.; Corradi, S.; Casciaro, B.; Vergine, V.; Lucantoni, F.; Cavinato, L.; Cammarone, S.; Loffredo, M. R.; Cappiello, F.; Calcaterra, A.; Erazo, S.; Ghirga, F.; Mori, M.; Imperi, F.; Ascenzioni, F.; Botta, B.
| Titolo | Data di pubblicazione | Autore(i) | File | Abstract |
|---|---|---|---|---|
| Esc peptides as novel potentiators of defective cystic fibrosis transmembrane conductance regulator: an unprecedented property of antimicrobial peptides | 1-gen-2022 | Ferrera, L.; Cappiello, F.; Loffredo, M. R.; Puglisi, E.; Casciaro, B.; Botta, B.; Galietta, L. J. V.; Mori, M.; Mangoni, M. L. | - | |
| Discovery of spirooxadiazoline oxindoles with dual-stage antimalarial activity | 1-gen-2022 | Lopes, E. A.; Mestre, R.; Fontinha, D.; Legac, J.; Pei, J. V.; Sanches-Vaz, M.; Mori, M.; Lehane, A. M.; Rosenthal, P. J.; Prudencio, M.; Santos, M. M. M. | - | |
| A selective competitive inhibitor of aldehyde dehydrogenase 1A3 hinders cancer cell growth, invasiveness and stemness in vitro | 1-gen-2021 | Gelardi, E. L. M.; Colombo, G.; Picarazzi, F.; Ferraris, D. M.; Mangione, A.; Petrarolo, G.; Aronica, E.; Rizzi, M.; Mori, M.; La Motta, C.; Garavaglia, S. | - | |
| Active Components from Cassia abbreviata Prevent HIV-1 Entry by Distinct Mechanisms of Action | 1-gen-2021 | Zheng, Yue; Yang, Xian-Wen; Schols, Dominique; Mori, Mattia; Botta, Bruno; Chevigné, Andy; Mulinge, Martin; Steinmetz, André; Schmit, Jean-Claude; Seguin-Devaux, Carole | - | |
| Design and Synthesis of Piperazine-Based Compounds Conjugated to Humanized Ferritin as Delivery System of siRNA in Cancer Cells | 1-gen-2021 | Pediconi, N.; Ghirga, F.; Del Plato, C.; Peruzzi, G.; Athanassopoulos, C. M.; Mori, M.; Crestoni, M. E.; Corinti, D.; Ugozzoli, F.; Massera, C.; Arcovito, A.; Botta, B.; Boffi, A.; Quaglio, D.; Baiocco, P. | - | |
| Sofosbuvir selects for drug-resistant amino acid variants in the zika virus RNA-dependent RNA-polymerase complex in vitro | 1-gen-2021 | Boccuto, A.; Dragoni, F.; Picarazzi, F.; Lai, A.; Ventura, C. D.; Veo, C.; Giammarino, F.; Saladini, F.; Zehender, G.; Zazzi, M.; Mori, M.; Vicenti, I. | - | |
| Identification of effective anticancer g-quadruplex-targeting chemotypes through the exploration of a high diversity library of natural compounds | 1-gen-2021 | Platella, C.; Ghirga, F.; Zizza, P.; Pompili, L.; Marzano, S.; Pagano, B.; Quaglio, D.; Vergine, V.; Cammarone, S.; Botta, B.; Biroccio, A.; Mori, M.; Montesarchio, D. | - | |
| Design and Synthesis of New Withaferin A Inspired Hedgehog Pathway Inhibitors | 1-gen-2021 | Bonandi, E.; Mori, M.; Infante, P.; Basili, I.; Di Marcotullio, L.; Calcaterra, A.; Catti, F.; Botta, B.; Passarella, D. | - | |
| Hepatic miR-144 Drives Fumarase Activity Preventing NRF2 Activation During Obesity | 1-gen-2021 | Azzimato, V.; Chen, P.; Barreby, E.; Morgantini, C.; Levi, L.; Vankova, A.; Jager, J.; Sulen, A.; Diotallevi, M.; Shen, J. X.; Miller, A.; Ellis, E.; Ryden, M.; Naslund, E.; Thorell, A.; Lauschke, V. M.; Channon, K. M.; Crabtree, M. J.; Haschemi, A.; Craige, S. M.; Mori, M.; Spallotta, F.; Aouadi, M. | - | |
