Sfoglia per Autore
Consensus screening for a challenging target: the quest for P-glycoprotein inhibitors
2024-01-01 Governa, Paolo; Biagi, Marco; Manetti, Fabrizio; Forli, Stefano
Early investigation of a novel SI306 theranostic prodrug for glioblastoma treatment
2024-01-01 Vagaggini, Chiara; Petroni, Debora; D'Agostino, Ilaria; Poggialini, Federica; Cavallini, Chiara; Cianciusi, Annarita; Salis, Annalisa; D'Antona, Lucia; Francesconi, Valeria; Manetti, Fabrizio; Damonte, Gianluca; Musumeci, Francesca; Menichetti, Luca; Dreassi, Elena; Carbone, Anna; Schenone, Silvia
Targeting GLI1 and GLI2 with small molecule inhibitors to suppress GLI-dependent transcription and tumor growth
2023-01-01 Maresca, Luisa; Crivaro, Enrica; Migliorini, Francesca; Anichini, Giulia; Giammona, Alessandro; Pepe, Sara; Poggialini, Federica; Vagaggini, Chiara; Giannini, Giuseppe; Sestini, Serena; Borgognoni, Lorenzo; Lapucci, Andrea; Dreassi, Elena; Taddei, Maurizio; Manetti, Fabrizio; Petricci, Elena; Stecca, Barbara
CanB, a Druggable Cellular Target in Mycobacterium tuberculosis
2023-01-01 Degiacomi, G; Gianibbi, B; Recchia, D; Stelitano, G; Truglio, Gi; Marra, P; Stamilla, A; Makarov, V; Chiarelli, Lr; Manetti, F; Pasca, Mr
Helichrysum stoechas (L.) Moench reduces body weight gain and modulates mood disorders via inhibition of silent information regulator 1 (SIRT1) by arzanol
2023-01-01 Borgonetti, Vittoria; Caroli, Clarissa; Governa, Paolo; Virginia, Brighenti; Pollastro, Federica; Franchini, Silvia; Manetti, Fabrizio; Les, Francisco; López, Victor; Pellati, Federica; Galeotti, Nicoletta
Effect of in vitro simulated digestion on the anti-Helicobacter Pylori activity of different Propolis extracts
2023-01-01 Governa, Paolo; Romagnoli, Giulia; Albanese, Paola; Rossi, Federico; Manetti, Fabrizio; Biagi, Marco
Zingiberene, a non-zinc-binding class I HDAC inhibitor: A novel strategy for the management of neuropathic pain
2023-01-01 Borgonetti, Vittoria; Governa, Paolo; Manetti, Fabrizio; Galeotti, Nicoletta
Antiviral Activity of Cannabidiolic Acid and Its Methyl Ester against SARS-CoV-2
2023-01-01 Tamburello, Martina; Salamone, Stefano; Anceschi, Lisa; Governa, Paolo; Brighenti, Virginia; Morellini, Alice; Rossini, Giada; Manetti, Fabrizio; Gallinella, Giorgio; Pollastro, Federica; Pellati, Federica
Cannabidiol-rich non-psychotropic Cannabis sativa L. oils attenuate peripheral neuropathy symptoms by regulation of CB2-mediated microglial neuroinflammation
2023-01-01 Borgonetti, Vittoria; Anceschi, Lisa; Brighenti, Virginia; Corsi, Lorenzo; Governa, Paolo; Manetti, Fabrizio; Pellati, Federica; Galeotti, Nicoletta
Investigation on the neuroprotective effect of a cannabidiol-enriched non-psychotropic Cannabis sativa L. extract in an in vitro model of excitotoxicity
2022-01-01 Borgonetti, Vittoria; Biagi, Marco; Galeotti, Nicoletta; Manetti, Fabrizio; Governa, Paolo
