Sfoglia per Autore
Early investigation of a novel SI306 theranostic prodrug for glioblastoma treatment
2024-01-01 Vagaggini, Chiara; Petroni, Debora; D'Agostino, Ilaria; Poggialini, Federica; Cavallini, Chiara; Cianciusi, Annarita; Salis, Annalisa; D'Antona, Lucia; Francesconi, Valeria; Manetti, Fabrizio; Damonte, Gianluca; Musumeci, Francesca; Menichetti, Luca; Dreassi, Elena; Carbone, Anna; Schenone, Silvia
Tenebrio molitor as a Simple and Cheap Preclinical Pharmacokinetic and Toxicity Model
2023-01-01 Brai, Annalaura; Poggialini, Federica; Vagaggini, Chiara; Pasqualini, Claudia; Simoni, Sauro; Francardi, Valeria; Dreassi, Elena
Biological Evaluation and In Vitro Characterization of ADME Profile of In-House Pyrazolo[3,4-d]pyrimidines as Dual Tyrosine Kinase Inhibitors Active against Glioblastoma Multiforme
2023-01-01 Poggialini, Federica; Vagaggini, Chiara; Brai, Annalaura; Pasqualini, Claudia; Crespan, Emmanuele; Maga, Giovanni; Perini, Cecilia; Cabella, Noemi; Botta, Lorenzo; Musumeci, Francesca; Frosini, Maria; Schenone, Silvia; Dreassi, Elena
Development and validation of derivatization-based LC-MS/MS method for quantification of short-chain fatty acids in human, rat, and mouse plasma
2023-01-01 Vagaggini, Chiara; Brai, Annalaura; Bonente, Denise; Lombardi, Jessica; Poggialini, Federica; Pasqualini, Claudia; Barone, Virginia; Nicoletti, Claudio; Bertelli, Eugenio; Dreassi, Elena
Brevundimonas aurantiaca M3d10, Isolated from the olive fly, produces hydroxylated astaxanthin
2023-01-01 Centini, Marisanna; Martinez-Sañudo, Isabel; Biagi, Marco; Dreassi, Elena; Mazzon, Luca; Marri, Laura
Triazolo[3,4- b]benzothiazole Scaffold as Versatile Nicotinamide Mimic Allowing Nanomolar Inhibition of Different PARP Enzymes
2023-01-01 Murthy, S.; Nizi, M. G.; Maksimainen, M. M.; Massari, S.; Alaviuhkola, J.; Lippok, B. E.; Vagaggini, C.; Sowa, S. T.; Galera-Prat, A.; Ashok, Y.; Venkannagari, H.; Prunskaite-Hyyrylainen, R.; Dreassi, E.; Luscher, B.; Korn, P.; Tabarrini, O.; Lehtio, L.
Use of distillery by-products as Tenebrio molitor mealworm feed supplement
2023-01-01 Brai, A.; Vagaggini, C.; Pasqualini, C.; Poggialini, F.; Tarchi, F.; Francardi, V.; Dreassi, E.
Efficient use of agricultural waste to naturally fortify Tenebrio molitor mealworms and evaluation of their nutraceutical properties
2023-01-01 Brai, A.; Poggialini, F.; Trivisani, C. I.; Vagaggini, C.; Tarchi, F.; Francardi, V.; Dreassi, E.
Discovery and Optimization of a Novel Macrocyclic Amidinourea Series Active as Acidic Mammalian Chitinase Inhibitors
2023-01-01 Balestri, Lorenzo Jacopo Ilic; Trivisani, Claudia Immacolata; Orofino, Francesco; Fiorucci, Diego; Truglio, Giuseppina Ivana; D'Agostino, Ilaria; Poggialini, Federica; Botta, Lorenzo; Docquier, Jean-Denis; Dreassi, Elena
Tyrosine Kinase Inhibitor Si409 Has In Vitro and In Vivo Anti-Tumor Activity Against Diffuse Large B-Cell Lymphoma
2023-01-01 Rango, E.; Di Maria, S.; Zamperini, C.; Poggialini, F.; Crespan, E.; Perini, C.; Sabetta, S.; Saponara, S.; Fusi, F.; Maga, G.; Angelucci, A.; Gaudio, E.; Berton, F.; Schenone, S.; Botta, L.; Dreassi, E.; Botta, M.
