Sfoglia per Autore
Multipurpose Iron-Chelating Ligands Inspired by Bioavailable Molecules
2024-01-01 Cini, Elena; Crisponi, Guido; Fantasia, Alessandra; Cappai, Rosita; Siciliano, Sofia; Florio, Giuseppe Di; Nurchi, Valeria M.; Corsini, Maddalena
Structural Characterization of Human Heat Shock Protein 90 N-Terminal Domain and Its Variants K112R and K112A in Complex with a Potent 1,2,3-Triazole-Based Inhibitor
2022-01-01 Tassone, Giusy; Mazzorana, Marco; Mangani, Stefano; Petricci, Elena; Cini, Elena; Giannini, Giuseppe; Pozzi, Cecilia; Maramai, Samuele
Quinolines and Oxazino-quinoline Derivatives as Small Molecule GLI1 Inhibitors Identified by Virtual Screening
2022-01-01 Manetti, Fabrizio; Maresca, Luisa; Crivaro, Enrica; Pepe, Sara; Cini, Elena; Singh, Snigdha; Governa, Paolo; Maramai, Samuele; Giannini, Giuseppe; Stecca, Barbara; Petricci, Elena
Synthesis, characterization, electrochemistry and in vitro cytotoxicity of a new “Triazole-Maltol” ligand and its platinum(II) complex
2022-01-01 Fusi, S.; Di Florio, G.; Margiotta, N.; Barbanente, A.; Cini, E.; Finetti, F.; Paradisi, L.; Trabalzini, L.; Fabrizi de Biani, F.; Corsini, M.
A pH-responsive crosslinker platform for antibody-drug conjugate (ADC) targeting delivery
2022-01-01 Migliorini, Francesca; Cini, Elena; Dreassi, Elena; Finetti, Federica; Ievoli, Giovanni; Macrì, Giulia; Petricci, Elena; Rango, Enrico; Trabalzini, Lorenza; Taddei, Maurizio
Synthesis of 2-Substitued Indoles via Pd-Catalysed Cyclization in an Aqueous Micellar Medium
2021-01-01 Siciliano, Sofia; Cini, Elena; Taddei, Maurizio; Vinciarelli, Giorgia
Antibody drug conjugates with hydroxamic acid cargos for histone deacetylase (HDAC) inhibition
2021-01-01 Cianferotti, C.; Faltoni, V.; Cini, E.; Ermini, E.; Migliorini, F.; Petricci, E.; Taddei, M.; Salvini, L.; Battistuzzi, G.; Milazzo, F. M.; Anastasi, A. M.; Chiapparino, C.; De Santis, R.; Giannini, G.
ErbB2 Targeted Epigenetic Modulation: Anti-tumor Efficacy of the ADC Trastuzumab-HDACi ST8176AA1
2020-01-01 Maria Milazzo, Ferdinando; Vesci, Loredana; Maria Anastasi, Anna; Chiapparino, Caterina; Rosi, Antonio; Giannini, Giuseppe; Taddei, Maurizio; Cini, Elena; Faltoni, Valentina; Petricci, Elena; Battistuzzi, Gianfranco; Salvini, Laura; Carollo, Valeria; De Santis, Rita
Metal Catalysis with Microwaves in Organic Synthesis: a Personal Account
2020-01-01 Petricci, E.; Cini, E.; Taddei, M.
In water alkylation of amines with alcohols through a borrowing hydrogen process catalysed by ruthenium nanoparticles
2020-01-01 Risi, Caterina; Calamante, Massimo; Cini, Elena; Faltoni, Valentina; Petricci, Elena; Rosati, Filippo; Taddei, Maurizio
In Water Markovnikov Hydration and One-Pot Reductive Hydroamination of Terminal Alkynes under Ruthenium Nanoparticle Catalysis
2020-01-01 Risi, C.; Cini, E.; Petricci, E.; Saponaro, S.; Taddei, M.
