Sfoglia per Autore
Omicron variants of SARS CoV-2 indicate a new antiviral strategy: Interfere with spike glycoprotein trimerization
2023-01-01 Niccolai, Neri; Trezza, Alfonso; Marchini, Federico; Bongini, Pietro; Bianchini, Monica; Santucci, Annalisa; Spiga, Ottavia; Visibelli, Anna
Dynamin-independent CaV1.2 and KCa1.1 channels regulation and vascular tone modulation by the mitochondrial fission inhibitors dynasore and dyngo-4a
2023-01-01 Ahmed, Amer; Trezza, Alfonso; Gentile, Mariangela; Paccagnini, Eugenio; Panti, Alice; Lupetti, Pietro; Spiga, Ottavia; Bova, Sergio; Fusi, Fabio
Functional, electrophysiology, and molecular dynamics analysis of quercetin-induced contraction of rat vascular musculature
2022-01-01 Trezza, A.; Spiga, O.; Mugnai, P.; Saponara, S.; Sgaragli, G.; Fusi, F.
Artificial intelligence-driven identification of morin analogues acting as CaV1.2 channel blockers: Synthesis and biological evaluation
2022-01-01 Carullo, G.; Falbo, F.; Ahmed, A.; Trezza, A.; Gianibbi, B.; Nicolotti, O.; Campiani, G.; Aiello, F.; Saponara, S.; Fusi, F.
Structural bioinformatic survey of protein-small molecule interfaces delineates the role of glycine in surface pocket formation
2022-01-01 Bongini, Pietro; Niccolai, Neri; Trezza, Alfonso; Mangiavacchi, Guido; Santucci, Annalisa; Spiga, Ottavia; Bianchini, Monica; Gardini, Simone
Novel Labdane Diterpenes-Based Synthetic Derivatives: Identification of a Bifunctional Vasodilator That Inhibits CaV1.2 and Stimulates KCa1.1 Channels
2022-01-01 Carullo, Gabriele; Saponara, Simona; Ahmed, Amer; Gorelli, Beatrice; Mazzotta, Sarah; Trezza, Alfonso; Gianibbi, Beatrice; Campiani, Giuseppe; Fusi, Fabio; Aiello, Francesca
Targeting neuronal calcium channels and GSK3β for Alzheimer's disease with naturally-inspired Diels-Alder adducts
2022-01-01 Bisi, Alessandra; Feoli, Alessandra; Trezza, Alfonso; Viejo, Lucia; Formaggio, Francesco; Bartolini, Manuela; Belluti, Federica; Gobbi, Silvia; Spiga, Ottavia; Caprini, Marco; de Los Rios, Cristobal; Castellano, Sabrina; Rampa, Angela
The drp-1-mediated mitochondrial fission inhibitor mdivi-1 impacts the function of ion channels and pathways underpinning vascular smooth muscle tone
2022-01-01 Ahmed, Amer; Trezza, Alfonso; Gentile, Mariangela; Paccagnini, Eugenio; Lupetti, Pietro; Spiga, Ottavia; Bova, Sergio; Fusi, Fabio
Pharmacological and In Silico Analysis of Oat Avenanthramides as EGFR Inhibitors: Effects on EGF-Induced Lung Cancer Cell Growth and Migration
2022-01-01 Trabalzini, Lorenza; Ercoli, Jasmine; Trezza, Alfonso; Schiavo, Irene; Macrì, Giulia; Moglia, Andrea; Spiga, Ottavia; Finetti, Federica
In Silico Multi-Target Approach Revealed Potential Lead Compounds as Scaffold for the Synthesis of Chemical Analogues Targeting SARS-CoV-2
2022-01-01 Trezza, Alfonso; Mugnaini, Claudia; Corelli, Federico; Santucci, Annalisa; Spiga, Ottavia
Vietnamese Dalbergia tonkinensis: A Promising Source of Mono- and Bifunctional Vasodilators
2022-01-01 Cuong, Nguyen Manh; Son, Ninh The; Nhan, Ngu Truong; Fukuyama, Yoshiyasu; Ahmed, Amer; Saponara, Simona; Trezza, Alfonso; Gianibbi, Beatrice; Vigni, Ginevra; Spiga, Ottavia; Fusi, Fabio
Multifaceted activity of polyciclic MDR revertant agents in drug-resistant leukemic cells: Role of the spacer
2021-01-01 Caciolla, Jessica; Picone, Giovanna; Farruggia, Giovanna; Valenti, Dario; Rampa, Angela; Malucelli, Emil; Belluti, Federica; Trezza, Alfonso; Spiga, Ottavia; Iotti, Stefano; Gobbi, Silvia; Cappadone, Concettina; Bisi, Alessandra
Structural Bioinformatics to unveil weaknesses of coronavirus spike glycoprotein stability
2021-01-01 Bongini, Pietro; Trezza, Alfonso; Bianchini, Monica; Spiga, Ottavia; Niccolai, Neri
2-hydroxy-4-(3,5,7-trihydroxy-4-oxo-4H-chromen-2-yl)phenyl(E)-3-(4-hydroxy-3-methoxyphenyl)acrylate: synthesis, in silico analysis and in vitro pharmacological evaluation
2021-01-01 Brizzi, A.; Trezza, A.; Spiga, O.; Maramai, S.; Scorzelli, F.; Saponara, S.; Fusi, F.