Progress towards Adjuvant Development: Focus on Antiviral Therapy
2023-01-01 Brai, A.; Poggialini, F.; Pasqualini, C.; Trivisani, C. I.; Vagaggini, C.; Dreassi, E.
Targeting GLI1 and GLI2 with small molecule inhibitors to suppress GLI-dependent transcription and tumor growth
2023-01-01 Maresca, Luisa; Crivaro, Enrica; Migliorini, Francesca; Anichini, Giulia; Giammona, Alessandro; Pepe, Sara; Poggialini, Federica; Vagaggini, Chiara; Giannini, Giuseppe; Sestini, Serena; Borgognoni, Lorenzo; Lapucci, Andrea; Dreassi, Elena; Taddei, Maurizio; Manetti, Fabrizio; Petricci, Elena; Stecca, Barbara
Privileged Scaffold Decoration for the Identification of the First Trisubstituted Triazine with Anti-SARS-CoV-2 Activity
2022-01-01 Cesarini, Silvia; Vicenti, Ilaria; Poggialini, Federica; Secchi, Massimiliano; Giammarino, Federica; Varasi, Ilenia; Lodola, Camilla; Zazzi, Maurizio; Dreassi, Elena; Maga, Giovanni; Botta, Lorenzo; Saladino, Raffaele
The impact of counterions in biological activity: case study of antibacterial alkylguanidino ureas
2022-01-01 Ardino, C.; Sannio, F.; Pasero, C.; Botta, L.; Dreassi, E.; Docquier, J. D.; D'Agostino, I.
A Greener Technique for Microwave-Assisted O-Silylation and Silyl Ether Deprotection of Uridine and Other Substrates
2022-01-01 Pasqualini, C.; Poggialini, F.; Vagaggini, C.; Brai, A.; Dreassi, E.
Serum Metabolomics and Proteomics to Study the Antihypertensive Effect of Protein Extracts from Tenebrio molitor
2022-01-01 Stella, Roberto; Peggion, Caterina; Bergantin, Caterina; Biancotto, Giancarlo; Frosini, Maria; Dreassi, Elena; Marcolongo, Paola; Aloisi, Anna Maria; Pessina, Federica
A pH-responsive crosslinker platform for antibody-drug conjugate (ADC) targeting delivery
2022-01-01 Migliorini, Francesca; Cini, Elena; Dreassi, Elena; Finetti, Federica; Ievoli, Giovanni; Macrì, Giulia; Petricci, Elena; Rango, Enrico; Trabalzini, Lorenza; Taddei, Maurizio
Antibacterial alkylguanidino ureas: Molecular simplification approach, searching for membrane-based MoA
2022-01-01 D'Agostino, I.; Ardino, C.; Poli, G.; Sannio, F.; Lucidi, M.; Poggialini, F.; Visaggio, D.; Rango, E.; Filippi, S.; Petricci, E.; Visca, P.; Botta, L.; Docquier, J. -D.; Dreassi, E.
Novel pyrazolo[3,4-d]pyrimidines as dual Src/Bcr-Abl kinase inhibitors: Synthesis and biological evaluation for chronic myeloid leukemia treatment
2022-01-01 Di Maria, S.; Picarazzi, F.; Mori, M.; Cianciusi, A.; Carbone, A.; Crespan, E.; Perini, C.; Sabetta, S.; Deplano, S.; Poggialini, F.; Molinari, A.; Aronne, R.; Maccioni, E.; Maga, G.; Angelucci, A.; Schenone, S.; Musumeci, F.; Dreassi, E.
