Sfoglia per Autore
Hypoxia as a driver of resistance to immunotherapy
2021-01-01 Kopecka, J.; Salaroglio, I. C.; Perez-Ruiz, E.; Sarmento-Ribeiro, A. B.; Saponara, S.; De Las Rivas, J.; Riganti, C.
Ritanserin blocks CaV1.2 channels in rat artery smooth muscles: electrophysiological, functional, and computational studies
2020-01-01 Fusi, F.; Trezza, A.; Sgaragli, G.; Spiga, O.; Saponara, S.; Bova, S.
Design, synthesis and pharmacological evaluation of ester-based quercetin derivatives as selective vascular KCa1.1 channel stimulators
2020-01-01 Carullo, G.; Ahmed, A.; Trezza, A.; Spiga, O.; Brizzi, A.; Saponara, S.; Fusi, F.; Aiello, F.
Vasorelaxant Effects Induced by Red Wine and Pomace Extracts of Magliocco Dolce cv
2020-01-01 Carullo, G.; Ahmed, A.; Fusi, F.; Sciubba, F.; Di Cocco, M. E.; Restuccia, D.; Spizzirri, U. G.; Saponara, S.; Aiello, F.
In vitro vascular toxicity assessment of NitDOX, a novel NO-releasing doxorubicin
2020-01-01 Durante, M.; Frosini, M.; Fusi, F.; Gamberucci, A.; Chegaev, K.; Rolando, B.; Riganti, C.; Fruttero, R.; Saponara, S.
Antihypertensive, cardio-and neuroprotective effects of Tenebrio molitor (Coleoptera: Tenebrionidae) defatted larvae in spontaneously hypertensive rats
2020-01-01 Pessina, F.; Frosini, M.; Marcolongo, P.; Fusi, F.; Saponara, S.; Gamberucci, A.; Valoti, M.; Giustarini, D.; Fiorenzani, P.; Gorelli, B.; Francardi, V.; Botta, M.; Dreassi, E.
Repurposing old drugs to fight multidrug resistant cancers
2020-01-01 Dinic, J.; Efferth, T.; Garcia-Sosa, A. T.; Grahovac, J.; Padron, J. M.; Pajeva, I.; Rizzolio, F.; Saponara, S.; Spengler, G.; Tsakovska, I.
The beneficial health effects of flavonoids on the cardiovascular system: focus on K+ channels
2020-01-01 Fusi, F; Trezza, A; Tramaglino, M; Sgaragli, G; Saponara, S; Spiga, O
The selective rat toxicant norbormide blocks KATP channels in smooth muscle cells but not in insulin-secreting cells
2019-01-01 Saponara, S.; Fusi, F.; Spiga, O.; Trezza, A.; Hopkins, B.; Brimble, M. A.; Rennison, D.; Bova, S.
Hyaluronated liposomes containing H2S-releasing doxorubicin are effective against P-glycoprotein-positive/doxorubicin-resistant osteosarcoma cells and xenografts
2019-01-01 Gazzano, E.; Buondonno, I.; Marengo, A.; Rolando, B.; Chegaev, K.; Kopecka, J.; Saponara, S.; Sorge, M.; Hattinger, C. M.; Gasco, A.; Fruttero, R.; Brancaccio, M.; Serra, M.; Stella, B.; Fattal, E.; Arpicco, S.; Riganti, C.
The multi-factorial nature of clinical multidrug resistance in cancer
2019-01-01 Assaraf, Yehuda G.; Brozovic, Anamaria; Cristina Gonçalves, Ana; Jurkovicova, Dana; Linē, Aija; Machuqueiro, Miguel; Saponara, Simona; Bela Sarmento-Ribeiro, Ana; R Xavier, Cristina P; Helena Vasconcelos, M
Vasoactivity of Mantonico and Pecorello grape pomaces on rat aorta rings: An insight into nutraceutical development
2019-01-01 Carullo, G.; Durante, M.; Sciubba, F.; Restuccia, D.; Spizzirri, U. G.; Ahmed, A.; Di Cocco, M. E.; Saponara S., ; Aiello, F.; Fusi, F.
