Sfoglia per Rivista
Design and Synthesis of New Transient Receptor Potential Vanilloid Type-1 (TRPV1) Channel Modulators: Identification, Molecular Modeling Analysis, and Pharmacological Characterization of the N-(4-Hydroxy-3-methoxybenzyl)-4-(thiophen-2-yl)butanamide, a Small Molecule Endowed with Agonist TRPV1 Activity and Protective Effects against Oxidative Stress
2016-01-01 Aiello, F.; Badolato, M.; Pessina, Federica; Sticozzi, C.; Maestrini, Vanessa; Aldinucci, C.; Luongo, L.; Guida, F.; Ligresti, A.; Artese, A.; Allarà, M.; Costa, G.; Frosini, Maria; Schiano Morello, A.; De Petrocellis, L.; Valacchi, G.; Alcaro, S.; Maione, S.; Di Marzo, V.; Corelli, Federico; Brizzi, Antonella
Exploiting the Power of Stereochemistry in Drug Action: 3-[(2S,6S,11S)-8-Hydroxy-6,11-dimethyl-1,4,5,6-tetrahydro-2,6-methano-3-benzazocin-3(2H)-yl]-N-phenylpropanamide as Potent Sigma-1 Receptor Antagonist
2020-01-01 Turnaturi, Rita; Pasquinucci, Lorella; Chiechio, Santina; Grasso, Margherita; Marrazzo, Agostino; Amata, Emanuele; Dichiara, Maria; Prezzavento, Orazio; Parenti, Carmela
Ionotropic Glutamate Receptor GluA2 in Complex with Bicyclic Pyrimidinedione-Based Compounds: When Small Compound Modifications Have Distinct Effects on Binding Interactions
2020-01-01 Frydenvang, Karla; Pickering, Darryl S; Kshirsagar, Giridhar U; Chemi, Giulia; Gemma, Sandra; Sprogøe, Desiree; Kærn, Anne Mette; Brogi, Simone; Campiani, Giuseppe; Butini, Stefania; Kastrup, Jette Sandholm
Retinitis pigmentosa and retinal degenerations: deciphering pathways and targets for drug discovery and development
2020-01-01 Carullo, G.; Federico, S.; Relitti, N.; Gemma, S.; Butini, S.; Campiani, G.
Selective Fatty Acid Amide Hydrolase Inhibitors as Potential Novel Antiepileptic Agents
2021-01-01 Grillo, Alessandro; Fezza, Filomena; Chemi, Giulia; Colangeli, Roberto; Brogi, Simone; Fazio, Domenico; Federico, Stefano; Papa, Alessandro; Relitti, Nicola; Di Maio, Roberto; Giorgi, Gianluca; Lamponi, Stefania; Valoti, Massimo; Gorelli, Beatrice; Saponara, Simona; Benedusi, Mascia; Pecorelli, Alessandra; Minetti, Patrizia; Valacchi, Giuseppe; Butini, Stefania; Campiani, Giuseppe; Gemma, Sandra; Maccarrone, Mauro; Di Giovanni, Giuseppe
Structural and molecular insight into Piperazine and Piperidine derivatives as Histamine H3 and Sigma-1 receptor antagonists with promising antinociceptive properties
2022-01-01 Szczepańska, Katarzyna; Podlewska, Sabina; Dichiara, Maria; Gentile, Davide; Patamia, Vincenzo; Rosier, Niklas; Mönnich, Denise; Ruiz Cantero M., Carmen; Karcz, Tadeusz; Łażewska, Dorota; Siwek, Agata; Pockes, Steffen; Cobos J., Enrique; Marrazzo, Agostino; Stark, Holger; Rescifina, Antonio; Bojarski J., Andrzej; Amata, Emanuele; Kieć-Kononowicz, Katarkyna
Synthesis, computational insights, and evaluation of novel sigma receptors ligands
2023-01-01 Dichiara, Maria; Ambrosio, FRANCESCA ALESSANDRA; Barbaraci, Carla; Gonzalez-Cano, Rafael; Costa, Giosuè.; Parenti, Carmela; Marrazzo, Agostino; Pasquinucci, Lorella; Cobos Enrique, J.; Alcaro, Stefano; Amata, Emanuele
Tuning Properties for Blood-Brain Barrier Permeation: A Statistics-Based Analysis
2020-01-01 Dichiara, Maria; Amata, Benedetto; Turnaturi, Rita; Marrazzo, Agostino; Amata, Emanuele
| Titolo | Data di pubblicazione | Autore(i) | File | Abstract |
|---|---|---|---|---|