Microwave Dielectric Heating for Solvent-free Organic Transformations
2019-01-01 Cini, Elena; Taddei, Maurizio
Stereoselective Synthesis of Sofosbuvir through Nucleoside Phosphorylation Controlled by Kinetic Resolution
2018-01-01 Cini, Elena; Barreca, Giuseppe; Carcone, Luca; Manetti, Fabrizio; Rasparini, Marcello; Taddei, Maurizio
Hedgehog pathway inhibitors of the acylthiourea and acylguanidine class show antitumor activity on colon cancer in vitro and in vivo
2018-01-01 Vesci, Loredana; Milazzo, Ferdinando Maria; Stasi, Maria Antonietta; Pace, Silvia; Manera, Francesco; Tallarico, Carlo; Cini, Elena; Petricci, Elena; Manetti, Fabrizio; De Santis, Rita; Giannini, Giuseppe
Antibody drug conjugates (ADCs) charged with HDAC inhibitor for targeted epigenetic modulation
2018-01-01 Cini, Elena; Faltoni, Valentina; Petricci, Elena; Taddei, Maurizio; Salvini, Laura; Giannini, Giuseppe; Vesci, Loredana; Milazzo, Ferdinando Maria; Anastasi, Anna Maria; Battistuzzi, Gianfranco; De Santis, Rita
Iron-Catalyzed Reductive Amination of Aldehydes in Isopropyl Alcohol/Water Media as Hydrogen Sources
2018-01-01 Petricci, Elena; Santillo, Niccolò; Castagnolo, Daniele; Cini, Elena; Taddei, Maurizio
Benzodiazepine scaffold as drug-like molecular simplification of FR235222: A chemical tool for exploring HDAC inhibition
2017-01-01 Randino, Rosario; Moronese, Ilaria; Cini, Elena; Bizzarro, Valentina; Persico, Marco; Grimaldi, Manuela; Scrima, Mario; D’Ursi, Anna Maria; Novellino, Ettore; Sobarzo Sánchez, Eduardo; Rastrelli, Luca; Fattorusso, Caterina; Petrella, Antonello; Rodriquez, Manuela; Taddei, Maurizio
Pd/C catalysis under microwave dielectric heating
2017-01-01 Cini, Elena; Petricci, Elena; Taddei, Maurizio
Nucleoside phosphoramidates useful for the treatment of viral infections and preparation thereof
2016-01-01 Barreca, Giuseppe; Rasparini, Marcello; Poggiali, Andrea; Carcone, Luca; Tufaro, Roberto Rocco; Marras, Giovanni; Taddei, Maurizio; Cini, Elena
Convergent Synthesis of the Renin Inhibitor Aliskiren Based on C5–C6 Disconnection and CO2H–NH2Equivalence
2016-01-01 Cini, Elena; Banfi, Luca; Barreca, Giuseppe; Carcone, Luca; Malpezzi, Luciana; Manetti, Fabrizio; Marras, Giovanni; Rasparini, Marcello; Riva, Renata; Roseblade, Stephen; Russo, Adele; Taddei, Maurizio; Vitale, Romina; Zanotti Gerosa, Antonio
Titolo | Data di pubblicazione | Autore(i) | File | Abstract |
---|---|---|---|---|
Multipurpose Iron-Chelating Ligands Inspired by Bioavailable Molecules | 1-gen-2024 | Cini, Elena; Crisponi, Guido; Fantasia, Alessandra; Cappai, Rosita; Siciliano, Sofia; Florio, Giuseppe Di; Nurchi, Valeria M.; Corsini, Maddalena | - | |
Structural Characterization of Human Heat Shock Protein 90 N-Terminal Domain and Its Variants K112R and K112A in Complex with a Potent 1,2,3-Triazole-Based Inhibitor | 1-gen-2022 | Tassone, Giusy; Mazzorana, Marco; Mangani, Stefano; Petricci, Elena; Cini, Elena; Giannini, Giuseppe; Pozzi, Cecilia; Maramai, Samuele | - | |
Quinolines and Oxazino-quinoline Derivatives as Small Molecule GLI1 Inhibitors Identified by Virtual Screening | 1-gen-2022 | Manetti, Fabrizio; Maresca, Luisa; Crivaro, Enrica; Pepe, Sara; Cini, Elena; Singh, Snigdha; Governa, Paolo; Maramai, Samuele; Giannini, Giuseppe; Stecca, Barbara; Petricci, Elena | - | |
Synthesis, characterization, electrochemistry and in vitro cytotoxicity of a new “Triazole-Maltol” ligand and its platinum(II) complex | 1-gen-2022 | Fusi, S.; Di Florio, G.; Margiotta, N.; Barbanente, A.; Cini, E.; Finetti, F.; Paradisi, L.; Trabalzini, L.; Fabrizi de Biani, F.; Corsini, M. | - | |
A pH-responsive crosslinker platform for antibody-drug conjugate (ADC) targeting delivery | 1-gen-2022 | Migliorini, Francesca; Cini, Elena; Dreassi, Elena; Finetti, Federica; Ievoli, Giovanni; Macrì, Giulia; Petricci, Elena; Rango, Enrico; Trabalzini, Lorenza; Taddei, Maurizio | - | |
