Sfoglia per Autore
A scaffold repositioning approach: dihydroBenzoImidazoTriazineDione (BITD) derivatives as selective ALDH1A1 inhibitors
2026-01-01 Bernardoni, Bianca Laura; D'Agostino, Ilaria; Siragusa, Sonia; Mori, Mattia; Garavaglia, Silvia; La Motta, Concettina
Functional and therapeutic effects of Glabrescione B delivery by liposomes on Hedgehog-dependent tumors
2026-01-01 Infante, Paola; Daniele, Raffaella; Bottero, Marta; Longo, Mariagrazia; Bufalieri, Francesca; Lospinoso Severini, Ludovica; Pesce, Cristiano; Fragassi, Agnese; Gabbia, Daniela; Navacci, Shirin; Basili, Irene; Adabbo, Gennaro; Cammarone, Silvia; Cianfoni, Gabriele; Ghirga, Francesca; Mori, Mattia; De Martin, Sara; Mancuso, Mariateresa; Caliceti, Paolo; Pazzaglia, Simonetta; Salmaso, Stefano; Di Marcotullio, Lucia
Protonation State-dependent Interaction of Polycationic Polymyxins with the Pseudomonas aeruginosa Outer Membrane Using Colistin A as a Model
2026-01-01 Cutarella, Luigi; Temprano, Alvaro G.; Tafi, Andrea; Mori, Mattia
Exploration of the aromatic abietane diterpenoid scaffold in the development of ArnT-mediated colistin resistance inhibitors
2026-01-01 Cammarone, Silvia; Pastore, Valentina; Ryzhuk, Mariya; Cristoferi, Martina; Speroni, Arianna; Imperi, Francesco; Corinti, Davide; Bonaccorsi Di Patti, Maria Carmela; Botta, Bruno; Quaglio, Deborah; Mori, Mattia; Ascenzioni, Fiorentina; Ghirga, Francesca
Discovery of a new selective ERAP1 inhibitor for Hedgehog-dependent cancer treatment
2026-01-01 Bufalieri, Francesca; Cucinotta, Antonino; Cammarone, Silvia; Agnoli, Francesca; Basili, Irene; Ferri, Giulia; Quaglio, Deborah; Caimano, Miriam; Capriotti, Anna Laura; Montone, Carmela Maria; Lospinoso Severini, Ludovica; Tempora, Patrizia; D'Amico, Silvia; Juretich, Francesca; Semrau, Marta S.; Navacci, Shirin; Conenna, Marilisa; Bordone, Rosa; Spallotta, Francesco; Garavaglia, Silvia; Storici, Paola; Ghirga, Francesca; Laganà, Aldo; Locatelli, Franco; Ayrault, Olivier; Infante, Paola; Botta, Bruno; Mori, Mattia; Fruci, Doriana; Di Marcotullio, Lucia
α-ketoglutarate/succinate ratio imbalance impairs thymine DNA glycosylase function and base excision repair process increasing susceptibility to pancreatic cancer
2026-01-01 Malatesta, Silvia; Vigiano Benedetti, Virginia; Salviati, Emanuela; Illi, Barbara; Manni, Isabella; Middonti, Emanuele; Rampioni Vinciguerra, Gian Luca; Licursi, Valerio; Troilo, Francesca; Colotti, Gianni; Cipolla, Lina; Sabbioneda, Simone; Perfetto, Livia; Piaggio, Giulia; Bussolino, Federico; Di Nicolantonio, Federica; Campiglia, Pietro; Sommella, Eduardo Maria; Mori, Mattia; Cencioni, Chiara; Spallotta, Francesco
Discovery of a Mixed and Prodrug-Like Inhibition Mechanism for Phosphocoumarins and Phosphoquinolinones against Human Carbonic Anhydrases
2026-01-01 Nocentini, Alessio; Giovannuzzi, Simone; Alterio, Vincenzo; Bonardi, Alessandro; Barons, Rudolfs; Zalubovskis, Raivis; Eldehna, Wagdy M.; Aronne, Rossella; Esposito, Davide; Luchinat, Enrico; De Simone, Giuseppina; Bartolucci, Gianluca; Gratteri, Paola; Mori, Mattia; Supuran, Claudiu T.
