Sfoglia per Autore
VA1213, a selective COX-2 inhibitor, exhibits antitumor activity by suppressing EGFR, AKT, and ERK1/2 phosphorylation
2026-01-01 Ciccone, Valerio; Cecchin, Claudia; Frosini, Maria; Saletti, Mario; Maramai, Samuele; Giuliani, Germano; Paolino, Marco; Cappelli, Andrea; Anzini, Maurizio; Donnini, Sandra; Morbidelli, Lucia
Drug enteric metabolism in gut microbiota-brain crosstalk
2025-01-01 Maramai, Samuele; Taddei, Maurizio; Castagnetti, Andrea; Viciani, Elisa; Koufi, Foteini-Dionysia; Neri, Irene; Boschetti, Elisa; Evangelisti, Camilla; Ratti, Stefano; Baldelli, Luca; Calandra-Buonaura, Giovanna; Cani, Ilaria; Cortelli, Pietro; Sambati, Luisa; Scorziello, Antonella; Taglialatela, Maurizio; Pardini, Matteo; Corsaro, Alessandro; Florio, Tullio; Giannini, Giuseppe
Use of imidazo[1,5-a]quinoline scaffold as the pharmacophore in the design of bivalent ligands of central benzodiazepine receptors
2025-01-01 Paolino, Marco; Saletti, Mario; Venditti, Jacopo; Castriconi, Federica; Giuliani, Germano; Maramai, Samuele; Toti, Alessandra; Ghelardini, Carla; Matucci, Rosanna; Villalobos, Narcy Alcazar; Anzini, Maurizio; Cappelli, Andrea
Evaluation of a New Riluzole‐Based Compound VA945 on Sodium and Potassium Conductances Expressed by SH-SY5Y-Derived Neurons
2025-01-01 Cazzola, J.; Talpo, F.; Faravelli, G.; Donati, C.; Maramai, S.; Saletti, M.; Giuliani, G.; Paolino, M.; Cappelli, A.; Anzini, M.; Sommi, P.; Vitali, A.; Sala, A.; Trucco, A.; Biella, G. R.; Spaiardi, P.
Indole-2-Carboxamide as an Effective Scaffold for the Design of New TRPV1 Agonists
2025-01-01 Maramai, Samuele; Mugnaini, Claudia; Paolino, Marco; Schiano Moriello, Aniello; De Petrocellis, Luciano; Corelli, Federico; Aiello, Francesca; Brizzi, Antonella
Light-mediated activation/deactivation control and in vitro ADME-Tox profiling of a donepezil-like Dual AChE/MAO-B Inhibitor
2025-01-01 Poggialini, Federica; Governa, Paolo; Vagaggini, Chiara; Maramai, Samuele; Lamponi, Stefania; Mugnaini, Claudia; Brizzi, Antonella; Purgatorio, Rosa; De Candia, Modesto; Catto, Marco; Dreassi, Elena; Manetti, Fabrizio; Corelli, Federico; Altomare, Cosimo Damiano; Cappelli, Andrea; Paolino, Marco
Catechol-O-methyltransferase (COMT)
2024-01-01 Tassone, Giusy; Carradori, Simone; Maramai, Samuele; D'Agostino, Ilaria
Novel multitarget directed ligands inspired by riluzole: A serendipitous synthesis of substituted benzo[b][1,4]thiazepines potentially useful as neuroprotective agents
2024-01-01 Maramai, S.; Saletti, M.; Paolino, M.; Giuliani, G.; Cazzola, J.; Spaiardi, P.; Talpo, F.; Frosini, M.; Pifferi, A.; Ballarotto, M.; Carotti, A.; Poggialini, F.; Vagaggini, C.; Dreassi, E.; Giorgi, G.; Dondio, G.; Cappelli, A.; Rosario Biella, G.; Anzini, M.
