Sfoglia per Autore
DNA and RNA polymerases
2024-01-01 Picarazzi, F.; Mori, M.
Perspectives in the treatment of antibiotic-resistant bacterial infections with active photodynamic partners within the framework of the EURESTOP COST Action (CA21145)
2024-01-01 Mori, Mattia; Dumoulin, Fabienne; Faustino, M. Amparo F.; Plaetzer, Kristjan
The Antiepileptic Drug Levetiracetam Inhibits Carbonic Anhydrase: In Vitro and In Silico Studies on Catalytically Active Human Isoforms
2024-01-01 Cutarella, L.; Mori, M.; Supuran, C. T.
Hedgehog Pathway Inhibition by Novel Small Molecules Impairs Melanoma Cell Migration and Invasion under Hypoxia
2024-01-01 Falsini, A.; Giuntini, G.; Mori, M.; Ghirga, F.; Quaglio, D.; Cucinotta, A.; Coppola, F.; Filippi, I.; Naldini, A.; Botta, B.; Carraro, F.
Exploring a New Generation of Pyrimidine and Pyridine Derivatives as Anti-Influenza Agents Targeting the Polymerase PA–PB1 Subunits Interaction
2024-01-01 Giacchello, Ilaria; Cianciusi, Annarita; Bertagnin, Chiara; Bonomini, Anna; Francesconi, Valeria; Mori, Mattia; Carbone, Anna; Musumeci, Francesca; Loregian, Arianna; Schenone, Silvia
Fragment-Based Interrogation of the 14–3–3/TAZ Protein–Protein Interaction
2024-01-01 Andlovic, Blaž; Valenti, Dario; Centorrino, Federica; Picarazzi, Francesca; Hristeva, Stanimira; Hiltmann, Malgorzata; Wolf, Alexander; Cantrelle, François-Xavier; Mori, Mattia; Landrieu, Isabelle; Levy, Laura M.; Klebl, Bert; Tzalis, Dimitrios; Genski, Thorsten; Eickhoff, Jan; Ottmann, Christian
The Rise of Bacterial G-Quadruplexes in Current Antimicrobial Discovery
2024-01-01 Ciaco, Stefano; Aronne, Rossella; Fiabane, Martina; Mori, Mattia
Novel 2,4-Dichloro-5-sulfamoylbenzoic Acid Oxime Esters: First Studies as Potential Human Carbonic Anhydrase Inhibitors
2024-01-01 Kilbile, Jaydeo T.; Sapkal, Suryakant B.; Renzi, Gioele; D'Agostino, Ilaria; Cutarella, Luigi; Mori, Mattia; De Filippis, Barbara; Islam, Imadul; Massardi, Maria Luisa; Somenza, Elena; Ronca, Roberto; Tamboli, Yasinalli; Carta, Fabrizio; Supuran, Claudiu T.
Solving the antibacterial resistance in Europe: The multipronged approach of the COST Action CA21145 EURESTOP
2024-01-01 Seguin-Devaux, Carole; Mestrovic, Tomislav; Arts, Jacobus J; Sen Karaman, Didem; Nativi, Cristina; Reichmann, Dana; Sahariah, Priyanka; Smani, Younes; Rijo, Patricia; Mori, Mattia
Cyclization of acyl thiosemicarbazides led to new Helicobacter pylori α‐carbonic anhydrase inhibitors
2024-01-01 Gumus, Arzu; D'Agostino, Ilaria; Puca, Valentina; Crocetta, Valentina; Carradori, Simone; Cutarella, Luigi; Mori, Mattia; Carta, Fabrizio; Angeli, Andrea; Capasso, Clemente; Supuran, Claudiu T.
Lasamide Containing Sulfonylpiperazines as Effective Agents for the Management of Glaucoma Associated Symptoms
2024-01-01 Kilbile, Jaydeo T.; Sapkal, Suryakant B.; Renzi, Gioele; D'Agostino, Ilaria; Boudjelal, Mohamed; Tamboli, Yasinalli; Cutarella, Luigi; Mori, Mattia; Sgambellone, Silvia; Villano, Serafina; Marri, Silvia; Lucarini, Laura; Carradori, Simone; Carta, Fabrizio; Supuran, Claudiu T.
