Sfoglia per Autore
Selective Delivery of Anticancer Natural G-Quadruplex Ligands by the AT11 Aptamer for Gastric Cancer Treatment
2026-01-01 Platella, Chiara; Trajkovski, Marko; Brancaccio, Mariarita; Di Palma, Rosita; Calcaterra, Andrea; Mori, Mattia; Falco, Geppino; Plavec, Janez; Montesarchio, Daniela
Protonation State-dependent Interaction of Polycationic Polymyxins with the Pseudomonas aeruginosa Outer Membrane Using Colistin A as a Model
2026-01-01 Cutarella, Luigi; Temprano, Alvaro G.; Tafi, Andrea; Mori, Mattia
Exploration of the aromatic abietane diterpenoid scaffold in the development of ArnT-mediated colistin resistance inhibitors
2026-01-01 Cammarone, Silvia; Pastore, Valentina; Ryzhuk, Mariya; Cristoferi, Martina; Speroni, Arianna; Imperi, Francesco; Corinti, Davide; Bonaccorsi Di Patti, Maria Carmela; Botta, Bruno; Quaglio, Deborah; Mori, Mattia; Ascenzioni, Fiorentina; Ghirga, Francesca
Discovery of a Mixed and Prodrug-Like Inhibition Mechanism for Phosphocoumarins and Phosphoquinolinones against Human Carbonic Anhydrases
2026-01-01 Nocentini, Alessio; Giovannuzzi, Simone; Alterio, Vincenzo; Bonardi, Alessandro; Barons, Rudolfs; Zalubovskis, Raivis; Eldehna, Wagdy M.; Aronne, Rossella; Esposito, Davide; Luchinat, Enrico; De Simone, Giuseppina; Bartolucci, Gianluca; Gratteri, Paola; Mori, Mattia; Supuran, Claudiu T.
Probing the Structure and Dynamics of Telomeric G-Quadruplexes with Thienoguanosine, a Fluorescent Analogue of Guanosine
2026-01-01 Singh, Pankhi; Mukherjee, Dipanjan; Hanser, Fabien; Tkach, Olha; Humbert, Nicolas; Avendano Avila, Constanza; Ciaco, Stefano; Martinez-Fernandez, Lara; Bansal, Sarthak; Kanj, Samuel; Bombarda, Elisa; Bourderioux, Aurélie; Dziuba, Dmytro; Tor, Yitzhak; Improta, Roberto; Mori, Mattia; Heddi, Brahim; Mély, Yves
α-ketoglutarate/succinate ratio imbalance impairs thymine DNA glycosylase function and base excision repair process increasing susceptibility to pancreatic cancer
2026-01-01 Malatesta, Silvia; Vigiano Benedetti, Virginia; Salviati, Emanuela; Illi, Barbara; Manni, Isabella; Middonti, Emanuele; Rampioni Vinciguerra, Gian Luca; Licursi, Valerio; Troilo, Francesca; Colotti, Gianni; Cipolla, Lina; Sabbioneda, Simone; Perfetto, Livia; Piaggio, Giulia; Bussolino, Federico; Di Nicolantonio, Federica; Campiglia, Pietro; Sommella, Eduardo Maria; Mori, Mattia; Cencioni, Chiara; Spallotta, Francesco
Discovery of a new selective ERAP1 inhibitor for Hedgehog-dependent cancer treatment
2026-01-01 Bufalieri, Francesca; Cucinotta, Antonino; Cammarone, Silvia; Agnoli, Francesca; Basili, Irene; Ferri, Giulia; Quaglio, Deborah; Caimano, Miriam; Capriotti, Anna Laura; Montone, Carmela Maria; Lospinoso Severini, Ludovica; Tempora, Patrizia; D'Amico, Silvia; Juretich, Francesca; Semrau, Marta S.; Navacci, Shirin; Conenna, Marilisa; Bordone, Rosa; Spallotta, Francesco; Garavaglia, Silvia; Storici, Paola; Ghirga, Francesca; Laganà, Aldo; Locatelli, Franco; Ayrault, Olivier; Infante, Paola; Botta, Bruno; Mori, Mattia; Fruci, Doriana; Di Marcotullio, Lucia
A scaffold repositioning approach: dihydroBenzoImidazoTriazineDione (BITD) derivatives as selective ALDH1A1 inhibitors
2026-01-01 Bernardoni, Bianca Laura; D'Agostino, Ilaria; Siragusa, Sonia; Mori, Mattia; Garavaglia, Silvia; La Motta, Concettina
