Sfoglia per Autore VAGAGGINI, CHIARA
Characterization of in vitro and in vivo properties of pharmacologically active compounds in a GLP-Like laboratory
2024-06-14 Vagaggini, Chiara
Serendipitous identification of azine anticancer agents using a privileged scaffold morphing strategy
2024-01-01 Cesarini, Silvia; Vicenti, Ilaria; Poggialini, Federica; Filippi, Silvia; Mancin, Eleonora; Fiaschi, Lia; De Marchi, Elisa; Giammarino, Federica; Vagaggini, Chiara; Bizzarri, Bruno Mattia; Saladino, Raffaele; Dreassi, Elena; Zazzi, Maurizio; Botta, Lorenzo
Infesting Seaweeds as a Novel Functional Food: Analysis of Nutrients, Antioxidants and ACE Inhibitory Effects
2024-01-01 Brai, Annalaura; Hasanaj, Anjeza; Vagaggini, Chiara; Poggialini, Federica; Dreassi, Elena
Design, synthesis, ADME and biological evaluation of benzylpiperidine and benzylpiperazine derivatives as novel reversible monoacylglycerol lipase (MAGL) inhibitors
2024-01-01 Di Stefano, M.; Masoni, S.; Bononi, G.; Poli, G.; Galati, S.; Gado, F.; Manzi, S.; Vagaggini, C.; Brai, A.; Caligiuri, I.; Asif, K.; Rizzolio, F.; Macchia, M.; Chicca, A.; Sodi, A.; Di Bussolo, V.; Minutolo, F.; Meier, P.; Gertsch, J.; Granchi, C.; Dreassi, E.; Tuccinardi, T.
Identification of Novel Non-Nucleoside Inhibitors of Zika Virus NS5 Protein Targeting MTase Activity
2024-01-01 Fiorucci, D.; Meaccini, M.; Poli, G.; Stincarelli, M. A.; Vagaggini, C.; Giannecchini, S.; Sutto-Ortiz, P.; Canard, B.; Decroly, E.; Dreassi, E.; Brai, A.; Botta, M.
Applying molecular hybridization to design a new class of pyrazolo[3,4-d]pyrimidines as Src inhibitors active in hepatocellular carcinoma
2024-01-01 Di Maria, Salvatore; Passannanti, Raffaele; Poggialini, Federica; Vagaggini, Chiara; Serafinelli, Alessia; Bianchi, Elena; Governa, Paolo; Botta, Lorenzo; Maga, Giovanni; Crespan, Emmanuele; Manetti, Fabrizio; Dreassi, Elena; Musumeci, Francesca; Carbone, Anna; Schenone, Silvia
Novel multitarget directed ligands inspired by riluzole: A serendipitous synthesis of substituted benzo[b][1,4]thiazepines potentially useful as neuroprotective agents
2024-01-01 Maramai, S.; Saletti, M.; Paolino, M.; Giuliani, G.; Cazzola, J.; Spaiardi, P.; Talpo, F.; Frosini, M.; Pifferi, A.; Ballarotto, M.; Carotti, A.; Poggialini, F.; Vagaggini, C.; Dreassi, E.; Giorgi, G.; Dondio, G.; Cappelli, A.; Rosario Biella, G.; Anzini, M.
A Facile Access to Green Fluorescent Albumin Derivatives
2024-01-01 Saletti, M.; Paolino, M.; Venditti, J.; Bonechi, C.; Giuliani, G.; Lamponi, S.; Tassone, G.; Boccia, A.; Botta, C.; Blancafort, L.; Poggialini, F.; Vagaggini, C.; Cappelli, A.
