Sfoglia per Autore
Synthesis and biological investigation of peptidomimetic SARS‐CoV‐2 main protease inhibitors bearing quinoline‐based heterocycles at P3
2025-01-01 Rossi, Sara; Deidda, Graziano; Fiaschi, Lia; Ibba, Roberta; Pieroni, Mariachiara; Dichiara, Maria; Carullo, Gabriele; Butini, Stefania; Ramunno, Anna; Brogi, Simone; Lolicato, Marco; Arrigoni, Cristina; Cabella, Noemi; Bavagnoli, Laura; Maga, Giovanni; Varasi, Ilenia; Biba, Camilla; Vicenti, Ilaria; Gemma, Sandra; Crespan, Emmanuele; Zazzi, Maurizio; Campiani, Giuseppe
Targeting N‐Methyl‐lysine Histone Demethylase KDM4 in Cancer: Natural Products Inhibitors as a Driving Force for Epigenetic Drug Discovery
2024-01-01 Cursaro, Ilaria; Milioni, Leonardo; Eslami, Kourosh; Sirous, Hajar; Carullo, Gabriele; Gemma, Sandra; Butini, Stefania; Campiani, Giuseppe
Enhancing Drug Discovery and Development through the Integration of Medicinal Chemistry, Chemical Biology, and Academia-Industry Partnerships: Insights from Roche’s Endocannabinoid System Projects
2024-01-01 Aebi, Johannes; Atz, Kenneth; Ametamey, Simon M.; Benz, Jörg; Blaising, Julie; Butini, Stefania; Campiani, Giuseppe; Carreira, Erick M.; Collin, Ludovic; De Lago, Eva; Gazzi, Thais; Gertsch, Jürg; Gobbi, Luca; Guba, Wolfgang; Fernández-Ruiz, Javier; Fingerle, Jürgen; Haider, Ahmed; He, Yingfang; Heitman, Laura H.; Honer, Michael; Hunziker, Daniel; Kuhn, Bernd; Maccarrone, Mauro; Märki, Hans Peter; Martin, Rainer E.; Mohr, Peter; Mu, Linjing; Nazaré, Marc; Nippa, David F.; Oddi, Sergio; O'Hara, Fionn; Pacher, Pal; Romero, Julian; Röver, Stephan; Rufer, Arne C.; Schibli, Roger; Schneider, Gisbert; Stepan, Antonia F.; Sykes, David A.; Ullmer, Christoph; Van der Stelt, Mario; Veprintsev, Dmitry B.; Wittwer, Matthias B.; Grether, Uwe
Spirotetrahydroisoquinoline-Based Histone Deacetylase Inhibitors as New Antifibrotic Agents: Biological Evaluation in Human Fibroblasts from Bronchoalveolar Lavages of Idiopathic Pulmonary Fibrosis Patients
2024-01-01 Fontana, Anna; Bergantini, Laura; Carullo, Gabriele; Scalvini, Laura; D'Alessandro, Miriana; Papulino, Chiara; Cameli, Paolo; Gangi, Sara; Vincenzi, Fabrizio; Varani, Katia; Contri, Chiara; Pasquini, Silvia; Pistocchi, Anna; Pezzotta, Alex; Carbone, Sabrina; Saponara, Simona; Gemma, Sandra; Altucci, Lucia; Benedetti, Rosaria; Lodola, Alessio; Mor, Marco; Bargagli, Elena; Butini, Stefania; Campiani, Giuseppe
Metalloenzyme Inhibitors against Zoonotic Infections: Focus on Leishmania and Schistosoma
2024-01-01 Rossi, Sara; Tudino, Valeria; Carullo, Gabriele; Butini, Stefania; Campiani, Giuseppe; Gemma, Sandra
Development of Epigenetic Modifiers with Therapeutic Potential in FMS-Related Tyrosine Kinase 3/Internal Tandem Duplication (FLT3/ITD) Acute Myeloid Leukemia and Other Blood Malignancies
2024-01-01 Carullo, Gabriele; Rossi, Sara; Giudice, Valentina; Pezzotta, Alex; Chianese, Ugo; Scala, Pasqualina; Carbone, Sabrina; Fontana, Anna; Panzeca, Giovanna; Pasquini, Silvia; Contri, Chiara; Gemma, Sandra; Ramunno, Anna; Saponara, Simona; Galvani, Francesca; Lodola, Alessio; Mor, Marco; Benedetti, Rosaria; Selleri, Carmine; Varani, Katia; Butini, Stefania; Altucci, Lucia; Vincenzi, Fabrizio; Pistocchi, Anna; Campiani, Giuseppe
Unlocking the potential of biostimulants in sustainable agriculture: Effect of wood distillate on the nutritional profiling of apples
2024-01-01 Fedeli, Riccardo; Dichiara, Maria; Carullo, Gabriele; Tudino, Valeria; Gemma, Sandra; Butini, Stefania; Campiani, Giuseppe; Loppi, Stefano
Synthetic derivatives of natural cinnamic acids as potential anti-colorectal cancer agents
2024-01-01 Falbo, F.; Gemma, S.; Koch, A.; Mazzotta, S.; Carullo, G.; Ramunno, A.; Butini, S.; Schneider-Stock, R.; Campiani, G.; Aiello, F.