Selective Delivery of Anticancer Natural G-Quadruplex Ligands by the AT11 Aptamer for Gastric Cancer Treatment
2026-01-01 Platella, Chiara; Trajkovski, Marko; Brancaccio, Mariarita; Di Palma, Rosita; Calcaterra, Andrea; Mori, Mattia; Falco, Geppino; Plavec, Janez; Montesarchio, Daniela
Probing the Structure and Dynamics of Telomeric G-Quadruplexes with Thienoguanosine, a Fluorescent Analogue of Guanosine
2026-01-01 Singh, Pankhi; Mukherjee, Dipanjan; Hanser, Fabien; Tkach, Olha; Humbert, Nicolas; Avendano Avila, Constanza; Ciaco, Stefano; Martinez-Fernandez, Lara; Bansal, Sarthak; Kanj, Samuel; Bombarda, Elisa; Bourderioux, Aurélie; Dziuba, Dmytro; Tor, Yitzhak; Improta, Roberto; Mori, Mattia; Heddi, Brahim; Mély, Yves
A novel noninvasive test based on near-infrared fluorescent cholephilic probes for hepatobiliary secretory function assessment
2025-01-01 Sanchez De Blas, Beatriz; Temprano, Alvaro G.; Cives-Losada, Candela; Briz, Oscar; Lozano, Elisa; Martinez-Chantar, Maria L.; Avila, Matias A.; Mori, Mattia; Ghallab, Ahmed; Hengstler, Jan G.; Perez-Melero, Concepción; Bermejo-Gonzalez, Francisco A.; Monte, Maria J.; Romero, Marta R.; Marin, Jose J. G.
Influenza a Virus Inhibition: Evaluating Computationally Identified Cyproheptadine Through In Vitro Assessment
2025-01-01 Glisic, Sanja; Stevanovic, Kristina; Perdih, Andrej; Bukreyeva, Natalya; Maruyama, Junki; Perovic, Vladimir; López-Serrano, Sergi; Darji, Ayub; Radosevic, Draginja; Sencanski, Milan; Veljkovic, Veljko; Botta, Bruno; Mori, Mattia; Paessler, Slobodan
The Production of Recombinant Azurin from Pseudomonas aeruginosa and Its Ability to Induce Apoptosis in Various Breast Cancer Cell Lines
2025-01-01 Kowalczyk, Tomasz; Merecz-Sadowska, Anna; Synowiec, Ewelina; Śliwiński, Tomasz; Piekarski, Janusz; Szemraj, Janusz; Mori, Mattia; Rijo, Patricia; Sitarek, Przemysław
Sustainable Joullié–Ugi and Continuous Flow Implementation Led to Novel Captopril-Inspired Broad-Spectrum Metallo-β-Lactamase Inhibitors
2025-01-01 Alfano, Antonella Ilenia; Pelliccia, Sveva; Barone, Simona; Cutarella, Luigi; Cancade, Sacha Michèle Idriss; Baia, Valerio; Cassese, Emilia; Russomanno, Pasquale; Messano, Nicolò; Frank, Denia; Weizel, Lilia; Rotter, Marco J.; Brunst, Steffen; Wichelhaus, Thomas A.; Proschak, Ewgenij; Tedesco, Daniele; Mori, Mattia; Docquier, Jean Denis; Summa, Vincenzo; Brindisi, Margherita
Development of nanovehicles for co-delivery of colistin and ArnT inhibitors
2025-01-01 Pastore, Valentina; Frison, Jessica; Pesce, Cristiano; Ryzhuk, Mariya; Garofalo, Mariangela; Cristoferi, Martina; Cammarone, Silvia; Fabrizio, Giorgia; Bonaccorsi Di Patti, Maria Carmela; Quaglio, Deborah; Ghirga, Francesca; Imperi, Francesco; Mori, Mattia; Caliceti, Paolo; Botta, Bruno; Ascenzioni, Fiorentina; Salmaso, Stefano
Biological Evaluation and Computational Modelling Studies on N-acyl Hydrazone and 2,5-Disubstituted 1,3,4-Oxadiazole Derivatives as Non-toxic Antimicrobial Agents
2025-01-01 Giray, Betul; Kaya, Nil; Fiabane, Martina; Buyuk, Ayse Seyma; Kucuk, Hatice Başpinar; Sardas, Semra; Mori, Mattia
Discovery of Indole-Based PDE5 Inhibitors: Synthesis and Pharmacological Evaluation
2025-01-01 Park, Shin-Young; Pham, Dang; Shukla, Param; Edward, Justin; John, Reshmi; Li, Addison; Hadjiargyrou, Michael; Mori, Mattia; Zuccarello, Elisa; Arancio, Ottavio; Fiorito, Jole
