Sfoglia per Autore
Targeting GLI1 and GLI2 with small molecule inhibitors to suppress GLI-dependent transcription and tumor growth
2023-01-01 Maresca, Luisa; Crivaro, Enrica; Migliorini, Francesca; Anichini, Giulia; Giammona, Alessandro; Pepe, Sara; Poggialini, Federica; Vagaggini, Chiara; Giannini, Giuseppe; Sestini, Serena; Borgognoni, Lorenzo; Lapucci, Andrea; Dreassi, Elena; Taddei, Maurizio; Manetti, Fabrizio; Petricci, Elena; Stecca, Barbara
Switching Mechanistic Pathways by Micellar Catalysis: A Highly Selective Rhodium Catalyst for the Hydroaminomethylation of Olefins with Anilines in Water
2023-01-01 Migliorini, F.; Monciatti, E.; Romagnoli, G.; Parisi, M. L.; Taubert, J.; Vogt, M.; Langer, R.; Petricci, E.
Structural Characterization of Human Heat Shock Protein 90 N-Terminal Domain and Its Variants K112R and K112A in Complex with a Potent 1,2,3-Triazole-Based Inhibitor
2022-01-01 Tassone, Giusy; Mazzorana, Marco; Mangani, Stefano; Petricci, Elena; Cini, Elena; Giannini, Giuseppe; Pozzi, Cecilia; Maramai, Samuele
Requirements for MRN endonuclease processing of topoisomerase II-mediated DNA damage in mammalian cells
2022-01-01 Sun, Yilun; Soans, Eroica; Mishina, Margarita; Petricci, Elena; Pommier, Yves; Nitiss, Karin C.; Nitiss, John L.
Quinolines and Oxazino-quinoline Derivatives as Small Molecule GLI1 Inhibitors Identified by Virtual Screening
2022-01-01 Manetti, Fabrizio; Maresca, Luisa; Crivaro, Enrica; Pepe, Sara; Cini, Elena; Singh, Snigdha; Governa, Paolo; Maramai, Samuele; Giannini, Giuseppe; Stecca, Barbara; Petricci, Elena
A pH-responsive crosslinker platform for antibody-drug conjugate (ADC) targeting delivery
2022-01-01 Migliorini, Francesca; Cini, Elena; Dreassi, Elena; Finetti, Federica; Ievoli, Giovanni; Macrì, Giulia; Petricci, Elena; Rango, Enrico; Trabalzini, Lorenza; Taddei, Maurizio
An Intramolecular Hydroaminomethylation-Based Approach to Pyrrolizidine Alkaloids under Microwave-Assisted Heating
2022-01-01 Petricci, Elena; Zurzolo, Simone; Matassini, Camilla; Maramai, Samuele; Cardona, Francesca; Goti, Andrea; Taddei, Maurizio
Survey on the Recent Advances in 4-Hydroxyphenylpyruvate Dioxygenase (HPPD) Inhibition by Diketone and Triketone Derivatives and Congeneric Compounds: Structural Analysis of HPPD/Inhibitor Complexes and Structure-Activity Relationship Considerations
2022-01-01 Governa, Paolo; Bernardini, Giulia; Braconi, Daniela; Manetti, Fabrizio; Santucci, Annalisa; Petricci, Elena
Antibacterial alkylguanidino ureas: Molecular simplification approach, searching for membrane-based MoA
2022-01-01 D'Agostino, I.; Ardino, C.; Poli, G.; Sannio, F.; Lucidi, M.; Poggialini, F.; Visaggio, D.; Rango, E.; Filippi, S.; Petricci, E.; Visca, P.; Botta, L.; Docquier, J. -D.; Dreassi, E.
A molecular spectroscopy approach for the investigation of early phase ochronotic pigment development in Alkaptonuria
2021-01-01 Bernini, A.; Petricci, E.; Atrei, A.; Baratto, M. C.; Manetti, F.; Santucci, A.