Upcycling Milk Industry Byproducts into Tenebrio molitor Larvae: Investigation on Fat, Protein, and Sugar Composition
2024-01-01 Brai, Annalaura; Neri, Cassia; Tarchi, Franca; Poggialini, Federica; Vagaggini, Chiara; Frosinini, Riccardo; Simoni, Sauro; Francardi, Valeria; Dreassi, Elena
Early investigation of a novel SI306 theranostic prodrug for glioblastoma treatment
2024-01-01 Vagaggini, Chiara; Petroni, Debora; D'Agostino, Ilaria; Poggialini, Federica; Cavallini, Chiara; Cianciusi, Annarita; Salis, Annalisa; D'Antona, Lucia; Francesconi, Valeria; Manetti, Fabrizio; Damonte, Gianluca; Musumeci, Francesca; Menichetti, Luca; Dreassi, Elena; Carbone, Anna; Schenone, Silvia
Inhibition of Pseudomonas aeruginosa Carbonic Anhydrases, Exploring Ciprofloxacin Functionalization Toward New Antibacterial Agents: An In-Depth Multidisciplinary Study
2024-01-01 Marinacci, B.; D'Agostino, I.; Angeli, A.; Carradori, S.; Melfi, F.; Grande, R.; Corsiani, M.; Ferraroni, M.; Agamennone, M.; Tondo, A. R.; Zara, S.; Puca, V.; Pellegrini, B.; Vagaggini, C.; Dreassi, E.; Patrauchan, M. A.; Capasso, C.; Nicolotti, O.; Carta, F.; Supuran, C. T.
Development and validation of derivatization-based LC-MS/MS method for quantification of short-chain fatty acids in human, rat, and mouse plasma
2023-01-01 Vagaggini, Chiara; Brai, Annalaura; Bonente, Denise; Lombardi, Jessica; Poggialini, Federica; Pasqualini, Claudia; Barone, Virginia; Nicoletti, Claudio; Bertelli, Eugenio; Dreassi, Elena
Exploiting fall foliage by-products to optimize Tenebrio molitor nutraceutical value
2023-01-01 Brai, A.; Provenzani, M. P.; Pasqualini, C.; Poggialini, F.; Vagaggini, C.; Tarchi, F.; Frosinini, R.; Francardi, V.; Simoni, S.; Dreassi, E.
THE REPLACEMENT OF FLOUR-BASED FEED WITH PELLETS REDUCES DUSTINESS AND IMPROVES TENEBRIO MOLITOR BREEDERS’ SAFETY
2023-01-01 Brai, A.; Tarchi, F.; Pasqualini, C.; Poggialini, F.; Vagaggini, C.; Frosinini, R.; Simoni, S.; Francardi, V.; Dreassi, E.
Biological Evaluation and In Vitro Characterization of ADME Profile of In-House Pyrazolo[3,4-d]pyrimidines as Dual Tyrosine Kinase Inhibitors Active against Glioblastoma Multiforme
2023-01-01 Poggialini, Federica; Vagaggini, Chiara; Brai, Annalaura; Pasqualini, Claudia; Crespan, Emmanuele; Maga, Giovanni; Perini, Cecilia; Cabella, Noemi; Botta, Lorenzo; Musumeci, Francesca; Frosini, Maria; Schenone, Silvia; Dreassi, Elena
Efficient use of agricultural waste to naturally fortify Tenebrio molitor mealworms and evaluation of their nutraceutical properties
2023-01-01 Brai, A.; Poggialini, F.; Trivisani, C. I.; Vagaggini, C.; Tarchi, F.; Francardi, V.; Dreassi, E.
Progress towards adjuvant development: focus on antiviral therapy
2023-01-01 Brai, A.; Poggialini, F.; Pasqualini, C.; Trivisani, C. I.; Vagaggini, C.; Dreassi, E.
Use of distillery by-products as Tenebrio molitor mealworm feed supplement
2023-01-01 Brai, A.; Vagaggini, C.; Pasqualini, C.; Poggialini, F.; Tarchi, F.; Francardi, V.; Dreassi, E.
Triazolo[3,4- b]benzothiazole scaffold as versatile nicotinamide mimic allowing nanomolar inhibition of different PARP enzymes
2023-01-01 Murthy, S.; Nizi, M. G.; Maksimainen, M. M.; Massari, S.; Alaviuhkola, J.; Lippok, B. E.; Vagaggini, C.; Sowa, S. T.; Galera-Prat, A.; Ashok, Y.; Venkannagari, H.; Prunskaite-Hyyrylainen, R.; Dreassi, E.; Luscher, B.; Korn, P.; Tabarrini, O.; Lehtio, L.