A novel potent class I HDAC inhibitor reverses the STAT4/p66Shc apoptotic defect in B cells from chronic lymphocytic leukemia patients
2024-01-01 Rossi, Sara; Tatangelo, Vanessa; Dichiara, Maria; Butini, Stefania; Gemma, Sandra; Brogi, Simone; Pasquini, Silvia; Cappello, Martina; Vincenzi, Fabrizio; Varani, Katia; Lopresti, Ludovica; Malchiodi, Margherita; Carrara, Chiara; Gozzetti, Alessandro; Bocchia, Monica; Marotta, Giuseppe; Patrussi, Laura; Carullo, Gabriele; Baldari, Cosima T.; Campiani, Giuseppe
Targeting Relevant HDACs to Support the Survival of Cone Photoreceptors in Inherited Retinal Diseases: Identification of a Potent Pharmacological Tool with In Vitro and In Vivo Efficacy
2024-01-01 Carullo, Gabriele; Orsini, Noemi; Piano, Ilaria; Pozzetti, Luca; Papa, Alessandro; Fontana, Anna; Napoli, Debora; Corsi, Francesca; Marco, Beatrice Di; Galante, Alessia; Marotta, Ludovica; Panzeca, Giovanna; O'Brien, Justine; Sanchez, Alicia Gomez; Doherty, Harry; Mahon, Niamh; Clarke, Leni; Contri, Chiara; Pasquini, Silvia; Gorelli, Beatrice; Saponara, Simona; Valoti, Massimo; Vincenzi, Fabrizio; Varani, Katia; Ramunno, Anna; Brogi, Simone; Butini, Stefania; Gemma, Sandra; Kennedy, Breandán N.; Gargini, Claudia; Strettoi, Enrica; Campiani, Giuseppe
Development of Potent and Selective Monoacylglycerol Lipase Inhibitors. SARs, Structural Analysis, and Biological Characterization
2024-01-01 Butini, Stefania; Grether, Uwe; Jung, Kwang-Mook; Ligresti, Alessia; Allarà, Marco; Postmus, Annemarieke G. J.; Maramai, Samuele; Brogi, Simone; Papa, Alessandro; Carullo, Gabriele; Sykes, David; Veprintsev, Dmitry; Federico, Stefano; Grillo, Alessandro; Di Guglielmo, Bruno; Ramunno, Anna; Stevens, Anna Floor; Heer, Dominik; Lamponi, Stefania; Gemma, Sandra; Benz, Jörg; Di Marzo, Vincenzo; van der Stelt, Mario; Piomelli, Daniele; Campiani, Giuseppe
Biostimulants for Sustainable Food Production: Effects of Wood Distillate to Fortify Chickpea Flour for Development of Functional Bakery Products
2024-01-01 Fedeli, Riccardo; Spizzirri, Umile Gianfranco; Aquino, Giovanna; Basilicata, Manuela Giovanna; Pepe, Giacomo; Campiglia, Pietro; Celletti, Silvia; Tudino, Valeria; Dichiara, Maria; Gemma, Sandra; Butini, Stefania; Carullo, Gabriele; Aiello, Francesca; Restuccia, Donatella; Campiani, Giuseppe; Loppi, Stefano
Traceability and authentication in agri-food production: A multivariate approach to the characterization of the Italian food excellence elephant garlic (Allium ampeloprasum L.), a vasoactive nutraceutical
2024-01-01 Carullo, G.; Borghini, F.; Fusi, F.; Saponara, S.; Fontana, A.; Pozzetti, L.; Fedeli, R.; Panti, A.; Gorelli, B.; Aquino, G.; Basilicata, M. G.; Pepe, G.; Campiglia, P.; Biagiotti, S.; Gemma, S.; Butini, S.; Pianezze, S.; Loppi, S.; Cavaglioni, A.; Perini, M.; Campiani, G.