Biomass Waste-Derived Pd-PiNe Catalyst for the Continuous-Flow Copper-Free Sonogashira Reaction in a CPME-Water Azeotropic Mixture
2021-01-01 Ferlin, F.; Valentini, F.; Sciosci, D.; Calamante, M.; Petricci, E.; Vaccaro, L.
Antibody drug conjugates with hydroxamic acid cargos for histone deacetylase (HDAC) inhibition
2021-01-01 Cianferotti, C.; Faltoni, V.; Cini, E.; Ermini, E.; Migliorini, F.; Petricci, E.; Taddei, M.; Salvini, L.; Battistuzzi, G.; Milazzo, F. M.; Anastasi, A. M.; Chiapparino, C.; De Santis, R.; Giannini, G.
Targeting non-canonical activation of GLI1 by the SOX2-BRD4 transcriptional complex improves the efficacy of HEDGEHOG pathway inhibition in melanoma
2021-01-01 Pietrobono, S.; Gaudio, E.; Gagliardi, S.; Zitani, M.; Carrassa, L.; Migliorini, F.; Petricci, E.; Manetti, F.; Makukhin, N.; Bond, A. G.; Paradise, B. D.; Ciulli, A.; Fernandez-Zapico, M. E.; Bertoni, F.; Stecca, B.
Micellar catalysis for sustainable hydroformylation
2021-01-01 Migliorini, F.; Dei, F.; Maramai, S.; Calamante, M.; Petricci, E.
The Antimalarial Mefloquine Shows Activity against Mycobacterium abscessus, Inhibiting Mycolic Acid Metabolism
2021-01-01 Degiacomi, Giulia; Chiarelli, Laurent Roberto; Recchia, Deborah; Petricci, Elena; Gianibbi, Beatrice; Fiscarelli, Ersilia Vita; Fattorini, Lanfranco; Manetti, Fabrizio; Pasca, Maria Rosalia
ErbB2 Targeted Epigenetic Modulation: Anti-tumor Efficacy of the ADC Trastuzumab-HDACi ST8176AA1
2020-01-01 Maria Milazzo, Ferdinando; Vesci, Loredana; Maria Anastasi, Anna; Chiapparino, Caterina; Rosi, Antonio; Giannini, Giuseppe; Taddei, Maurizio; Cini, Elena; Faltoni, Valentina; Petricci, Elena; Battistuzzi, Gianfranco; Salvini, Laura; Carollo, Valeria; De Santis, Rita
Novel textile dye obtained through transformation of 2-amino-3-methoxybenzoic acid by free and immobilised laccase from a Pleurotus ostreatus strain
2020-01-01 Wlizlo, K.; Polak, J.; Jarosz-Wilkolazka, A.; Pogni, R.; Petricci, E.
Pharmacophore-Based Virtual Screening for Identification of Negative Modulators of GLI1 as Potential Anticancer Agents
2020-01-01 Manetti, Fabrizio; Stecca, Barbara; Santini, Roberta; Maresca, Luisa; Giannini, Giuseppe; Taddei, Maurizio; Petricci, Elena
Structure and bioactive properties of novel textile dyes synthesised by fungal laccase
2020-01-01 Polak, J.; Wlizlo, K.; Pogni, R.; Petricci, E.; Graz, M.; Szalapata, K.; Osinska-jaroszuk, M.; Kapral-piotrowska, J.; Pawlikowska-pawlega, B.; Jarosz-wilkolazka, A.
In Water Markovnikov Hydration and One-Pot Reductive Hydroamination of Terminal Alkynes under Ruthenium Nanoparticle Catalysis
2020-01-01 Risi, C.; Cini, E.; Petricci, E.; Saponaro, S.; Taddei, M.
