Sfoglia per Autore
Peptaibol Analogs Show Potent Antibacterial Activity against Multidrug Resistant Opportunistic Pathogens
2023-01-01 Dalla Torre, Chiara; Sannio, Filomena; Battistella, Mattia; Docquier, Jean-Denis; De Zotti, Marta
Benzenesulfonamide derivatives as Vibrio cholerae carbonic anhydrases inhibitors: a computational-aided insight in the structural rigidity-activity relationships
2023-01-01 Fantacuzzi, Marialuigia; D'Agostino, Ilaria; Carradori, Simone; Liguori, Francesco; Carta, Fabrizio; Agamennone, Mariangela; Angeli, Andrea; Sannio, Filomena; Docquier, Jean-Denis; Capasso, Clemente; Supuran, Claudiu T
Zidovudine-β-Lactam Pronucleoside Strategy for Selective Delivery into Gram-Negative Bacteria Triggered by β-Lactamases
2023-01-01 Rosales-Hurtado, Miyanou; Sannio, Filomena; Lari, Lindita; Verdirosa, Federica; Feller, Georges; Carretero, Elodie; Vo-Hoang, Yen; Licznar-Fajardo, Patricia; Docquier, Jean-Denis; Gavara, Laurent
Nucleoside Derivatives of 2,6-Diaminopurine Antivirals: Base-Modified Nucleosides with Broad-Spectrum Antimicrobial Properties
2023-01-01 Grazia Martina, Maria; Giammarino, Federica; Vicenti, Ilaria; Groaz, Elisabetta; Rozenski, Jef; Incerti, Matteo; Sannio, Filomena; Docquier, Jean Denis; Zazzi, Maurizio; Radi, Marco
Lunaemycins, New Cyclic Hexapeptide Antibiotics from the Cave Moonmilk-Dweller Streptomyces lunaelactis MM109T
2023-01-01 Martinet, Loïc; Naômé, Aymeric; Rezende, Lucas C D; Tellatin, Déborah; Pignon, Bernard; Docquier, Jean-Denis; Sannio, Filomena; Baiwir, Dominique; Mazzucchelli, Gabriel; Frédérich, Michel; Rigali, Sébastien
Chemical Optimization of Selective Pseudomonas aeruginosa LasB Elastase Inhibitors and Their Impact on LasB-Mediated Activation of IL-1β in Cellular and Animal Infection Models
2023-01-01 Everett, Martin J; Davies, David T; Leiris, Simon; Sprynski, Nicolas; Llanos, Agustina; Castandet, Jérôme M; Lozano, Clarisse; Larock, Christopher N; Larock, Doris L; Corsica, Giuseppina; Docquier, Jean-Denis; Pallin, Thomas D; Cridland, Andrew; Blench, Toby; Zalacain, Magdalena; Lemonnier, Marc
Discovery and Optimization of a Novel Macrocyclic Amidinourea Series Active as Acidic Mammalian Chitinase Inhibitors
2023-01-01 Balestri, Lorenzo Jacopo Ilic; Trivisani, Claudia Immacolata; Orofino, Francesco; Fiorucci, Diego; Truglio, Giuseppina Ivana; D'Agostino, Ilaria; Poggialini, Federica; Botta, Lorenzo; Docquier, Jean-Denis; Dreassi, Elena
Discovering NDM-1 inhibitors using molecular substructure embeddings representations
2023-01-01 Papastergiou, Thomas; Azé, Jérôme; Bringay, Sandra; Louet, Maxime; Poncelet, Pascal; Rosales-Hurtado, Miyanou; Vo-Hoang, Yen; Licznar-Fajardo, Patricia; Docquier, Jean-Denis; Gavara, Laurent
Towards Innovative Antibacterial Correctors for Cystic Fibrosis Targeting the Lung Microbiome with a Multifunctional Effect
2022-01-01 Martina, Maria Grazia; Sannio, Filomena; Crespan, Emmanuele; Pavone, Marialaura; Simoncini, Alice; Barbieri, Francesca; Perini, Cecilia; Pesce, Emanuela; Maga, Giovanni; Pedemonte, Nicoletta; Docquier, Jean-Denis; Radi, Marco
