Sfoglia per Autore
Synthesis, 1 structural properties, and pharmacological evaluation of 2-(acylamino)thiophene-3-carboxamides and analogues thereof
2014-01-01 Mugnaini, Claudia; Pedani, Valentina; Giunta, D.; Sechi, B.; Solinas, M.; Casti, A.; Castelli, M. P.; Giorgi, Gianluca; Corelli, Federico
New fluoroquinolones active against fluoroquinolones-resistant Mycobacterium tuberculosis strains
2013-01-01 Guerrini, Valentina; De Rosa, M.; Pasquini, S.; Mugnaini, Claudia; Brizzi, Antonella; Cuppone, Anna Maria; Pozzi, Gianni; Corelli, Federico
Synthesis and pharmacological characterization of 2-(acylamino)thiophene derivatives as metabolically stable, orally effective, positive allosteric modulators of the GABAB receptor
2013-01-01 Mugnaini, Claudia; Pedani, Valentina; Casu, Angelo; Lobina, Carla; Casti, Alberto; Maccioni, Paola; Porcu, Alessandra; Giunta, Daniela; Lamponi, Stefania; Solinas, Maurizio; Dragoni, Stefania; Valoti, Massimo; Colombo, Giancarlo; Castelli, Maria Paola; Gessa, Gian Luigi; Corelli, Federico
Characterization of COR627 and COR628, two novel positive allosteric modulators of the GABA B receptor
2012-01-01 Castelli, M. P.; Casu, A.; Casti, P.; Lobina, C.; Carai, M. A. M.; Colombo, G.; Solinas, M.; Giunta, D.; Mugnaini, Claudia; Pasquini, Serena; Tafi, Andrea; Brogi, Simone; Gessa, G. L.; Corelli, Federico
The bioisosteric concept applied to cannabinoid ligands
2012-01-01 Mugnaini, Claudia; Pasquini, Serena; Corelli, Federico
Investigations on the 4-quinolone-3-carboxylic acid motif part 5: modulation of the physicochemical profile of a set of potent and selective cannabinoid-2 receptor ligands through a bioisosteric approach
2012-01-01 Mugnaini, Claudia; Nocerino, S.; Pedani, Valentina; Pasquini, Serena; Tafi, Andrea; De Chiaro, M.; Bellucci, L.; Valoti, Massimo; Guida, F.; Luongo, L.; Dragoni, Stefania; Ligresti, A.; Rosenberg, A.; Bolognini, D.; Cascio, M. G.; Pertwee, R. G.; Moaddel, R.; Maione, S.; Di Marzo, V.; Corelli, Federico
Investigations on the 4-Quinolone-3-carboxylic Acid Motif. 6. Synthesis and Pharmacological Evaluation of 7-Substituted 4-Quinolone-3-carboxamide Derivatives as High Affinity Ligands for Cannabinoid Receptors
2012-01-01 Pasquini, Serena; De Rosa, Maria; Ligresti, A.; Mugnaini, Claudia; Brizzi, Antonella; Caradonna, N. P.; Cascio, M. G.; Bolognini, D.; Pertwee, R. G.; Di Marzo, V.; Corelli, Federico
Comparison of the effect of the positive allosteric modulator of the GABAb receptor, GS39783, on alcohol self-administration in three different lines of alcohol-preferring rats
2012-01-01 Maccioni, P.; Zaru, A.; Loi, B.; Lobina, C.; Carai, M. A. M.; Gessa, G. L.; Capra, A.; Mugnaini, Claudia; Pasquini, Serena; Corelli, Federico; Hyytiä, P.; Lumeng, L.; Colombo, G.