Development of Potent and Selective Monoacylglycerol Lipase Inhibitors. SARs, Structural Analysis, and Biological Characterization
2024-01-01 Butini, Stefania; Grether, Uwe; Jung, Kwang-Mook; Ligresti, Alessia; Allarà, Marco; Postmus, Annemarieke G. J.; Maramai, Samuele; Brogi, Simone; Papa, Alessandro; Carullo, Gabriele; Sykes, David; Veprintsev, Dmitry; Federico, Stefano; Grillo, Alessandro; Di Guglielmo, Bruno; Ramunno, Anna; Stevens, Anna Floor; Heer, Dominik; Lamponi, Stefania; Gemma, Sandra; Benz, Jörg; Di Marzo, Vincenzo; van der Stelt, Mario; Piomelli, Daniele; Campiani, Giuseppe
Exploiting the bile acid binding protein as transporter of a Cholic Acid/Mirin bioconjugate for potential applications in liver cancer therapy
2024-01-01 Tassone, Giusy; Maramai, Samuele; Paolino, Marco; Lamponi, Stefania; Poggialini, Federica; Dreassi, Elena; Petricci, Elena; Alcaro, Stefano; Pozzi, Cecilia; Romeo, Isabella
Therapeutic potential for coxib-nitric oxide releasing hybrids in cancer treatment
2023-01-01 Giordani, Antonio; Poce, Giovanna; Consalvi, Sara; Maramai, Samuele; Saletti, Mario; Rossi, Antonietta; Patrignani, Paola; Biava, Mariangela; Anzini, Maurizio
In Silico-Guided Rational Drug Design and Synthesis of Novel 4-(Thiophen-2-yl)butanamides as Potent and Selective TRPV1 Agonists
2023-01-01 Romeo, Isabella; Brizzi, Antonella; Pessina, Federica; Ambrosio, Francesca Alessandra; Aiello, Francesca; Belardo, Carmela; Carullo, Gabriele; Costa, Giosuè; De Petrocellis, Luciano; Frosini, Maria; Luongo, Livio; Maramai, Samuele; Paolino, Marco; Moriello, Aniello Schiano; Mugnaini, Claudia; Scorzelli, Francesco; Maione, Sabatino; Corelli, Federico; Di Marzo, Vincenzo; Alcaro, Stefano; Artese, Anna
Macroreticular POLITAG-Pd(0) for the waste minimized hydrogenation/reductive amination of phenols using formic acid as hydrogen source
2023-01-01 Valentini, F.; Di Erasmo, B.; Ciancuti, C.; Rossi, S.; Maramai, S.; Taddei, M.; Vaccaro, L.
Lipoic/Capsaicin-Related Amides: Synthesis and Biological Characterization of New TRPV1 Agonists Endowed with Protective Properties against Oxidative Stress
2022-01-01 Brizzi, Antonella; Maramai, Samuele; Aiello, Francesca; Baratto, Maria Camilla; Corelli, Federico; Mugnaini, Claudia; Paolino, Marco; Scorzelli, Francesco; Aldinucci, Carlo; De Petrocellis, Luciano; Signorini, Cinzia; Pessina, Federica
Inhibition of monoacylglycerol lipase by NSD1819 as an effective strategy for the endocannabinoid system modulation against neuroinflammation-related disorders
2022-01-01 Micheli, Laura; Maramai, Samuele; Toti, Alessandra; Ferrara, Valentina; Ciampi, Clara; Di Cesare Mannelli, Lorenzo; Ghelardini, Carla
Structural characterization of human heat shock protein 90 N-Terminal domain and its variants K112R and K112A in complex with a potent 1,2,3-Triazole-based inhibitor
2022-01-01 Tassone, Giusy; Mazzorana, Marco; Mangani, Stefano; Petricci, Elena; Cini, Elena; Giannini, Giuseppe; Pozzi, Cecilia; Maramai, Samuele