A fragment-based drug discovery strategy applied to the identification of NDM-1 β-lactamase inhibitors
2022-01-01 Caburet, Jérémy; Boucherle, Benjamin; Bourdillon, Sofiane; Simoncelli, Giorgia; Verdirosa, Federica; Docquier, Jean-Denis; Moreau, Yohann; Krimm, Isabelle; Crouzy, Serge; Peuchmaur, Marine
A Clinical Study Provides the First Direct Evidence That Interindividual Variations in Fecal β-Lactamase Activity Affect the Gut Mycobiota Dynamics in Response to β-Lactam Antibiotics
2022-01-01 Delavy, Margot; Burdet, Charles; Sertour, Natacha; Devente, Savannah; Docquier, Jean-Denis; Grall, Nathalie; Volant, Stevenn; Ghozlane, Amine; Duval, Xavier; Mentré, France; D'Enfert, Christophe; Bougnoux, Marie-Elisabeth
Antibacterial alkylguanidino ureas: Molecular simplification approach, searching for membrane-based MoA
2022-01-01 D'Agostino, I.; Ardino, C.; Poli, G.; Sannio, F.; Lucidi, M.; Poggialini, F.; Visaggio, D.; Rango, E.; Filippi, S.; Petricci, E.; Visca, P.; Botta, L.; Docquier, J. -D.; Dreassi, E.
Editorial: Structural and Biochemical Aspects of the Interaction of β-Lactamases With State-of-the-Art Inhibitors
2022-01-01 Papp-Wallace, Krisztina M; Docquier, Jean-Denis; Kerff, Frederic; Power, Pablo
Optimization of 1,2,4-Triazole-3-thiones toward Broad-Spectrum Metallo-β-lactamase Inhibitors Showing Potent Synergistic Activity on VIM- and NDM-1-Producing Clinical Isolates
2022-01-01 Legru, Alice; Verdirosa, Federica; Vo-Hoang, Yen; Tassone, Giusy; Vascon, Filippo; Thomas, Caitlyn A; Sannio, Filomena; Corsica, Giuseppina; Benvenuti, Manuela; Feller, Georges; Coulon, Rémi; Marcoccia, Francesca; Devente, Savannah Rowane; Bouajila, Ezeddine; Piveteau, Catherine; Leroux, Florence; Deprez-Poulain, Rebecca; Deprez, Benoît; Licznar-Fajardo, Patricia; Crowder, Michael W; Cendron, Laura; Pozzi, Cecilia; Mangani, Stefano; Docquier, Jean-Denis; Hernandez, Jean-François; Gavara, Laurent
1,2,4-Triazole-3-thione analogues with an arylakyl group at position 4 as metallo-β-lactamase inhibitors
2022-01-01 Gavara, Laurent; Verdirosa, Federica; Sevaille, Laurent; Legru, Alice; Corsica, Giuseppina; Nauton, Lionel; Sandra Mercuri, Paola; Sannio, Filomena; De Luca, Filomena; Hadjadj, Margot; Cerboni, Giulia; Vo Hoang, Yen; Licznar-Fajardo, Patricia; Galleni, Moreno; Docquier, Jean-Denis; Hernandez, Jean-François
1,2,4-Triazole-3-Thione Analogues with a 2-Ethylbenzoic Acid at Position 4 as VIM-type Metallo-β-Lactamase Inhibitors
2022-01-01 Verdirosa, Federica; Gavara, Laurent; Sevaille, Laurent; Tassone, Giusy; Corsica, Giuseppina; Legru, Alice; Feller, Georges; Chelini, Giulia; Mercuri, Paola Sandra; Tanfoni, Silvia; Sannio, Filomena; Benvenuti, Manuela; Cerboni, Giulia; De Luca, Filomena; Bouajila, Ezeddine; Vo Hoang, Yen; Licznar-Fajardo, Patricia; Galleni, Moreno; Pozzi, Cecilia; Mangani, Stefano; Docquier, Jean-Denis; Hernandez, Jean-François
The impact of counterions in biological activity: case study of antibacterial alkylguanidino ureas
2022-01-01 Ardino, C.; Sannio, F.; Pasero, C.; Botta, L.; Dreassi, E.; Docquier, J. D.; D'Agostino, I.