Titolo | Data di pubblicazione | Autore(i) | File | Abstract |
---|---|---|---|---|
Targeting GLI1 and GLI2 with small molecule inhibitors to suppress GLI-dependent transcription and tumor growth | 1-gen-2023 | Maresca, Luisa; Crivaro, Enrica; Migliorini, Francesca; Anichini, Giulia; Giammona, Alessandro; Pepe, Sara; Poggialini, Federica; Vagaggini, Chiara; Giannini, Giuseppe; Sestini, Serena; Borgognoni, Lorenzo; Lapucci, Andrea; Dreassi, Elena; Taddei, Maurizio; Manetti, Fabrizio; Petricci, Elena; Stecca, Barbara | - | |
Switching Mechanistic Pathways by Micellar Catalysis: A Highly Selective Rhodium Catalyst for the Hydroaminomethylation of Olefins with Anilines in Water | 1-gen-2023 | Migliorini, F.; Monciatti, E.; Romagnoli, G.; Parisi, M. L.; Taubert, J.; Vogt, M.; Langer, R.; Petricci, E. | - | |
Structural Characterization of Human Heat Shock Protein 90 N-Terminal Domain and Its Variants K112R and K112A in Complex with a Potent 1,2,3-Triazole-Based Inhibitor | 1-gen-2022 | Tassone, Giusy; Mazzorana, Marco; Mangani, Stefano; Petricci, Elena; Cini, Elena; Giannini, Giuseppe; Pozzi, Cecilia; Maramai, Samuele | - | |
Requirements for MRN endonuclease processing of topoisomerase II-mediated DNA damage in mammalian cells | 1-gen-2022 | Sun, Yilun; Soans, Eroica; Mishina, Margarita; Petricci, Elena; Pommier, Yves; Nitiss, Karin C.; Nitiss, John L. | - | |
Quinolines and Oxazino-quinoline Derivatives as Small Molecule GLI1 Inhibitors Identified by Virtual Screening | 1-gen-2022 | Manetti, Fabrizio; Maresca, Luisa; Crivaro, Enrica; Pepe, Sara; Cini, Elena; Singh, Snigdha; Governa, Paolo; Maramai, Samuele; Giannini, Giuseppe; Stecca, Barbara; Petricci, Elena | - | |
A pH-responsive crosslinker platform for antibody-drug conjugate (ADC) targeting delivery | 1-gen-2022 | Migliorini, Francesca; Cini, Elena; Dreassi, Elena; Finetti, Federica; Ievoli, Giovanni; Macrì, Giulia; Petricci, Elena; Rango, Enrico; Trabalzini, Lorenza; Taddei, Maurizio | - | |
An Intramolecular Hydroaminomethylation-Based Approach to Pyrrolizidine Alkaloids under Microwave-Assisted Heating | 1-gen-2022 | Petricci, Elena; Zurzolo, Simone; Matassini, Camilla; Maramai, Samuele; Cardona, Francesca; Goti, Andrea; Taddei, Maurizio | - | |
Survey on the Recent Advances in 4-Hydroxyphenylpyruvate Dioxygenase (HPPD) Inhibition by Diketone and Triketone Derivatives and Congeneric Compounds: Structural Analysis of HPPD/Inhibitor Complexes and Structure-Activity Relationship Considerations | 1-gen-2022 | Governa, Paolo; Bernardini, Giulia; Braconi, Daniela; Manetti, Fabrizio; Santucci, Annalisa; Petricci, Elena | - | |
Antibacterial alkylguanidino ureas: Molecular simplification approach, searching for membrane-based MoA | 1-gen-2022 | D'Agostino, I.; Ardino, C.; Poli, G.; Sannio, F.; Lucidi, M.; Poggialini, F.; Visaggio, D.; Rango, E.; Filippi, S.; Petricci, E.; Visca, P.; Botta, L.; Docquier, J. -D.; Dreassi, E. | - | |
