Sfoglia per Titolo
Novel Potent 5-HT3 Receptor Ligands Based on the Pyrrolidone Structure. Effects of the Quaternization of the Basic Nitrogen on the Interaction with 5-HT3 Receptor
2002-01-01 Cappelli, Andrea; Gallelli, A.; Braile, C.; Anzini, Maurizio; Vomero, Salvatore; Mennuni, L.; Makovec, F; Menziani, M. C.; De Benedetti, P. G.; Donati, Alessandro; Giorgi, Gianluca
Novel potent 5-HT3 receptor ligands based on the pyrrolidone structure: synthesis, biological evaluation, and computational rationalization of the ligand-receptor interaction modalities
2002-01-01 Cappelli, A.; Anzini, M.; Vomero, S.; Mennuni, L.; Makovec, F.; Doucet, E.; Hamon, M.; Menziani, M. C.; De Benedetti, P. G.; Giorgi, G.; Ghelardini, C.; Collina, S.
Novel Potent and Selective 5-HT3 Receptor Antagonists Based on Arylpiperazine Skeleton: Synthesis, Structure, Biological Activity and CoMFA Studies
1995-01-01 Anzini, Maurizio; Cappelli, Andrea; Vomero, Salvatore; Giorgi, Gianluca; Langer, T.; Hamon, M.; Merahi, N.; Emerit, B. M.; Cagnotto, A.; Skorupska, M.; Mennini, T.; Pinto, J. C.
Novel Potent and Selective Agonists of the GPR55 Receptor Based on the 3-Benzylquinolin-2(1H)-One Scaffold
2022-01-01 Ceni, C.; Benko, M. J.; Mohamed, K. A.; Poli, G.; Di Stefano, M.; Tuccinardi, T.; Digiacomo, M.; Valoti, M.; Laprairie, R. B.; Macchia, M.; Bertini, S.
Novel Potent and Selective Central 5-HT3 Receptor Ligands Provided with Different Intrinsic Efficacy. 2. Molecular Basis of the Intrinsic Efficacy of Arylpiperazine Derivatives at the Central 5-HT3 Receptors
1999-01-01 Cappelli, Andrea; Anzini, Maurizio; Vomero, Salvatore; Canullo, L.; Mennuni, L.; Makovec, F.; Doucet, E.; Hamon, M.; Menziani, M. C.; DE BENEDETTI, P. G.; Bruni, G.; Romeo, M. R.; Giorgi, Gianluca; Donati, Alessandro
Novel potent and selective central 5-HT3 receptor ligands provided with different intrinsic efficacy. I. Mapping the central 5-HT3 recceptor binding site by arylpiperazine derivatives
1998-01-01 Cappelli, Andrea; Anzini, Maurizio; Vomero, Salvatore; Mennuni, L.; Makovec, F.; Doucet, E.; Hamon, M.; Bruni, G.; Romeo, M. R.; Menziani, M. C.; De Benedetti, P. G.; Langer, T.
A novel potent class I HDAC inhibitor reverses the STAT4/p66Shc apoptotic defect in B cells from chronic lymphocytic leukemia patients
2024-01-01 Rossi, Sara; Tatangelo, Vanessa; Dichiara, Maria; Butini, Stefania; Gemma, Sandra; Brogi, Simone; Pasquini, Silvia; Cappello, Martina; Vincenzi, Fabrizio; Varani, Katia; Lopresti, Ludovica; Malchiodi, Margherita; Carrara, Chiara; Gozzetti, Alessandro; Bocchia, Monica; Marotta, Giuseppe; Patrussi, Laura; Carullo, Gabriele; Baldari, Cosima T.; Campiani, Giuseppe
The novel potent multidrug resistance inhibitors N,N-bis(cyclohexanol)amine aryl esters are devoid of vascular effects
2011-01-01 Saponara, Simona; Gorelli, B; Tzankova, V; Martelli, C; Teodori, E; Sgaragli, G; Fusi, Fabio
Novel Primers-Probe Sets for Detection and Identification of Mycobacteria by PCR-Microarray Assay
2012-01-01 Lazzeri, E.; Santoro, F.; Oggioni, M. R.; Iannelli, F.; Pozzi, G.