Optimization of Pyrazole Compounds as Antibiotic Adjuvants Active against Colistin- and Carbapenem-Resistant Acinetobacter baumannii
2022-01-01 Sannio, Filomena; Brizzi, Antonella; Del Prete, Rosita; Avigliano, Marialuce; Simone, Tiziana; Pagli, Carlotta; Ferraro, Teresa; De Luca, Filomena; Paolino, Marco; Corelli, Federico; Mugnaini, Claudia; Docquier, Jean-Denis
4-Alkyl-1,2,4-triazole-3-thione analogues as metallo-β-lactamase inhibitors
2021-01-01 Gavara, Laurent; Legru, Alice; Verdirosa, Federica; Sevaille, Laurent; Nauton, Lionel; Corsica, Giuseppina; Mercuri, Paola Sandra; Sannio, Filomena; Feller, Georges; Coulon, Rémi; De Luca, Filomena; Cerboni, Giulia; Tanfoni, Silvia; Chelini, Giulia; Galleni, Moreno; Docquier, Jean-Denis; Hernandez, Jean-François
1,2,4-Triazole-3-thione compounds with a 4-ethyl alkyl/aryl sulfide substituent are broad-spectrum metallo-β-lactamase inhibitors with re-sensitization activity
2021-01-01 Legru, Alice; Verdirosa, Federica; Hernandez, Jean-François; Tassone, Giusy; Sannio, Filomena; Benvenuti, Manuela; Conde, Pierre-Alexis; Bossis, Guillaume; Thomas, Caitlyn A; Crowder, Michael W; Dillenberger, Melissa; Becker, Katja; Pozzi, Cecilia; Mangani, Stefano; Docquier, Jean-Denis; Gavara, Laurent
Titolo | Data di pubblicazione | Autore(i) | File | Abstract |
---|---|---|---|---|
Peptaibol Analogs Show Potent Antibacterial Activity against Multidrug Resistant Opportunistic Pathogens | 1-gen-2023 | Dalla Torre, Chiara; Sannio, Filomena; Battistella, Mattia; Docquier, Jean-Denis; De Zotti, Marta | - | |
Benzenesulfonamide derivatives as Vibrio cholerae carbonic anhydrases inhibitors: a computational-aided insight in the structural rigidity-activity relationships | 1-gen-2023 | Fantacuzzi, Marialuigia; D'Agostino, Ilaria; Carradori, Simone; Liguori, Francesco; Carta, Fabrizio; Agamennone, Mariangela; Angeli, Andrea; Sannio, Filomena; Docquier, Jean-Denis; Capasso, Clemente; Supuran, Claudiu T | - | |
Zidovudine-β-Lactam Pronucleoside Strategy for Selective Delivery into Gram-Negative Bacteria Triggered by β-Lactamases | 1-gen-2023 | Rosales-Hurtado, Miyanou; Sannio, Filomena; Lari, Lindita; Verdirosa, Federica; Feller, Georges; Carretero, Elodie; Vo-Hoang, Yen; Licznar-Fajardo, Patricia; Docquier, Jean-Denis; Gavara, Laurent | - | |
Nucleoside Derivatives of 2,6-Diaminopurine Antivirals: Base-Modified Nucleosides with Broad-Spectrum Antimicrobial Properties | 1-gen-2023 | Grazia Martina, Maria; Giammarino, Federica; Vicenti, Ilaria; Groaz, Elisabetta; Rozenski, Jef; Incerti, Matteo; Sannio, Filomena; Docquier, Jean Denis; Zazzi, Maurizio; Radi, Marco | - | |
Lunaemycins, New Cyclic Hexapeptide Antibiotics from the Cave Moonmilk-Dweller Streptomyces lunaelactis MM109T | 1-gen-2023 | Martinet, Loïc; Naômé, Aymeric; Rezende, Lucas C D; Tellatin, Déborah; Pignon, Bernard; Docquier, Jean-Denis; Sannio, Filomena; Baiwir, Dominique; Mazzucchelli, Gabriel; Frédérich, Michel; Rigali, Sébastien | - | |
