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Titolo Data di pubblicazione Autore(i) File Abstract
1,2,4-Triazole-3-thione analogues with an arylakyl group at position 4 as metallo-β-lactamase inhibitors 1-gen-2022 Gavara, Laurent; Verdirosa, Federica; Sevaille, Laurent; Legru, Alice; Corsica, Giuseppina; Nauton, Lionel; Sandra Mercuri, Paola; Sannio, Filomena; De Luca, Filomena; Hadjadj, Margot; Cerboni, Giulia; Vo Hoang, Yen; Licznar-Fajardo, Patricia; Galleni, Moreno; Docquier, Jean-Denis; Hernandez, Jean-François -
1,2,4-Triazole-3-Thione Analogues with a 2-Ethylbenzoic Acid at Position 4 as VIM-type Metallo-β-Lactamase Inhibitors 1-gen-2022 Verdirosa, Federica; Gavara, Laurent; Sevaille, Laurent; Tassone, Giusy; Corsica, Giuseppina; Legru, Alice; Feller, Georges; Chelini, Giulia; Mercuri, Paola Sandra; Tanfoni, Silvia; Sannio, Filomena; Benvenuti, Manuela; Cerboni, Giulia; De Luca, Filomena; Bouajila, Ezeddine; Vo Hoang, Yen; Licznar-Fajardo, Patricia; Galleni, Moreno; Pozzi, Cecilia; Mangani, Stefano; Docquier, Jean-Denis; Hernandez, Jean-François -
Optimization of Pyrazole Compounds as Antibiotic Adjuvants Active against Colistin- and Carbapenem-Resistant Acinetobacter baumannii 1-gen-2022 Sannio, Filomena; Brizzi, Antonella; Del Prete, Rosita; Avigliano, Marialuce; Simone, Tiziana; Pagli, Carlotta; Ferraro, Teresa; De Luca, Filomena; Paolino, Marco; Corelli, Federico; Mugnaini, Claudia; Docquier, Jean-Denis -
4-Alkyl-1,2,4-triazole-3-thione analogues as metallo-β-lactamase inhibitors 1-gen-2021 Gavara, Laurent; Legru, Alice; Verdirosa, Federica; Sevaille, Laurent; Nauton, Lionel; Corsica, Giuseppina; Mercuri, Paola Sandra; Sannio, Filomena; Feller, Georges; Coulon, Rémi; De Luca, Filomena; Cerboni, Giulia; Tanfoni, Silvia; Chelini, Giulia; Galleni, Moreno; Docquier, Jean-Denis; Hernandez, Jean-François -
Discovery of Taniborbactam (VNRX-5133): A Broad-Spectrum Serine- And Metallo-β-lactamase Inhibitor for Carbapenem-Resistant Bacterial Infections 1-gen-2020 Liu, B.; Trout, R. E. L.; Chu, G. -H.; Mcgarry, D.; Jackson, R. W.; Hamrick, J. C.; Daigle, D. M.; Cusick, S. M.; Pozzi, C.; De Luca, F.; Benvenuti, M.; Mangani, S.; Docquier, J. -D.; Weiss, W. J.; Pevear, D. C.; Xerri, L.; Burns, C. J. -
Amino acid replacement at position 228 induces fluctuation in the Ω-loop of KPC-3 and reduces the affinity against oxyimino cephalosporins: Kinetic and molecular dynamics studies 1-gen-2020 Piccirilli, A.; Brisdelli, F.; Docquier, J. D.; Aschi, M.; Cherubini, S.; De Luca, F.; Matagne, A.; Amicosante, G.; Perilli, M. -
VNRX-5133 (Taniborbactam), a broad-spectrum inhibitor of serine- And metallo-β-lactamases, restores activity of cefepime in enterobacterales and Pseudomonas aeruginosa 1-gen-2020 Hamrick, J. C.; Docquier, J. -D.; Uehara, T.; Myers, C. L.; Six, D. A.; Chatwin, C. L.; John, K. J.; Vernacchio, S. F.; Cusick, S. M.; Trout, R. E. L.; Pozzi, C.; De Luca, F.; Benvenuti, M.; Mangani, S.; Liu, B.; Jackson, R. W.; Moeck, G.; Xerri, L.; Burns, C. J.; Pevear, D. C.; Daigle, D. M. -
Virtual screening identifies broad-spectrum β-lactamase inhibitors with activity on clinically relevant serine- and metallo-carbapenemases 1-gen-2020 Spyrakis, F.; Santucci, M.; Maso, L.; Cross, S.; Gianquinto, E.; Sannio, F.; Verdirosa, F.; De Luca, F.; Docquier, J. D.; Cendron, L.; Tondi, D.; Venturelli, A.; Cruciani, G.; Costi, M. P. -
4-Amino-1,2,4-triazole-3-thione-derived Schiff bases as metallo-β-lactamase inhibitors 1-gen-2020 Gavara, L.; Sevaille, L.; De Luca, F.; Mercuri, P.; Bebrone, C.; Feller, G.; Legru, A.; Cerboni, G.; Tanfoni, S.; Baud, D.; Cutolo, G.; Bestgen, B.; Chelini, G.; Verdirosa, F.; Sannio, F.; Pozzi, C.; Benvenuti, M.; Kwapien, K.; Fischer, M.; Becker, K.; Frere, J. -M.; Mangani, S.; Gresh, N.; Berthomieu, D.; Galleni, M.; Docquier, Jd; Hernandez, J. -F. -
Screen of Unfocused Libraries Identified Compounds with Direct or Synergistic Antibacterial Activity 1-gen-2020 Mugnaini, C.; Sannio, F.; Brizzi, A.; Del Prete, R.; Simone, T.; Ferraro, T.; De Luca, F.; Corelli, F.; Docquier, J. D. -