Nutritionally enriched tomatoes (Solanum lycopersicum L.) grown with wood distillate: chemical and biological characterization for quality assessment
2023-01-01 Fedeli, Riccardo; Marotta, Ludovica; Frattaruolo, Luca; Panti, Alice; Carullo, Gabriele; Fusi, Fabio; Saponara, Simona; Gemma, Sandra; Butini, Stefania; Cappello, Anna Rita; Vannini, Andrea; Campiani, Giuseppe; Loppi, Stefano
Pioneering first-in-class FAAH-HDAC inhibitors as potential multitarget neuroprotective agents
2023-01-01 Papa, Alessandro; Cursaro, Ilaria; Pozzetti, Luca; Contri, Chiara; Cappello, Martina; Pasquini, Silvia; Carullo, Gabriele; Ramunno, Anna; Gemma, Sandra; Varani, Katia; Butini, Stefania; Campiani, Giuseppe; Vincenzi, Fabrizio
Development of potent and selective FAAH inhibitors with improved drug-like properties as potential tools to treat neuroinflammatory conditions
2023-01-01 Papa, Alessandro; Pasquini, Silvia; Galvani, Francesca; Cammarota, Mariarosaria; Contri, Chiara; Carullo, Gabriele; Gemma, Sandra; Ramunno, Anna; Lamponi, Stefania; Gorelli, Beatrice; Saponara, Simona; Varani, Katia; Mor, Marco; Campiani, Giuseppe; Boscia, Francesca; Vincenzi, Fabrizio; Lodola, Alessio; Butini, Stefania
Development of quinazolinone derivatives as modulators of virulence factors of Pseudomonas aeruginosa Cystic Fibrosis strains
2023-01-01 Carullo, Gabriele; Di Bonaventura, Giovanni; Rossi, Sara; Lupetti, Veronica; Tudino, Valeria; Brogi, Simone; Butini, Stefania; Campiani, Giuseppe; Gemma, Sandra; Pompilio, Arianna
Total Synthesis of the Natural Chalcone Lophirone E, Synthetic Studies toward Benzofuran and Indole-Based Analogues, and Investigation of Anti-Leishmanial Activity
2022-01-01 Pozzetti, L.; Ibba, R.; Rossi, S.; Taglialatela-Scafati, O.; Taramelli, D.; Basilico, N.; D'Alessandro, S.; Parapini, S.; Butini, S.; Campiani, G.; Gemma, S.