The antimicrobial potential of adarotene derivatives against Staphylococcus aureus strains
2024-01-01 Princiotto, Salvatore; Casciaro, Bruno; G. Temprano, Alvaro; Musso, Loana; Sacchi, Francesca; Loffredo, Maria Rosa; Cappiello, Floriana; Sacco, Federica; Raponi, Giammarco; Fernandez, Virginia Perez; Iucci, Teresa; Mangoni, Maria Luisa; Mori, Mattia; Dallavalle, Sabrina; Pisano, Claudio
Azobenzenesulfonamide Carbonic Anhydrase Inhibitors as New Weapons to Fight Helicobacter pylori: Synthesis, Bioactivity Evaluation, In Vivo Toxicity, and Computational Studies
2024-01-01 Giampietro, Letizia; Marinacci, Beatrice; Della Valle, Alice; D'Agostino, Ilaria; Lauro, Aldo; Mori, Mattia; Carradori, Simone; Ammazzalorso, Alessandra; De Filippis, Barbara; Maccallini, Cristina; Angeli, Andrea; Capasso, Clemente; Francati, Santolo; Mollica, Adriano; Grande, Rossella; Supuran, Claudiu T.
Recent developments of agents targeting Vibrio cholerae: patents and literature data
2024-01-01 Melfi, Francesco; Carradori, Simone; Mencarelli, Noemi; Campestre, Cristina; Granese, Arianna; Mori, Mattia
Inhibition of adenovirus transport from the endosome to the cell nucleus by rotenone
2024-01-01 Balsera-Manzanero, María; Ghirga, Francesca; Ruiz-Molina, Ana; Mori, Mattia; Pachón, Jerónimo; Botta, Bruno; Cordero, Elisa; Quaglio, Deborah; Sánchez-Céspedes, Javier
Exploring the Antiviral Potential of Natural Compounds against Influenza: A Combined Computational and Experimental Approach
2024-01-01 Perovic, Vladimir; Stevanovic, Kristina; Bukreyeva, Natalya; Paessler, Slobodan; Maruyama, Junki; López-Serrano, Sergi; Darji, Ayub; Sencanski, Milan; Radosevic, Draginja; Berardozzi, Simone; Botta, Bruno; Mori, Mattia; Glisic, Sanja
Inhibitors of UHRF1 base flipping activity showing cytotoxicity against cancer cells
2023-01-01 Ciaco, Stefano; Mazzoleni, Viola; Javed, Aqib; Eiler, Sylvia; Ruff, Marc; Mousli, Marc; Mori, Mattia; Mély, Yves
Exploring the potential of anthraquinone-based hybrids for identifying a novel generation of antagonists for the Smoothened receptor in HH-dependent tumour
2023-01-01 Quaglio, Deborah; Infante, Paola; Cammarone, Silvia; Lamelza, Lara; Conenna, Marilisa; Ghirga, Francesca; Adabbo, Gennaro; Pisano, Luca; Di Marcotullio, Lucia; Botta, Bruno; Mori, Mattia
Antimalarial drugs: what's new in the patents?