Harder than Metal: Challenging Antimicrobial Resistance with Metallo-β-lactamase Inhibitors
2025-01-01 De Falco, Antonietta; Alfano, Antonella Ilenia; Cutarella, Luigi; Mori, Mattia; Brindisi, Margherita
Functional and therapeutic effects of Glabrescione B delivery by liposomes on Hedgehog-dependent tumors
2025-01-01 Infante, Paola; Daniele, Raffaella; Bottero, Marta; Longo, Mariagrazia; Bufalieri, Francesca; Lospinoso Severini, Ludovica; Pesce, Cristiano; Fragassi, Agnese; Gabbia, Daniela; Navacci, Shirin; Basili, Irene; Adabbo, Gennaro; Cammarone, Silvia; Cianfoni, Gabriele; Ghirga, Francesca; Mori, Mattia; De Martin, Sara; Mancuso, Mariateresa; Caliceti, Paolo; Pazzaglia, Simonetta; Salmaso, Stefano; Di Marcotullio, Lucia
Plectranthus‐derived Abietanes as Protein Kinase C‐δ Activators: In Silico Design, Human Serum Albumin Interaction, and Stability Evaluation
2025-01-01 Isca, Vera M. S.; Nikolić, Milan; Filipović, Nenad; Mori, Mattia; Rijo, Patricia
Retargeting Gram-Positive-Only Adarotene-Derived Antibacterials to Broad-Spectrum Antibiotics
2025-01-01 Princiotto, Salvatore; Cutarella, Luigi; Fortuna, Alessandra; Mellini, Marta; Casciaro, Bruno; Loffredo, Maria Rosa; Temprano, Alvaro G.; Cappiello, Floriana; Leoni, Livia; Mangoni, Maria Luisa; Mori, Mattia; Musso, Loana; Sacchi, Francesca; Pinna, Cecilia; Rampioni, Giordano; Dallavalle, Sabrina; Pisano, Claudio
Decoding the base flipping mechanism of the SET- and RING-associated (SRA) domain of the epigenetic UHRF1 protein
2025-01-01 Mukherjee, Dipanjan; Ciaco, Stefano; Martinez-Fernandez, Lara; Gavvala, Krishna; Bombarda, Elisa; Bourdérioux, Aurélie; Dziuba, Dmytro; Hanser, Fabien; Humbert, Nicolas; Javed, Aqib; Mousli, Marc; Singh, Pankhi; Tor, Yitzhak; Improta, Roberto; Mori, Mattia; Mély, Yves
The dual-site agonist for human M2 muscarinic receptors Iper-8-naphtalimide induces mitochondrial dysfunction in Saccharomyces cerevisiae
2025-01-01 Cirigliano, Angela; Amelina, Antonia; Passarini, Elena; Ricelli, Alessandra; Balasco, Nicole; Mori, Mattia; Botta, Bruno; De Stefano, Maria Egle; Papotto, Claudio; Guerriero, Claudia; Tata, Ada Maria; Rinaldi, Teresa
Biological Evaluation and Computational Modelling Studies on N-acyl Hydrazone and 2,5-Disubstituted 1,3,4-Oxadiazole Derivatives as Non-toxic Antimicrobial Agents
2025-01-01 Giray, Betul; Kaya, Nil; Fiabane, Martina; Buyuk, Ayse Seyma; Kucuk, Hatice Başpinar; Sardas, Semra; Mori, Mattia
Structure-Based Ligandability Exploration of a G-Quadruplex-Forming Sequence from the Pseudomonas aeruginosa Genome
2025-01-01 Fiabane, Martina; Platella, Chiara; Diaco, Fabiana; Biancucci, Cristiano; Calcaterra, Andrea; Musumeci, Domenica; Antonelli, Guido; Turriziani, Ombretta; Botta, Bruno; Montesarchio, Daniela; Mori, Mattia
Design, synthesis, molecular modelling investigation and biological studies of novel human carbonic anhydrase inhibitors based on coumalic acid
2025-01-01 Pontecorvi, Virginia; Angeli, Andrea; Cutarella, Luigi; Mori, Mattia; Secci, Daniela; Coluccia, Michele; Carradori, Simone; Troiani, Anna; Pepi, Federico; Salvitti, Chiara; Di Noi, Alessia; Spano, Mattia; Arrighi, Francesca; De Falco, Elena; Bordin, Antonella; Berrino, Emanuela; Granese, Arianna; Chimenti, Paola; Guglielmi, Paolo; Supuran, Claudiu T.