Quinolines and Oxazino-quinoline derivatives as small molecule GLI1 inhibitors identified by virtual screening
2022-01-01 Manetti, Fabrizio; Maresca, Luisa; Crivaro, Enrica; Pepe, Sara; Cini, Elena; Singh, Snigdha; Governa, Paolo; Maramai, Samuele; Giannini, Giuseppe; Stecca, Barbara; Petricci, Elena
Design, synthesis and biological evaluation of light-driven on-off multitarget AChE and MAO-B inhibitors
2022-01-01 Paolino, Marco; Rullo, Mariagrazia; Maramai, Samuele; de Candia, Modesto; Pisani, Leonardo; Catto, Marco; Mugnaini, Claudia; Brizzi, Antonella; Cappelli, Andrea; Olivucci, Massimo; Corelli, Federico; Altomare, Cosimo D
Novel analgesic/anti-inflammatory agents: 1,5-Diarylpyrrole nitrooxyethyl sulfides and related compounds as Cyclooxygenase-2 inhibitors containing a nitric oxide donor moiety endowed with vasorelaxant properties
2022-01-01 Saletti, Mario; Maramai, Samuele; Reale, Annalisa; Paolino, Marco; Brogi, Simone; Di Capua, Angela; Cappelli, Andrea; Giorgi, Gianluca; D'Avino, Danilo; Rossi, Antonietta; Ghelardini, Carla; Di Cesare Mannelli, Lorenzo; Sardella, Roccaldo; Carotti, Andrea; Woelkart, Gerald; Klösch, Burkhard; Bigogno, Chiara; Dondio, Giulio; Anzini, Maurizio
An Intramolecular Hydroaminomethylation-Based Approach to Pyrrolizidine Alkaloids under Microwave-Assisted Heating
2022-01-01 Petricci, Elena; Zurzolo, Simone; Matassini, Camilla; Maramai, Samuele; Cardona, Francesca; Goti, Andrea; Taddei, Maurizio
| Titolo | Data di pubblicazione | Autore(i) | File | Abstract |
|---|---|---|---|---|
| VA1213, a selective COX-2 inhibitor, exhibits antitumor activity by suppressing EGFR, AKT, and ERK1/2 phosphorylation | 1-gen-2026 | Ciccone, Valerio; Cecchin, Claudia; Frosini, Maria; Saletti, Mario; Maramai, Samuele; Giuliani, Germano; Paolino, Marco; Cappelli, Andrea; Anzini, Maurizio; Donnini, Sandra; Morbidelli, Lucia | - | |
| Drug enteric metabolism in gut microbiota-brain crosstalk | 1-gen-2025 | Maramai, Samuele; Taddei, Maurizio; Castagnetti, Andrea; Viciani, Elisa; Koufi, Foteini-Dionysia; Neri, Irene; Boschetti, Elisa; Evangelisti, Camilla; Ratti, Stefano; Baldelli, Luca; Calandra-Buonaura, Giovanna; Cani, Ilaria; Cortelli, Pietro; Sambati, Luisa; Scorziello, Antonella; Taglialatela, Maurizio; Pardini, Matteo; Corsaro, Alessandro; Florio, Tullio; Giannini, Giuseppe | - | |
| Use of imidazo[1,5-a]quinoline scaffold as the pharmacophore in the design of bivalent ligands of central benzodiazepine receptors | 1-gen-2025 | Paolino, Marco; Saletti, Mario; Venditti, Jacopo; Castriconi, Federica; Giuliani, Germano; Maramai, Samuele; Toti, Alessandra; Ghelardini, Carla; Matucci, Rosanna; Villalobos, Narcy Alcazar; Anzini, Maurizio; Cappelli, Andrea | - | |
| Evaluation of a New Riluzole‐Based Compound VA945 on Sodium and Potassium Conductances Expressed by SH-SY5Y-Derived Neurons | 1-gen-2025 | Cazzola, J.; Talpo, F.; Faravelli, G.; Donati, C.; Maramai, S.; Saletti, M.; Giuliani, G.; Paolino, M.; Cappelli, A.; Anzini, M.; Sommi, P.; Vitali, A.; Sala, A.; Trucco, A.; Biella, G. R.; Spaiardi, P. | - | |