Negative chronotropism, positive inotropism and lusitropism of 3,5-di-t-butyl-4-hydroxyanisole (DTBHA) on rat heart preparations occur through reduction of RyR2 Ca2+ leak
2018-01-01 Pessina, Federica; Gamberucci, Alessandra; Chen, Jialin; Liu, Boyin; Vangheluwe, Peter; Gorelli, Beatrice; Lorenzini, Stefania; Spiga, Ottavia; Trezza, Alfonso; Sgaragli, Giampietro; Saponara, Simona
Antimalarial agents against both sexual and asexual parasites stages: structure-activity relationships and biological studies of the Malaria Box compound 1-[5-(4-bromo-2-chlorophenyl)furan-2-yl]- N -[(piperidin-4-yl)methyl]methanamine (MMV019918) and analogues
2018-01-01 Vallone, Alessandra; D'Alessandro, Sarah; Brogi, Simone; Brindisi, Margherita; Chemi, Giulia; Alfano, Gloria; Lamponi, Stefania; Lee, Soon Goo; Jez, Joseph M.; Koolen, Karin J. M.; Dechering, Koen J.; Saponara, Simona; Fusi, Fabio; Gorelli, Beatrice; Taramelli, Donatella; Parapini, Silvia; Caldelari, Reto; Campiani, Giuseppe; Gemma, Sandra; Butini, Stefania
New NO- and H2S-releasing doxorubicins as targeted therapy against chemoresistance in castration-resistant prostate cancer: in vitro and in vivo evaluations
2018-01-01 Bigagli, Elisabetta; Luceri, Cristina; DE ANGIOLETTI, Maria; Chegaev, Konstantin; D’Ambrosio, Mario; Riganti, Chiara; Gazzano, Elena; Saponara, Simona; Longini, Mariangela; Luceri, Francesca; Cinci, Lorenzo
Interference measurements and failure analysis of patch-clamp laboratory instrumentation for electrophysiology tests
2018-01-01 Saponara, S.; Fusi, F.; Saponara, S.; Macucci, M.; Groza, V
Folate-targeted liposomal nitrooxy-doxorubicin: an effective tool against P-glycoprotein-positive and folate receptor-positive tumors
2018-01-01 Gazzano, Elena; Rolando, Barbara; Chegaev, Konstantin; Salaroglio, Iris C.; Kopecka, Joanna; Pedrini, Isabella; Saponara, Simona; Sorge, Matteo; Buondonno, Ilaria; Stella, Barbara; Marengo, Alessandro; Valoti, Massimo; Brancaccio, Mara; Fruttero, Roberta; Gasco, Alberto; Arpicco, Silvia; Riganti, Chiara
From in silico to in vitro: A trip to reveal flavonoid binding on the Rattus norvegicus Kir6.1 ATP-sensitive inward rectifier potassium channel
2018-01-01 Trezza, Alfonso; Cicaloni, Vittoria; Porciatti, Piera; Langella, Andrea; Fusi, Fabio; Saponara, Simona; Spiga, Ottavia
The surge of flavonoids as novel, fine regulators of cardiovascular Cav channels
2017-01-01 Fusi, Fabio; Spiga, Ottavia; Trezza, Alfonso; Sgaragli, Giampietro; Saponara, Simona
Failure Effect Analysis of Patch-Clamp Electronic Instrumentation in Electrophysiology Experiments
2017-01-01 Saponara, Sergio; Fusi, Fabio; Saponara, Simona; Macucci, Massimo
Titolo | Data di pubblicazione | Autore(i) | File | Abstract |
---|---|---|---|---|
Hypoxia as a driver of resistance to immunotherapy | 1-gen-2021 | Kopecka, J.; Salaroglio, I. C.; Perez-Ruiz, E.; Sarmento-Ribeiro, A. B.; Saponara, S.; De Las Rivas, J.; Riganti, C. | - | |