Novel promoters and coding first exons in DLG2 linked to developmental disorders and intellectual disability
2017-01-01 Reggiani, Claudio; Coppens, Sandra; Sekhara, Tayeb; Dimov, Ivan; Pichon, Bruno; Lufin, Nicolas; Addor, Marie-Claude; Belligni, Elga Fabia; Digilio, Maria Cristina; Faletra, Flavio; Ferrero, Giovanni Battista; Gerard, Marion; Isidor, Bertrand; Joss, Shelagh; Niel-Bütschi, Florence; Perrone, Maria Dolores; Petit, Florence; Renieri, Alessandra; Romana, Serge; Topa, Alexandra; Vermeesch, Joris Robert; Lenaerts, Tom; Casimir, Georges; Abramowicz, Marc; Bontempi, Gianluca; Vilain, Catheline; Deconinck, Nicolas; Smits, Guillaume
A novel protein from the serum of Python sebae, structurally homologous with type-γ phospholipase A2 inhibitor, displays antitumour activity
2011-01-01 Donnini, Sandra; Finetti, Federica; Francese, S; Boscaro, F; Dani, Fr; Maset, F; Frasson, R; Palmieri, M; Pazzagli, M; De Filippis, V; Garaci, E; Ziche, Marina
The novel pseudo-compound transposon Tn7086 carries aminoglycoside resistance genes in Enterococcus faecalis
2026-01-01 Colombini, Lorenzo; Tirziu, Mariana; De Giorgi, Stefano; Cuppone, Anna Maria; Sangiorgio, Giuseppe; Bonomo, Carmelo; Bongiorno, Dafne; Stefani, Stefania; Ricci, Susanna; Pozzi, Gianni; Santoro, Francesco; Iannelli, Francesco
Novel PTEN mutations in neurodevelopmental disorders and macrocephaly
2009-01-01 Orrico, A.; Galli, L.; Buoni, S.; Orsi, A.; Vonella, G.; Sorrentino, V.
Novel pyrazolo[3,4-d]pyrimidines as dual Src/Bcr-Abl kinase inhibitors: synthesis and biological evaluation for chronic myeloid leukemia treatment
2022-01-01 Di Maria, S.; Picarazzi, F.; Mori, M.; Cianciusi, A.; Carbone, A.; Crespan, E.; Perini, C.; Sabetta, S.; Deplano, S.; Poggialini, F.; Molinari, A.; Aronne, R.; Maccioni, E.; Maga, G.; Angelucci, A.; Schenone, S.; Musumeci, F.; Dreassi, E.
Novel pyrrolo-1,5-benzoxazepine compounds display significant activity against resistant chronic myeloid leukaemia cells in vitro, in ex vivo patient samples and in vivo
2010-01-01 Bright, S. A.; Mcelligott, A. M.; O'Connell, J. W.; O'Connor, L; Carroll, P; Campiani, Giuseppe; Deininger, M. W.; Conneally, E; Lawler, M; Williams, D. C.; Zisterer, D. M.
The novel pyrrolo-1,5-benzoxazepine, PBOX-15, synergistically enhances the apoptotic efficacy of imatinib in gastrointestinal stromal tumours; suggested mechanism of action of PBOX-15
2016-01-01 Kinsella, Paula; Greene, Lisa M; Bright, Sandra A; Pollock, Jade K; Butini, Stefania; Campiani, Giuseppe; Bauer, Sebastian; Williams, D. Clive; Zisterer, Daniela M.
The novel pyrrolo-1,5-benzoxazepine, PBOX-21, potentiates the apoptotic efficacy of STI571 (imatinib mesylate) in human chronic myeloid leukaemia cells
2009-01-01 Bright, S. A.; Greene, L. M.; Greene, T. F.; Campiani, Giuseppe; Butini, Stefania; Brindisi, Margherita; Lawler, M.; Meegan, M. J.; Wilòiams, D. C.; Zisterer, D. M.
The novel pyrrolo-1,5-benzoxazepine, PBOX-6, synergistically enhances the apoptotic effects of carboplatin in drug sensitive and multidrug resistant neuroblastoma cells
2014-01-01 Lennon, Jennifer C.; Bright, Sandra A.; Carroll, Eilis; Butini, Stefania; Campiani, Giuseppe; O'Meara, Anne; Williams, D. Clive; Zisterer, Daniela M.
Novel quinolone-based potent and selective HDAC6 inhibitors: synthesis, molecular modeling studies and biological investigation
2021-01-01 Relitti, N.; Saraswati, A. P.; Chemi, G.; Brindisi, M.; Brogi, S.; Herp, D.; Schmidtkunz, K.; Saccoccia, F.; Ruberti, G.; Ulivieri, C.; Vanni, F.; Sarno, F.; Altucci, L.; Lamponi, S.; Jung, M.; Gemma, S.; Butini, S.; Campiani, G.