Design, Synthesis, and Pharmacological Characterization of Indole-3-ylacetamides, Indole-3-yloxoacetamides, and Indole-3-ylcarboxamides: Potent and Selective CB2 Cannabinoid Receptor Inverse Agonists
2012-01-01 Pasquini, Serena; Mugnaini, Claudia; Ligresti, A.; Tafi, Andrea; Brogi, Simone; Falciani, C.; Pedani, Valentina; Pesco, N.; Guida, F.; Luongo, L.; Varani, K.; Borea, P. A.; Maione, S.; Di Marzo, V.; Corelli, Federico
A novel CB2 agonist, COR167, potently protects rat brain cortical slices against OGD and reperfusion injury
2012-01-01 Contartese, Antonella; Valoti, Massimo; Corelli, Federico; Pasquini, Serena; Mugnaini, Claudia; Pessina, Federica; Aldinucci, Carlo; Sgaragli, GIAN PIETRO; Frosini, Maria
Investigations on the 4-Quinolone-3-carboxylic Acid Motif. 4. Identification of New Potent and Selective Ligands for the Cannabinoid Type 2 Receptor with Diverse Substitution Patterns and Antihyperalgesic Effects in Mice
2011-01-01 Pasquini, Serena; De Rosa, Maria; Pedani, Valentina; Mugnaini, Claudia; Guida, F.; Luongo, L.; De Chiaro, M; Maione, S.; Dragoni, Stefania; Frosini, Maria; Ligresti, A.; Di Marzo, V.; Corelli, Federico
Three-Dimensional Quantitative Structure-Selectivity Relationships (3D-QSSR) Analysis Guided Rational Design of a Highly Selective Ligand for the Cannabinoid Receptor 2
2011-01-01 Brogi, Simone; Corelli, Federico; Di Marzo, Vincenzo; Ligresti, Alessia; Mugnaini, Claudia; Pasquini, Serena; Tafi, Andrea
Development and characterization of immobilized cannabinoid receptor (CB1/CB2) open tubular column for on-line screening
2011-01-01 Moaddel, R.; Rosenberg, A.; Spelman, K.; Frazier, J.; Frazier, C.; Nocerino, S.; Brizzi, Antonella; Mugnaini, Claudia; Wainer, I. W.
Regioselective functionalization of quinolin-4(1H)-ones via sequential palladium-catalyzed reactions
2011-01-01 Mugnaini, Claudia; Falciani, Chiara; De Rosa, Maria; Brizzi, Antonella; Pasquini, Serena; Corelli, Federico
Activation of the GABAB receptor prevents nicotine-induced locomotor stimulation in mice
2011-01-01 Lobina, C.; Carai, M. A. M.; Froestl, W.; Mugnaini, Claudia; Pasquini, Serena; Corelli, Federico; G. e. s. s. a. G., L.; Colombo, G.
Reduction by the positive allosteric modulator of the GABAB receptor, GS39783, of alcohol self-administration in Sardinian alcohol-preferring rats exposed to the “sipper” procedure
2010-01-01 Maccioni, P.; Flore, P.; Carai, M. A. M.; Mugnaini, Claudia; Pasquini, Serena; Corelli, Federico; Gessa, G. L.; Colombo, G.
Investigations on the 4-Quinolone-3-carboxylic Acid Motif. 3. Synthesis, Structure-Affinity Relationships, and Pharmacological Characterization of 6-Substituted 4-Quinolone-3-carboxamides as Highly Selective Cannabinoid-2 Receptor Ligands
2010-01-01 Pasquini, Serena; Ligresti, A.; Mugnaini, Claudia; Semeraro, Teresa; Cicione, L.; De Rosa, Maria; Guida, F.; Luongo, L.; De Chiaro, M.; Cascio, M. G.; Bolognini, D.; Marini, P.; Pertwee, R.; Maione, S.; Di Marzo, V.; Corelli, Federico
The 4-Quinolone-3-carboxylic Acid Motif as a Multivalent Scaffold in Medicinal Chemistry
2009-01-01 Mugnaini, Claudia; Pasquini, Serena; Corelli, Federico
Rapid combinatorial access to a library of 1,5-disubstituted-3-indole-N-alkylacetamides as CB2 receptor ligands
2009-01-01 Pasquini, Serena; Mugnaini, Claudia; Brizzi, Antonella; Ligresti, A.; Di Marzo, V.; Ghiron, C.; Corelli, Federico
Synthesis and biological evaluation of guanidino compounds endowed with subnanomolar affinity as competitive inhibitors of maize polyamine oxidase
