Sfoglia per Autore
Synthetic derivatives of natural cinnamic acids as potential anti-colorectal cancer agents
2024-01-01 Falbo, F; Gemma, S; Koch, A; Mazzotta, S; Carullo, G; Ramunno, A; Butini, S; Schneider-Stock, R; Campiani, G; Aiello, F
Development of Potent and Selective Monoacylglycerol Lipase Inhibitors. SARs, Structural Analysis, and Biological Characterization
2024-01-01 Butini, Stefania; Grether, Uwe; Jung, Kwang-Mook; Ligresti, Alessia; Allarà, Marco; Postmus, Annemarieke G. J.; Maramai, Samuele; Brogi, Simone; Papa, Alessandro; Carullo, Gabriele; Sykes, David; Veprintsev, Dmitry; Federico, Stefano; Grillo, Alessandro; Di Guglielmo, Bruno; Ramunno, Anna; Stevens, Anna Floor; Heer, Dominik; Lamponi, Stefania; Gemma, Sandra; Benz, Jörg; Di Marzo, Vincenzo; van der Stelt, Mario; Piomelli, Daniele; Campiani, Giuseppe
Traceability and authentication in agri-food production: A multivariate approach to the characterization of the Italian food excellence elephant garlic (Allium ampeloprasum L.), a vasoactive nutraceutical
2024-01-01 Carullo, G.; Borghini, F.; Fusi, F.; Saponara, S.; Fontana, A.; Pozzetti, L.; Fedeli, R.; Panti, A.; Gorelli, B.; Aquino, G.; Basilicata, M. G.; Pepe, G.; Campiglia, P.; Biagiotti, S.; Gemma, S.; Butini, S.; Pianezze, S.; Loppi, S.; Cavaglioni, A.; Perini, M.; Campiani, G.
Development of Quinazolinone Derivatives as Modulators of Virulence Factors of Pseudomonas aeruginosa Cystic Fibrosis Strains
2023-01-01 Carullo, Gabriele; Di Bonaventura, Giovanni; Rossi, Sara; Lupetti, Veronica; Tudino, Valeria; Brogi, Simone; Butini, Stefania; Campiani, Giuseppe; Gemma, Sandra; Pompilio, Arianna
Nutritionally enriched tomatoes (Solanum lycopersicum L.) grown with wood distillate: chemical and biological characterization for quality assessment
2023-01-01 Fedeli, Riccardo; Marotta, Ludovica; Frattaruolo, Luca; Panti, Alice; Carullo, Gabriele; Fusi, Fabio; Saponara, Simona; Gemma, Sandra; Butini, Stefania; Cappello, Anna Rita; Vannini, Andrea; Campiani, Giuseppe; Loppi, Stefano
Pioneering first-in-class FAAH-HDAC inhibitors as potential multitarget neuroprotective agents
2023-01-01 Papa, Alessandro; Cursaro, Ilaria; Pozzetti, Luca; Contri, Chiara; Cappello, Martina; Pasquini, Silvia; Carullo, Gabriele; Ramunno, Anna; Gemma, Sandra; Varani, Katia; Butini, Stefania; Campiani, Giuseppe; Vincenzi, Fabrizio
The green chemistry of chalcones: Valuable sources of privileged core structures for drug discovery
2022-01-01 Marotta, Ludovica; Rossi, Sara; Ibba, Roberta; Brogi, Simone; Calderone, Vincenzo; Butini, Stefania; Campiani, Giuseppe; Gemma, Sandra
Total Synthesis of the Natural Chalcone Lophirone E, Synthetic Studies toward Benzofuran and Indole-Based Analogues, and Investigation of Anti-Leishmanial Activity
2022-01-01 Pozzetti, L.; Ibba, R.; Rossi, S.; Taglialatela-Scafati, O.; Taramelli, D.; Basilico, N.; D'Alessandro, S.; Parapini, S.; Butini, S.; Campiani, G.; Gemma, S.
A Therapeutic Perspective of HDAC8 in Different Diseases: An Overview of Selective Inhibitors
2022-01-01 Fontana, A.; Cursaro, I.; Carullo, G.; Gemma, S.; Butini, S.; Campiani, G.