Antibacterial activity of tamoxifen derivatives against methicillin-resistant Staphylococcus aureus
2025-01-01 Molina Panadero, Irene; Falcón Torres, Javier; Hmadcha, Abdelkrim; Princiotto, Salvatore; Cutarella, Luigi; Mori, Mattia; Dallavalle, Sabrina; Christodoulou, Michael S.; Smani, Younes
Esc peptides and derivatives potentiate the activity of CFTR with gating defects and display antipseudomonal activity in cystic fibrosis-like lung disease
2025-01-01 Ferrera, Loretta; Cappiello, Floriana; Venturini, Arianna; Lu, Hexin; Casciaro, Bruno; Cappella, Giacomo; Bontempi, Giulio; Corrente, Alessandra; Strippoli, Raffaele; Zara, Federico; Di, Y. Peter; Galietta, Luis J. V.; Mori, Mattia; Mangoni, Maria Luisa
Design, synthesis, molecular modelling investigation and biological studies of novel human carbonic anhydrase inhibitors based on coumalic acid
2025-01-01 Pontecorvi, Virginia; Angeli, Andrea; Cutarella, Luigi; Mori, Mattia; Secci, Daniela; Coluccia, Michele; Carradori, Simone; Troiani, Anna; Pepi, Federico; Salvitti, Chiara; Di Noi, Alessia; Spano, Mattia; Arrighi, Francesca; De Falco, Elena; Bordin, Antonella; Berrino, Emanuela; Granese, Arianna; Chimenti, Paola; Guglielmi, Paolo; Supuran, Claudiu T.
Structure-Based Ligandability Exploration of a G-Quadruplex-Forming Sequence from the Pseudomonas aeruginosa Genome
2025-01-01 Fiabane, Martina; Platella, Chiara; Diaco, Fabiana; Biancucci, Cristiano; Calcaterra, Andrea; Musumeci, Domenica; Antonelli, Guido; Turriziani, Ombretta; Botta, Bruno; Montesarchio, Daniela; Mori, Mattia
| Titolo | Data di pubblicazione | Autore(i) | File | Abstract |
|---|---|---|---|---|
| A scaffold repositioning approach: dihydroBenzoImidazoTriazineDione (BITD) derivatives as selective ALDH1A1 inhibitors | 1-gen-2026 | Bernardoni, Bianca Laura; D'Agostino, Ilaria; Siragusa, Sonia; Mori, Mattia; Garavaglia, Silvia; La Motta, Concettina | - | |
| Functional and therapeutic effects of Glabrescione B delivery by liposomes on Hedgehog-dependent tumors | 1-gen-2026 | Infante, Paola; Daniele, Raffaella; Bottero, Marta; Longo, Mariagrazia; Bufalieri, Francesca; Lospinoso Severini, Ludovica; Pesce, Cristiano; Fragassi, Agnese; Gabbia, Daniela; Navacci, Shirin; Basili, Irene; Adabbo, Gennaro; Cammarone, Silvia; Cianfoni, Gabriele; Ghirga, Francesca; Mori, Mattia; De Martin, Sara; Mancuso, Mariateresa; Caliceti, Paolo; Pazzaglia, Simonetta; Salmaso, Stefano; Di Marcotullio, Lucia | - | |
| Protonation State-dependent Interaction of Polycationic Polymyxins with the Pseudomonas aeruginosa Outer Membrane Using Colistin A as a Model | 1-gen-2026 | Cutarella, Luigi; Temprano, Alvaro G.; Tafi, Andrea; Mori, Mattia | - | |
| Exploration of the aromatic abietane diterpenoid scaffold in the development of ArnT-mediated colistin resistance inhibitors | 1-gen-2026 | Cammarone, Silvia; Pastore, Valentina; Ryzhuk, Mariya; Cristoferi, Martina; Speroni, Arianna; Imperi, Francesco; Corinti, Davide; Bonaccorsi Di Patti, Maria Carmela; Botta, Bruno; Quaglio, Deborah; Mori, Mattia; Ascenzioni, Fiorentina; Ghirga, Francesca | - | |