In Silico Analysis of Peptide-Based Derivatives Containing Bifunctional Warheads Engaging Prime and Non-Prime Subsites to Covalent Binding SARS-CoV-2 Main Protease (Mpro)
2022-01-01 Brogi, Simone; Rossi, Sara; Ibba, Roberta; Butini, Stefania; Calderone, Vincenzo; Campiani, Giuseppe; Gemma, Sandra
Bronchoalveolar-Lavage-Derived Fibroblast Cell Line (B-LSDM7) as a new protocol for investigating the mechanisms of idiopathic pulmonary fibrosis
2022-01-01 Bergantini, Laura; D'Alessandro, Miriana; Gangi, Sara; Cavallaro, Dalila; Campiani, Giuseppe; Butini, Stefania; Landi, Claudia; Bini, Luca; Cameli, Paolo; Bargagli, Elena
| Titolo | Data di pubblicazione | Autore(i) | File | Abstract |
|---|---|---|---|---|
| Synthesis and biological investigation of peptidomimetic SARS‐CoV‐2 main protease inhibitors bearing quinoline‐based heterocycles at P3 | 1-gen-2025 | Rossi, Sara; Deidda, Graziano; Fiaschi, Lia; Ibba, Roberta; Pieroni, Mariachiara; Dichiara, Maria; Carullo, Gabriele; Butini, Stefania; Ramunno, Anna; Brogi, Simone; Lolicato, Marco; Arrigoni, Cristina; Cabella, Noemi; Bavagnoli, Laura; Maga, Giovanni; Varasi, Ilenia; Biba, Camilla; Vicenti, Ilaria; Gemma, Sandra; Crespan, Emmanuele; Zazzi, Maurizio; Campiani, Giuseppe | - | |
| Targeting N‐Methyl‐lysine Histone Demethylase KDM4 in Cancer: Natural Products Inhibitors as a Driving Force for Epigenetic Drug Discovery | 1-gen-2024 | Cursaro, Ilaria; Milioni, Leonardo; Eslami, Kourosh; Sirous, Hajar; Carullo, Gabriele; Gemma, Sandra; Butini, Stefania; Campiani, Giuseppe | - | |
| Enhancing Drug Discovery and Development through the Integration of Medicinal Chemistry, Chemical Biology, and Academia-Industry Partnerships: Insights from Roche’s Endocannabinoid System Projects | 1-gen-2024 | Aebi, Johannes; Atz, Kenneth; Ametamey, Simon M.; Benz, Jörg; Blaising, Julie; Butini, Stefania; Campiani, Giuseppe; Carreira, Erick M.; Collin, Ludovic; De Lago, Eva; Gazzi, Thais; Gertsch, Jürg; Gobbi, Luca; Guba, Wolfgang; Fernández-Ruiz, Javier; Fingerle, Jürgen; Haider, Ahmed; He, Yingfang; Heitman, Laura H.; Honer, Michael; Hunziker, Daniel; Kuhn, Bernd; Maccarrone, Mauro; Märki, Hans Peter; Martin, Rainer E.; Mohr, Peter; Mu, Linjing; Nazaré, Marc; Nippa, David F.; Oddi, Sergio; O'Hara, Fionn; Pacher, Pal; Romero, Julian; Röver, Stephan; Rufer, Arne C.; Schibli, Roger; Schneider, Gisbert; Stepan, Antonia F.; Sykes, David A.; Ullmer, Christoph; Van der Stelt, Mario; Veprintsev, Dmitry B.; Wittwer, Matthias B.; Grether, Uwe | - | |
| Spirotetrahydroisoquinoline-Based Histone Deacetylase Inhibitors as New Antifibrotic Agents: Biological Evaluation in Human Fibroblasts from Bronchoalveolar Lavages of Idiopathic Pulmonary Fibrosis Patients | 1-gen-2024 | Fontana, Anna; Bergantini, Laura; Carullo, Gabriele; Scalvini, Laura; D'Alessandro, Miriana; Papulino, Chiara; Cameli, Paolo; Gangi, Sara; Vincenzi, Fabrizio; Varani, Katia; Contri, Chiara; Pasquini, Silvia; Pistocchi, Anna; Pezzotta, Alex; Carbone, Sabrina; Saponara, Simona; Gemma, Sandra; Altucci, Lucia; Benedetti, Rosaria; Lodola, Alessio; Mor, Marco; Bargagli, Elena; Butini, Stefania; Campiani, Giuseppe | - | |
| Metalloenzyme Inhibitors against Zoonotic Infections: Focus on Leishmania and Schistosoma | 1-gen-2024 | Rossi, Sara; Tudino, Valeria; Carullo, Gabriele; Butini, Stefania; Campiani, Giuseppe; Gemma, Sandra | - | |