A molecular spectroscopy approach for the investigation of early phase ochronotic pigment development in Alkaptonuria | 1-gen-2021 | Bernini, A.; Petricci, E.; Atrei, A.; Baratto, M. C.; Manetti, F.; Santucci, A. | - | |
Biomass Waste-Derived Pd-PiNe Catalyst for the Continuous-Flow Copper-Free Sonogashira Reaction in a CPME-Water Azeotropic Mixture | 1-gen-2021 | Ferlin, F.; Valentini, F.; Sciosci, D.; Calamante, M.; Petricci, E.; Vaccaro, L. | - | |
Antibody drug conjugates with hydroxamic acid cargos for histone deacetylase (HDAC) inhibition | 1-gen-2021 | Cianferotti, C.; Faltoni, V.; Cini, E.; Ermini, E.; Migliorini, F.; Petricci, E.; Taddei, M.; Salvini, L.; Battistuzzi, G.; Milazzo, F. M.; Anastasi, A. M.; Chiapparino, C.; De Santis, R.; Giannini, G. | - | |
Targeting non-canonical activation of GLI1 by the SOX2-BRD4 transcriptional complex improves the efficacy of HEDGEHOG pathway inhibition in melanoma | 1-gen-2021 | Pietrobono, S.; Gaudio, E.; Gagliardi, S.; Zitani, M.; Carrassa, L.; Migliorini, F.; Petricci, E.; Manetti, F.; Makukhin, N.; Bond, A. G.; Paradise, B. D.; Ciulli, A.; Fernandez-Zapico, M. E.; Bertoni, F.; Stecca, B. | - | |
Micellar catalysis for sustainable hydroformylation | 1-gen-2021 | Migliorini, F.; Dei, F.; Maramai, S.; Calamante, M.; Petricci, E. | - | |
The Antimalarial Mefloquine Shows Activity against Mycobacterium abscessus, Inhibiting Mycolic Acid Metabolism | 1-gen-2021 | Degiacomi, Giulia; Chiarelli, Laurent Roberto; Recchia, Deborah; Petricci, Elena; Gianibbi, Beatrice; Fiscarelli, Ersilia Vita; Fattorini, Lanfranco; Manetti, Fabrizio; Pasca, Maria Rosalia | - | |
ErbB2 Targeted Epigenetic Modulation: Anti-tumor Efficacy of the ADC Trastuzumab-HDACi ST8176AA1 | 1-gen-2020 | Maria Milazzo, Ferdinando; Vesci, Loredana; Maria Anastasi, Anna; Chiapparino, Caterina; Rosi, Antonio; Giannini, Giuseppe; Taddei, Maurizio; Cini, Elena; Faltoni, Valentina; Petricci, Elena; Battistuzzi, Gianfranco; Salvini, Laura; Carollo, Valeria; De Santis, Rita | - | |
Novel textile dye obtained through transformation of 2-amino-3-methoxybenzoic acid by free and immobilised laccase from a Pleurotus ostreatus strain | 1-gen-2020 | Wlizlo, K.; Polak, J.; Jarosz-Wilkolazka, A.; Pogni, R.; Petricci, E. | - | |
Pharmacophore-Based Virtual Screening for Identification of Negative Modulators of GLI1 as Potential Anticancer Agents | 1-gen-2020 | Manetti, Fabrizio; Stecca, Barbara; Santini, Roberta; Maresca, Luisa; Giannini, Giuseppe; Taddei, Maurizio; Petricci, Elena | - | |
Structure and bioactive properties of novel textile dyes synthesised by fungal laccase | 1-gen-2020 | Polak, J.; Wlizlo, K.; Pogni, R.; Petricci, E.; Graz, M.; Szalapata, K.; Osinska-jaroszuk, M.; Kapral-piotrowska, J.; Pawlikowska-pawlega, B.; Jarosz-wilkolazka, A. | - | |
In Water Markovnikov Hydration and One-Pot Reductive Hydroamination of Terminal Alkynes under Ruthenium Nanoparticle Catalysis | 1-gen-2020 | Risi, C.; Cini, E.; Petricci, E.; Saponaro, S.; Taddei, M. | - |
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