2009-01-01 Manetti, Fabrizio; Cona, A.; Angeli, L.; Mugnaini, Claudia; Raffi, F.; Capone, C.; Dreassi, Elena; Zizzari, A. T.; Tisi, A.; Federico, R.; Botta, Maurizio
| Titolo | Data di pubblicazione | Autore(i) | File | Abstract |
|---|---|---|---|---|
| Synthesis, 1 structural properties, and pharmacological evaluation of 2-(acylamino)thiophene-3-carboxamides and analogues thereof | 1-gen-2014 | Mugnaini, Claudia; Pedani, Valentina; Giunta, D.; Sechi, B.; Solinas, M.; Casti, A.; Castelli, M. P.; Giorgi, Gianluca; Corelli, Federico | - | |
| New fluoroquinolones active against fluoroquinolones-resistant Mycobacterium tuberculosis strains | 1-gen-2013 | Guerrini, Valentina; De Rosa, M.; Pasquini, S.; Mugnaini, Claudia; Brizzi, Antonella; Cuppone, Anna Maria; Pozzi, Gianni; Corelli, Federico | - | |
| Synthesis and pharmacological characterization of 2-(acylamino)thiophene derivatives as metabolically stable, orally effective, positive allosteric modulators of the GABAB receptor | 1-gen-2013 | Mugnaini, Claudia; Pedani, Valentina; Casu, Angelo; Lobina, Carla; Casti, Alberto; Maccioni, Paola; Porcu, Alessandra; Giunta, Daniela; Lamponi, Stefania; Solinas, Maurizio; Dragoni, Stefania; Valoti, Massimo; Colombo, Giancarlo; Castelli, Maria Paola; Gessa, Gian Luigi; Corelli, Federico | - | |
| Characterization of COR627 and COR628, two novel positive allosteric modulators of the GABA B receptor | 1-gen-2012 | Castelli, M. P.; Casu, A.; Casti, P.; Lobina, C.; Carai, M. A. M.; Colombo, G.; Solinas, M.; Giunta, D.; Mugnaini, Claudia; Pasquini, Serena; Tafi, Andrea; Brogi, Simone; Gessa, G. L.; Corelli, Federico | - | |
| The bioisosteric concept applied to cannabinoid ligands | 1-gen-2012 | Mugnaini, Claudia; Pasquini, Serena; Corelli, Federico | - | |
| Investigations on the 4-quinolone-3-carboxylic acid motif part 5: modulation of the physicochemical profile of a set of potent and selective cannabinoid-2 receptor ligands through a bioisosteric approach | 1-gen-2012 | Mugnaini, Claudia; Nocerino, S.; Pedani, Valentina; Pasquini, Serena; Tafi, Andrea; De Chiaro, M.; Bellucci, L.; Valoti, Massimo; Guida, F.; Luongo, L.; Dragoni, Stefania; Ligresti, A.; Rosenberg, A.; Bolognini, D.; Cascio, M. G.; Pertwee, R. G.; Moaddel, R.; Maione, S.; Di Marzo, V.; Corelli, Federico | - | |
| Investigations on the 4-Quinolone-3-carboxylic Acid Motif. 6. Synthesis and Pharmacological Evaluation of 7-Substituted 4-Quinolone-3-carboxamide Derivatives as High Affinity Ligands for Cannabinoid Receptors | 1-gen-2012 | Pasquini, Serena; De Rosa, Maria; Ligresti, A.; Mugnaini, Claudia; Brizzi, Antonella; Caradonna, N. P.; Cascio, M. G.; Bolognini, D.; Pertwee, R. G.; Di Marzo, V.; Corelli, Federico | - | |
| Comparison of the effect of the positive allosteric modulator of the GABAb receptor, GS39783, on alcohol self-administration in three different lines of alcohol-preferring rats | 1-gen-2012 | Maccioni, P.; Zaru, A.; Loi, B.; Lobina, C.; Carai, M. A. M.; Gessa, G. L.; Capra, A.; Mugnaini, Claudia; Pasquini, Serena; Corelli, Federico; Hyytiä, P.; Lumeng, L.; Colombo, G. | - | |
| Design, Synthesis, and Pharmacological Characterization of Indole-3-ylacetamides, Indole-3-yloxoacetamides, and Indole-3-ylcarboxamides: Potent and Selective CB2 Cannabinoid Receptor Inverse Agonists | 1-gen-2012 | Pasquini, Serena; Mugnaini, Claudia; Ligresti, A.; Tafi, Andrea; Brogi, Simone; Falciani, C.; Pedani, Valentina; Pesco, N.; Guida, F.; Luongo, L.; Varani, K.; Borea, P. A.; Maione, S.; Di Marzo, V.; Corelli, Federico | - | |