| Discovery of a new selective ERAP1 inhibitor for Hedgehog-dependent cancer treatment | 1-gen-2026 | Bufalieri, Francesca; Cucinotta, Antonino; Cammarone, Silvia; Agnoli, Francesca; Basili, Irene; Ferri, Giulia; Quaglio, Deborah; Caimano, Miriam; Capriotti, Anna Laura; Montone, Carmela Maria; Lospinoso Severini, Ludovica; Tempora, Patrizia; D'Amico, Silvia; Juretich, Francesca; Semrau, Marta S.; Navacci, Shirin; Conenna, Marilisa; Bordone, Rosa; Spallotta, Francesco; Garavaglia, Silvia; Storici, Paola; Ghirga, Francesca; Laganà, Aldo; Locatelli, Franco; Ayrault, Olivier; Infante, Paola; Botta, Bruno; Mori, Mattia; Fruci, Doriana; Di Marcotullio, Lucia | - | |
| α-ketoglutarate/succinate ratio imbalance impairs thymine DNA glycosylase function and base excision repair process increasing susceptibility to pancreatic cancer | 1-gen-2026 | Malatesta, Silvia; Vigiano Benedetti, Virginia; Salviati, Emanuela; Illi, Barbara; Manni, Isabella; Middonti, Emanuele; Rampioni Vinciguerra, Gian Luca; Licursi, Valerio; Troilo, Francesca; Colotti, Gianni; Cipolla, Lina; Sabbioneda, Simone; Perfetto, Livia; Piaggio, Giulia; Bussolino, Federico; Di Nicolantonio, Federica; Campiglia, Pietro; Sommella, Eduardo Maria; Mori, Mattia; Cencioni, Chiara; Spallotta, Francesco | - | |
| Discovery of a Mixed and Prodrug-Like Inhibition Mechanism for Phosphocoumarins and Phosphoquinolinones against Human Carbonic Anhydrases | 1-gen-2026 | Nocentini, Alessio; Giovannuzzi, Simone; Alterio, Vincenzo; Bonardi, Alessandro; Barons, Rudolfs; Zalubovskis, Raivis; Eldehna, Wagdy M.; Aronne, Rossella; Esposito, Davide; Luchinat, Enrico; De Simone, Giuseppina; Bartolucci, Gianluca; Gratteri, Paola; Mori, Mattia; Supuran, Claudiu T. | - | |
| Selective Delivery of Anticancer Natural G-Quadruplex Ligands by the AT11 Aptamer for Gastric Cancer Treatment | 1-gen-2026 | Platella, Chiara; Trajkovski, Marko; Brancaccio, Mariarita; Di Palma, Rosita; Calcaterra, Andrea; Mori, Mattia; Falco, Geppino; Plavec, Janez; Montesarchio, Daniela | - | |
| Probing the Structure and Dynamics of Telomeric G-Quadruplexes with Thienoguanosine, a Fluorescent Analogue of Guanosine | 1-gen-2026 | Singh, Pankhi; Mukherjee, Dipanjan; Hanser, Fabien; Tkach, Olha; Humbert, Nicolas; Avendano Avila, Constanza; Ciaco, Stefano; Martinez-Fernandez, Lara; Bansal, Sarthak; Kanj, Samuel; Bombarda, Elisa; Bourderioux, Aurélie; Dziuba, Dmytro; Tor, Yitzhak; Improta, Roberto; Mori, Mattia; Heddi, Brahim; Mély, Yves | - | |
| A novel noninvasive test based on near-infrared fluorescent cholephilic probes for hepatobiliary secretory function assessment | 1-gen-2025 | Sanchez De Blas, Beatriz; Temprano, Alvaro G.; Cives-Losada, Candela; Briz, Oscar; Lozano, Elisa; Martinez-Chantar, Maria L.; Avila, Matias A.; Mori, Mattia; Ghallab, Ahmed; Hengstler, Jan G.; Perez-Melero, Concepción; Bermejo-Gonzalez, Francisco A.; Monte, Maria J.; Romero, Marta R.; Marin, Jose J. G. | - | |
| Influenza a Virus Inhibition: Evaluating Computationally Identified Cyproheptadine Through In Vitro Assessment | 1-gen-2025 | Glisic, Sanja; Stevanovic, Kristina; Perdih, Andrej; Bukreyeva, Natalya; Maruyama, Junki; Perovic, Vladimir; López-Serrano, Sergi; Darji, Ayub; Radosevic, Draginja; Sencanski, Milan; Veljkovic, Veljko; Botta, Bruno; Mori, Mattia; Paessler, Slobodan | - | |
| The Production of Recombinant Azurin from Pseudomonas aeruginosa and Its Ability to Induce Apoptosis in Various Breast Cancer Cell Lines | 1-gen-2025 | Kowalczyk, Tomasz; Merecz-Sadowska, Anna; Synowiec, Ewelina; Śliwiński, Tomasz; Piekarski, Janusz; Szemraj, Janusz; Mori, Mattia; Rijo, Patricia; Sitarek, Przemysław | - | |