| Glabrescione B delivery by self-assembling micelles efficiently inhibits tumor growth in preclinical models of Hedgehog-dependent medulloblastoma | 1-gen-2021 | Infante, P.; Malfanti, A.; Quaglio, D.; Balducci, S.; De Martin, S.; Bufalieri, F.; Mastrotto, F.; Basili, I.; Garofalo, M.; Lospinoso Severini, L.; Mori, M.; Manni, I.; Moretti, M.; Nicoletti, C.; Piaggio, G.; Caliceti, P.; Botta, B.; Ghirga, F.; Salmaso, S.; Di Marcotullio, L. | - | |
| INHIBITORS OF ANTIBIOTIC RESISTANCE MEDIATED BY ARN T | 1-gen-2020 | Imperi, Francesco; Ascenzioni, Fiorentina; Mori, Mattia; Ghirga, Francesca; Quaglio, Deborah; Corradi, Silvia; LO SCIUTO, Alessandra; Botta, Bruno; Calcaterra, Andrea; Stefanelli, Roberta | - | |
| Dual smo/braf inhibition by flavonolignans from silybum marianum† | 1-gen-2020 | Diukendjieva, A.; Zaharieva, M. M.; Mori, M.; Alov, P.; Tsakovska, I.; Pencheva, T.; Najdenski, H.; Kren, V.; Felici, C.; Bufalieri, F.; Di Marcotullio, L.; Botta, B.; Botta, M.; Pajeva, I. | - | |
| Evaluation of sofosbuvir activity and resistance profile against West Nile virus in vitro. | 1-gen-2020 | Dragoni, F; Boccuto, A; Picarazzi, F; Giannini, A; Giammarino, F; Saladini, F; Mori, M; Mastrangelo, E; Zazzi, M; Vicenti, I. | - | |
| Targeting the RdRp of Emerging RNA Viruses: The Structure-Based Drug Design Challenge | 1-gen-2020 | Picarazzi, F.; Vicenti, I.; Saladini, F.; Zazzi, M.; Mori, M. | - | |
| What makes thienoguanosine an outstanding fluorescent DNA probe? | 1-gen-2020 | Mely, Y.; Kuchlyan, J.; Martinez-Fernandez, L.; Mori, M.; Gavvala, K.; Ciaco, S.; Boudier, C.; Richert, L.; Didier, P.; Tor, Y.; Improta, R. | - | |
| In Memory of Maurizio Botta: His Vision of Medicinal Chemistry | 1-gen-2020 | Botta, Lorenzo; Mori, Mattia | - | |
| Discovery of small molecule inhibitors of Leishmania braziliensis Hsp90 chaperone | 1-gen-2020 | Batista, F. A. H.; Ramos, S. L.; Tassone, G.; Leitao, A.; Montanari, C. A.; Botta, M.; Mori, M.; Borges, J. C. | - | |
| Structural Elucidation and Antimicrobial Characterization of Novel Diterpenoids from Fabiana densa var. ramulosa | 1-gen-2020 | Quaglio, D.; Corradi, S.; Erazo, S.; Vergine, V.; Berardozzi, S.; Sciubba, F.; Cappiello, F.; Crestoni, M. E.; Ascenzioni, F.; Imperi, F.; Delle Monache, F.; Mori, M.; Loffredo, M. R.; Ghirga, F.; Casciaro, B.; Botta, B.; Mangoni, M. L. | - | |
| Experimental and Computational Druggability Exploration of the 14-3-3ζ/SOS1pS1161PPI Interface | 1-gen-2020 | Ballone, A.; Picarazzi, F.; Prosser, C.; Davis, J.; Ottmann, C.; Mori, M. | - | |
| Ent-Beyerane Diterpenes as a Key Platform for the Development of ArnT-Mediated Colistin Resistance Inhibitors | 1-gen-2020 | Quaglio, D.; Mangoni, M. L.; Stefanelli, R.; Corradi, S.; Casciaro, B.; Vergine, V.; Lucantoni, F.; Cavinato, L.; Cammarone, S.; Loffredo, M. R.; Cappiello, F.; Calcaterra, A.; Erazo, S.; Ghirga, F.; Mori, M.; Imperi, F.; Ascenzioni, F.; Botta, B. | - |
Legenda icone
- file ad accesso aperto
- file disponibili sulla rete interna
- file disponibili agli utenti autorizzati
- file disponibili solo agli amministratori
- file sotto embargo
- nessun file disponibile