Design and synthesis of multifunctional microtubule targeting agents endowed with dual pro-apoptotic and anti-autophagic efficacy
2022-01-01 Campiani, Giuseppe; Khan, Tuhina; Ulivieri, Cristina; Staiano, Leopoldo; Papulino, Chiara; Magnano, Stefania; Nathwani, Seema; Ramunno, Anna; Lucena-Agell, Daniel; Relitti, Nicola; Federico, Stefano; Pozzetti, Luca; Carullo, Gabriele; Casagni, Alice; Brogi, Simone; Vanni, Francesca; Galatello, Paola; Ghanim, Magda; Mccabe, Niamh; Lamponi, Stefania; Valoti, Massimo; Ibrahim, Ola; O'Sullivan, Jeffrey; Turkington, Richard; Kelly, Vincent P.; Vanwemmel, Ruben; Díaz, J. Fernando; Gemma, Sandra; Zisterer, Daniela; Altucci, Lucia; De Matteis, Antonella; Butini, Stefania; Benedetti, Rosaria
Synthesis of Unsymmetrical Squaramides as Allosteric GSK-3β Inhibitors Promoting β-Catenin-Mediated Transcription of TCF/LEF in Retinal Pigment Epithelial Cells
2022-01-01 Carullo, Gabriele; Bottoni, Laura; Pasquini, Silvia; Papa, Alessandro; Contri, Chiara; Brogi, Simone; Calderone, Vincenzo; Orlandini, Maurizio; Gemma, Sandra; Varani, Katia; Butini, Stefania; Galvagni, Federico; Vincenzi, Fabrizio; Campiani, Giuseppe
Azetidin-2-one-based small molecules as dual hHDAC6/HDAC8 inhibitors: Investigation of their mechanism of action and impact of dual inhibition profile on cell viability
2022-01-01 Federico, S.; Khan, T.; Fontana, A.; Brogi, S.; Benedetti, R.; Sarno, F.; Carullo, G.; Pezzotta, A.; Saraswati, A. P.; Passaro, E.; Pozzetti, L.; Papa, A.; Relitti, N.; Gemma, S.; Butini, S.; Pistocchi, A.; Ramunno, A.; Vincenzi, F.; Varani, K.; Tatangelo, V.; Patrussi, L.; Baldari, C. T.; Saponara, S.; Gorelli, B.; Lamponi, S.; Valoti, M.; Saccoccia, F.; Giannaccari, M.; Ruberti, G.; Herp, D.; Jung, M.; Altucci, L.; Campiani, G.
Covalent reversible inhibitors of cysteine proteases containing the nitrile warhead: recent advancement in the field of viral and parasitic diseases
2022-01-01 Brogi, S.; Ibba, R.; Rossi, S.; Butini, S.; Calderone, V.; Gemma, S.; Campiani, G.
Design and Synthesis of Oligopeptidic Parvulin Inhibitors
2022-01-01 Relitti, N.; Prasanth Saraswati, A.; Carullo, G.; Papa, A.; Monti, A.; Benedetti, R.; Passaro, E.; Brogi, S.; Calderone, V.; Butini, S.; Gemma, S.; Altucci, L.; Campiani, G.; Doti, N.
