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Mostrati risultati da 1 a 20 di 172
Titolo Data di pubblicazione Autore(i) File Abstract
Structure-Based Ligandability Exploration of a G-Quadruplex-Forming Sequence from the Pseudomonas aeruginosa Genome 1-gen-2025 Fiabane, Martina; Platella, Chiara; Diaco, Fabiana; Biancucci, Cristiano; Calcaterra, Andrea; Musumeci, Domenica; Antonelli, Guido; Turriziani, Ombretta; Botta, Bruno; Montesarchio, Daniela; Mori, Mattia -
Influenza a Virus Inhibition: Evaluating Computationally Identified Cyproheptadine Through In Vitro Assessment 1-gen-2025 Glisic, Sanja; Stevanovic, Kristina; Perdih, Andrej; Bukreyeva, Natalya; Maruyama, Junki; Perovic, Vladimir; López-Serrano, Sergi; Darji, Ayub; Radosevic, Draginja; Sencanski, Milan; Veljkovic, Veljko; Botta, Bruno; Mori, Mattia; Paessler, Slobodan -
The Production of Recombinant Azurin from Pseudomonas aeruginosa and Its Ability to Induce Apoptosis in Various Breast Cancer Cell Lines 1-gen-2025 Kowalczyk, Tomasz; Merecz-Sadowska, Anna; Synowiec, Ewelina; Śliwiński, Tomasz; Piekarski, Janusz; Szemraj, Janusz; Mori, Mattia; Rijo, Patricia; Sitarek, Przemysław -
A novel noninvasive test based on near-infrared fluorescent cholephilic probes for hepatobiliary secretory function assessment 1-gen-2025 Sanchez De Blas, Beatriz; Temprano, Alvaro G.; Cives-Losada, Candela; Briz, Oscar; Lozano, Elisa; Martinez-Chantar, Maria L.; Avila, Matias A.; Mori, Mattia; Ghallab, Ahmed; Hengstler, Jan G.; Perez-Melero, Concepción; Bermejo-Gonzalez, Francisco A.; Monte, Maria J.; Romero, Marta R.; Marin, Jose J. G. -
Development of nanovehicles for co-delivery of colistin and ArnT inhibitors 1-gen-2025 Pastore, Valentina; Frison, Jessica; Pesce, Cristiano; Ryzhuk, Mariya; Garofalo, Mariangela; Cristoferi, Martina; Cammarone, Silvia; Fabrizio, Giorgia; Bonaccorsi Di Patti, Maria Carmela; Quaglio, Deborah; Ghirga, Francesca; Imperi, Francesco; Mori, Mattia; Caliceti, Paolo; Botta, Bruno; Ascenzioni, Fiorentina; Salmaso, Stefano -
Discovery of Indole-Based PDE5 Inhibitors: Synthesis and Pharmacological Evaluation 1-gen-2025 Park, Shin-Young; Pham, Dang; Shukla, Param; Edward, Justin; John, Reshmi; Li, Addison; Hadjiargyrou, Michael; Mori, Mattia; Zuccarello, Elisa; Arancio, Ottavio; Fiorito, Jole -
Antibacterial activity of tamoxifen derivatives against methicillin-resistant Staphylococcus aureus 1-gen-2025 Molina Panadero, Irene; Falcón Torres, Javier; Hmadcha, Abdelkrim; Princiotto, Salvatore; Cutarella, Luigi; Mori, Mattia; Dallavalle, Sabrina; Christodoulou, Michael S.; Smani, Younes -
Sustainable Joullié–Ugi and Continuous Flow Implementation Led to Novel Captopril-Inspired Broad-Spectrum Metallo-β-Lactamase Inhibitors 1-gen-2025 Alfano, Antonella Ilenia; Pelliccia, Sveva; Barone, Simona; Cutarella, Luigi; Cancade, Sacha Michèle Idriss; Baia, Valerio; Cassese, Emilia; Russomanno, Pasquale; Messano, Nicolò; Frank, Denia; Weizel, Lilia; Rotter, Marco J.; Brunst, Steffen; Wichelhaus, Thomas A.; Proschak, Ewgenij; Tedesco, Daniele; Mori, Mattia; Docquier, Jean Denis; Summa, Vincenzo; Brindisi, Margherita -
A scaffold repositioning approach: dihydroBenzoImidazoTriazineDione (BITD) derivatives as selective ALDH1A1 inhibitors 1-gen-2025 Bernardoni, Bianca Laura; D'Agostino, Ilaria; Siragusa, Sonia; Mori, Mattia; Garavaglia, Silvia; La Motta, Concettina -