2023-01-01 Lopes, Elizabeth A; Santos, Maria M M; Mori, Mattia
Natural flavonoid derivatives have pan-Coronavirus antiviral activity
2023-01-01 Mori, Mattia; Quaglio, Deborah; Calcaterra, Andrea; Ghirga, Francesca; Sorrentino, Leonardo; Cammarone, Silvia; Fracella, Matteo; D'Auria, Alessandra; Frasca, Federica; Criscuolo, Elena; Clementi, Nicola; Mancini, Nicasio; Botta, Bruno; Antonelli, Guido; Pierangeli, Alessandra; Scagnolari, Carolina
Titolo | Data di pubblicazione | Autore(i) | File | Abstract |
---|---|---|---|---|
DNA and RNA polymerases | 1-gen-2024 | Picarazzi, F.; Mori, M. | - | |
Perspectives in the treatment of antibiotic-resistant bacterial infections with active photodynamic partners within the framework of the EURESTOP COST Action (CA21145) | 1-gen-2024 | Mori, Mattia; Dumoulin, Fabienne; Faustino, M. Amparo F.; Plaetzer, Kristjan | - | |
The Antiepileptic Drug Levetiracetam Inhibits Carbonic Anhydrase: In Vitro and In Silico Studies on Catalytically Active Human Isoforms | 1-gen-2024 | Cutarella, L.; Mori, M.; Supuran, C. T. | - | |
Hedgehog Pathway Inhibition by Novel Small Molecules Impairs Melanoma Cell Migration and Invasion under Hypoxia | 1-gen-2024 | Falsini, A.; Giuntini, G.; Mori, M.; Ghirga, F.; Quaglio, D.; Cucinotta, A.; Coppola, F.; Filippi, I.; Naldini, A.; Botta, B.; Carraro, F. | - | |
Exploring a New Generation of Pyrimidine and Pyridine Derivatives as Anti-Influenza Agents Targeting the Polymerase PA–PB1 Subunits Interaction | 1-gen-2024 | Giacchello, Ilaria; Cianciusi, Annarita; Bertagnin, Chiara; Bonomini, Anna; Francesconi, Valeria; Mori, Mattia; Carbone, Anna; Musumeci, Francesca; Loregian, Arianna; Schenone, Silvia | - | |
Fragment-Based Interrogation of the 14–3–3/TAZ Protein–Protein Interaction | 1-gen-2024 | Andlovic, Blaž; Valenti, Dario; Centorrino, Federica; Picarazzi, Francesca; Hristeva, Stanimira; Hiltmann, Malgorzata; Wolf, Alexander; Cantrelle, François-Xavier; Mori, Mattia; Landrieu, Isabelle; Levy, Laura M.; Klebl, Bert; Tzalis, Dimitrios; Genski, Thorsten; Eickhoff, Jan; Ottmann, Christian | - | |
The Rise of Bacterial G-Quadruplexes in Current Antimicrobial Discovery | 1-gen-2024 | Ciaco, Stefano; Aronne, Rossella; Fiabane, Martina; Mori, Mattia | - | |
Novel 2,4-Dichloro-5-sulfamoylbenzoic Acid Oxime Esters: First Studies as Potential Human Carbonic Anhydrase Inhibitors | 1-gen-2024 | Kilbile, Jaydeo T.; Sapkal, Suryakant B.; Renzi, Gioele; D'Agostino, Ilaria; Cutarella, Luigi; Mori, Mattia; De Filippis, Barbara; Islam, Imadul; Massardi, Maria Luisa; Somenza, Elena; Ronca, Roberto; Tamboli, Yasinalli; Carta, Fabrizio; Supuran, Claudiu T. | - | |
Solving the antibacterial resistance in Europe: The multipronged approach of the COST Action CA21145 EURESTOP | 1-gen-2024 | Seguin-Devaux, Carole; Mestrovic, Tomislav; Arts, Jacobus J; Sen Karaman, Didem; Nativi, Cristina; Reichmann, Dana; Sahariah, Priyanka; Smani, Younes; Rijo, Patricia; Mori, Mattia | - | |
Cyclization of acyl thiosemicarbazides led to new Helicobacter pylori α‐carbonic anhydrase inhibitors | 1-gen-2024 | Gumus, Arzu; D'Agostino, Ilaria; Puca, Valentina; Crocetta, Valentina; Carradori, Simone; Cutarella, Luigi; Mori, Mattia; Carta, Fabrizio; Angeli, Andrea; Capasso, Clemente; Supuran, Claudiu T. | - | |