A novel ray tracing algorithm for scenarios comprising pre-ordered multiple planar reflectors, straight wedges, and vertexes
2014-01-01 Puggelli, Federico; Carluccio, Giorgio; Albani, Matteo
| Titolo | Data di pubblicazione | Autore(i) | File | Abstract |
|---|---|---|---|---|
| Novel Potent 5-HT3 Receptor Ligands Based on the Pyrrolidone Structure. Effects of the Quaternization of the Basic Nitrogen on the Interaction with 5-HT3 Receptor | 1-gen-2002 | Cappelli, Andrea; Gallelli, A.; Braile, C.; Anzini, Maurizio; Vomero, Salvatore; Mennuni, L.; Makovec, F; Menziani, M. C.; De Benedetti, P. G.; Donati, Alessandro; Giorgi, Gianluca | - | |
| Novel potent 5-HT3 receptor ligands based on the pyrrolidone structure: synthesis, biological evaluation, and computational rationalization of the ligand-receptor interaction modalities | 1-gen-2002 | Cappelli, A.; Anzini, M.; Vomero, S.; Mennuni, L.; Makovec, F.; Doucet, E.; Hamon, M.; Menziani, M. C.; De Benedetti, P. G.; Giorgi, G.; Ghelardini, C.; Collina, S. | - | |
| Novel Potent and Selective 5-HT3 Receptor Antagonists Based on Arylpiperazine Skeleton: Synthesis, Structure, Biological Activity and CoMFA Studies | 1-gen-1995 | Anzini, Maurizio; Cappelli, Andrea; Vomero, Salvatore; Giorgi, Gianluca; Langer, T.; Hamon, M.; Merahi, N.; Emerit, B. M.; Cagnotto, A.; Skorupska, M.; Mennini, T.; Pinto, J. C. | - | |
| Novel Potent and Selective Agonists of the GPR55 Receptor Based on the 3-Benzylquinolin-2(1H)-One Scaffold | 1-gen-2022 | Ceni, C.; Benko, M. J.; Mohamed, K. A.; Poli, G.; Di Stefano, M.; Tuccinardi, T.; Digiacomo, M.; Valoti, M.; Laprairie, R. B.; Macchia, M.; Bertini, S. | - | |
| Novel Potent and Selective Central 5-HT3 Receptor Ligands Provided with Different Intrinsic Efficacy. 2. Molecular Basis of the Intrinsic Efficacy of Arylpiperazine Derivatives at the Central 5-HT3 Receptors | 1-gen-1999 | Cappelli, Andrea; Anzini, Maurizio; Vomero, Salvatore; Canullo, L.; Mennuni, L.; Makovec, F.; Doucet, E.; Hamon, M.; Menziani, M. C.; DE BENEDETTI, P. G.; Bruni, G.; Romeo, M. R.; Giorgi, Gianluca; Donati, Alessandro | - | |
| Novel potent and selective central 5-HT3 receptor ligands provided with different intrinsic efficacy. I. Mapping the central 5-HT3 recceptor binding site by arylpiperazine derivatives | 1-gen-1998 | Cappelli, Andrea; Anzini, Maurizio; Vomero, Salvatore; Mennuni, L.; Makovec, F.; Doucet, E.; Hamon, M.; Bruni, G.; Romeo, M. R.; Menziani, M. C.; De Benedetti, P. G.; Langer, T. | - | |
| A novel potent class I HDAC inhibitor reverses the STAT4/p66Shc apoptotic defect in B cells from chronic lymphocytic leukemia patients | 1-gen-2024 | Rossi, Sara; Tatangelo, Vanessa; Dichiara, Maria; Butini, Stefania; Gemma, Sandra; Brogi, Simone; Pasquini, Silvia; Cappello, Martina; Vincenzi, Fabrizio; Varani, Katia; Lopresti, Ludovica; Malchiodi, Margherita; Carrara, Chiara; Gozzetti, Alessandro; Bocchia, Monica; Marotta, Giuseppe; Patrussi, Laura; Carullo, Gabriele; Baldari, Cosima T.; Campiani, Giuseppe | - | |
| The novel potent multidrug resistance inhibitors N,N-bis(cyclohexanol)amine aryl esters are devoid of vascular effects | 1-gen-2011 | Saponara, Simona; Gorelli, B; Tzankova, V; Martelli, C; Teodori, E; Sgaragli, G; Fusi, Fabio | - | |
| Novel Primers-Probe Sets for Detection and Identification of Mycobacteria by PCR-Microarray Assay | 1-gen-2012 | Lazzeri, E.; Santoro, F.; Oggioni, M. R.; Iannelli, F.; Pozzi, G. | - | |
| Novel promoters and coding first exons in DLG2 linked to developmental disorders and intellectual disability | 1-gen-2017 | Reggiani, Claudio; Coppens, Sandra; Sekhara, Tayeb; Dimov, Ivan; Pichon, Bruno; Lufin, Nicolas; Addor, Marie-Claude; Belligni, Elga Fabia; Digilio, Maria Cristina; Faletra, Flavio; Ferrero, Giovanni Battista; Gerard, Marion; Isidor, Bertrand; Joss, Shelagh; Niel-Bütschi, Florence; Perrone, Maria Dolores; Petit, Florence; Renieri, Alessandra; Romana, Serge; Topa, Alexandra; Vermeesch, Joris Robert; Lenaerts, Tom; Casimir, Georges; Abramowicz, Marc; Bontempi, Gianluca; Vilain, Catheline; Deconinck, Nicolas; Smits, Guillaume | - | |