Flavonoids and hERG channels: Friends or foes?
2021-01-01 Saponara, S.; Fusi, F.; Iovinelli, D.; Ahmed, A.; Trezza, A.; Spiga, O.; Sgaragli, G.; Valoti, M.
A multitarget semi-synthetic derivative of the flavonoid morin with improved in vitro vasorelaxant activity: Role of CaV1.2 and KCa1.1 channels
2021-01-01 Carullo, G.; Ahmed, A.; Trezza, A.; Spiga, O.; Brizzi, A.; Saponara, S.; Fusi, F.; Aiello, F.
Potential roles of protease inhibitors in anticancer therapy
2020-01-01 Trezza, A.; Cicaloni, V.; Pettini, F.; Spiga, O.
Ritanserin blocks CaV1.2 channels in rat artery smooth muscles: electrophysiological, functional, and computational studies
2020-01-01 Fusi, F.; Trezza, A.; Sgaragli, G.; Spiga, O.; Saponara, S.; Bova, S.
An integrated drug repurposing strategy for the rapid identification of potential SARS-CoV-2 viral inhibitors
2020-01-01 Trezza, A.; Iovinelli, D.; Santucci, A.; Prischi, F.; Spiga, O.
A possible strategy to fight COVID-19: Interfering with spike glycoprotein trimerization
2020-01-01 Bongini, Pietro; Trezza, Alfonso; Bianchini, Monica; Spiga, Ottavia; Niccolai, Neri
Titolo | Data di pubblicazione | Autore(i) | File | Abstract |
---|---|---|---|---|
Omicron variants of SARS CoV-2 indicate a new antiviral strategy: Interfere with spike glycoprotein trimerization | 1-gen-2023 | Niccolai, Neri; Trezza, Alfonso; Marchini, Federico; Bongini, Pietro; Bianchini, Monica; Santucci, Annalisa; Spiga, Ottavia; Visibelli, Anna | - | |
Dynamin-independent CaV1.2 and KCa1.1 channels regulation and vascular tone modulation by the mitochondrial fission inhibitors dynasore and dyngo-4a | 1-gen-2023 | Ahmed, Amer; Trezza, Alfonso; Gentile, Mariangela; Paccagnini, Eugenio; Panti, Alice; Lupetti, Pietro; Spiga, Ottavia; Bova, Sergio; Fusi, Fabio | - | |
Functional, electrophysiology, and molecular dynamics analysis of quercetin-induced contraction of rat vascular musculature | 1-gen-2022 | Trezza, A.; Spiga, O.; Mugnai, P.; Saponara, S.; Sgaragli, G.; Fusi, F. | - | |
Artificial intelligence-driven identification of morin analogues acting as CaV1.2 channel blockers: Synthesis and biological evaluation | 1-gen-2022 | Carullo, G.; Falbo, F.; Ahmed, A.; Trezza, A.; Gianibbi, B.; Nicolotti, O.; Campiani, G.; Aiello, F.; Saponara, S.; Fusi, F. | - | |
Structural bioinformatic survey of protein-small molecule interfaces delineates the role of glycine in surface pocket formation | 1-gen-2022 | Bongini, Pietro; Niccolai, Neri; Trezza, Alfonso; Mangiavacchi, Guido; Santucci, Annalisa; Spiga, Ottavia; Bianchini, Monica; Gardini, Simone | - | |
Novel Labdane Diterpenes-Based Synthetic Derivatives: Identification of a Bifunctional Vasodilator That Inhibits CaV1.2 and Stimulates KCa1.1 Channels | 1-gen-2022 | Carullo, Gabriele; Saponara, Simona; Ahmed, Amer; Gorelli, Beatrice; Mazzotta, Sarah; Trezza, Alfonso; Gianibbi, Beatrice; Campiani, Giuseppe; Fusi, Fabio; Aiello, Francesca | - | |
Targeting neuronal calcium channels and GSK3β for Alzheimer's disease with naturally-inspired Diels-Alder adducts | 1-gen-2022 | Bisi, Alessandra; Feoli, Alessandra; Trezza, Alfonso; Viejo, Lucia; Formaggio, Francesco; Bartolini, Manuela; Belluti, Federica; Gobbi, Silvia; Spiga, Ottavia; Caprini, Marco; de Los Rios, Cristobal; Castellano, Sabrina; Rampa, Angela | - | |
