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Titolo Data di pubblicazione Autore(i) File Abstract
Reduction by the positive allosteric modulator of the GABAB receptor, GS39783, of alcohol self-administration in Sardinian alcohol-preferring rats exposed to the “sipper” procedure 1-gen-2010 Maccioni, P.; Flore, P.; Carai, M. A. M.; Mugnaini, Claudia; Pasquini, Serena; Corelli, Federico; Gessa, G. L.; Colombo, G. -
Rapid combinatorial access to a library of 1,5-disubstituted-3-indole-N-alkylacetamides as CB2 receptor ligands 1-gen-2009 Pasquini, Serena; Mugnaini, Claudia; Brizzi, Antonella; Ligresti, A.; Di Marzo, V.; Ghiron, C.; Corelli, Federico -
The 4-Quinolone-3-carboxylic Acid Motif as a Multivalent Scaffold in Medicinal Chemistry 1-gen-2009 Mugnaini, Claudia; Pasquini, Serena; Corelli, Federico -
Synthesis and biological evaluation of guanidino compounds endowed with subnanomolar affinity as competitive inhibitors of maize polyamine oxidase 1-gen-2009 Manetti, Fabrizio; Cona, A.; Angeli, L.; Mugnaini, Claudia; Raffi, F.; Capone, C.; Dreassi, Elena; Zizzari, A. T.; Tisi, A.; Federico, R.; Botta, Maurizio -
Investigations on the 4-Quinolone-3-carboxylic Acid Motif. 2. Synthesis and Structure-Activity Relationship of Potent and Selective Cannabinoid-2 Receptor Agonists Endowed with Analgesic Activity in Vivo 1-gen-2008 Pasquini, Serena; Botta, Lorenzo; Semeraro, Teresa; Mugnaini, Claudia; Ligresti, A.; Palazzo, E.; Maione, S.; Di Marzo, V.; Corelli, Federico -
Practical synthesis of novel purine analogues as Hsp90 inhibitors. 1-gen-2008 Semeraro, T; Mugnaini, Claudia; Manetti, Fabrizio; Pasquini, S; Corelli, Federico -
Preparation of a set of 4,5-dihydro-3H-pyrrolo[3,2-d]pyrimidin-4-ones as potential Hsp90 ligands 1-gen-2008 Semeraro, Teresa; Mugnaini, Claudia; Corelli, Federico -
Investigations on the 4-Quinolone-3-carboxylic Acid Motif. 1. Synthesis and Structure-Activity Relationship of a Class of Human Immunodeficiency Virus type 1 Integrase Inhibitors 1-gen-2008 Pasquini, Serena; Mugnaini, Claudia; Tintori, Cristina; Botta, Maurizio; Trejos, A.; Arvela, R. K.; Larhed, M.; Vitvrouw, M.; Michiels, M.; Christ, F.; Debyser, Z.; Corelli, Federico -
Toward novel HIV-1 integrase binding inhibitors: molecular modeling, synthesis, and biological studies 1-gen-2007 Mugnaini, Claudia; Rajamaki, S.; Tintori, Cristina; Corelli, Federico; Massa, Silvio; Witvrouw, M.; Debyser, Z.; Veljkovic, V.; Botta, Maurizio -
Synthesis and biological evaluation of 4-alkylamino-6-(2-hydroxyethyl)-2-methylthiopyrimidines as a new ribella virus inhibitors 1-gen-2007 Mugnaini, Claudia; Petricci, Elena; Botta, Maurizio; Corelli, Federico; Mastromarino, P.; Giorgi, Gianluca -
Dihydro-alkylthio-benzyl-oxopyrimidines as Inhibitors of Reverse Transcriptase: Synthesis and Rationalization of the Biological Data on Both Wild-Type Enzyme and Relevant Clinical Mutants 1-gen-2007 Mugnaini, Claudia; Alongi, M; Togninelli, A; Gevariya, H; Brizzi, Antonella; Manetti, Fabrizio; Bernardini, C; Angeli, L; Tafi, Andrea; Bellucci, L; Corelli, Federico; Massa, Silvio; Maga, G; Samuele, A; Facchini, M; CLOTET CODINA, I; ARMAND UGON, M; ESTE J., A; Botta, Maurizio -
Simplified Analogs Of Immucillin-G Retain Potent Human Purine Nucleoside Phosphorylase Inhibitory Activity 1-gen-2006 Semeraro, T; Alvarez, R; Botta, Maurizio; Ghiron, C; Lossani, A; Manetti, Fabrizio; Mugnaini, Claudia; Focher, F; Corelli, Federico -
Simplified Analogues of Immucillin-G Retain Potent Human Purine Nucleoside Phosphorylase Inhibitory Activity 1-gen-2006 Semeraro, T; Lossani, A; Botta, Maurizio; Ghiron, C; Alvarez, R; Manetti, Fabrizio; Mugnaini, Claudia; Valensin, S; Focher, F; Corelli, Federico -
Synthesis and biological investigation of S-aryl-S-DABO derivatives as HIV-1 inhibitors 1-gen-2006 Mugnaini, Claudia; Manetti, Fabrizio; EST J., A; Clotet Codina, I.; Maga, G.; Cancio, R.; Botta, Maurizio; Corelli, Federico -
Towards new methodologies for the synthesis of biologically interesting 6-substituted pyrimidines and 4(3H)-pyrimidinones 1-gen-2006 Petricci, Elena; Mugnaini, Claudia; Botta, Maurizio; Togninelli, A.; Bernardini, C.; Manetti, Fabrizio; Parlato, M. C.; Renzulli, M. L.; Alongi, M.; Falciani, C.; Corelli, Federico; Botta, M. -
Solution-phase parallel synthesis of S-DABO analogues 1-gen-2006 Togninelli, A.; Carmi, C.; Petricci, E.; Mugnaini, C.; Massa, S.; Corelli, F.; Botta, M. -
Combinatorial chemistry as a tool for targeting different stages of the replicative HIV-1 cycle 1-gen-2005 Mugnaini, Claudia; Petricci, Elena; Corelli, Federico; Botta, Maurizio -
Parallel Solution-Phase and Microwave-Assisted Synthesis of New S-DABO Derivatives Endowed with Subnanomolar Anti-HIV-1 Activity 1-gen-2005 Manetti, Fabrizio; Este, J. A.; CLOTET CODINA, I.; ARMAND UGON, M.; Maga, G.; Crespan, E.; Cancio, R.; Mugnaini, Claudia; Bernardini, C.; Togninelli, A.; Carmi, C.; Alongi, M.; Petricci, Elena; Massa, S.; Corelli, Federico; Botta, Maurizio -
Synthesis of reactive cytidine derivatives as building blocks for cross-linking oligonucleotides 1-gen-2005 Radi, Marco; Mugnaini, Claudia; Petricci, Elena; Corelli, Federico; Botta, Maurizio -
A new linker for anchoring/masking primary amines on solid support 1-gen-2005 Paladino, A.; Mugnaini, Claudia; Botta, Maurizio; Corelli, Federico -
Mostrati risultati da 61 a 80 di 90
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