Biological Evaluation and Computational Modelling Studies on N-acyl Hydrazone and 2,5-Disubstituted 1,3,4-Oxadiazole Derivatives as Non-toxic Antimicrobial Agents 1-gen-2025 Giray, Betul; Kaya, Nil; Fiabane, Martina; Buyuk, Ayse Seyma; Kucuk, Hatice Başpinar; Sardas, Semra; Mori, Mattia -
Esc peptides and derivatives potentiate the activity of CFTR with gating defects and display antipseudomonal activity in cystic fibrosis-like lung disease 1-gen-2025 Ferrera, Loretta; Cappiello, Floriana; Venturini, Arianna; Lu, Hexin; Casciaro, Bruno; Cappella, Giacomo; Bontempi, Giulio; Corrente, Alessandra; Strippoli, Raffaele; Zara, Federico; Di, Y. Peter; Galietta, Luis J. V.; Mori, Mattia; Mangoni, Maria Luisa -
Design, synthesis, molecular modelling investigation and biological studies of novel human carbonic anhydrase inhibitors based on coumalic acid 1-gen-2025 Pontecorvi, Virginia; Angeli, Andrea; Cutarella, Luigi; Mori, Mattia; Secci, Daniela; Coluccia, Michele; Carradori, Simone; Troiani, Anna; Pepi, Federico; Salvitti, Chiara; Di Noi, Alessia; Spano, Mattia; Arrighi, Francesca; De Falco, Elena; Bordin, Antonella; Berrino, Emanuela; Granese, Arianna; Chimenti, Paola; Guglielmi, Paolo; Supuran, Claudiu T. -
DNA and RNA polymerases 1-gen-2024 Picarazzi, F.; Mori, M. -
Perspectives in the treatment of antibiotic-resistant bacterial infections with active photodynamic partners within the framework of the EURESTOP COST Action (CA21145) 1-gen-2024 Mori, Mattia; Dumoulin, Fabienne; Faustino, M. Amparo F.; Plaetzer, Kristjan -
Hedgehog Pathway Inhibition by Novel Small Molecules Impairs Melanoma Cell Migration and Invasion under Hypoxia 1-gen-2024 Falsini, A.; Giuntini, G.; Mori, M.; Ghirga, F.; Quaglio, D.; Cucinotta, A.; Coppola, F.; Filippi, I.; Naldini, A.; Botta, B.; Carraro, F. -
Novel 2,4-Dichloro-5-sulfamoylbenzoic Acid Oxime Esters: First Studies as Potential Human Carbonic Anhydrase Inhibitors 1-gen-2024 Kilbile, Jaydeo T.; Sapkal, Suryakant B.; Renzi, Gioele; D'Agostino, Ilaria; Cutarella, Luigi; Mori, Mattia; De Filippis, Barbara; Islam, Imadul; Massardi, Maria Luisa; Somenza, Elena; Ronca, Roberto; Tamboli, Yasinalli; Carta, Fabrizio; Supuran, Claudiu T. -
Cyclization of acyl thiosemicarbazides led to new Helicobacter pylori α‐carbonic anhydrase inhibitors 1-gen-2024 Gumus, Arzu; D'Agostino, Ilaria; Puca, Valentina; Crocetta, Valentina; Carradori, Simone; Cutarella, Luigi; Mori, Mattia; Carta, Fabrizio; Angeli, Andrea; Capasso, Clemente; Supuran, Claudiu T. -
Solving the antibacterial resistance in Europe: The multipronged approach of the COST Action CA21145 EURESTOP 1-gen-2024 Seguin-Devaux, Carole; Mestrovic, Tomislav; Arts, Jacobus J; Sen Karaman, Didem; Nativi, Cristina; Reichmann, Dana; Sahariah, Priyanka; Smani, Younes; Rijo, Patricia; Mori, Mattia -
Fragment-Based Interrogation of the 14–3–3/TAZ Protein–Protein Interaction 1-gen-2024 Andlovic, Blaž; Valenti, Dario; Centorrino, Federica; Picarazzi, Francesca; Hristeva, Stanimira; Hiltmann, Malgorzata; Wolf, Alexander; Cantrelle, François-Xavier; Mori, Mattia; Landrieu, Isabelle; Levy, Laura M.; Klebl, Bert; Tzalis, Dimitrios; Genski, Thorsten; Eickhoff, Jan; Ottmann, Christian -
Exploring a New Generation of Pyrimidine and Pyridine Derivatives as Anti-Influenza Agents Targeting the Polymerase PA–PB1 Subunits Interaction 1-gen-2024 Giacchello, Ilaria; Cianciusi, Annarita; Bertagnin, Chiara; Bonomini, Anna; Francesconi, Valeria; Mori, Mattia; Carbone, Anna; Musumeci, Francesca; Loregian, Arianna; Schenone, Silvia -
Mostrati risultati da 1 a 20 di 172
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