SAR Studies Leading to the Identification of a Novel Series of Metallo-β-lactamase Inhibitors for the Treatment of Carbapenem-Resistant Enterobacteriaceae Infections That Display Efficacy in an Animal Infection Model 1-gen-2019 Leiris, Simon; Coelho, Alicia; Castandet, Jérôme; Bayet, Maëlle; Lozano, Clarisse; Bougnon, Juliette; Bousquet, Justine; Everett, Martin; Lemonnier, Marc; Sprynski, Nicolas; Zalacain, Magdalena; Pallin, Thomas David; Cramp, Michael C.; Jennings, Neil; Raphy, Gilles; Jones, Mark W.; Pattipati, Ramesh; Shankar, Battu; Sivasubrahmanyam, Relangi; Soodhagani, Ashok K.; Juventhala, Ramakrishna R.; Pottabathini, Narender; Pothukanuri, Srinivasu; Benvenuti, Manuela; Pozzi, Cecilia; Mangani, Stefano; De Luca, Filomena; Cerboni, Giulia; Docquier, Jean-Denis; Davies, David T. -
Alkyl-guanidine Compounds as Potent Broad-Spectrum Antibacterial Agents: Chemical Library Extension and Biological Characterization 1-gen-2018 Pasero, Carolina; D'Agostino, Ilaria; De Luca, Filomena; Zamperini, Claudio; Deodato, Davide; Truglio, Giuseppina I.; Sannio, Filomena; DEL PRETE, Rosita; Ferraro, Teresa; Visaggio, Daniela; Mancini, Arianna; Guglielmi, Mario B.; Visca, Paolo; Docquier, Jean-Denis; Botta, Maurizio -
Boric acid and acetate anion binding to subclass B3 metallo-β-lactamase BJP-1 provides clues for mechanism of action and inhibitor design 1-gen-2018 Di Pisa, Flavio; Pozzi, Cecilia; Benvenuti, Manuela; Docquier, Jean-Denis; De Luca, Filomena; Mangani, Stefano -
Discovery of a Novel Metallo-β-Lactamase Inhibitor that Potentiates Meropenem Activity against Carbapenem-Resistant Enterobacteriaceae 1-gen-2018 Everett, Martin; Sprynski, Nicolas; Coelho, Alicia; Castandet, Jérôme; Bayet, Maëlle; Bougnon, Juliette; Lozano, Clarisse; Davies, David T; Leiris, Simon; Zalacain, Magdalena; Morrissey, Ian; Magnet, Sophie; Holden, Kirsty; Warn, Peter; De Luca, Filomena; Docquier, Jean-Denis; Lemonnier, Marc -
Atomic-Resolution Structure of a Class C β-Lactamase and Its Complex with Avibactam 1-gen-2018 Pozzi, Cecilia; Di Pisa, Flavio; De Luca, Filomena; Benvenuti, Manuela; Docquier, Jean Denis; Mangani, Stefano -
Chryseobacterium gleum in a man with prostatectomy in Senegal: A case report and review of the literature 1-gen-2017 Arouna, O; DE LUCA, Filomena; Camara, M.; Fall, B.; Fall, B.; Ba Diallo, A.; Docquier, JEAN DENIS; Mboup, S. -
1,2,4-Triazole-3-thione compounds as inhibitors of di-zinc metallo-β-lactamases 1-gen-2017 Sevaille, Laurent; Gavara, Laurent; Bebrone, Carine; DE LUCA, Filomena; Nauton, Lionel; Achard, Maud; Mercuri, Paola; Tanfoni, Silvia; Borgianni, Luisa; Guyon, Carole; Lonjon, Pauline; Turan Zitouni, Gülhan; Dzieciolowski, Julia; Becker, Katja; Bénard, Lionel; Condon, Ciaran; Maillard, Ludovic; Martinez, Jean; Frère, Jean Marie; Dideberg, Otto; Galleni, Moreno; Docquier, JEAN DENIS; Hernandez, Jean François -
Design and synthesis of a novel inhibitor of T. Viride chitinase through an in silico target fishing protocol 1-gen-2017 Maccari, Giorgio; Deodato, Davide; Fiorucci, Diego; Orofino, Francesco; Truglio, Giuseppina I.; Pasero, Carolina; Martini, Riccardo; De Luca, Filomena; Docquier, Jean-Denis; Botta, Maurizio -
Identification, synthesis and biological activity of alkyl-guanidine oligomers as potent antibacterial agents 1-gen-2017 Zamperini, C.; Maccari, G.; Deodato, D.; Pasero, Carolina; D'Agostino, Ilaria; Orofino, Francesco; De Luca, F.; Dreassi, E.; Docquier, J. D.; Botta, M. -
Computational and biological profile of boronic acids for the detection of bacterial serine- and metallo-beta-lactamases 1-gen-2017 Santucci, Matteo; Spyrakis, Francesca; Cross, Simon; Quotadamo, Antonio; Farina, Davide; Tondi, Donatella; De Luca, Filomena; Docquier, Jean-Denis; Prieto, Ana Isabel; Ibacache, Claudia; Blázquez, Jesús; Venturelli, Alberto; Cruciani, Gabriele; Costi, Maria Paola -
Mostrati risultati da 1 a 20 di 42
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