In Silico Analysis of Peptide-Based Derivatives Containing Bifunctional Warheads Engaging Prime and Non-Prime Subsites to Covalent Binding SARS-CoV-2 Main Protease (Mpro)
2022-01-01 Brogi, Simone; Rossi, Sara; Ibba, Roberta; Butini, Stefania; Calderone, Vincenzo; Campiani, Giuseppe; Gemma, Sandra
Development of potent and selective FAAH inhibitors with improved drug-like properties as potential tools to treat neuroinflammatory conditions
2022-01-01 Papa, Alessandro; Pasquini, Silvia; Galvani, Francesca; Cammarota, Mariarosaria; Contri, Chiara; Carullo, Gabriele; Gemma, Sandra; Ramunno, Anna; Lamponi, Stefania; Gorelli, Beatrice; Saponara, Simona; Varani, Katia; Mor, Marco; Campiani, Giuseppe; Boscia, Francesca; Vincenzi, Fabrizio; Lodola, Alessio; Butini, Stefania
Bronchoalveolar-Lavage-Derived Fibroblast Cell Line (B-LSDM7) as a New Protocol for Investigating the Mechanisms of Idiopathic Pulmonary Fibrosis
2022-01-01 Bergantini, Laura; D'Alessandro, Miriana; Gangi, Sara; Cavallaro, Dalila; Campiani, Giuseppe; Butini, Stefania; Landi, Claudia; Bini, Luca; Cameli, Paolo; Bargagli, Elena
Crystal structures of Schistosoma mansoni histone deacetylase 8 reveal a novel binding site for allosteric inhibitors
2022-01-01 Saccoccia, Fulvio; Pozzetti, Luca; Gimmelli, Roberto; Butini, Stefania; Guidi, Alessandra; Papoff, Giuliana; Giannaccari, Marialaura; Brogi, Simone; Scognamiglio, Viviana; Gemma, Sandra; Ruberti, Giovina; Campiani, Giuseppe
Optimization of Potent and Specific Trypanothione Reductase Inhibitors: A Structure-Based Drug Discovery Approach
2022-01-01 Battista, Theo; Federico, Stefano; Brogi, Simone; Pozzetti, Luca; Khan, Tuhina; Butini, Stefania; Ramunno, Anna; Fiorentino, Eleonora; Orsini, Stefania; Di Muccio, Trentina; Fiorillo, Annarita; Exertier, Cécile; Di Risola, Daniel; Colotti, Gianni; Gemma, Sandra; Ilari, Andrea; Campiani, Giuseppe
Extra Virgin Olive Oil Extracts of Indigenous Southern Tuscany Cultivar Act as Anti-Inflammatory and Vasorelaxant Nutraceuticals
2022-01-01 Pozzetti, L.; Ferrara, F.; Marotta, L.; Gemma, S.; Butini, S.; Benedusi, M.; Fusi, F.; Ahmed, A.; Pomponi, S.; Ferrari, S.; Perini, M.; Ramunno, A.; Pepe, G.; Campiglia, P.; Valacchi, G.; Carullo, G.; Campiani, G.
Titolo | Data di pubblicazione | Autore(i) | File | Abstract |
---|---|---|---|---|
Synthetic derivatives of natural cinnamic acids as potential anti-colorectal cancer agents | 1-gen-2024 | Falbo, F; Gemma, S; Koch, A; Mazzotta, S; Carullo, G; Ramunno, A; Butini, S; Schneider-Stock, R; Campiani, G; Aiello, F | - | |
Development of Potent and Selective Monoacylglycerol Lipase Inhibitors. SARs, Structural Analysis, and Biological Characterization | 1-gen-2024 | Butini, Stefania; Grether, Uwe; Jung, Kwang-Mook; Ligresti, Alessia; Allarà, Marco; Postmus, Annemarieke G. J.; Maramai, Samuele; Brogi, Simone; Papa, Alessandro; Carullo, Gabriele; Sykes, David; Veprintsev, Dmitry; Federico, Stefano; Grillo, Alessandro; Di Guglielmo, Bruno; Ramunno, Anna; Stevens, Anna Floor; Heer, Dominik; Lamponi, Stefania; Gemma, Sandra; Benz, Jörg; Di Marzo, Vincenzo; van der Stelt, Mario; Piomelli, Daniele; Campiani, Giuseppe | - | |