| Development of Epigenetic Modifiers with Therapeutic Potential in FMS-Related Tyrosine Kinase 3/Internal Tandem Duplication (FLT3/ITD) Acute Myeloid Leukemia and Other Blood Malignancies | 1-gen-2024 | Carullo, Gabriele; Rossi, Sara; Giudice, Valentina; Pezzotta, Alex; Chianese, Ugo; Scala, Pasqualina; Carbone, Sabrina; Fontana, Anna; Panzeca, Giovanna; Pasquini, Silvia; Contri, Chiara; Gemma, Sandra; Ramunno, Anna; Saponara, Simona; Galvani, Francesca; Lodola, Alessio; Mor, Marco; Benedetti, Rosaria; Selleri, Carmine; Varani, Katia; Butini, Stefania; Altucci, Lucia; Vincenzi, Fabrizio; Pistocchi, Anna; Campiani, Giuseppe | - | |
| Unlocking the potential of biostimulants in sustainable agriculture: Effect of wood distillate on the nutritional profiling of apples | 1-gen-2024 | Fedeli, Riccardo; Dichiara, Maria; Carullo, Gabriele; Tudino, Valeria; Gemma, Sandra; Butini, Stefania; Campiani, Giuseppe; Loppi, Stefano | - | |
| Synthetic derivatives of natural cinnamic acids as potential anti-colorectal cancer agents | 1-gen-2024 | Falbo, F.; Gemma, S.; Koch, A.; Mazzotta, S.; Carullo, G.; Ramunno, A.; Butini, S.; Schneider-Stock, R.; Campiani, G.; Aiello, F. | - | |
| A novel potent class I HDAC inhibitor reverses the STAT4/p66Shc apoptotic defect in B cells from chronic lymphocytic leukemia patients | 1-gen-2024 | Rossi, Sara; Tatangelo, Vanessa; Dichiara, Maria; Butini, Stefania; Gemma, Sandra; Brogi, Simone; Pasquini, Silvia; Cappello, Martina; Vincenzi, Fabrizio; Varani, Katia; Lopresti, Ludovica; Malchiodi, Margherita; Carrara, Chiara; Gozzetti, Alessandro; Bocchia, Monica; Marotta, Giuseppe; Patrussi, Laura; Carullo, Gabriele; Baldari, Cosima T.; Campiani, Giuseppe | - | |
| Targeting Relevant HDACs to Support the Survival of Cone Photoreceptors in Inherited Retinal Diseases: Identification of a Potent Pharmacological Tool with In Vitro and In Vivo Efficacy | 1-gen-2024 | Carullo, Gabriele; Orsini, Noemi; Piano, Ilaria; Pozzetti, Luca; Papa, Alessandro; Fontana, Anna; Napoli, Debora; Corsi, Francesca; Marco, Beatrice Di; Galante, Alessia; Marotta, Ludovica; Panzeca, Giovanna; O'Brien, Justine; Sanchez, Alicia Gomez; Doherty, Harry; Mahon, Niamh; Clarke, Leni; Contri, Chiara; Pasquini, Silvia; Gorelli, Beatrice; Saponara, Simona; Valoti, Massimo; Vincenzi, Fabrizio; Varani, Katia; Ramunno, Anna; Brogi, Simone; Butini, Stefania; Gemma, Sandra; Kennedy, Breandán N.; Gargini, Claudia; Strettoi, Enrica; Campiani, Giuseppe | - | |
| Development of Potent and Selective Monoacylglycerol Lipase Inhibitors. SARs, Structural Analysis, and Biological Characterization | 1-gen-2024 | Butini, Stefania; Grether, Uwe; Jung, Kwang-Mook; Ligresti, Alessia; Allarà, Marco; Postmus, Annemarieke G. J.; Maramai, Samuele; Brogi, Simone; Papa, Alessandro; Carullo, Gabriele; Sykes, David; Veprintsev, Dmitry; Federico, Stefano; Grillo, Alessandro; Di Guglielmo, Bruno; Ramunno, Anna; Stevens, Anna Floor; Heer, Dominik; Lamponi, Stefania; Gemma, Sandra; Benz, Jörg; Di Marzo, Vincenzo; van der Stelt, Mario; Piomelli, Daniele; Campiani, Giuseppe | - | |
| Biostimulants for Sustainable Food Production: Effects of Wood Distillate to Fortify Chickpea Flour for Development of Functional Bakery Products | 1-gen-2024 | Fedeli, Riccardo; Spizzirri, Umile Gianfranco; Aquino, Giovanna; Basilicata, Manuela Giovanna; Pepe, Giacomo; Campiglia, Pietro; Celletti, Silvia; Tudino, Valeria; Dichiara, Maria; Gemma, Sandra; Butini, Stefania; Carullo, Gabriele; Aiello, Francesca; Restuccia, Donatella; Campiani, Giuseppe; Loppi, Stefano | - | |