The Veterinary Anti-Parasitic Selamectin Is a Novel Inhibitor of the Mycobacterium tuberculosis DprE1 Enzyme
2022-01-01 Ezquerra-Aznárez, José Manuel; Degiacomi, Giulia; Gašparovič, Henrich; Stelitano, Giovanni; Sammartino, Josè Camilla; Korduláková, Jana; Governa, Paolo; Manetti, Fabrizio; Pasca, Maria Rosalia; Chiarelli, Laurent Roberto; Ramón-García, Santiago
Quinolines and Oxazino-quinoline Derivatives as Small Molecule GLI1 Inhibitors Identified by Virtual Screening
2022-01-01 Manetti, Fabrizio; Maresca, Luisa; Crivaro, Enrica; Pepe, Sara; Cini, Elena; Singh, Snigdha; Governa, Paolo; Maramai, Samuele; Giannini, Giuseppe; Stecca, Barbara; Petricci, Elena
Synthesis and biological activity evaluation of 3-(hetero) arylideneindolin-2-ones as potential c-Src inhibitors
2022-01-01 Princiotto, Salvatore; Musso, Loana; Manetti, Fabrizio; Marcellini, Valentina; Maga, Giovanni; Crespan, Emmanuele; Perini, Cecilia; Zaffaroni, Nadia; Beretta, Giovanni Luca; Dallavalle, Sabrina
Recent research results have converted gp120 binders to a therapeutic option for the treatment of HIV-1 infection. A medicinal chemistry point of view
2022-01-01 Governa, Paolo; Manetti, Fabrizio
Structural Rigidification of N-Aryl-pyrroles into Indoles Active against Intracellular and Drug-Resistant Mycobacteria
2022-01-01 Semenya, Dorothy; Touitou, Meir; Ribeiro, Camila Maringolo; Pavan, Fernando Rogerio; Pisano, Luca; Singh, Vinayak; Chibale, Kelly; Bano, Georg; Toscani, Anita; Manetti, Fabrizio; Gianibbi, Beatrice; Castagnolo, Daniele
Effects of in vitro simulated digestion on the antioxidant activity of different Camellia sinensis (L.) Kuntze leaves extracts
2022-01-01 Governa, Paolo; Manetti, Fabrizio; Miraldi, Elisabetta; Biagi, Marco
Survey on the Recent Advances in 4-Hydroxyphenylpyruvate Dioxygenase (HPPD) Inhibition by Diketone and Triketone Derivatives and Congeneric Compounds: Structural Analysis of HPPD/Inhibitor Complexes and Structure-Activity Relationship Considerations
2022-01-01 Governa, Paolo; Bernardini, Giulia; Braconi, Daniela; Manetti, Fabrizio; Santucci, Annalisa; Petricci, Elena
Non-psychotropic Cannabis sativa L. phytocomplex modulates microglial inflammatory response through CB2 receptors-, endocannabinoids-, and NF-κB-mediated signaling
2022-01-01 Borgonetti, V.; Benatti, C.; Governa, P.; Isoldi, G.; Pellati, F.; Alboni, S.; Tascedda, F.; Montopoli, M.; Galeotti, N.; Manetti, F.; Miraldi, E.; Biagi, M.; Rigillo, G.
Conformational insights into the C-terminal mutations of human rhodopsin in retinitis pigmentosa
2022-01-01 Picarazzi, Francesca; Manetti, Fabrizio; Marigo, Valeria; Mori, Mattia
Tapping into the antitubercular potential of 2,5-dimethylpyrroles: A structure-activity relationship interrogation
2022-01-01 Semenya, D.; Touitou, M.; Masci, D.; Ribeiro, C. M.; Pavan, F. R.; Dos Santos Fernandes, G. F.; Gianibbi, B.; Manetti, F.; Castagnolo, D.