Chemical Optimization of Selective Pseudomonas aeruginosa LasB Elastase Inhibitors and Their Impact on LasB-Mediated Activation of IL-1β in Cellular and Animal Infection Models | 1-gen-2023 | Everett, Martin J; Davies, David T; Leiris, Simon; Sprynski, Nicolas; Llanos, Agustina; Castandet, Jérôme M; Lozano, Clarisse; Larock, Christopher N; Larock, Doris L; Corsica, Giuseppina; Docquier, Jean-Denis; Pallin, Thomas D; Cridland, Andrew; Blench, Toby; Zalacain, Magdalena; Lemonnier, Marc | - | |
Discovery and Optimization of a Novel Macrocyclic Amidinourea Series Active as Acidic Mammalian Chitinase Inhibitors | 1-gen-2023 | Balestri, Lorenzo Jacopo Ilic; Trivisani, Claudia Immacolata; Orofino, Francesco; Fiorucci, Diego; Truglio, Giuseppina Ivana; D'Agostino, Ilaria; Poggialini, Federica; Botta, Lorenzo; Docquier, Jean-Denis; Dreassi, Elena | - | |
Discovering NDM-1 inhibitors using molecular substructure embeddings representations | 1-gen-2023 | Papastergiou, Thomas; Azé, Jérôme; Bringay, Sandra; Louet, Maxime; Poncelet, Pascal; Rosales-Hurtado, Miyanou; Vo-Hoang, Yen; Licznar-Fajardo, Patricia; Docquier, Jean-Denis; Gavara, Laurent | - | |
Towards Innovative Antibacterial Correctors for Cystic Fibrosis Targeting the Lung Microbiome with a Multifunctional Effect | 1-gen-2022 | Martina, Maria Grazia; Sannio, Filomena; Crespan, Emmanuele; Pavone, Marialaura; Simoncini, Alice; Barbieri, Francesca; Perini, Cecilia; Pesce, Emanuela; Maga, Giovanni; Pedemonte, Nicoletta; Docquier, Jean-Denis; Radi, Marco | - | |
A fragment-based drug discovery strategy applied to the identification of NDM-1 β-lactamase inhibitors | 1-gen-2022 | Caburet, Jérémy; Boucherle, Benjamin; Bourdillon, Sofiane; Simoncelli, Giorgia; Verdirosa, Federica; Docquier, Jean-Denis; Moreau, Yohann; Krimm, Isabelle; Crouzy, Serge; Peuchmaur, Marine | - | |
A Clinical Study Provides the First Direct Evidence That Interindividual Variations in Fecal β-Lactamase Activity Affect the Gut Mycobiota Dynamics in Response to β-Lactam Antibiotics | 1-gen-2022 | Delavy, Margot; Burdet, Charles; Sertour, Natacha; Devente, Savannah; Docquier, Jean-Denis; Grall, Nathalie; Volant, Stevenn; Ghozlane, Amine; Duval, Xavier; Mentré, France; D'Enfert, Christophe; Bougnoux, Marie-Elisabeth | - | |
Antibacterial alkylguanidino ureas: Molecular simplification approach, searching for membrane-based MoA | 1-gen-2022 | D'Agostino, I.; Ardino, C.; Poli, G.; Sannio, F.; Lucidi, M.; Poggialini, F.; Visaggio, D.; Rango, E.; Filippi, S.; Petricci, E.; Visca, P.; Botta, L.; Docquier, J. -D.; Dreassi, E. | - | |
Editorial: Structural and Biochemical Aspects of the Interaction of β-Lactamases With State-of-the-Art Inhibitors | 1-gen-2022 | Papp-Wallace, Krisztina M; Docquier, Jean-Denis; Kerff, Frederic; Power, Pablo | - | |