Reversible Monoacylglycerol Lipase Inhibitors: Discovery of a New Class of Benzylpiperidine Derivatives
2022-01-01 Bononi, Giulia; Di Stefano, Miriana; Poli, Giulio; Ortore, Gabriella; Meier, Philip; Masetto, Francesca; Caligiuri, Isabella; Rizzolio, Flavio; Macchia, Marco; Chicca, Andrea; Avan, Amir; Giovannetti, Elisa; Vagaggini, Chiara; Brai, Annalaura; Dreassi, Elena; Valoti, Massimo; Minutolo, Filippo; Granchi, Carlotta; Gertsch, Jürg; Tuccinardi, Tiziano
| Titolo | Data di pubblicazione | Autore(i) | File | Abstract |
|---|---|---|---|---|
| Early investigation of a novel SI306 theranostic prodrug for glioblastoma treatment | 1-gen-2024 | Vagaggini, Chiara; Petroni, Debora; D'Agostino, Ilaria; Poggialini, Federica; Cavallini, Chiara; Cianciusi, Annarita; Salis, Annalisa; D'Antona, Lucia; Francesconi, Valeria; Manetti, Fabrizio; Damonte, Gianluca; Musumeci, Francesca; Menichetti, Luca; Dreassi, Elena; Carbone, Anna; Schenone, Silvia | - | |
| Tenebrio molitor as a Simple and Cheap Preclinical Pharmacokinetic and Toxicity Model | 1-gen-2023 | Brai, Annalaura; Poggialini, Federica; Vagaggini, Chiara; Pasqualini, Claudia; Simoni, Sauro; Francardi, Valeria; Dreassi, Elena | - | |
| Biological Evaluation and In Vitro Characterization of ADME Profile of In-House Pyrazolo[3,4-d]pyrimidines as Dual Tyrosine Kinase Inhibitors Active against Glioblastoma Multiforme | 1-gen-2023 | Poggialini, Federica; Vagaggini, Chiara; Brai, Annalaura; Pasqualini, Claudia; Crespan, Emmanuele; Maga, Giovanni; Perini, Cecilia; Cabella, Noemi; Botta, Lorenzo; Musumeci, Francesca; Frosini, Maria; Schenone, Silvia; Dreassi, Elena | - | |
| Development and validation of derivatization-based LC-MS/MS method for quantification of short-chain fatty acids in human, rat, and mouse plasma | 1-gen-2023 | Vagaggini, Chiara; Brai, Annalaura; Bonente, Denise; Lombardi, Jessica; Poggialini, Federica; Pasqualini, Claudia; Barone, Virginia; Nicoletti, Claudio; Bertelli, Eugenio; Dreassi, Elena | - | |
| Brevundimonas aurantiaca M3d10, Isolated from the olive fly, produces hydroxylated astaxanthin | 1-gen-2023 | Centini, Marisanna; Martinez-Sañudo, Isabel; Biagi, Marco; Dreassi, Elena; Mazzon, Luca; Marri, Laura | - | |
| Triazolo[3,4- b]benzothiazole Scaffold as Versatile Nicotinamide Mimic Allowing Nanomolar Inhibition of Different PARP Enzymes | 1-gen-2023 | Murthy, S.; Nizi, M. G.; Maksimainen, M. M.; Massari, S.; Alaviuhkola, J.; Lippok, B. E.; Vagaggini, C.; Sowa, S. T.; Galera-Prat, A.; Ashok, Y.; Venkannagari, H.; Prunskaite-Hyyrylainen, R.; Dreassi, E.; Luscher, B.; Korn, P.; Tabarrini, O.; Lehtio, L. | - | |
| Use of distillery by-products as Tenebrio molitor mealworm feed supplement | 1-gen-2023 | Brai, A.; Vagaggini, C.; Pasqualini, C.; Poggialini, F.; Tarchi, F.; Francardi, V.; Dreassi, E. | - | |
| Efficient use of agricultural waste to naturally fortify Tenebrio molitor mealworms and evaluation of their nutraceutical properties | 1-gen-2023 | Brai, A.; Poggialini, F.; Trivisani, C. I.; Vagaggini, C.; Tarchi, F.; Francardi, V.; Dreassi, E. | - | |
| Discovery and Optimization of a Novel Macrocyclic Amidinourea Series Active as Acidic Mammalian Chitinase Inhibitors | 1-gen-2023 | Balestri, Lorenzo Jacopo Ilic; Trivisani, Claudia Immacolata; Orofino, Francesco; Fiorucci, Diego; Truglio, Giuseppina Ivana; D'Agostino, Ilaria; Poggialini, Federica; Botta, Lorenzo; Docquier, Jean-Denis; Dreassi, Elena | - | |