Ritanserin blocks CaV1.2 channels in rat artery smooth muscles: electrophysiological, functional, and computational studies | 1-gen-2020 | Fusi, F.; Trezza, A.; Sgaragli, G.; Spiga, O.; Saponara, S.; Bova, S. | - | |
Design, synthesis and pharmacological evaluation of ester-based quercetin derivatives as selective vascular KCa1.1 channel stimulators | 1-gen-2020 | Carullo, G.; Ahmed, A.; Trezza, A.; Spiga, O.; Brizzi, A.; Saponara, S.; Fusi, F.; Aiello, F. | - | |
Vasorelaxant Effects Induced by Red Wine and Pomace Extracts of Magliocco Dolce cv | 1-gen-2020 | Carullo, G.; Ahmed, A.; Fusi, F.; Sciubba, F.; Di Cocco, M. E.; Restuccia, D.; Spizzirri, U. G.; Saponara, S.; Aiello, F. | - | |
In vitro vascular toxicity assessment of NitDOX, a novel NO-releasing doxorubicin | 1-gen-2020 | Durante, M.; Frosini, M.; Fusi, F.; Gamberucci, A.; Chegaev, K.; Rolando, B.; Riganti, C.; Fruttero, R.; Saponara, S. | - | |
Antihypertensive, cardio-and neuroprotective effects of Tenebrio molitor (Coleoptera: Tenebrionidae) defatted larvae in spontaneously hypertensive rats | 1-gen-2020 | Pessina, F.; Frosini, M.; Marcolongo, P.; Fusi, F.; Saponara, S.; Gamberucci, A.; Valoti, M.; Giustarini, D.; Fiorenzani, P.; Gorelli, B.; Francardi, V.; Botta, M.; Dreassi, E. | - | |
Repurposing old drugs to fight multidrug resistant cancers | 1-gen-2020 | Dinic, J.; Efferth, T.; Garcia-Sosa, A. T.; Grahovac, J.; Padron, J. M.; Pajeva, I.; Rizzolio, F.; Saponara, S.; Spengler, G.; Tsakovska, I. | - | |
The beneficial health effects of flavonoids on the cardiovascular system: focus on K+ channels | 1-gen-2020 | Fusi, F; Trezza, A; Tramaglino, M; Sgaragli, G; Saponara, S; Spiga, O | - | |
The selective rat toxicant norbormide blocks KATP channels in smooth muscle cells but not in insulin-secreting cells | 1-gen-2019 | Saponara, S.; Fusi, F.; Spiga, O.; Trezza, A.; Hopkins, B.; Brimble, M. A.; Rennison, D.; Bova, S. | - | |
Hyaluronated liposomes containing H2S-releasing doxorubicin are effective against P-glycoprotein-positive/doxorubicin-resistant osteosarcoma cells and xenografts | 1-gen-2019 | Gazzano, E.; Buondonno, I.; Marengo, A.; Rolando, B.; Chegaev, K.; Kopecka, J.; Saponara, S.; Sorge, M.; Hattinger, C. M.; Gasco, A.; Fruttero, R.; Brancaccio, M.; Serra, M.; Stella, B.; Fattal, E.; Arpicco, S.; Riganti, C. | - | |
The multi-factorial nature of clinical multidrug resistance in cancer | 1-gen-2019 | Assaraf, Yehuda G.; Brozovic, Anamaria; Cristina Gonçalves, Ana; Jurkovicova, Dana; Linē, Aija; Machuqueiro, Miguel; Saponara, Simona; Bela Sarmento-Ribeiro, Ana; R Xavier, Cristina P; Helena Vasconcelos, M | - | |
Vasoactivity of Mantonico and Pecorello grape pomaces on rat aorta rings: An insight into nutraceutical development | 1-gen-2019 | Carullo, G.; Durante, M.; Sciubba, F.; Restuccia, D.; Spizzirri, U. G.; Ahmed, A.; Di Cocco, M. E.; Saponara S., ; Aiello, F.; Fusi, F. | - | |