| Design and Synthesis of New Transient Receptor Potential Vanilloid Type-1 (TRPV1) Channel Modulators: Identification, Molecular Modeling Analysis, and Pharmacological Characterization of the N-(4-Hydroxy-3-methoxybenzyl)-4-(thiophen-2-yl)butanamide, a Small Molecule Endowed with Agonist TRPV1 Activity and Protective Effects against Oxidative Stress | 1-gen-2016 | Aiello, F.; Badolato, M.; Pessina, Federica; Sticozzi, C.; Maestrini, Vanessa; Aldinucci, C.; Luongo, L.; Guida, F.; Ligresti, A.; Artese, A.; Allarà, M.; Costa, G.; Frosini, Maria; Schiano Morello, A.; De Petrocellis, L.; Valacchi, G.; Alcaro, S.; Maione, S.; Di Marzo, V.; Corelli, Federico; Brizzi, Antonella | - | |
| Exploiting the Power of Stereochemistry in Drug Action: 3-[(2S,6S,11S)-8-Hydroxy-6,11-dimethyl-1,4,5,6-tetrahydro-2,6-methano-3-benzazocin-3(2H)-yl]-N-phenylpropanamide as Potent Sigma-1 Receptor Antagonist | 1-gen-2020 | Turnaturi, Rita; Pasquinucci, Lorella; Chiechio, Santina; Grasso, Margherita; Marrazzo, Agostino; Amata, Emanuele; Dichiara, Maria; Prezzavento, Orazio; Parenti, Carmela | - | |
| Ionotropic Glutamate Receptor GluA2 in Complex with Bicyclic Pyrimidinedione-Based Compounds: When Small Compound Modifications Have Distinct Effects on Binding Interactions | 1-gen-2020 | Frydenvang, Karla; Pickering, Darryl S; Kshirsagar, Giridhar U; Chemi, Giulia; Gemma, Sandra; Sprogøe, Desiree; Kærn, Anne Mette; Brogi, Simone; Campiani, Giuseppe; Butini, Stefania; Kastrup, Jette Sandholm | - | |
| Retinitis pigmentosa and retinal degenerations: deciphering pathways and targets for drug discovery and development | 1-gen-2020 | Carullo, G.; Federico, S.; Relitti, N.; Gemma, S.; Butini, S.; Campiani, G. | - | |
| Selective Fatty Acid Amide Hydrolase Inhibitors as Potential Novel Antiepileptic Agents | 1-gen-2021 | Grillo, Alessandro; Fezza, Filomena; Chemi, Giulia; Colangeli, Roberto; Brogi, Simone; Fazio, Domenico; Federico, Stefano; Papa, Alessandro; Relitti, Nicola; Di Maio, Roberto; Giorgi, Gianluca; Lamponi, Stefania; Valoti, Massimo; Gorelli, Beatrice; Saponara, Simona; Benedusi, Mascia; Pecorelli, Alessandra; Minetti, Patrizia; Valacchi, Giuseppe; Butini, Stefania; Campiani, Giuseppe; Gemma, Sandra; Maccarrone, Mauro; Di Giovanni, Giuseppe | - | |
| Structural and molecular insight into Piperazine and Piperidine derivatives as Histamine H3 and Sigma-1 receptor antagonists with promising antinociceptive properties | 1-gen-2022 | Szczepańska, Katarzyna; Podlewska, Sabina; Dichiara, Maria; Gentile, Davide; Patamia, Vincenzo; Rosier, Niklas; Mönnich, Denise; Ruiz Cantero M., Carmen; Karcz, Tadeusz; Łażewska, Dorota; Siwek, Agata; Pockes, Steffen; Cobos J., Enrique; Marrazzo, Agostino; Stark, Holger; Rescifina, Antonio; Bojarski J., Andrzej; Amata, Emanuele; Kieć-Kononowicz, Katarkyna | - | |
| Synthesis, computational insights, and evaluation of novel sigma receptors ligands | 1-gen-2023 | Dichiara, Maria; Ambrosio, FRANCESCA ALESSANDRA; Barbaraci, Carla; Gonzalez-Cano, Rafael; Costa, Giosuè.; Parenti, Carmela; Marrazzo, Agostino; Pasquinucci, Lorella; Cobos Enrique, J.; Alcaro, Stefano; Amata, Emanuele | - | |
| Tuning Properties for Blood-Brain Barrier Permeation: A Statistics-Based Analysis | 1-gen-2020 | Dichiara, Maria; Amata, Benedetto; Turnaturi, Rita; Marrazzo, Agostino; Amata, Emanuele | - |
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