Tenebrio molitor as a Simple and Cheap Preclinical Pharmacokinetic and Toxicity Model
2023-01-01 Brai, Annalaura; Poggialini, Federica; Vagaggini, Chiara; Pasqualini, Claudia; Simoni, Sauro; Francardi, Valeria; Dreassi, Elena
Titolo | Data di pubblicazione | Autore(i) | File | Abstract |
---|---|---|---|---|
Characterization of in vitro and in vivo properties of pharmacologically active compounds in a GLP-Like laboratory | 14-giu-2024 | Vagaggini, Chiara | - | |
Serendipitous identification of azine anticancer agents using a privileged scaffold morphing strategy | 1-gen-2024 | Cesarini, Silvia; Vicenti, Ilaria; Poggialini, Federica; Filippi, Silvia; Mancin, Eleonora; Fiaschi, Lia; De Marchi, Elisa; Giammarino, Federica; Vagaggini, Chiara; Bizzarri, Bruno Mattia; Saladino, Raffaele; Dreassi, Elena; Zazzi, Maurizio; Botta, Lorenzo | - | |
Infesting Seaweeds as a Novel Functional Food: Analysis of Nutrients, Antioxidants and ACE Inhibitory Effects | 1-gen-2024 | Brai, Annalaura; Hasanaj, Anjeza; Vagaggini, Chiara; Poggialini, Federica; Dreassi, Elena | - | |
Design, synthesis, ADME and biological evaluation of benzylpiperidine and benzylpiperazine derivatives as novel reversible monoacylglycerol lipase (MAGL) inhibitors | 1-gen-2024 | Di Stefano, M.; Masoni, S.; Bononi, G.; Poli, G.; Galati, S.; Gado, F.; Manzi, S.; Vagaggini, C.; Brai, A.; Caligiuri, I.; Asif, K.; Rizzolio, F.; Macchia, M.; Chicca, A.; Sodi, A.; Di Bussolo, V.; Minutolo, F.; Meier, P.; Gertsch, J.; Granchi, C.; Dreassi, E.; Tuccinardi, T. | - | |
Identification of Novel Non-Nucleoside Inhibitors of Zika Virus NS5 Protein Targeting MTase Activity | 1-gen-2024 | Fiorucci, D.; Meaccini, M.; Poli, G.; Stincarelli, M. A.; Vagaggini, C.; Giannecchini, S.; Sutto-Ortiz, P.; Canard, B.; Decroly, E.; Dreassi, E.; Brai, A.; Botta, M. | - | |
Applying molecular hybridization to design a new class of pyrazolo[3,4-d]pyrimidines as Src inhibitors active in hepatocellular carcinoma | 1-gen-2024 | Di Maria, Salvatore; Passannanti, Raffaele; Poggialini, Federica; Vagaggini, Chiara; Serafinelli, Alessia; Bianchi, Elena; Governa, Paolo; Botta, Lorenzo; Maga, Giovanni; Crespan, Emmanuele; Manetti, Fabrizio; Dreassi, Elena; Musumeci, Francesca; Carbone, Anna; Schenone, Silvia | - | |
Novel multitarget directed ligands inspired by riluzole: A serendipitous synthesis of substituted benzo[b][1,4]thiazepines potentially useful as neuroprotective agents | 1-gen-2024 | Maramai, S.; Saletti, M.; Paolino, M.; Giuliani, G.; Cazzola, J.; Spaiardi, P.; Talpo, F.; Frosini, M.; Pifferi, A.; Ballarotto, M.; Carotti, A.; Poggialini, F.; Vagaggini, C.; Dreassi, E.; Giorgi, G.; Dondio, G.; Cappelli, A.; Rosario Biella, G.; Anzini, M. | - | |
A Facile Access to Green Fluorescent Albumin Derivatives | 1-gen-2024 | Saletti, M.; Paolino, M.; Venditti, J.; Bonechi, C.; Giuliani, G.; Lamponi, S.; Tassone, G.; Boccia, A.; Botta, C.; Blancafort, L.; Poggialini, F.; Vagaggini, C.; Cappelli, A. | - | |
Upcycling Milk Industry Byproducts into Tenebrio molitor Larvae: Investigation on Fat, Protein, and Sugar Composition | 1-gen-2024 | Brai, Annalaura; Neri, Cassia; Tarchi, Franca; Poggialini, Federica; Vagaggini, Chiara; Frosinini, Riccardo; Simoni, Sauro; Francardi, Valeria; Dreassi, Elena | - | |