| A novel protein from the serum of Python sebae, structurally homologous with type-γ phospholipase A2 inhibitor, displays antitumour activity | 1-gen-2011 | Donnini, Sandra; Finetti, Federica; Francese, S; Boscaro, F; Dani, Fr; Maset, F; Frasson, R; Palmieri, M; Pazzagli, M; De Filippis, V; Garaci, E; Ziche, Marina | - | |
| The novel pseudo-compound transposon Tn7086 carries aminoglycoside resistance genes in Enterococcus faecalis | 1-gen-2026 | Colombini, Lorenzo; Tirziu, Mariana; De Giorgi, Stefano; Cuppone, Anna Maria; Sangiorgio, Giuseppe; Bonomo, Carmelo; Bongiorno, Dafne; Stefani, Stefania; Ricci, Susanna; Pozzi, Gianni; Santoro, Francesco; Iannelli, Francesco | - | |
| Novel PTEN mutations in neurodevelopmental disorders and macrocephaly | 1-gen-2009 | Orrico, A.; Galli, L.; Buoni, S.; Orsi, A.; Vonella, G.; Sorrentino, V. | - | |
| Novel pyrazolo[3,4-d]pyrimidines as dual Src/Bcr-Abl kinase inhibitors: synthesis and biological evaluation for chronic myeloid leukemia treatment | 1-gen-2022 | Di Maria, S.; Picarazzi, F.; Mori, M.; Cianciusi, A.; Carbone, A.; Crespan, E.; Perini, C.; Sabetta, S.; Deplano, S.; Poggialini, F.; Molinari, A.; Aronne, R.; Maccioni, E.; Maga, G.; Angelucci, A.; Schenone, S.; Musumeci, F.; Dreassi, E. | - | |
| Novel pyrrolo-1,5-benzoxazepine compounds display significant activity against resistant chronic myeloid leukaemia cells in vitro, in ex vivo patient samples and in vivo | 1-gen-2010 | Bright, S. A.; Mcelligott, A. M.; O'Connell, J. W.; O'Connor, L; Carroll, P; Campiani, Giuseppe; Deininger, M. W.; Conneally, E; Lawler, M; Williams, D. C.; Zisterer, D. M. | - | |
| The novel pyrrolo-1,5-benzoxazepine, PBOX-15, synergistically enhances the apoptotic efficacy of imatinib in gastrointestinal stromal tumours; suggested mechanism of action of PBOX-15 | 1-gen-2016 | Kinsella, Paula; Greene, Lisa M; Bright, Sandra A; Pollock, Jade K; Butini, Stefania; Campiani, Giuseppe; Bauer, Sebastian; Williams, D. Clive; Zisterer, Daniela M. | - | |
| The novel pyrrolo-1,5-benzoxazepine, PBOX-21, potentiates the apoptotic efficacy of STI571 (imatinib mesylate) in human chronic myeloid leukaemia cells | 1-gen-2009 | Bright, S. A.; Greene, L. M.; Greene, T. F.; Campiani, Giuseppe; Butini, Stefania; Brindisi, Margherita; Lawler, M.; Meegan, M. J.; Wilòiams, D. C.; Zisterer, D. M. | - | |
| The novel pyrrolo-1,5-benzoxazepine, PBOX-6, synergistically enhances the apoptotic effects of carboplatin in drug sensitive and multidrug resistant neuroblastoma cells | 1-gen-2014 | Lennon, Jennifer C.; Bright, Sandra A.; Carroll, Eilis; Butini, Stefania; Campiani, Giuseppe; O'Meara, Anne; Williams, D. Clive; Zisterer, Daniela M. | - | |
| Novel quinolone-based potent and selective HDAC6 inhibitors: synthesis, molecular modeling studies and biological investigation | 1-gen-2021 | Relitti, N.; Saraswati, A. P.; Chemi, G.; Brindisi, M.; Brogi, S.; Herp, D.; Schmidtkunz, K.; Saccoccia, F.; Ruberti, G.; Ulivieri, C.; Vanni, F.; Sarno, F.; Altucci, L.; Lamponi, S.; Jung, M.; Gemma, S.; Butini, S.; Campiani, G. | - | |
| A novel ray tracing algorithm for scenarios comprising pre-ordered multiple planar reflectors, straight wedges, and vertexes | 1-gen-2014 | Puggelli, Federico; Carluccio, Giorgio; Albani, Matteo | - |
Legenda icone
- file ad accesso aperto
- file disponibili sulla rete interna
- file disponibili agli utenti autorizzati
- file disponibili solo agli amministratori
- file sotto embargo
- nessun file disponibile