Lasamide Containing Sulfonylpiperazines as Effective Agents for the Management of Glaucoma Associated Symptoms | 1-gen-2024 | Kilbile, Jaydeo T.; Sapkal, Suryakant B.; Renzi, Gioele; D'Agostino, Ilaria; Boudjelal, Mohamed; Tamboli, Yasinalli; Cutarella, Luigi; Mori, Mattia; Sgambellone, Silvia; Villano, Serafina; Marri, Silvia; Lucarini, Laura; Carradori, Simone; Carta, Fabrizio; Supuran, Claudiu T. | - | |
The antimicrobial potential of adarotene derivatives against Staphylococcus aureus strains | 1-gen-2024 | Princiotto, Salvatore; Casciaro, Bruno; G. Temprano, Alvaro; Musso, Loana; Sacchi, Francesca; Loffredo, Maria Rosa; Cappiello, Floriana; Sacco, Federica; Raponi, Giammarco; Fernandez, Virginia Perez; Iucci, Teresa; Mangoni, Maria Luisa; Mori, Mattia; Dallavalle, Sabrina; Pisano, Claudio | - | |
Azobenzenesulfonamide Carbonic Anhydrase Inhibitors as New Weapons to Fight Helicobacter pylori: Synthesis, Bioactivity Evaluation, In Vivo Toxicity, and Computational Studies | 1-gen-2024 | Giampietro, Letizia; Marinacci, Beatrice; Della Valle, Alice; D'Agostino, Ilaria; Lauro, Aldo; Mori, Mattia; Carradori, Simone; Ammazzalorso, Alessandra; De Filippis, Barbara; Maccallini, Cristina; Angeli, Andrea; Capasso, Clemente; Francati, Santolo; Mollica, Adriano; Grande, Rossella; Supuran, Claudiu T. | - | |
Recent developments of agents targeting Vibrio cholerae: patents and literature data | 1-gen-2024 | Melfi, Francesco; Carradori, Simone; Mencarelli, Noemi; Campestre, Cristina; Granese, Arianna; Mori, Mattia | - | |
Inhibition of adenovirus transport from the endosome to the cell nucleus by rotenone | 1-gen-2024 | Balsera-Manzanero, María; Ghirga, Francesca; Ruiz-Molina, Ana; Mori, Mattia; Pachón, Jerónimo; Botta, Bruno; Cordero, Elisa; Quaglio, Deborah; Sánchez-Céspedes, Javier | - | |
Exploring the Antiviral Potential of Natural Compounds against Influenza: A Combined Computational and Experimental Approach | 1-gen-2024 | Perovic, Vladimir; Stevanovic, Kristina; Bukreyeva, Natalya; Paessler, Slobodan; Maruyama, Junki; López-Serrano, Sergi; Darji, Ayub; Sencanski, Milan; Radosevic, Draginja; Berardozzi, Simone; Botta, Bruno; Mori, Mattia; Glisic, Sanja | - | |
Inhibitors of UHRF1 base flipping activity showing cytotoxicity against cancer cells | 1-gen-2023 | Ciaco, Stefano; Mazzoleni, Viola; Javed, Aqib; Eiler, Sylvia; Ruff, Marc; Mousli, Marc; Mori, Mattia; Mély, Yves | - | |
Exploring the potential of anthraquinone-based hybrids for identifying a novel generation of antagonists for the Smoothened receptor in HH-dependent tumour | 1-gen-2023 | Quaglio, Deborah; Infante, Paola; Cammarone, Silvia; Lamelza, Lara; Conenna, Marilisa; Ghirga, Francesca; Adabbo, Gennaro; Pisano, Luca; Di Marcotullio, Lucia; Botta, Bruno; Mori, Mattia | - | |
Antimalarial drugs: what's new in the patents? | 1-gen-2023 | Lopes, Elizabeth A; Santos, Maria M M; Mori, Mattia | - | |
Natural flavonoid derivatives have pan-Coronavirus antiviral activity | 1-gen-2023 | Mori, Mattia; Quaglio, Deborah; Calcaterra, Andrea; Ghirga, Francesca; Sorrentino, Leonardo; Cammarone, Silvia; Fracella, Matteo; D'Auria, Alessandra; Frasca, Federica; Criscuolo, Elena; Clementi, Nicola; Mancini, Nicasio; Botta, Bruno; Antonelli, Guido; Pierangeli, Alessandra; Scagnolari, Carolina | - |
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