| Sustainable Joullié–Ugi and Continuous Flow Implementation Led to Novel Captopril-Inspired Broad-Spectrum Metallo-β-Lactamase Inhibitors | 1-gen-2025 | Alfano, Antonella Ilenia; Pelliccia, Sveva; Barone, Simona; Cutarella, Luigi; Cancade, Sacha Michèle Idriss; Baia, Valerio; Cassese, Emilia; Russomanno, Pasquale; Messano, Nicolò; Frank, Denia; Weizel, Lilia; Rotter, Marco J.; Brunst, Steffen; Wichelhaus, Thomas A.; Proschak, Ewgenij; Tedesco, Daniele; Mori, Mattia; Docquier, Jean Denis; Summa, Vincenzo; Brindisi, Margherita | - | |
| Development of nanovehicles for co-delivery of colistin and ArnT inhibitors | 1-gen-2025 | Pastore, Valentina; Frison, Jessica; Pesce, Cristiano; Ryzhuk, Mariya; Garofalo, Mariangela; Cristoferi, Martina; Cammarone, Silvia; Fabrizio, Giorgia; Bonaccorsi Di Patti, Maria Carmela; Quaglio, Deborah; Ghirga, Francesca; Imperi, Francesco; Mori, Mattia; Caliceti, Paolo; Botta, Bruno; Ascenzioni, Fiorentina; Salmaso, Stefano | - | |
| Biological Evaluation and Computational Modelling Studies on N-acyl Hydrazone and 2,5-Disubstituted 1,3,4-Oxadiazole Derivatives as Non-toxic Antimicrobial Agents | 1-gen-2025 | Giray, Betul; Kaya, Nil; Fiabane, Martina; Buyuk, Ayse Seyma; Kucuk, Hatice Başpinar; Sardas, Semra; Mori, Mattia | - | |
| Discovery of Indole-Based PDE5 Inhibitors: Synthesis and Pharmacological Evaluation | 1-gen-2025 | Park, Shin-Young; Pham, Dang; Shukla, Param; Edward, Justin; John, Reshmi; Li, Addison; Hadjiargyrou, Michael; Mori, Mattia; Zuccarello, Elisa; Arancio, Ottavio; Fiorito, Jole | - | |
| Antibacterial activity of tamoxifen derivatives against methicillin-resistant Staphylococcus aureus | 1-gen-2025 | Molina Panadero, Irene; Falcón Torres, Javier; Hmadcha, Abdelkrim; Princiotto, Salvatore; Cutarella, Luigi; Mori, Mattia; Dallavalle, Sabrina; Christodoulou, Michael S.; Smani, Younes | - | |
| Esc peptides and derivatives potentiate the activity of CFTR with gating defects and display antipseudomonal activity in cystic fibrosis-like lung disease | 1-gen-2025 | Ferrera, Loretta; Cappiello, Floriana; Venturini, Arianna; Lu, Hexin; Casciaro, Bruno; Cappella, Giacomo; Bontempi, Giulio; Corrente, Alessandra; Strippoli, Raffaele; Zara, Federico; Di, Y. Peter; Galietta, Luis J. V.; Mori, Mattia; Mangoni, Maria Luisa | - | |
| Design, synthesis, molecular modelling investigation and biological studies of novel human carbonic anhydrase inhibitors based on coumalic acid | 1-gen-2025 | Pontecorvi, Virginia; Angeli, Andrea; Cutarella, Luigi; Mori, Mattia; Secci, Daniela; Coluccia, Michele; Carradori, Simone; Troiani, Anna; Pepi, Federico; Salvitti, Chiara; Di Noi, Alessia; Spano, Mattia; Arrighi, Francesca; De Falco, Elena; Bordin, Antonella; Berrino, Emanuela; Granese, Arianna; Chimenti, Paola; Guglielmi, Paolo; Supuran, Claudiu T. | - | |
| Structure-Based Ligandability Exploration of a G-Quadruplex-Forming Sequence from the Pseudomonas aeruginosa Genome | 1-gen-2025 | Fiabane, Martina; Platella, Chiara; Diaco, Fabiana; Biancucci, Cristiano; Calcaterra, Andrea; Musumeci, Domenica; Antonelli, Guido; Turriziani, Ombretta; Botta, Bruno; Montesarchio, Daniela; Mori, Mattia | - |
Legenda icone
- file ad accesso aperto
- file disponibili sulla rete interna
- file disponibili agli utenti autorizzati
- file disponibili solo agli amministratori
- file sotto embargo
- nessun file disponibile