Antibacterial activity of tamoxifen derivatives against methicillin-resistant Staphylococcus aureus
2025-01-01 Molina Panadero, Irene; Falcón Torres, Javier; Hmadcha, Abdelkrim; Princiotto, Salvatore; Cutarella, Luigi; Mori, Mattia; Dallavalle, Sabrina; Christodoulou, Michael S.; Smani, Younes
Sustainable Joullié–Ugi and Continuous Flow Implementation Led to Novel Captopril-Inspired Broad-Spectrum Metallo-β-Lactamase Inhibitors
2025-01-01 Alfano, Antonella Ilenia; Pelliccia, Sveva; Barone, Simona; Cutarella, Luigi; Cancade, Sacha Michèle Idriss; Baia, Valerio; Cassese, Emilia; Russomanno, Pasquale; Messano, Nicolò; Frank, Denia; Weizel, Lilia; Rotter, Marco J.; Brunst, Steffen; Wichelhaus, Thomas A.; Proschak, Ewgenij; Tedesco, Daniele; Mori, Mattia; Docquier, Jean Denis; Summa, Vincenzo; Brindisi, Margherita
A novel noninvasive test based on near-infrared fluorescent cholephilic probes for hepatobiliary secretory function assessment
2025-01-01 Sanchez De Blas, Beatriz; Temprano, Alvaro G.; Cives-Losada, Candela; Briz, Oscar; Lozano, Elisa; Martinez-Chantar, Maria L.; Avila, Matias A.; Mori, Mattia; Ghallab, Ahmed; Hengstler, Jan G.; Perez-Melero, Concepción; Bermejo-Gonzalez, Francisco A.; Monte, Maria J.; Romero, Marta R.; Marin, Jose J. G.
| Titolo | Data di pubblicazione | Autore(i) | File | Abstract |
|---|---|---|---|---|
| Selective Delivery of Anticancer Natural G-Quadruplex Ligands by the AT11 Aptamer for Gastric Cancer Treatment | 1-gen-2026 | Platella, Chiara; Trajkovski, Marko; Brancaccio, Mariarita; Di Palma, Rosita; Calcaterra, Andrea; Mori, Mattia; Falco, Geppino; Plavec, Janez; Montesarchio, Daniela | - | |
| Protonation State-dependent Interaction of Polycationic Polymyxins with the Pseudomonas aeruginosa Outer Membrane Using Colistin A as a Model | 1-gen-2026 | Cutarella, Luigi; Temprano, Alvaro G.; Tafi, Andrea; Mori, Mattia | - | |
| Exploration of the aromatic abietane diterpenoid scaffold in the development of ArnT-mediated colistin resistance inhibitors | 1-gen-2026 | Cammarone, Silvia; Pastore, Valentina; Ryzhuk, Mariya; Cristoferi, Martina; Speroni, Arianna; Imperi, Francesco; Corinti, Davide; Bonaccorsi Di Patti, Maria Carmela; Botta, Bruno; Quaglio, Deborah; Mori, Mattia; Ascenzioni, Fiorentina; Ghirga, Francesca | - | |
| Discovery of a Mixed and Prodrug-Like Inhibition Mechanism for Phosphocoumarins and Phosphoquinolinones against Human Carbonic Anhydrases | 1-gen-2026 | Nocentini, Alessio; Giovannuzzi, Simone; Alterio, Vincenzo; Bonardi, Alessandro; Barons, Rudolfs; Zalubovskis, Raivis; Eldehna, Wagdy M.; Aronne, Rossella; Esposito, Davide; Luchinat, Enrico; De Simone, Giuseppina; Bartolucci, Gianluca; Gratteri, Paola; Mori, Mattia; Supuran, Claudiu T. | - | |
| Probing the Structure and Dynamics of Telomeric G-Quadruplexes with Thienoguanosine, a Fluorescent Analogue of Guanosine | 1-gen-2026 | Singh, Pankhi; Mukherjee, Dipanjan; Hanser, Fabien; Tkach, Olha; Humbert, Nicolas; Avendano Avila, Constanza; Ciaco, Stefano; Martinez-Fernandez, Lara; Bansal, Sarthak; Kanj, Samuel; Bombarda, Elisa; Bourderioux, Aurélie; Dziuba, Dmytro; Tor, Yitzhak; Improta, Roberto; Mori, Mattia; Heddi, Brahim; Mély, Yves | - | |