Traceability and authentication in agri-food production: A multivariate approach to the characterization of the Italian food excellence elephant garlic (Allium ampeloprasum L.), a vasoactive nutraceutical | 1-gen-2024 | Carullo, G.; Borghini, F.; Fusi, F.; Saponara, S.; Fontana, A.; Pozzetti, L.; Fedeli, R.; Panti, A.; Gorelli, B.; Aquino, G.; Basilicata, M. G.; Pepe, G.; Campiglia, P.; Biagiotti, S.; Gemma, S.; Butini, S.; Pianezze, S.; Loppi, S.; Cavaglioni, A.; Perini, M.; Campiani, G. | - | |
Development of Quinazolinone Derivatives as Modulators of Virulence Factors of Pseudomonas aeruginosa Cystic Fibrosis Strains | 1-gen-2023 | Carullo, Gabriele; Di Bonaventura, Giovanni; Rossi, Sara; Lupetti, Veronica; Tudino, Valeria; Brogi, Simone; Butini, Stefania; Campiani, Giuseppe; Gemma, Sandra; Pompilio, Arianna | - | |
Nutritionally enriched tomatoes (Solanum lycopersicum L.) grown with wood distillate: chemical and biological characterization for quality assessment | 1-gen-2023 | Fedeli, Riccardo; Marotta, Ludovica; Frattaruolo, Luca; Panti, Alice; Carullo, Gabriele; Fusi, Fabio; Saponara, Simona; Gemma, Sandra; Butini, Stefania; Cappello, Anna Rita; Vannini, Andrea; Campiani, Giuseppe; Loppi, Stefano | - | |
Pioneering first-in-class FAAH-HDAC inhibitors as potential multitarget neuroprotective agents | 1-gen-2023 | Papa, Alessandro; Cursaro, Ilaria; Pozzetti, Luca; Contri, Chiara; Cappello, Martina; Pasquini, Silvia; Carullo, Gabriele; Ramunno, Anna; Gemma, Sandra; Varani, Katia; Butini, Stefania; Campiani, Giuseppe; Vincenzi, Fabrizio | - | |
The green chemistry of chalcones: Valuable sources of privileged core structures for drug discovery | 1-gen-2022 | Marotta, Ludovica; Rossi, Sara; Ibba, Roberta; Brogi, Simone; Calderone, Vincenzo; Butini, Stefania; Campiani, Giuseppe; Gemma, Sandra | - | |
Total Synthesis of the Natural Chalcone Lophirone E, Synthetic Studies toward Benzofuran and Indole-Based Analogues, and Investigation of Anti-Leishmanial Activity | 1-gen-2022 | Pozzetti, L.; Ibba, R.; Rossi, S.; Taglialatela-Scafati, O.; Taramelli, D.; Basilico, N.; D'Alessandro, S.; Parapini, S.; Butini, S.; Campiani, G.; Gemma, S. | - | |
A Therapeutic Perspective of HDAC8 in Different Diseases: An Overview of Selective Inhibitors | 1-gen-2022 | Fontana, A.; Cursaro, I.; Carullo, G.; Gemma, S.; Butini, S.; Campiani, G. | - | |
Design and synthesis of multifunctional microtubule targeting agents endowed with dual pro-apoptotic and anti-autophagic efficacy | 1-gen-2022 | Campiani, Giuseppe; Khan, Tuhina; Ulivieri, Cristina; Staiano, Leopoldo; Papulino, Chiara; Magnano, Stefania; Nathwani, Seema; Ramunno, Anna; Lucena-Agell, Daniel; Relitti, Nicola; Federico, Stefano; Pozzetti, Luca; Carullo, Gabriele; Casagni, Alice; Brogi, Simone; Vanni, Francesca; Galatello, Paola; Ghanim, Magda; Mccabe, Niamh; Lamponi, Stefania; Valoti, Massimo; Ibrahim, Ola; O'Sullivan, Jeffrey; Turkington, Richard; Kelly, Vincent P.; Vanwemmel, Ruben; Díaz, J. Fernando; Gemma, Sandra; Zisterer, Daniela; Altucci, Lucia; De Matteis, Antonella; Butini, Stefania; Benedetti, Rosaria | - | |
Synthesis of Unsymmetrical Squaramides as Allosteric GSK-3β Inhibitors Promoting β-Catenin-Mediated Transcription of TCF/LEF in Retinal Pigment Epithelial Cells | 1-gen-2022 | Carullo, Gabriele; Bottoni, Laura; Pasquini, Silvia; Papa, Alessandro; Contri, Chiara; Brogi, Simone; Calderone, Vincenzo; Orlandini, Maurizio; Gemma, Sandra; Varani, Katia; Butini, Stefania; Galvagni, Federico; Vincenzi, Fabrizio; Campiani, Giuseppe | - | |