Synthesis of 2-Substitued Indoles via Pd-Catalysed Cyclization in an Aqueous Micellar Medium | 1-gen-2021 | Siciliano, Sofia; Cini, Elena; Taddei, Maurizio; Vinciarelli, Giorgia | - | |
Antibody drug conjugates with hydroxamic acid cargos for histone deacetylase (HDAC) inhibition | 1-gen-2021 | Cianferotti, C.; Faltoni, V.; Cini, E.; Ermini, E.; Migliorini, F.; Petricci, E.; Taddei, M.; Salvini, L.; Battistuzzi, G.; Milazzo, F. M.; Anastasi, A. M.; Chiapparino, C.; De Santis, R.; Giannini, G. | - | |
ErbB2 Targeted Epigenetic Modulation: Anti-tumor Efficacy of the ADC Trastuzumab-HDACi ST8176AA1 | 1-gen-2020 | Maria Milazzo, Ferdinando; Vesci, Loredana; Maria Anastasi, Anna; Chiapparino, Caterina; Rosi, Antonio; Giannini, Giuseppe; Taddei, Maurizio; Cini, Elena; Faltoni, Valentina; Petricci, Elena; Battistuzzi, Gianfranco; Salvini, Laura; Carollo, Valeria; De Santis, Rita | - | |
Metal Catalysis with Microwaves in Organic Synthesis: a Personal Account | 1-gen-2020 | Petricci, E.; Cini, E.; Taddei, M. | - | |
In water alkylation of amines with alcohols through a borrowing hydrogen process catalysed by ruthenium nanoparticles | 1-gen-2020 | Risi, Caterina; Calamante, Massimo; Cini, Elena; Faltoni, Valentina; Petricci, Elena; Rosati, Filippo; Taddei, Maurizio | - | |
In Water Markovnikov Hydration and One-Pot Reductive Hydroamination of Terminal Alkynes under Ruthenium Nanoparticle Catalysis | 1-gen-2020 | Risi, C.; Cini, E.; Petricci, E.; Saponaro, S.; Taddei, M. | - | |
Microwave Dielectric Heating for Solvent-free Organic Transformations | 1-gen-2019 | Cini, Elena; Taddei, Maurizio | - | |
Stereoselective Synthesis of Sofosbuvir through Nucleoside Phosphorylation Controlled by Kinetic Resolution | 1-gen-2018 | Cini, Elena; Barreca, Giuseppe; Carcone, Luca; Manetti, Fabrizio; Rasparini, Marcello; Taddei, Maurizio | - | |
Hedgehog pathway inhibitors of the acylthiourea and acylguanidine class show antitumor activity on colon cancer in vitro and in vivo | 1-gen-2018 | Vesci, Loredana; Milazzo, Ferdinando Maria; Stasi, Maria Antonietta; Pace, Silvia; Manera, Francesco; Tallarico, Carlo; Cini, Elena; Petricci, Elena; Manetti, Fabrizio; De Santis, Rita; Giannini, Giuseppe | - | |
Antibody drug conjugates (ADCs) charged with HDAC inhibitor for targeted epigenetic modulation | 1-gen-2018 | Cini, Elena; Faltoni, Valentina; Petricci, Elena; Taddei, Maurizio; Salvini, Laura; Giannini, Giuseppe; Vesci, Loredana; Milazzo, Ferdinando Maria; Anastasi, Anna Maria; Battistuzzi, Gianfranco; De Santis, Rita | - | |
Iron-Catalyzed Reductive Amination of Aldehydes in Isopropyl Alcohol/Water Media as Hydrogen Sources | 1-gen-2018 | Petricci, Elena; Santillo, Niccolò; Castagnolo, Daniele; Cini, Elena; Taddei, Maurizio | - | |
Benzodiazepine scaffold as drug-like molecular simplification of FR235222: A chemical tool for exploring HDAC inhibition | 1-gen-2017 | Randino, Rosario; Moronese, Ilaria; Cini, Elena; Bizzarro, Valentina; Persico, Marco; Grimaldi, Manuela; Scrima, Mario; D’Ursi, Anna Maria; Novellino, Ettore; Sobarzo Sánchez, Eduardo; Rastrelli, Luca; Fattorusso, Caterina; Petrella, Antonello; Rodriquez, Manuela; Taddei, Maurizio | - | |
Pd/C catalysis under microwave dielectric heating | 1-gen-2017 | Cini, Elena; Petricci, Elena; Taddei, Maurizio | - | |
Nucleoside phosphoramidates useful for the treatment of viral infections and preparation thereof | 1-gen-2016 | Barreca, Giuseppe; Rasparini, Marcello; Poggiali, Andrea; Carcone, Luca; Tufaro, Roberto Rocco; Marras, Giovanni; Taddei, Maurizio; Cini, Elena | - | |
Convergent Synthesis of the Renin Inhibitor Aliskiren Based on C5–C6 Disconnection and CO2H–NH2Equivalence | 1-gen-2016 | Cini, Elena; Banfi, Luca; Barreca, Giuseppe; Carcone, Luca; Malpezzi, Luciana; Manetti, Fabrizio; Marras, Giovanni; Rasparini, Marcello; Riva, Renata; Roseblade, Stephen; Russo, Adele; Taddei, Maurizio; Vitale, Romina; Zanotti Gerosa, Antonio | - |
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