The drp-1-mediated mitochondrial fission inhibitor mdivi-1 impacts the function of ion channels and pathways underpinning vascular smooth muscle tone | 1-gen-2022 | Ahmed, Amer; Trezza, Alfonso; Gentile, Mariangela; Paccagnini, Eugenio; Lupetti, Pietro; Spiga, Ottavia; Bova, Sergio; Fusi, Fabio | - | |
Pharmacological and In Silico Analysis of Oat Avenanthramides as EGFR Inhibitors: Effects on EGF-Induced Lung Cancer Cell Growth and Migration | 1-gen-2022 | Trabalzini, Lorenza; Ercoli, Jasmine; Trezza, Alfonso; Schiavo, Irene; Macrì, Giulia; Moglia, Andrea; Spiga, Ottavia; Finetti, Federica | - | |
In Silico Multi-Target Approach Revealed Potential Lead Compounds as Scaffold for the Synthesis of Chemical Analogues Targeting SARS-CoV-2 | 1-gen-2022 | Trezza, Alfonso; Mugnaini, Claudia; Corelli, Federico; Santucci, Annalisa; Spiga, Ottavia | - | |
Vietnamese Dalbergia tonkinensis: A Promising Source of Mono- and Bifunctional Vasodilators | 1-gen-2022 | Cuong, Nguyen Manh; Son, Ninh The; Nhan, Ngu Truong; Fukuyama, Yoshiyasu; Ahmed, Amer; Saponara, Simona; Trezza, Alfonso; Gianibbi, Beatrice; Vigni, Ginevra; Spiga, Ottavia; Fusi, Fabio | - | |
Multifaceted activity of polyciclic MDR revertant agents in drug-resistant leukemic cells: Role of the spacer | 1-gen-2021 | Caciolla, Jessica; Picone, Giovanna; Farruggia, Giovanna; Valenti, Dario; Rampa, Angela; Malucelli, Emil; Belluti, Federica; Trezza, Alfonso; Spiga, Ottavia; Iotti, Stefano; Gobbi, Silvia; Cappadone, Concettina; Bisi, Alessandra | - | |
Structural Bioinformatics to unveil weaknesses of coronavirus spike glycoprotein stability | 1-gen-2021 | Bongini, Pietro; Trezza, Alfonso; Bianchini, Monica; Spiga, Ottavia; Niccolai, Neri | - | |
2-hydroxy-4-(3,5,7-trihydroxy-4-oxo-4H-chromen-2-yl)phenyl(E)-3-(4-hydroxy-3-methoxyphenyl)acrylate: synthesis, in silico analysis and in vitro pharmacological evaluation | 1-gen-2021 | Brizzi, A.; Trezza, A.; Spiga, O.; Maramai, S.; Scorzelli, F.; Saponara, S.; Fusi, F. | - | |
Flavonoids and hERG channels: Friends or foes? | 1-gen-2021 | Saponara, S.; Fusi, F.; Iovinelli, D.; Ahmed, A.; Trezza, A.; Spiga, O.; Sgaragli, G.; Valoti, M. | - | |
A multitarget semi-synthetic derivative of the flavonoid morin with improved in vitro vasorelaxant activity: Role of CaV1.2 and KCa1.1 channels | 1-gen-2021 | Carullo, G.; Ahmed, A.; Trezza, A.; Spiga, O.; Brizzi, A.; Saponara, S.; Fusi, F.; Aiello, F. | - | |
Potential roles of protease inhibitors in anticancer therapy | 1-gen-2020 | Trezza, A.; Cicaloni, V.; Pettini, F.; Spiga, O. | - | |
Ritanserin blocks CaV1.2 channels in rat artery smooth muscles: electrophysiological, functional, and computational studies | 1-gen-2020 | Fusi, F.; Trezza, A.; Sgaragli, G.; Spiga, O.; Saponara, S.; Bova, S. | - | |
An integrated drug repurposing strategy for the rapid identification of potential SARS-CoV-2 viral inhibitors | 1-gen-2020 | Trezza, A.; Iovinelli, D.; Santucci, A.; Prischi, F.; Spiga, O. | - | |
A possible strategy to fight COVID-19: Interfering with spike glycoprotein trimerization | 1-gen-2020 | Bongini, Pietro; Trezza, Alfonso; Bianchini, Monica; Spiga, Ottavia; Niccolai, Neri | - |
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