Optimization of 1,2,4-Triazole-3-thiones toward Broad-Spectrum Metallo-β-lactamase Inhibitors Showing Potent Synergistic Activity on VIM- and NDM-1-Producing Clinical Isolates | 1-gen-2022 | Legru, Alice; Verdirosa, Federica; Vo-Hoang, Yen; Tassone, Giusy; Vascon, Filippo; Thomas, Caitlyn A; Sannio, Filomena; Corsica, Giuseppina; Benvenuti, Manuela; Feller, Georges; Coulon, Rémi; Marcoccia, Francesca; Devente, Savannah Rowane; Bouajila, Ezeddine; Piveteau, Catherine; Leroux, Florence; Deprez-Poulain, Rebecca; Deprez, Benoît; Licznar-Fajardo, Patricia; Crowder, Michael W; Cendron, Laura; Pozzi, Cecilia; Mangani, Stefano; Docquier, Jean-Denis; Hernandez, Jean-François; Gavara, Laurent | - | |
1,2,4-Triazole-3-thione analogues with an arylakyl group at position 4 as metallo-β-lactamase inhibitors | 1-gen-2022 | Gavara, Laurent; Verdirosa, Federica; Sevaille, Laurent; Legru, Alice; Corsica, Giuseppina; Nauton, Lionel; Sandra Mercuri, Paola; Sannio, Filomena; De Luca, Filomena; Hadjadj, Margot; Cerboni, Giulia; Vo Hoang, Yen; Licznar-Fajardo, Patricia; Galleni, Moreno; Docquier, Jean-Denis; Hernandez, Jean-François | - | |
1,2,4-Triazole-3-Thione Analogues with a 2-Ethylbenzoic Acid at Position 4 as VIM-type Metallo-β-Lactamase Inhibitors | 1-gen-2022 | Verdirosa, Federica; Gavara, Laurent; Sevaille, Laurent; Tassone, Giusy; Corsica, Giuseppina; Legru, Alice; Feller, Georges; Chelini, Giulia; Mercuri, Paola Sandra; Tanfoni, Silvia; Sannio, Filomena; Benvenuti, Manuela; Cerboni, Giulia; De Luca, Filomena; Bouajila, Ezeddine; Vo Hoang, Yen; Licznar-Fajardo, Patricia; Galleni, Moreno; Pozzi, Cecilia; Mangani, Stefano; Docquier, Jean-Denis; Hernandez, Jean-François | - | |
The impact of counterions in biological activity: case study of antibacterial alkylguanidino ureas | 1-gen-2022 | Ardino, C.; Sannio, F.; Pasero, C.; Botta, L.; Dreassi, E.; Docquier, J. D.; D'Agostino, I. | - | |
Optimization of Pyrazole Compounds as Antibiotic Adjuvants Active against Colistin- and Carbapenem-Resistant Acinetobacter baumannii | 1-gen-2022 | Sannio, Filomena; Brizzi, Antonella; Del Prete, Rosita; Avigliano, Marialuce; Simone, Tiziana; Pagli, Carlotta; Ferraro, Teresa; De Luca, Filomena; Paolino, Marco; Corelli, Federico; Mugnaini, Claudia; Docquier, Jean-Denis | - | |
4-Alkyl-1,2,4-triazole-3-thione analogues as metallo-β-lactamase inhibitors | 1-gen-2021 | Gavara, Laurent; Legru, Alice; Verdirosa, Federica; Sevaille, Laurent; Nauton, Lionel; Corsica, Giuseppina; Mercuri, Paola Sandra; Sannio, Filomena; Feller, Georges; Coulon, Rémi; De Luca, Filomena; Cerboni, Giulia; Tanfoni, Silvia; Chelini, Giulia; Galleni, Moreno; Docquier, Jean-Denis; Hernandez, Jean-François | - | |
1,2,4-Triazole-3-thione compounds with a 4-ethyl alkyl/aryl sulfide substituent are broad-spectrum metallo-β-lactamase inhibitors with re-sensitization activity | 1-gen-2021 | Legru, Alice; Verdirosa, Federica; Hernandez, Jean-François; Tassone, Giusy; Sannio, Filomena; Benvenuti, Manuela; Conde, Pierre-Alexis; Bossis, Guillaume; Thomas, Caitlyn A; Crowder, Michael W; Dillenberger, Melissa; Becker, Katja; Pozzi, Cecilia; Mangani, Stefano; Docquier, Jean-Denis; Gavara, Laurent | - |
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