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Mostrati risultati da 1 a 20 di 194
Titolo Data di pubblicazione Autore(i) File Abstract
In Silico-Guided Rational Drug Design and Synthesis of Novel 4-(Thiophen-2-yl)butanamides as Potent and Selective TRPV1 Agonists 1-gen-2023 Romeo, Isabella; Brizzi, Antonella; Pessina, Federica; Ambrosio, Francesca Alessandra; Aiello, Francesca; Belardo, Carmela; Carullo, Gabriele; Costa, Giosuè; De Petrocellis, Luciano; Frosini, Maria; Luongo, Livio; Maramai, Samuele; Paolino, Marco; Moriello, Aniello Schiano; Mugnaini, Claudia; Scorzelli, Francesco; Maione, Sabatino; Corelli, Federico; Di Marzo, Vincenzo; Alcaro, Stefano; Artese, Anna -
Synthesis of pyrazolo[1,5-a]pyrimidine ring as a possible bioisosteric replacement of the 5-(1H-pyrrol-1-yl)pyrazole scaffold 1-gen-2022 Mugnaini, Claudia; Pasculini, Livia; Pagli, Carlotta; Brizzi, Antonella; Paolino, Marco; Gianibbi, Beatrice; Corelli, Federico -
Lipoic/Capsaicin-Related Amides: Synthesis and Biological Characterization of New TRPV1 Agonists Endowed with Protective Properties against Oxidative Stress 1-gen-2022 Brizzi, Antonella; Maramai, Samuele; Aiello, Francesca; Baratto, Maria Camilla; Corelli, Federico; Mugnaini, Claudia; Paolino, Marco; Scorzelli, Francesco; Aldinucci, Carlo; De Petrocellis, Luciano; Signorini, Cinzia; Pessina, Federica -
Optimization of Pyrazole Compounds as Antibiotic Adjuvants Active against Colistin- and Carbapenem-Resistant Acinetobacter baumannii 1-gen-2022 Sannio, Filomena; Brizzi, Antonella; Del Prete, Rosita; Avigliano, Marialuce; Simone, Tiziana; Pagli, Carlotta; Ferraro, Teresa; De Luca, Filomena; Paolino, Marco; Corelli, Federico; Mugnaini, Claudia; Docquier, Jean-Denis -
Design, synthesis and biological evaluation of light-driven on-off multitarget AChE and MAO-B inhibitors 1-gen-2022 Paolino, Marco; Rullo, Mariagrazia; Maramai, Samuele; de Candia, Modesto; Pisani, Leonardo; Catto, Marco; Mugnaini, Claudia; Brizzi, Antonella; Cappelli, Andrea; Olivucci, Massimo; Corelli, Federico; Altomare, Cosimo D -
In silico multi-target approach revealed potential lead compounds as scaffold for the synthesis of chemical analogues targeting SARS-CoV-2 1-gen-2022 Trezza, Alfonso; Mugnaini, Claudia; Corelli, Federico; Santucci, Annalisa; Spiga, Ottavia -
Computational drug repurposing for the identification of SARS-CoV-2 main protease inhibitors 1-gen-2021 Fiorucci, Diego; Milletti, Eva; Orofino, Francesco; Brizzi, Antonella; Mugnaini, Claudia; Corelli, Federico -
Suppressing effect of the novel positive allosteric modulator of the GABAB receptor, COR659, on locomotor hyperactivity induced by different drugs of abuse 1-gen-2021 Lobina, Carla; Maccioni, Paola; Lorrai, Irene; Zaru, Alessandro; Collu, Maria; Carai, Mauro A. M.; Brizzi, Antonella; Mugnaini, Claudia; Luigi Gessa, Gian; Corelli, Federico; Colombo, Giancarlo -
Has a “Chemical Magic” Opened up New Prospects for Glaucoma? 1-gen-2021 Corelli, Federico -
Viral Envelope Membrane: A Special Entry Pathway and a Promising Drug Target 1-gen-2021 Palombi, Nastasja; Brai, Annalaura; Gerace, Martina; DI MARIA, Salvatore; Orofino, Francesco; Corelli, Federico -