| Traceability and authentication in agri-food production: A multivariate approach to the characterization of the Italian food excellence elephant garlic (Allium ampeloprasum L.), a vasoactive nutraceutical | 1-gen-2024 | Carullo, G.; Borghini, F.; Fusi, F.; Saponara, S.; Fontana, A.; Pozzetti, L.; Fedeli, R.; Panti, A.; Gorelli, B.; Aquino, G.; Basilicata, M. G.; Pepe, G.; Campiglia, P.; Biagiotti, S.; Gemma, S.; Butini, S.; Pianezze, S.; Loppi, S.; Cavaglioni, A.; Perini, M.; Campiani, G. | - | |
| Nutritionally enriched tomatoes (Solanum lycopersicum L.) grown with wood distillate: chemical and biological characterization for quality assessment | 1-gen-2023 | Fedeli, Riccardo; Marotta, Ludovica; Frattaruolo, Luca; Panti, Alice; Carullo, Gabriele; Fusi, Fabio; Saponara, Simona; Gemma, Sandra; Butini, Stefania; Cappello, Anna Rita; Vannini, Andrea; Campiani, Giuseppe; Loppi, Stefano | - | |
| Pioneering first-in-class FAAH-HDAC inhibitors as potential multitarget neuroprotective agents | 1-gen-2023 | Papa, Alessandro; Cursaro, Ilaria; Pozzetti, Luca; Contri, Chiara; Cappello, Martina; Pasquini, Silvia; Carullo, Gabriele; Ramunno, Anna; Gemma, Sandra; Varani, Katia; Butini, Stefania; Campiani, Giuseppe; Vincenzi, Fabrizio | - | |
| Development of potent and selective FAAH inhibitors with improved drug-like properties as potential tools to treat neuroinflammatory conditions | 1-gen-2023 | Papa, Alessandro; Pasquini, Silvia; Galvani, Francesca; Cammarota, Mariarosaria; Contri, Chiara; Carullo, Gabriele; Gemma, Sandra; Ramunno, Anna; Lamponi, Stefania; Gorelli, Beatrice; Saponara, Simona; Varani, Katia; Mor, Marco; Campiani, Giuseppe; Boscia, Francesca; Vincenzi, Fabrizio; Lodola, Alessio; Butini, Stefania | - | |
| Development of quinazolinone derivatives as modulators of virulence factors of Pseudomonas aeruginosa Cystic Fibrosis strains | 1-gen-2023 | Carullo, Gabriele; Di Bonaventura, Giovanni; Rossi, Sara; Lupetti, Veronica; Tudino, Valeria; Brogi, Simone; Butini, Stefania; Campiani, Giuseppe; Gemma, Sandra; Pompilio, Arianna | - | |
| Total Synthesis of the Natural Chalcone Lophirone E, Synthetic Studies toward Benzofuran and Indole-Based Analogues, and Investigation of Anti-Leishmanial Activity | 1-gen-2022 | Pozzetti, L.; Ibba, R.; Rossi, S.; Taglialatela-Scafati, O.; Taramelli, D.; Basilico, N.; D'Alessandro, S.; Parapini, S.; Butini, S.; Campiani, G.; Gemma, S. | - | |
| In Silico Analysis of Peptide-Based Derivatives Containing Bifunctional Warheads Engaging Prime and Non-Prime Subsites to Covalent Binding SARS-CoV-2 Main Protease (Mpro) | 1-gen-2022 | Brogi, Simone; Rossi, Sara; Ibba, Roberta; Butini, Stefania; Calderone, Vincenzo; Campiani, Giuseppe; Gemma, Sandra | - | |
| Bronchoalveolar-Lavage-Derived Fibroblast Cell Line (B-LSDM7) as a new protocol for investigating the mechanisms of idiopathic pulmonary fibrosis | 1-gen-2022 | Bergantini, Laura; D'Alessandro, Miriana; Gangi, Sara; Cavallaro, Dalila; Campiani, Giuseppe; Butini, Stefania; Landi, Claudia; Bini, Luca; Cameli, Paolo; Bargagli, Elena | - |
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