| α-ketoglutarate/succinate ratio imbalance impairs thymine DNA glycosylase function and base excision repair process increasing susceptibility to pancreatic cancer | 1-gen-2026 | Malatesta, Silvia; Vigiano Benedetti, Virginia; Salviati, Emanuela; Illi, Barbara; Manni, Isabella; Middonti, Emanuele; Rampioni Vinciguerra, Gian Luca; Licursi, Valerio; Troilo, Francesca; Colotti, Gianni; Cipolla, Lina; Sabbioneda, Simone; Perfetto, Livia; Piaggio, Giulia; Bussolino, Federico; Di Nicolantonio, Federica; Campiglia, Pietro; Sommella, Eduardo Maria; Mori, Mattia; Cencioni, Chiara; Spallotta, Francesco | - | |
| Discovery of a new selective ERAP1 inhibitor for Hedgehog-dependent cancer treatment | 1-gen-2026 | Bufalieri, Francesca; Cucinotta, Antonino; Cammarone, Silvia; Agnoli, Francesca; Basili, Irene; Ferri, Giulia; Quaglio, Deborah; Caimano, Miriam; Capriotti, Anna Laura; Montone, Carmela Maria; Lospinoso Severini, Ludovica; Tempora, Patrizia; D'Amico, Silvia; Juretich, Francesca; Semrau, Marta S.; Navacci, Shirin; Conenna, Marilisa; Bordone, Rosa; Spallotta, Francesco; Garavaglia, Silvia; Storici, Paola; Ghirga, Francesca; Laganà, Aldo; Locatelli, Franco; Ayrault, Olivier; Infante, Paola; Botta, Bruno; Mori, Mattia; Fruci, Doriana; Di Marcotullio, Lucia | - | |
| A scaffold repositioning approach: dihydroBenzoImidazoTriazineDione (BITD) derivatives as selective ALDH1A1 inhibitors | 1-gen-2026 | Bernardoni, Bianca Laura; D'Agostino, Ilaria; Siragusa, Sonia; Mori, Mattia; Garavaglia, Silvia; La Motta, Concettina | - | |
| Harder than Metal: Challenging Antimicrobial Resistance with Metallo-β-lactamase Inhibitors | 1-gen-2025 | De Falco, Antonietta; Alfano, Antonella Ilenia; Cutarella, Luigi; Mori, Mattia; Brindisi, Margherita | - | |
| Functional and therapeutic effects of Glabrescione B delivery by liposomes on Hedgehog-dependent tumors | 1-gen-2025 | Infante, Paola; Daniele, Raffaella; Bottero, Marta; Longo, Mariagrazia; Bufalieri, Francesca; Lospinoso Severini, Ludovica; Pesce, Cristiano; Fragassi, Agnese; Gabbia, Daniela; Navacci, Shirin; Basili, Irene; Adabbo, Gennaro; Cammarone, Silvia; Cianfoni, Gabriele; Ghirga, Francesca; Mori, Mattia; De Martin, Sara; Mancuso, Mariateresa; Caliceti, Paolo; Pazzaglia, Simonetta; Salmaso, Stefano; Di Marcotullio, Lucia | - | |
| Plectranthus‐derived Abietanes as Protein Kinase C‐δ Activators: In Silico Design, Human Serum Albumin Interaction, and Stability Evaluation | 1-gen-2025 | Isca, Vera M. S.; Nikolić, Milan; Filipović, Nenad; Mori, Mattia; Rijo, Patricia | - | |
| Retargeting Gram-Positive-Only Adarotene-Derived Antibacterials to Broad-Spectrum Antibiotics | 1-gen-2025 | Princiotto, Salvatore; Cutarella, Luigi; Fortuna, Alessandra; Mellini, Marta; Casciaro, Bruno; Loffredo, Maria Rosa; Temprano, Alvaro G.; Cappiello, Floriana; Leoni, Livia; Mangoni, Maria Luisa; Mori, Mattia; Musso, Loana; Sacchi, Francesca; Pinna, Cecilia; Rampioni, Giordano; Dallavalle, Sabrina; Pisano, Claudio | - | |