| Tyrosine Kinase Inhibitor Si409 Has In Vitro and In Vivo Anti-Tumor Activity Against Diffuse Large B-Cell Lymphoma | 1-gen-2023 | Rango, E.; Di Maria, S.; Zamperini, C.; Poggialini, F.; Crespan, E.; Perini, C.; Sabetta, S.; Saponara, S.; Fusi, F.; Maga, G.; Angelucci, A.; Gaudio, E.; Berton, F.; Schenone, S.; Botta, L.; Dreassi, E.; Botta, M. | - | |
| Progress towards Adjuvant Development: Focus on Antiviral Therapy | 1-gen-2023 | Brai, A.; Poggialini, F.; Pasqualini, C.; Trivisani, C. I.; Vagaggini, C.; Dreassi, E. | - | |
| Targeting GLI1 and GLI2 with small molecule inhibitors to suppress GLI-dependent transcription and tumor growth | 1-gen-2023 | Maresca, Luisa; Crivaro, Enrica; Migliorini, Francesca; Anichini, Giulia; Giammona, Alessandro; Pepe, Sara; Poggialini, Federica; Vagaggini, Chiara; Giannini, Giuseppe; Sestini, Serena; Borgognoni, Lorenzo; Lapucci, Andrea; Dreassi, Elena; Taddei, Maurizio; Manetti, Fabrizio; Petricci, Elena; Stecca, Barbara | - | |
| Privileged Scaffold Decoration for the Identification of the First Trisubstituted Triazine with Anti-SARS-CoV-2 Activity | 1-gen-2022 | Cesarini, Silvia; Vicenti, Ilaria; Poggialini, Federica; Secchi, Massimiliano; Giammarino, Federica; Varasi, Ilenia; Lodola, Camilla; Zazzi, Maurizio; Dreassi, Elena; Maga, Giovanni; Botta, Lorenzo; Saladino, Raffaele | - | |
| The impact of counterions in biological activity: case study of antibacterial alkylguanidino ureas | 1-gen-2022 | Ardino, C.; Sannio, F.; Pasero, C.; Botta, L.; Dreassi, E.; Docquier, J. D.; D'Agostino, I. | - | |
| A Greener Technique for Microwave-Assisted O-Silylation and Silyl Ether Deprotection of Uridine and Other Substrates | 1-gen-2022 | Pasqualini, C.; Poggialini, F.; Vagaggini, C.; Brai, A.; Dreassi, E. | - | |
| Serum Metabolomics and Proteomics to Study the Antihypertensive Effect of Protein Extracts from Tenebrio molitor | 1-gen-2022 | Stella, Roberto; Peggion, Caterina; Bergantin, Caterina; Biancotto, Giancarlo; Frosini, Maria; Dreassi, Elena; Marcolongo, Paola; Aloisi, Anna Maria; Pessina, Federica | - | |
| A pH-responsive crosslinker platform for antibody-drug conjugate (ADC) targeting delivery | 1-gen-2022 | Migliorini, Francesca; Cini, Elena; Dreassi, Elena; Finetti, Federica; Ievoli, Giovanni; Macrì, Giulia; Petricci, Elena; Rango, Enrico; Trabalzini, Lorenza; Taddei, Maurizio | - | |
| Antibacterial alkylguanidino ureas: Molecular simplification approach, searching for membrane-based MoA | 1-gen-2022 | D'Agostino, I.; Ardino, C.; Poli, G.; Sannio, F.; Lucidi, M.; Poggialini, F.; Visaggio, D.; Rango, E.; Filippi, S.; Petricci, E.; Visca, P.; Botta, L.; Docquier, J. -D.; Dreassi, E. | - | |
| Novel pyrazolo[3,4-d]pyrimidines as dual Src/Bcr-Abl kinase inhibitors: Synthesis and biological evaluation for chronic myeloid leukemia treatment | 1-gen-2022 | Di Maria, S.; Picarazzi, F.; Mori, M.; Cianciusi, A.; Carbone, A.; Crespan, E.; Perini, C.; Sabetta, S.; Deplano, S.; Poggialini, F.; Molinari, A.; Aronne, R.; Maccioni, E.; Maga, G.; Angelucci, A.; Schenone, S.; Musumeci, F.; Dreassi, E. | - | |
| Reversible Monoacylglycerol Lipase Inhibitors: Discovery of a New Class of Benzylpiperidine Derivatives | 1-gen-2022 | Bononi, Giulia; Di Stefano, Miriana; Poli, Giulio; Ortore, Gabriella; Meier, Philip; Masetto, Francesca; Caligiuri, Isabella; Rizzolio, Flavio; Macchia, Marco; Chicca, Andrea; Avan, Amir; Giovannetti, Elisa; Vagaggini, Chiara; Brai, Annalaura; Dreassi, Elena; Valoti, Massimo; Minutolo, Filippo; Granchi, Carlotta; Gertsch, Jürg; Tuccinardi, Tiziano | - |
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