| Titolo | Data di pubblicazione | Autore(i) | File | Abstract |
|---|---|---|---|---|
| Consensus screening for a challenging target: the quest for P-glycoprotein inhibitors | 1-gen-2024 | Governa, Paolo; Biagi, Marco; Manetti, Fabrizio; Forli, Stefano | - | |
| Early investigation of a novel SI306 theranostic prodrug for glioblastoma treatment | 1-gen-2024 | Vagaggini, Chiara; Petroni, Debora; D'Agostino, Ilaria; Poggialini, Federica; Cavallini, Chiara; Cianciusi, Annarita; Salis, Annalisa; D'Antona, Lucia; Francesconi, Valeria; Manetti, Fabrizio; Damonte, Gianluca; Musumeci, Francesca; Menichetti, Luca; Dreassi, Elena; Carbone, Anna; Schenone, Silvia | - | |
| Targeting GLI1 and GLI2 with small molecule inhibitors to suppress GLI-dependent transcription and tumor growth | 1-gen-2023 | Maresca, Luisa; Crivaro, Enrica; Migliorini, Francesca; Anichini, Giulia; Giammona, Alessandro; Pepe, Sara; Poggialini, Federica; Vagaggini, Chiara; Giannini, Giuseppe; Sestini, Serena; Borgognoni, Lorenzo; Lapucci, Andrea; Dreassi, Elena; Taddei, Maurizio; Manetti, Fabrizio; Petricci, Elena; Stecca, Barbara | - | |
| CanB, a Druggable Cellular Target in Mycobacterium tuberculosis | 1-gen-2023 | Degiacomi, G; Gianibbi, B; Recchia, D; Stelitano, G; Truglio, Gi; Marra, P; Stamilla, A; Makarov, V; Chiarelli, Lr; Manetti, F; Pasca, Mr | - | |
| Helichrysum stoechas (L.) Moench reduces body weight gain and modulates mood disorders via inhibition of silent information regulator 1 (SIRT1) by arzanol | 1-gen-2023 | Borgonetti, Vittoria; Caroli, Clarissa; Governa, Paolo; Virginia, Brighenti; Pollastro, Federica; Franchini, Silvia; Manetti, Fabrizio; Les, Francisco; López, Victor; Pellati, Federica; Galeotti, Nicoletta | - | |
| Effect of in vitro simulated digestion on the anti-Helicobacter Pylori activity of different Propolis extracts | 1-gen-2023 | Governa, Paolo; Romagnoli, Giulia; Albanese, Paola; Rossi, Federico; Manetti, Fabrizio; Biagi, Marco | - | |
| Zingiberene, a non-zinc-binding class I HDAC inhibitor: A novel strategy for the management of neuropathic pain | 1-gen-2023 | Borgonetti, Vittoria; Governa, Paolo; Manetti, Fabrizio; Galeotti, Nicoletta | - | |
| Antiviral Activity of Cannabidiolic Acid and Its Methyl Ester against SARS-CoV-2 | 1-gen-2023 | Tamburello, Martina; Salamone, Stefano; Anceschi, Lisa; Governa, Paolo; Brighenti, Virginia; Morellini, Alice; Rossini, Giada; Manetti, Fabrizio; Gallinella, Giorgio; Pollastro, Federica; Pellati, Federica | - | |
| Cannabidiol-rich non-psychotropic Cannabis sativa L. oils attenuate peripheral neuropathy symptoms by regulation of CB2-mediated microglial neuroinflammation | 1-gen-2023 | Borgonetti, Vittoria; Anceschi, Lisa; Brighenti, Virginia; Corsi, Lorenzo; Governa, Paolo; Manetti, Fabrizio; Pellati, Federica; Galeotti, Nicoletta | - | |
| Investigation on the neuroprotective effect of a cannabidiol-enriched non-psychotropic Cannabis sativa L. extract in an in vitro model of excitotoxicity | 1-gen-2022 | Borgonetti, Vittoria; Biagi, Marco; Galeotti, Nicoletta; Manetti, Fabrizio; Governa, Paolo | - | |