COR758, a negative allosteric modulator of GABAB receptors 1-gen-2021 Porcu, Alessandra; Mostallino, Rafaela; Serra, Valeria; Melis, Miriam; Sogos, Valeria; Beggiato, Sarah; Ferraro, Luca; Manetti, Fabrizio; Gianibbi, Beatrice; Bettler, Bernhard; Corelli, Federico; Mugnaini, Claudia; Castelli, M. Paola -
The GABAB receptor positive allosteric modulator COR659: in vitro metabolism, in vivo pharmacokinetics in rats, synthesis and pharmacological characterization of metabolically protected derivatives 1-gen-2020 Ferlenghi, Francesca; Maccioni, Paola; Mugnaini, Claudia; Brizzi, Antonella; Fara, Federica; Mostallino, Rafaela; M Paola, Castelli; Colombo, Giancarlo; Mor, Marco; Vacondio, Federica; Corelli, Federico -
Design, synthesis, and physicochemical and pharmacological profiling of 7‐Hydroxy-5-oxopyrazolo[4,3‐b]pyridine-6-carboxamide derivatives with antiosteoarthritic activity in vivo 1-gen-2020 Mugnaini, Claudia; Kostrzewa, Magdalena; Bryk, Marta; Mokhtar Mahmoud, Ali; Brizzi, Antonella; Lamponi, Stefania; Giorgi, Gianluca; Ferlenghi, Francesca; Vacondio, Federica; Maccioni, Paola; Colombo, Giancarlo; Mor, Marco; Starowicz, Katarzyna; Di Marzo, Vincenzo; Ligresti, Alessia; Corelli, Federico -
Structure optimization of positive allosteric modulators of GABAB receptors led to the unexpected discovery of antagonists/potential negative allosteric modulators 1-gen-2020 Mugnaini, Claudia; Brizzi, Antonella; Mostallino, Rafaela; Paola Castelli, Maria; Corelli, Federico -
Differential effects of saikosaponins on alcohol and chocolate self-administration in rats. 1-gen-2020 Maccioni, Paola; Lorrai1, Irene; Fara, Federica; Carai, Mauro A. M.; Luigi Gessa, Gian; Chin4 Jung Hwan Lee, Young-Won; Cheol Kwon, Hak; Corelli, Federico; Colombo, Giancarlo -
Screen of unfocused libraries identified compounds with direct or synergistic antibacterial activity 1-gen-2020 Mugnaini, C.; Sannio, F.; Brizzi, A.; Del Prete, R.; Simone, T.; Ferraro, T.; De Luca, F.; Corelli, F.; Docquier, J. D. -
New synthesis of N1- and N2-substituted pyrazolo[4,3-b]pyridine-5-one derivatives as CB2 receptor ligands 1-gen-2020 Mugnaini, Claudia; Brizzi, Antonella; Vinciarelli, Giorgia; Paolino, Marco; Corelli, Federico -
Synthetic bioactive olivetol-related amides: the influence of the phenolic group in cannabinoid receptor activity 1-gen-2020 Brizzi, Antonella; Aiello, Francesca; Boccella, Serena; Grazia Cascio, Maria; De Petrocellis, Luciano; Frosini, Maria; Gado, Francesca; Ligresti, Alessia; Luongo, Livio; Marini, Pietro; Mugnaini, Claudia; Pessina, Federica; Corelli, Federico; Maione, Sabatino; Manera, Clementina; Pertwee, Roger G.; Di Marzo, Vincenzo -
A novel highly selective cannabinoid CB2 agonist reduces in vitro growth and TGF-beta release of human glial cell tumors 1-gen-2019 Cioni, Chiara; Tassi, Maristella; Marotta, Giuseppe; Mugnaini, Claudia; Corelli, Federico; Annunziata, Pasquale -
Suppressing effect of CMPPE, a new positive allosteric modulator of the GABAB receptor, on alcohol self-administration and reinstatement of alcohol seeking in rats 1-gen-2019 Maccioni, Paola; Fara, Federica; Lorrai, Irene; Acciaro, Carla; Mugnaini, Claudia; Corelli, Federico; Colombo, Giancarlo -
Mostrati risultati da 1 a 20 di 194
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