Negative chronotropism, positive inotropism and lusitropism of 3,5-di-t-butyl-4-hydroxyanisole (DTBHA) on rat heart preparations occur through reduction of RyR2 Ca2+ leak | 1-gen-2018 | Pessina, Federica; Gamberucci, Alessandra; Chen, Jialin; Liu, Boyin; Vangheluwe, Peter; Gorelli, Beatrice; Lorenzini, Stefania; Spiga, Ottavia; Trezza, Alfonso; Sgaragli, Giampietro; Saponara, Simona | - | |
Antimalarial agents against both sexual and asexual parasites stages: structure-activity relationships and biological studies of the Malaria Box compound 1-[5-(4-bromo-2-chlorophenyl)furan-2-yl]- N -[(piperidin-4-yl)methyl]methanamine (MMV019918) and analogues | 1-gen-2018 | Vallone, Alessandra; D'Alessandro, Sarah; Brogi, Simone; Brindisi, Margherita; Chemi, Giulia; Alfano, Gloria; Lamponi, Stefania; Lee, Soon Goo; Jez, Joseph M.; Koolen, Karin J. M.; Dechering, Koen J.; Saponara, Simona; Fusi, Fabio; Gorelli, Beatrice; Taramelli, Donatella; Parapini, Silvia; Caldelari, Reto; Campiani, Giuseppe; Gemma, Sandra; Butini, Stefania | - | |
New NO- and H2S-releasing doxorubicins as targeted therapy against chemoresistance in castration-resistant prostate cancer: in vitro and in vivo evaluations | 1-gen-2018 | Bigagli, Elisabetta; Luceri, Cristina; DE ANGIOLETTI, Maria; Chegaev, Konstantin; D’Ambrosio, Mario; Riganti, Chiara; Gazzano, Elena; Saponara, Simona; Longini, Mariangela; Luceri, Francesca; Cinci, Lorenzo | - | |
Interference measurements and failure analysis of patch-clamp laboratory instrumentation for electrophysiology tests | 1-gen-2018 | Saponara, S.; Fusi, F.; Saponara, S.; Macucci, M.; Groza, V | - | |
Folate-targeted liposomal nitrooxy-doxorubicin: an effective tool against P-glycoprotein-positive and folate receptor-positive tumors | 1-gen-2018 | Gazzano, Elena; Rolando, Barbara; Chegaev, Konstantin; Salaroglio, Iris C.; Kopecka, Joanna; Pedrini, Isabella; Saponara, Simona; Sorge, Matteo; Buondonno, Ilaria; Stella, Barbara; Marengo, Alessandro; Valoti, Massimo; Brancaccio, Mara; Fruttero, Roberta; Gasco, Alberto; Arpicco, Silvia; Riganti, Chiara | - | |
From in silico to in vitro: A trip to reveal flavonoid binding on the Rattus norvegicus Kir6.1 ATP-sensitive inward rectifier potassium channel | 1-gen-2018 | Trezza, Alfonso; Cicaloni, Vittoria; Porciatti, Piera; Langella, Andrea; Fusi, Fabio; Saponara, Simona; Spiga, Ottavia | - | |
The surge of flavonoids as novel, fine regulators of cardiovascular Cav channels | 1-gen-2017 | Fusi, Fabio; Spiga, Ottavia; Trezza, Alfonso; Sgaragli, Giampietro; Saponara, Simona | - | |
Failure Effect Analysis of Patch-Clamp Electronic Instrumentation in Electrophysiology Experiments | 1-gen-2017 | Saponara, Sergio; Fusi, Fabio; Saponara, Simona; Macucci, Massimo | - |
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