| Indole-2-Carboxamide as an Effective Scaffold for the Design of New TRPV1 Agonists | 1-gen-2025 | Maramai, Samuele; Mugnaini, Claudia; Paolino, Marco; Schiano Moriello, Aniello; De Petrocellis, Luciano; Corelli, Federico; Aiello, Francesca; Brizzi, Antonella | - | |
| Light-mediated activation/deactivation control and in vitro ADME-Tox profiling of a donepezil-like Dual AChE/MAO-B Inhibitor | 1-gen-2025 | Poggialini, Federica; Governa, Paolo; Vagaggini, Chiara; Maramai, Samuele; Lamponi, Stefania; Mugnaini, Claudia; Brizzi, Antonella; Purgatorio, Rosa; De Candia, Modesto; Catto, Marco; Dreassi, Elena; Manetti, Fabrizio; Corelli, Federico; Altomare, Cosimo Damiano; Cappelli, Andrea; Paolino, Marco | - | |
| Catechol-O-methyltransferase (COMT) | 1-gen-2024 | Tassone, Giusy; Carradori, Simone; Maramai, Samuele; D'Agostino, Ilaria | - | |
| Novel multitarget directed ligands inspired by riluzole: A serendipitous synthesis of substituted benzo[b][1,4]thiazepines potentially useful as neuroprotective agents | 1-gen-2024 | Maramai, S.; Saletti, M.; Paolino, M.; Giuliani, G.; Cazzola, J.; Spaiardi, P.; Talpo, F.; Frosini, M.; Pifferi, A.; Ballarotto, M.; Carotti, A.; Poggialini, F.; Vagaggini, C.; Dreassi, E.; Giorgi, G.; Dondio, G.; Cappelli, A.; Rosario Biella, G.; Anzini, M. | - | |
| Development of Potent and Selective Monoacylglycerol Lipase Inhibitors. SARs, Structural Analysis, and Biological Characterization | 1-gen-2024 | Butini, Stefania; Grether, Uwe; Jung, Kwang-Mook; Ligresti, Alessia; Allarà, Marco; Postmus, Annemarieke G. J.; Maramai, Samuele; Brogi, Simone; Papa, Alessandro; Carullo, Gabriele; Sykes, David; Veprintsev, Dmitry; Federico, Stefano; Grillo, Alessandro; Di Guglielmo, Bruno; Ramunno, Anna; Stevens, Anna Floor; Heer, Dominik; Lamponi, Stefania; Gemma, Sandra; Benz, Jörg; Di Marzo, Vincenzo; van der Stelt, Mario; Piomelli, Daniele; Campiani, Giuseppe | - | |
| Exploiting the bile acid binding protein as transporter of a Cholic Acid/Mirin bioconjugate for potential applications in liver cancer therapy | 1-gen-2024 | Tassone, Giusy; Maramai, Samuele; Paolino, Marco; Lamponi, Stefania; Poggialini, Federica; Dreassi, Elena; Petricci, Elena; Alcaro, Stefano; Pozzi, Cecilia; Romeo, Isabella | - | |
| Therapeutic potential for coxib-nitric oxide releasing hybrids in cancer treatment | 1-gen-2023 | Giordani, Antonio; Poce, Giovanna; Consalvi, Sara; Maramai, Samuele; Saletti, Mario; Rossi, Antonietta; Patrignani, Paola; Biava, Mariangela; Anzini, Maurizio | - | |
| In Silico-Guided Rational Drug Design and Synthesis of Novel 4-(Thiophen-2-yl)butanamides as Potent and Selective TRPV1 Agonists | 1-gen-2023 | Romeo, Isabella; Brizzi, Antonella; Pessina, Federica; Ambrosio, Francesca Alessandra; Aiello, Francesca; Belardo, Carmela; Carullo, Gabriele; Costa, Giosuè; De Petrocellis, Luciano; Frosini, Maria; Luongo, Livio; Maramai, Samuele; Paolino, Marco; Moriello, Aniello Schiano; Mugnaini, Claudia; Scorzelli, Francesco; Maione, Sabatino; Corelli, Federico; Di Marzo, Vincenzo; Alcaro, Stefano; Artese, Anna | - | |