Azetidin-2-one-based small molecules as dual hHDAC6/HDAC8 inhibitors: Investigation of their mechanism of action and impact of dual inhibition profile on cell viability | 1-gen-2022 | Federico, S.; Khan, T.; Fontana, A.; Brogi, S.; Benedetti, R.; Sarno, F.; Carullo, G.; Pezzotta, A.; Saraswati, A. P.; Passaro, E.; Pozzetti, L.; Papa, A.; Relitti, N.; Gemma, S.; Butini, S.; Pistocchi, A.; Ramunno, A.; Vincenzi, F.; Varani, K.; Tatangelo, V.; Patrussi, L.; Baldari, C. T.; Saponara, S.; Gorelli, B.; Lamponi, S.; Valoti, M.; Saccoccia, F.; Giannaccari, M.; Ruberti, G.; Herp, D.; Jung, M.; Altucci, L.; Campiani, G. | - | |
Covalent reversible inhibitors of cysteine proteases containing the nitrile warhead: recent advancement in the field of viral and parasitic diseases | 1-gen-2022 | Brogi, S.; Ibba, R.; Rossi, S.; Butini, S.; Calderone, V.; Gemma, S.; Campiani, G. | - | |
Design and Synthesis of Oligopeptidic Parvulin Inhibitors | 1-gen-2022 | Relitti, N.; Prasanth Saraswati, A.; Carullo, G.; Papa, A.; Monti, A.; Benedetti, R.; Passaro, E.; Brogi, S.; Calderone, V.; Butini, S.; Gemma, S.; Altucci, L.; Campiani, G.; Doti, N. | - | |
In Silico Analysis of Peptide-Based Derivatives Containing Bifunctional Warheads Engaging Prime and Non-Prime Subsites to Covalent Binding SARS-CoV-2 Main Protease (Mpro) | 1-gen-2022 | Brogi, Simone; Rossi, Sara; Ibba, Roberta; Butini, Stefania; Calderone, Vincenzo; Campiani, Giuseppe; Gemma, Sandra | - | |
Development of potent and selective FAAH inhibitors with improved drug-like properties as potential tools to treat neuroinflammatory conditions | 1-gen-2022 | Papa, Alessandro; Pasquini, Silvia; Galvani, Francesca; Cammarota, Mariarosaria; Contri, Chiara; Carullo, Gabriele; Gemma, Sandra; Ramunno, Anna; Lamponi, Stefania; Gorelli, Beatrice; Saponara, Simona; Varani, Katia; Mor, Marco; Campiani, Giuseppe; Boscia, Francesca; Vincenzi, Fabrizio; Lodola, Alessio; Butini, Stefania | - | |
Bronchoalveolar-Lavage-Derived Fibroblast Cell Line (B-LSDM7) as a New Protocol for Investigating the Mechanisms of Idiopathic Pulmonary Fibrosis | 1-gen-2022 | Bergantini, Laura; D'Alessandro, Miriana; Gangi, Sara; Cavallaro, Dalila; Campiani, Giuseppe; Butini, Stefania; Landi, Claudia; Bini, Luca; Cameli, Paolo; Bargagli, Elena | - | |
Crystal structures of Schistosoma mansoni histone deacetylase 8 reveal a novel binding site for allosteric inhibitors | 1-gen-2022 | Saccoccia, Fulvio; Pozzetti, Luca; Gimmelli, Roberto; Butini, Stefania; Guidi, Alessandra; Papoff, Giuliana; Giannaccari, Marialaura; Brogi, Simone; Scognamiglio, Viviana; Gemma, Sandra; Ruberti, Giovina; Campiani, Giuseppe | - | |
Optimization of Potent and Specific Trypanothione Reductase Inhibitors: A Structure-Based Drug Discovery Approach | 1-gen-2022 | Battista, Theo; Federico, Stefano; Brogi, Simone; Pozzetti, Luca; Khan, Tuhina; Butini, Stefania; Ramunno, Anna; Fiorentino, Eleonora; Orsini, Stefania; Di Muccio, Trentina; Fiorillo, Annarita; Exertier, Cécile; Di Risola, Daniel; Colotti, Gianni; Gemma, Sandra; Ilari, Andrea; Campiani, Giuseppe | - | |
Extra Virgin Olive Oil Extracts of Indigenous Southern Tuscany Cultivar Act as Anti-Inflammatory and Vasorelaxant Nutraceuticals | 1-gen-2022 | Pozzetti, L.; Ferrara, F.; Marotta, L.; Gemma, S.; Butini, S.; Benedusi, M.; Fusi, F.; Ahmed, A.; Pomponi, S.; Ferrari, S.; Perini, M.; Ramunno, A.; Pepe, G.; Campiglia, P.; Valacchi, G.; Carullo, G.; Campiani, G. | - |
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