| Decoding the base flipping mechanism of the SET- and RING-associated (SRA) domain of the epigenetic UHRF1 protein | 1-gen-2025 | Mukherjee, Dipanjan; Ciaco, Stefano; Martinez-Fernandez, Lara; Gavvala, Krishna; Bombarda, Elisa; Bourdérioux, Aurélie; Dziuba, Dmytro; Hanser, Fabien; Humbert, Nicolas; Javed, Aqib; Mousli, Marc; Singh, Pankhi; Tor, Yitzhak; Improta, Roberto; Mori, Mattia; Mély, Yves | - | |
| The dual-site agonist for human M2 muscarinic receptors Iper-8-naphtalimide induces mitochondrial dysfunction in Saccharomyces cerevisiae | 1-gen-2025 | Cirigliano, Angela; Amelina, Antonia; Passarini, Elena; Ricelli, Alessandra; Balasco, Nicole; Mori, Mattia; Botta, Bruno; De Stefano, Maria Egle; Papotto, Claudio; Guerriero, Claudia; Tata, Ada Maria; Rinaldi, Teresa | - | |
| Biological Evaluation and Computational Modelling Studies on N-acyl Hydrazone and 2,5-Disubstituted 1,3,4-Oxadiazole Derivatives as Non-toxic Antimicrobial Agents | 1-gen-2025 | Giray, Betul; Kaya, Nil; Fiabane, Martina; Buyuk, Ayse Seyma; Kucuk, Hatice Başpinar; Sardas, Semra; Mori, Mattia | - | |
| Structure-Based Ligandability Exploration of a G-Quadruplex-Forming Sequence from the Pseudomonas aeruginosa Genome | 1-gen-2025 | Fiabane, Martina; Platella, Chiara; Diaco, Fabiana; Biancucci, Cristiano; Calcaterra, Andrea; Musumeci, Domenica; Antonelli, Guido; Turriziani, Ombretta; Botta, Bruno; Montesarchio, Daniela; Mori, Mattia | - | |
| Design, synthesis, molecular modelling investigation and biological studies of novel human carbonic anhydrase inhibitors based on coumalic acid | 1-gen-2025 | Pontecorvi, Virginia; Angeli, Andrea; Cutarella, Luigi; Mori, Mattia; Secci, Daniela; Coluccia, Michele; Carradori, Simone; Troiani, Anna; Pepi, Federico; Salvitti, Chiara; Di Noi, Alessia; Spano, Mattia; Arrighi, Francesca; De Falco, Elena; Bordin, Antonella; Berrino, Emanuela; Granese, Arianna; Chimenti, Paola; Guglielmi, Paolo; Supuran, Claudiu T. | - | |
| Antibacterial activity of tamoxifen derivatives against methicillin-resistant Staphylococcus aureus | 1-gen-2025 | Molina Panadero, Irene; Falcón Torres, Javier; Hmadcha, Abdelkrim; Princiotto, Salvatore; Cutarella, Luigi; Mori, Mattia; Dallavalle, Sabrina; Christodoulou, Michael S.; Smani, Younes | - | |
| Sustainable Joullié–Ugi and Continuous Flow Implementation Led to Novel Captopril-Inspired Broad-Spectrum Metallo-β-Lactamase Inhibitors | 1-gen-2025 | Alfano, Antonella Ilenia; Pelliccia, Sveva; Barone, Simona; Cutarella, Luigi; Cancade, Sacha Michèle Idriss; Baia, Valerio; Cassese, Emilia; Russomanno, Pasquale; Messano, Nicolò; Frank, Denia; Weizel, Lilia; Rotter, Marco J.; Brunst, Steffen; Wichelhaus, Thomas A.; Proschak, Ewgenij; Tedesco, Daniele; Mori, Mattia; Docquier, Jean Denis; Summa, Vincenzo; Brindisi, Margherita | - | |
| A novel noninvasive test based on near-infrared fluorescent cholephilic probes for hepatobiliary secretory function assessment | 1-gen-2025 | Sanchez De Blas, Beatriz; Temprano, Alvaro G.; Cives-Losada, Candela; Briz, Oscar; Lozano, Elisa; Martinez-Chantar, Maria L.; Avila, Matias A.; Mori, Mattia; Ghallab, Ahmed; Hengstler, Jan G.; Perez-Melero, Concepción; Bermejo-Gonzalez, Francisco A.; Monte, Maria J.; Romero, Marta R.; Marin, Jose J. G. | - |
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