| Macroreticular POLITAG-Pd(0) for the waste minimized hydrogenation/reductive amination of phenols using formic acid as hydrogen source | 1-gen-2023 | Valentini, F.; Di Erasmo, B.; Ciancuti, C.; Rossi, S.; Maramai, S.; Taddei, M.; Vaccaro, L. | - | |
| Lipoic/Capsaicin-Related Amides: Synthesis and Biological Characterization of New TRPV1 Agonists Endowed with Protective Properties against Oxidative Stress | 1-gen-2022 | Brizzi, Antonella; Maramai, Samuele; Aiello, Francesca; Baratto, Maria Camilla; Corelli, Federico; Mugnaini, Claudia; Paolino, Marco; Scorzelli, Francesco; Aldinucci, Carlo; De Petrocellis, Luciano; Signorini, Cinzia; Pessina, Federica | - | |
| Inhibition of monoacylglycerol lipase by NSD1819 as an effective strategy for the endocannabinoid system modulation against neuroinflammation-related disorders | 1-gen-2022 | Micheli, Laura; Maramai, Samuele; Toti, Alessandra; Ferrara, Valentina; Ciampi, Clara; Di Cesare Mannelli, Lorenzo; Ghelardini, Carla | - | |
| Structural characterization of human heat shock protein 90 N-Terminal domain and its variants K112R and K112A in complex with a potent 1,2,3-Triazole-based inhibitor | 1-gen-2022 | Tassone, Giusy; Mazzorana, Marco; Mangani, Stefano; Petricci, Elena; Cini, Elena; Giannini, Giuseppe; Pozzi, Cecilia; Maramai, Samuele | - | |
| Quinolines and Oxazino-quinoline derivatives as small molecule GLI1 inhibitors identified by virtual screening | 1-gen-2022 | Manetti, Fabrizio; Maresca, Luisa; Crivaro, Enrica; Pepe, Sara; Cini, Elena; Singh, Snigdha; Governa, Paolo; Maramai, Samuele; Giannini, Giuseppe; Stecca, Barbara; Petricci, Elena | - | |
| Design, synthesis and biological evaluation of light-driven on-off multitarget AChE and MAO-B inhibitors | 1-gen-2022 | Paolino, Marco; Rullo, Mariagrazia; Maramai, Samuele; de Candia, Modesto; Pisani, Leonardo; Catto, Marco; Mugnaini, Claudia; Brizzi, Antonella; Cappelli, Andrea; Olivucci, Massimo; Corelli, Federico; Altomare, Cosimo D | - | |
| Novel analgesic/anti-inflammatory agents: 1,5-Diarylpyrrole nitrooxyethyl sulfides and related compounds as Cyclooxygenase-2 inhibitors containing a nitric oxide donor moiety endowed with vasorelaxant properties | 1-gen-2022 | Saletti, Mario; Maramai, Samuele; Reale, Annalisa; Paolino, Marco; Brogi, Simone; Di Capua, Angela; Cappelli, Andrea; Giorgi, Gianluca; D'Avino, Danilo; Rossi, Antonietta; Ghelardini, Carla; Di Cesare Mannelli, Lorenzo; Sardella, Roccaldo; Carotti, Andrea; Woelkart, Gerald; Klösch, Burkhard; Bigogno, Chiara; Dondio, Giulio; Anzini, Maurizio | - | |
| An Intramolecular Hydroaminomethylation-Based Approach to Pyrrolizidine Alkaloids under Microwave-Assisted Heating | 1-gen-2022 | Petricci, Elena; Zurzolo, Simone; Matassini, Camilla; Maramai, Samuele; Cardona, Francesca; Goti, Andrea; Taddei, Maurizio | - |
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