| A novel CB2 agonist, COR167, potently protects rat brain cortical slices against OGD and reperfusion injury | 1-gen-2012 | Contartese, Antonella; Valoti, Massimo; Corelli, Federico; Pasquini, Serena; Mugnaini, Claudia; Pessina, Federica; Aldinucci, Carlo; Sgaragli, GIAN PIETRO; Frosini, Maria | - | |
| Investigations on the 4-Quinolone-3-carboxylic Acid Motif. 4. Identification of New Potent and Selective Ligands for the Cannabinoid Type 2 Receptor with Diverse Substitution Patterns and Antihyperalgesic Effects in Mice | 1-gen-2011 | Pasquini, Serena; De Rosa, Maria; Pedani, Valentina; Mugnaini, Claudia; Guida, F.; Luongo, L.; De Chiaro, M; Maione, S.; Dragoni, Stefania; Frosini, Maria; Ligresti, A.; Di Marzo, V.; Corelli, Federico | - | |
| Three-Dimensional Quantitative Structure-Selectivity Relationships (3D-QSSR) Analysis Guided Rational Design of a Highly Selective Ligand for the Cannabinoid Receptor 2 | 1-gen-2011 | Brogi, Simone; Corelli, Federico; Di Marzo, Vincenzo; Ligresti, Alessia; Mugnaini, Claudia; Pasquini, Serena; Tafi, Andrea | - | |
| Development and characterization of immobilized cannabinoid receptor (CB1/CB2) open tubular column for on-line screening | 1-gen-2011 | Moaddel, R.; Rosenberg, A.; Spelman, K.; Frazier, J.; Frazier, C.; Nocerino, S.; Brizzi, Antonella; Mugnaini, Claudia; Wainer, I. W. | - | |
| Regioselective functionalization of quinolin-4(1H)-ones via sequential palladium-catalyzed reactions | 1-gen-2011 | Mugnaini, Claudia; Falciani, Chiara; De Rosa, Maria; Brizzi, Antonella; Pasquini, Serena; Corelli, Federico | - | |
| Activation of the GABAB receptor prevents nicotine-induced locomotor stimulation in mice | 1-gen-2011 | Lobina, C.; Carai, M. A. M.; Froestl, W.; Mugnaini, Claudia; Pasquini, Serena; Corelli, Federico; G. e. s. s. a. G., L.; Colombo, G. | - | |
| Reduction by the positive allosteric modulator of the GABAB receptor, GS39783, of alcohol self-administration in Sardinian alcohol-preferring rats exposed to the “sipper” procedure | 1-gen-2010 | Maccioni, P.; Flore, P.; Carai, M. A. M.; Mugnaini, Claudia; Pasquini, Serena; Corelli, Federico; Gessa, G. L.; Colombo, G. | - | |
| Investigations on the 4-Quinolone-3-carboxylic Acid Motif. 3. Synthesis, Structure-Affinity Relationships, and Pharmacological Characterization of 6-Substituted 4-Quinolone-3-carboxamides as Highly Selective Cannabinoid-2 Receptor Ligands | 1-gen-2010 | Pasquini, Serena; Ligresti, A.; Mugnaini, Claudia; Semeraro, Teresa; Cicione, L.; De Rosa, Maria; Guida, F.; Luongo, L.; De Chiaro, M.; Cascio, M. G.; Bolognini, D.; Marini, P.; Pertwee, R.; Maione, S.; Di Marzo, V.; Corelli, Federico | - | |
| The 4-Quinolone-3-carboxylic Acid Motif as a Multivalent Scaffold in Medicinal Chemistry | 1-gen-2009 | Mugnaini, Claudia; Pasquini, Serena; Corelli, Federico | - | |
| Rapid combinatorial access to a library of 1,5-disubstituted-3-indole-N-alkylacetamides as CB2 receptor ligands | 1-gen-2009 | Pasquini, Serena; Mugnaini, Claudia; Brizzi, Antonella; Ligresti, A.; Di Marzo, V.; Ghiron, C.; Corelli, Federico | - | |
| Synthesis and biological evaluation of guanidino compounds endowed with subnanomolar affinity as competitive inhibitors of maize polyamine oxidase | 1-gen-2009 | Manetti, Fabrizio; Cona, A.; Angeli, L.; Mugnaini, Claudia; Raffi, F.; Capone, C.; Dreassi, Elena; Zizzari, A. T.; Tisi, A.; Federico, R.; Botta, Maurizio | - |
Legenda icone
- file ad accesso aperto
- file disponibili sulla rete interna
- file disponibili agli utenti autorizzati
- file disponibili solo agli amministratori
- file sotto embargo
- nessun file disponibile