Early investigation of a novel SI306 theranostic prodrug for glioblastoma treatment | 1-gen-2024 | Vagaggini, Chiara; Petroni, Debora; D'Agostino, Ilaria; Poggialini, Federica; Cavallini, Chiara; Cianciusi, Annarita; Salis, Annalisa; D'Antona, Lucia; Francesconi, Valeria; Manetti, Fabrizio; Damonte, Gianluca; Musumeci, Francesca; Menichetti, Luca; Dreassi, Elena; Carbone, Anna; Schenone, Silvia | - | |
Inhibition of Pseudomonas aeruginosa Carbonic Anhydrases, Exploring Ciprofloxacin Functionalization Toward New Antibacterial Agents: An In-Depth Multidisciplinary Study | 1-gen-2024 | Marinacci, B.; D'Agostino, I.; Angeli, A.; Carradori, S.; Melfi, F.; Grande, R.; Corsiani, M.; Ferraroni, M.; Agamennone, M.; Tondo, A. R.; Zara, S.; Puca, V.; Pellegrini, B.; Vagaggini, C.; Dreassi, E.; Patrauchan, M. A.; Capasso, C.; Nicolotti, O.; Carta, F.; Supuran, C. T. | - | |
Development and validation of derivatization-based LC-MS/MS method for quantification of short-chain fatty acids in human, rat, and mouse plasma | 1-gen-2023 | Vagaggini, Chiara; Brai, Annalaura; Bonente, Denise; Lombardi, Jessica; Poggialini, Federica; Pasqualini, Claudia; Barone, Virginia; Nicoletti, Claudio; Bertelli, Eugenio; Dreassi, Elena | - | |
Exploiting fall foliage by-products to optimize Tenebrio molitor nutraceutical value | 1-gen-2023 | Brai, A.; Provenzani, M. P.; Pasqualini, C.; Poggialini, F.; Vagaggini, C.; Tarchi, F.; Frosinini, R.; Francardi, V.; Simoni, S.; Dreassi, E. | - | |
THE REPLACEMENT OF FLOUR-BASED FEED WITH PELLETS REDUCES DUSTINESS AND IMPROVES TENEBRIO MOLITOR BREEDERS’ SAFETY | 1-gen-2023 | Brai, A.; Tarchi, F.; Pasqualini, C.; Poggialini, F.; Vagaggini, C.; Frosinini, R.; Simoni, S.; Francardi, V.; Dreassi, E. | - | |
Biological Evaluation and In Vitro Characterization of ADME Profile of In-House Pyrazolo[3,4-d]pyrimidines as Dual Tyrosine Kinase Inhibitors Active against Glioblastoma Multiforme | 1-gen-2023 | Poggialini, Federica; Vagaggini, Chiara; Brai, Annalaura; Pasqualini, Claudia; Crespan, Emmanuele; Maga, Giovanni; Perini, Cecilia; Cabella, Noemi; Botta, Lorenzo; Musumeci, Francesca; Frosini, Maria; Schenone, Silvia; Dreassi, Elena | - | |
Efficient use of agricultural waste to naturally fortify Tenebrio molitor mealworms and evaluation of their nutraceutical properties | 1-gen-2023 | Brai, A.; Poggialini, F.; Trivisani, C. I.; Vagaggini, C.; Tarchi, F.; Francardi, V.; Dreassi, E. | - | |
Progress towards adjuvant development: focus on antiviral therapy | 1-gen-2023 | Brai, A.; Poggialini, F.; Pasqualini, C.; Trivisani, C. I.; Vagaggini, C.; Dreassi, E. | - | |
Use of distillery by-products as Tenebrio molitor mealworm feed supplement | 1-gen-2023 | Brai, A.; Vagaggini, C.; Pasqualini, C.; Poggialini, F.; Tarchi, F.; Francardi, V.; Dreassi, E. | - | |
Triazolo[3,4- b]benzothiazole scaffold as versatile nicotinamide mimic allowing nanomolar inhibition of different PARP enzymes | 1-gen-2023 | Murthy, S.; Nizi, M. G.; Maksimainen, M. M.; Massari, S.; Alaviuhkola, J.; Lippok, B. E.; Vagaggini, C.; Sowa, S. T.; Galera-Prat, A.; Ashok, Y.; Venkannagari, H.; Prunskaite-Hyyrylainen, R.; Dreassi, E.; Luscher, B.; Korn, P.; Tabarrini, O.; Lehtio, L. | - | |
Tenebrio molitor as a Simple and Cheap Preclinical Pharmacokinetic and Toxicity Model | 1-gen-2023 | Brai, Annalaura; Poggialini, Federica; Vagaggini, Chiara; Pasqualini, Claudia; Simoni, Sauro; Francardi, Valeria; Dreassi, Elena | - |
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