| The Veterinary Anti-Parasitic Selamectin Is a Novel Inhibitor of the Mycobacterium tuberculosis DprE1 Enzyme | 1-gen-2022 | Ezquerra-Aznárez, José Manuel; Degiacomi, Giulia; Gašparovič, Henrich; Stelitano, Giovanni; Sammartino, Josè Camilla; Korduláková, Jana; Governa, Paolo; Manetti, Fabrizio; Pasca, Maria Rosalia; Chiarelli, Laurent Roberto; Ramón-García, Santiago | - | |
| Quinolines and Oxazino-quinoline Derivatives as Small Molecule GLI1 Inhibitors Identified by Virtual Screening | 1-gen-2022 | Manetti, Fabrizio; Maresca, Luisa; Crivaro, Enrica; Pepe, Sara; Cini, Elena; Singh, Snigdha; Governa, Paolo; Maramai, Samuele; Giannini, Giuseppe; Stecca, Barbara; Petricci, Elena | - | |
| Synthesis and biological activity evaluation of 3-(hetero) arylideneindolin-2-ones as potential c-Src inhibitors | 1-gen-2022 | Princiotto, Salvatore; Musso, Loana; Manetti, Fabrizio; Marcellini, Valentina; Maga, Giovanni; Crespan, Emmanuele; Perini, Cecilia; Zaffaroni, Nadia; Beretta, Giovanni Luca; Dallavalle, Sabrina | - | |
| Recent research results have converted gp120 binders to a therapeutic option for the treatment of HIV-1 infection. A medicinal chemistry point of view | 1-gen-2022 | Governa, Paolo; Manetti, Fabrizio | - | |
| Structural Rigidification of N-Aryl-pyrroles into Indoles Active against Intracellular and Drug-Resistant Mycobacteria | 1-gen-2022 | Semenya, Dorothy; Touitou, Meir; Ribeiro, Camila Maringolo; Pavan, Fernando Rogerio; Pisano, Luca; Singh, Vinayak; Chibale, Kelly; Bano, Georg; Toscani, Anita; Manetti, Fabrizio; Gianibbi, Beatrice; Castagnolo, Daniele | - | |
| Effects of in vitro simulated digestion on the antioxidant activity of different Camellia sinensis (L.) Kuntze leaves extracts | 1-gen-2022 | Governa, Paolo; Manetti, Fabrizio; Miraldi, Elisabetta; Biagi, Marco | - | |
| Survey on the Recent Advances in 4-Hydroxyphenylpyruvate Dioxygenase (HPPD) Inhibition by Diketone and Triketone Derivatives and Congeneric Compounds: Structural Analysis of HPPD/Inhibitor Complexes and Structure-Activity Relationship Considerations | 1-gen-2022 | Governa, Paolo; Bernardini, Giulia; Braconi, Daniela; Manetti, Fabrizio; Santucci, Annalisa; Petricci, Elena | - | |
| Non-psychotropic Cannabis sativa L. phytocomplex modulates microglial inflammatory response through CB2 receptors-, endocannabinoids-, and NF-κB-mediated signaling | 1-gen-2022 | Borgonetti, V.; Benatti, C.; Governa, P.; Isoldi, G.; Pellati, F.; Alboni, S.; Tascedda, F.; Montopoli, M.; Galeotti, N.; Manetti, F.; Miraldi, E.; Biagi, M.; Rigillo, G. | - | |
| Conformational insights into the C-terminal mutations of human rhodopsin in retinitis pigmentosa | 1-gen-2022 | Picarazzi, Francesca; Manetti, Fabrizio; Marigo, Valeria; Mori, Mattia | - | |
| Tapping into the antitubercular potential of 2,5-dimethylpyrroles: A structure-activity relationship interrogation | 1-gen-2022 | Semenya, D.; Touitou, M.; Masci, D.; Ribeiro, C. M.; Pavan, F. R.; Dos Santos Fernandes, G. F.; Gianibbi, B.; Manetti, F.; Castagnolo, D. | - |
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