Sfoglia per Rivista ACS CHEMICAL BIOLOGY
Development of a multiplexed activity-based protein profiling assay to evaluate activity of endocannabinoid hydrolase inhibitors
2018-01-01 Janssen, Antonius P A; Van der Vliet, Daan; Bakker, Alexander T; Jiang, Ming; Grimm, Sebastian H; Campiani, Giuseppe; Butini, Stefania; van der Stelt, Mario
Functional and structural characterization of 2-amino-4-phenylthiazole inhibitors of the HIV-1 nucleocapsid protein with antiviral activity
2014-01-01 Mori, Mattia; Nucci, Alessandro; Lang, M. C.; Humbert, N.; Boudier, C.; Debaene, F.; Sanglier Cianferani, S.; Catala, M.; Schult Dietrich, P.; Dietrich, U.; Tisné, C.; Mely, Y.; Botta, Maurizio
Hit Recycling: Discovery of a Potent Carbonic Anhydrase Inhibitor by in Silico Target Fishing
2015-01-01 Mori, Mattia; Cau, Ylenia; Vignaroli, Giulia; Laurenzana, Ilaria; Caivano, Antonella; Vullo, Daniela; Supuran, Claudiu T.; Botta, Maurizio
Identification of Phosphate-Containing Compounds as New Inhibitors of 14-3-3/c-Abl Protein-Protein Interaction
2020-01-01 Iralde-Lorente, Leire; Tassone, Giusy; Clementi, Letizia; Franci, Lorenzo; Munier, Claire C; Cau, Ylenia; Mori, Mattia; Chiariello, Mario; Angelucci, Adriano; Perry, Matthew W D; Pozzi, Cecilia; Mangani, Stefano; Botta, Maurizio
Loop electrostatics modulates the intersubunit interactions in ferritin
2014-01-01 Bernacchioni, Caterina; Ghini, Veronica; Pozzi, Cecilia; DI PISA, Flavio; Theil, Elizabeth C.; Turano, Paola
Molecular Basis of Selective Inhibition and Slow Reversibility of Avibactam against Class D Carbapenemases: A Structure-Guided Study of OXA-24 and OXA-48.
2015-01-01 Lahiri, Sd; Mangani, Stefano; Jahić, H; Benvenuti, M; Durand Reville, Tf; DE LUCA, Filomena; Ehmann, De; Rossolini, GIAN MARIA; Alm, Ra; Docquier, JEAN DENIS
Structure-Based Identification of HIV-1 Nucleocapsid Protein Inhibitors Active against Wild-Type and Drug-Resistant HIV-1 Strains
2018-01-01 Mori, Mattia; Kovalenko, Lesia; Malancona, Savina; Saladini, Francesco; De Forni, Davide; Pires, Manuel; Humbert, Nicolas; Real, Eleonore; Botzanowski, Thomas; Cianférani, Sarah; Giannini, Alessia; Dasso Lang, Maria Chiara; Cugia, Giulia; Poddesu, Barbara; Lori, Franco; Zazzi, Maurizio; Harper, Steven; Summa, Vincenzo; Mely, Yves; Botta, Maurizio
Titolo | Data di pubblicazione | Autore(i) | File | Abstract |
---|---|---|---|---|
Development of a multiplexed activity-based protein profiling assay to evaluate activity of endocannabinoid hydrolase inhibitors | 1-gen-2018 | Janssen, Antonius P A; Van der Vliet, Daan; Bakker, Alexander T; Jiang, Ming; Grimm, Sebastian H; Campiani, Giuseppe; Butini, Stefania; van der Stelt, Mario | - | |
Functional and structural characterization of 2-amino-4-phenylthiazole inhibitors of the HIV-1 nucleocapsid protein with antiviral activity | 1-gen-2014 | Mori, Mattia; Nucci, Alessandro; Lang, M. C.; Humbert, N.; Boudier, C.; Debaene, F.; Sanglier Cianferani, S.; Catala, M.; Schult Dietrich, P.; Dietrich, U.; Tisné, C.; Mely, Y.; Botta, Maurizio | - | |
Hit Recycling: Discovery of a Potent Carbonic Anhydrase Inhibitor by in Silico Target Fishing | 1-gen-2015 | Mori, Mattia; Cau, Ylenia; Vignaroli, Giulia; Laurenzana, Ilaria; Caivano, Antonella; Vullo, Daniela; Supuran, Claudiu T.; Botta, Maurizio | - | |
Identification of Phosphate-Containing Compounds as New Inhibitors of 14-3-3/c-Abl Protein-Protein Interaction | 1-gen-2020 | Iralde-Lorente, Leire; Tassone, Giusy; Clementi, Letizia; Franci, Lorenzo; Munier, Claire C; Cau, Ylenia; Mori, Mattia; Chiariello, Mario; Angelucci, Adriano; Perry, Matthew W D; Pozzi, Cecilia; Mangani, Stefano; Botta, Maurizio | - | |
Loop electrostatics modulates the intersubunit interactions in ferritin | 1-gen-2014 | Bernacchioni, Caterina; Ghini, Veronica; Pozzi, Cecilia; DI PISA, Flavio; Theil, Elizabeth C.; Turano, Paola | - | |
Molecular Basis of Selective Inhibition and Slow Reversibility of Avibactam against Class D Carbapenemases: A Structure-Guided Study of OXA-24 and OXA-48. | 1-gen-2015 | Lahiri, Sd; Mangani, Stefano; Jahić, H; Benvenuti, M; Durand Reville, Tf; DE LUCA, Filomena; Ehmann, De; Rossolini, GIAN MARIA; Alm, Ra; Docquier, JEAN DENIS | - | |
Structure-Based Identification of HIV-1 Nucleocapsid Protein Inhibitors Active against Wild-Type and Drug-Resistant HIV-1 Strains | 1-gen-2018 | Mori, Mattia; Kovalenko, Lesia; Malancona, Savina; Saladini, Francesco; De Forni, Davide; Pires, Manuel; Humbert, Nicolas; Real, Eleonore; Botzanowski, Thomas; Cianférani, Sarah; Giannini, Alessia; Dasso Lang, Maria Chiara; Cugia, Giulia; Poddesu, Barbara; Lori, Franco; Zazzi, Maurizio; Harper, Steven; Summa, Vincenzo; Mely, Yves; Botta, Maurizio | - |
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